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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2280 products of "Membrane Transporter/Ion Channel"

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  • NYX-2925
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    NYX-2925

    CAS:
    <p>NYX-2925, an oral NMDAR modulator, enhances Src in mPFC. No CAMKII impact or addictive/sedative effects. Useful for CNS disorder studies.</p>
    Formula:C14H23N3O4
    Color and Shape:Solid
    Molecular weight:297.35

    Ref: TM-T73359

  • Opakalim
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    Opakalim

    CAS:
    <p>Opakalim is an activator of potassium channels (potassium channel) and exhibits anticonvulsant activity.</p>
    Formula:C18H22F2N4O
    Color and Shape:Solid
    Molecular weight:348.39

    Ref: TM-T206117

  • GABA-IN-4
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    GABA-IN-4

    CAS:
    <p>GABA-IN-4 (Compound 17) is a derivative of N-(indol-3-ylglyoxylyl)benzylamine. It exhibits high affinity for the benzodiazepine receptor (BzR), the binding site within the GABAA receptor complex, with a Ki value of 67 nM. Benzodiazepines are widely used as anxiolytic, sedative-hypnotic, and anticonvulsant agents.</p>
    Formula:C17H13ClN2O2
    Color and Shape:Solid
    Molecular weight:312.75

    Ref: TM-T205501

  • CRM1-IN-3
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    CRM1-IN-3

    CAS:
    <p>CRM1-IN-3 (B28), a noncovalent inhibitor of CRM1, is utilized in the research of protein localization and tumor studies [1].</p>
    Formula:C26H26ClN3O3
    Color and Shape:Solid
    Molecular weight:463.96

    Ref: TM-T86090

  • Suloctidil HCl
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    Suloctidil HCl

    CAS:
    <p>Suloctidil HCl is a peripheral vascular dilator.</p>
    Formula:C20H36ClNOS
    Color and Shape:Solid
    Molecular weight:374.02

    Ref: TM-T0712L

  • Sp-8-Br-cGMPS
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    Sp-8-Br-cGMPS

    CAS:
    <p>Sp-8-Br-cGMPS, an analogue of cGMP, acts as an agonist for cGMP gated cation channels (CNG channels) with an EC50 of 106.5 μM. While Sp-8-Br-cGMPS can induce currents, it does not stabilize channel open states as effectively as a full agonist.</p>
    Formula:C10H11BrN5O6PS
    Color and Shape:Solid
    Molecular weight:440.17

    Ref: TM-T88734

  • 3-Bromoamphetamine hydrochloride
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    3-Bromoamphetamine hydrochloride

    CAS:
    <p>3-Bromoamphetamine hydrochloride is a para-substituted amphetamine that functions as a monoamine releaser.</p>
    Formula:C9H13BrClN
    Color and Shape:Solid
    Molecular weight:250.563

    Ref: TM-T206868

  • (2S,3S,11bR)-Dihydrotetrabenazine
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    (2S,3S,11bR)-Dihydrotetrabenazine

    CAS:
    <p>(2S,3S,11bR)-Dihydrotetrabenazine ((2S,3S,11bR)-DHTBZ) is a highly selective inhibitor of vesicular monoamine transporter 2 (VMAT2) with a Ki value of 593 nM. It suppresses the vesicular transport of monoamine neurotransmitters, such as dopamine and serotonin, leading to reduced release into the synaptic cleft. This compound holds potential for research in Huntington's disease and other hyperkinetic movement disorders.</p>
    Formula:C19H29NO3
    Color and Shape:Solid
    Molecular weight:319.44

    Ref: TM-T207440

  • Zilvetrigine
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    Zilvetrigine

    CAS:
    <p>Zilvetrigine is a sodium channel (sodium channel) blocker. It can be used as an analgesic.</p>
    Formula:C20H20ClN3O2
    Color and Shape:Solid
    Molecular weight:369.845

    Ref: TM-T205304

  • NMDA agonist 1
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    NMDA agonist 1

    CAS:
    <p>NMDA agonist 1 (compound 42d) is a potent NMDA agonist with a Ki value of 96 nM. It acts as a partial agonist of the GluN1/GluN2B complex, exhibiting an EC50 value of 78 nM.</p>
    Formula:C12H13N3O3S
    Color and Shape:Solid
    Molecular weight:279.315

    Ref: TM-T204880

  • Tamitinol
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    Tamitinol

    CAS:
    <p>Tamitinol is a neurotropic drug. It has been found to help symptoms of obsessive rumination in conjunction with maprotiline.</p>
    Formula:C12H20N2OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:240.37

    Ref: TM-T24852

  • CymitQuimica logo
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    Cav 3.2 inhibitor 2

    <p>Cav 3.2 inhibitor 2 blocks T-type Ca2+ channels (IC50=0.09339 μM) and reduces mouse somatic/visceral pain. Used for intractable pain studies.</p>
    Formula:C32H37F2N3O
    Color and Shape:Solid
    Molecular weight:517.65

    Ref: TM-T63606

  • CymitQuimica logo
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    KCa2 channel modulator 2

    Compound 2q is a potent, subtype-selective K/Ca 2 modulator, effective on human K Ca 2.3 and rat K Ca 2.2a with EC50s of 0.60 μM and 0.64 μM.
    Formula:C16H15ClFN5
    Color and Shape:Solid
    Molecular weight:331.78

    Ref: TM-T60986

  • CymitQuimica logo
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    PDE1-IN-4

    <p>PDE1-IN-4: inhibits PDE1C/A/B with IC50s 10/145/354 nM, may help study idiopathic pulmonary fibrosis.</p>
    Formula:C33H33N3O4
    Color and Shape:Solid
    Molecular weight:535.63

    Ref: TM-T63776

  • CymitQuimica logo
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    GABAA receptor agonist 2

    <p>Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.</p>
    Formula:C22H36O5
    Color and Shape:Solid
    Molecular weight:380.52

    Ref: TM-T61625

  • YY-23
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    YY-23

    CAS:
    <p>YY-23 is a selective NMDAR (containing GluN2C or GluN2D) inhibitor. By inhibiting NMDARs with GluN2D on GABAergic interneurons in the prefrontal cortex, YY-23 suppresses GABAergic neurotransmission and enhances excitatory transmission. YY-23 exhibits antidepressant activity and is useful for neurological disease research.</p>
    Formula:C33H54O8
    Color and Shape:Solid
    Molecular weight:578.777

    Ref: TM-T206120

  • S-8510 phosphate
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    S-8510 phosphate

    CAS:
    <p>S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).</p>
    Formula:C12H13N4O6P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:340.23

    Ref: TM-T12792

  • Leualacin
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    Leualacin

    CAS:
    <p>Leualacin is a novel calcium blocker from Hapsidospora irregularis.</p>
    Formula:C31H47N3O7
    Purity:98%
    Color and Shape:Solid
    Molecular weight:573.72

    Ref: TM-T25674

  • Antidepressant agent 9
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    Antidepressant agent 9

    CAS:
    <p>Antidepressant agent 9 (Compound 24) is an orally active inhibitor of NMDAR and SERT, with IC50 values of 3.50 μM and 1044 nM, respectively. It exhibits good metabolic stability and plasma exposure, and demonstrates antidepressant-like effects in the forced swim test in mice.</p>
    Formula:C17H24N2
    Color and Shape:Solid
    Molecular weight:256.386

    Ref: TM-T205640

  • Suzetrigine
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    Suzetrigine

    CAS:
    <p>Suzetrigine (VX-548) is an oral NaV1.8 inhibitor with analgesic properties for acute pain research.</p>
    Formula:C21H20F5N3O4
    Purity:98.08% - 99.27%
    Color and Shape:Solid
    Molecular weight:473.39

    Ref: TM-T69552