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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • BGT1-IN-1
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    BGT1-IN-1

    CAS:
    BGT1-IN-1 (compound 9) is an effective inhibitor of BGT1, demonstrating IC50 values of 13.9 µM for hBGT1 and 58.3 µM for GAT3. It exhibits no cytotoxic effects and possesses neuroprotective activity.
    Formula:C6H9NO2
    Color and Shape:Solid
    Molecular weight:127.14

    Ref: TM-T200935

  • CFTR corrector 17
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    CFTR corrector 17

    CAS:
    CFTRcorrector 17 (example 17) is a regulator of the cystic fibrosis transmembrane conductance regulator (CFTR). It is utilized in the study of diseases mediated by CFTR.
    Formula:C18H15FN2O2
    Color and Shape:Solid
    Molecular weight:310.32

    Ref: TM-T201013

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    (R)-KMH-233

    CAS:
    <p>(R)-KMH-233 is an isomer of KMH-233, which can serve as a reference compound in experiments. KMH-233 functions as a potent, reversible, and selective inhibitor of L-type amino acid transporter 1 (LAT1), effectively hindering the uptake of LAT1 substrate, l-leucine (IC50=18 μM), and also inhibiting cell growth. Even at a low concentration of 25 μM, KMH-233 significantly enhances the efficacy of Bestatin and cisplatin.</p>
    Formula:C32H25N7O5
    Molecular weight:587.58

    Ref: TM-TYD-02664

  • EF1502 free base
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    EF1502 free base

    CAS:
    <p>EF1502 is a potent and selective GABA transporter inhibitor.</p>
    Formula:C22H26N2O2S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:414.58

    Ref: TM-T27241

  • Tamitinol
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    Tamitinol

    CAS:
    <p>Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.</p>
    Formula:C12H20N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:240.37

    Ref: TM-T24852

  • ZK 93426 hydrochloride
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    ZK 93426 hydrochloride

    CAS:
    <p>benzodiazepine receptor antagonist,competitive</p>
    Formula:C18H21ClN2O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:348.82

    Ref: TM-T23562

  • Leualacin
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    Leualacin

    CAS:
    <p>Leualacin is a novel calcium blocker from Hapsidospora irregularis.</p>
    Formula:C31H47N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.72

    Ref: TM-T25674

  • CAD204520
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    CAD204520

    CAS:
    <p>CAD204520 functions as an inhibitor of SERCA (IC50 = 0.34 μM), specifically targeting mutations in the wild-type NOTCH1 protein associated with T-cell acute lymphoblastic leukemia (T-ALL) and mantle cell lymphoma (MCL).</p>
    Formula:C23H32F3N3O2
    Color and Shape:Solid
    Molecular weight:439.51

    Ref: TM-T200097

  • Detajmium
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    Detajmium

    CAS:
    Detajmium is an anti-arrhythmia compound. It is an Na(+)-channel-blocking drug with an extremely long recovery from use-dependent sodium channel block.
    Formula:C27H42N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.64

    Ref: TM-T25312

  • AP-6
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    AP-6

    CAS:
    AP-6, a selective TMEM175 inhibitor, enhances lysosomal macromolecular catabolism by acutely inhibiting TMEM175, thus speeding up macrophage and other digestive activities. This compound holds potential for use in Parkinson's disease research due to its role in modulating lysosomal function.
    Formula:C16H14N4
    Color and Shape:Solid
    Molecular weight:262.31

    Ref: TM-T200356

  • AN-988
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    AN-988

    CAS:
    <p>AN-988 (compound 6) is a covalent CRM1 inhibitor.</p>
    Formula:C22H22N2O4S
    Color and Shape:Solid
    Molecular weight:410.49

    Ref: TM-T200424

  • Fletazepam
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    Fletazepam

    CAS:
    Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.
    Formula:C17H13ClF4N2
    Color and Shape:Solid
    Molecular weight:356.74

    Ref: TM-T201147

  • Butein tetramethyl ether
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    Butein tetramethyl ether

    CAS:
    <p>Butein tetramethyl ether (Compound 20) is a potent and selective inhibitor of breast cancer resistance protein / ATP-binding cassette sub-family G member 2 (BCRP/ABCG2). It inhibits MCF-7 MX and MDCKBCRP cells with IC50 values of 2.2 μM and 1.03 μM, respectively. Butein tetramethyl ether holds potential for cancer research.</p>
    Formula:C19H20O5
    Color and Shape:Solid
    Molecular weight:328.359

    Ref: TM-T204268

  • 3-Methoxy PCE hydrochloride
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    3-Methoxy PCE hydrochloride

    CAS:
    3-Methoxy PCE (3-MEO PCE) hydrochloride is an arylcyclohexylamine compound that functions as an NMDA receptor antagonist with a pKi value of 7.22.
    Formula:C15H24ClNO
    Color and Shape:Solid
    Molecular weight:269.81

    Ref: TM-T204329

  • Mibefradil dihydrochloride hydrate
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    Mibefradil dihydrochloride hydrate

    CAS:
    <p>Mibefradil dihydrochloride hydrate is a long-acting antihypertensive blocking high-voltage L calcium channels.</p>
    Formula:C29H42Cl2FN3O4
    Color and Shape:Solid
    Molecular weight:586.57

    Ref: TM-T64151

  • LY 235959
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    LY 235959

    CAS:
    <p>LY 235959 is a NMDA receptor antagonist.</p>
    Formula:C11H20NO5P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:277.25

    Ref: TM-T22944

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    CRM1 degrader 1

    <p>CRM1 degrader 1 (1l) is a low-toxic CRM1 degrader that induces apoptosis in gastric carcinoma and selectively inhibits the proliferation of gastric cancer[1].</p>
    Formula:C16H20O3
    Color and Shape:Solid
    Molecular weight:260.33

    Ref: TM-T60416

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    PF-06305591 dihydrate

    <p>PF-06305591 dihydrate is a potent and highly selective voltage gated sodium channel NaV1.8 blocker (IC 50 = 15 nM) with an excellent preclinical in vitro ADME</p>
    Formula:C15H26N4O3
    Color and Shape:Solid
    Molecular weight:310.39

    Ref: TM-T60761

  • Unoprostone
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    Unoprostone

    CAS:
    <p>Unoprostone is a prostaglandin F2α analogs (PGAs), and reduces intraocular pressure and is used topically for glaucoma or ocular hypertension.</p>
    Formula:C22H38O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:382.53

    Ref: TM-T13955

  • P2X4-IN-1
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    P2X4-IN-1

    CAS:
    <p>P2X4-IN-1 is an orally active P2X4 inhibitor. P2X4-IN-1 is applicable in research focused on disease prevention.</p>
    Formula:C18H14ClN5O3S
    Color and Shape:Solid
    Molecular weight:415.85

    Ref: TM-T207340