Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(336 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2290 products of "Membrane Transporter/Ion Channel"
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Way 125971
CAS:<p>Way 125971 is a bioactive chemcial.</p>Formula:C22H28N4O5S2Color and Shape:SolidMolecular weight:492.61LY393615
<p>LY393615 (NCC1048) is a novel blocker of both neuronal Ca²⁺ (calcium) and Na⁺ (sodium) channels, exhibiting half-maximal inhibitory concentrations (IC₅₀) of 1.9</p>Purity:98%Color and Shape:Odour SolidA 80915A
CAS:<p>A80915A: Semi-naphthoquinone antibiotic, blocks gastric (H(+)-K+)-ATPase; potency varies with enzyme conformation; K+ reduces binding rate.</p>Formula:C26H31Cl3O5Color and Shape:SolidMolecular weight:529.88AZD-3161
CAS:<p>AZD-3161 is a sodium channel regulator for pain.</p>Formula:C23H21F3N4O4Color and Shape:SolidMolecular weight:474.43(R)-Funapide
CAS:<p>(R)-Funapide ((R)-TV 45070), the less active R-enantiomer of Funapide, acts as a potent Nav1.7 sodium channel blocker, primarily utilized in pain research [1].</p>Formula:C22H14F3NO5Color and Shape:SolidMolecular weight:429.35LY 274614
CAS:<p>LY 274614 is a structurally novel systemically active competitive NMDA receptor antagonist.</p>Formula:C11H20NO5PColor and Shape:SolidMolecular weight:277.25Chlorotoxin TFA
<p>Chlorotoxin TFA, a scorpion venom peptide, blocks chloride channels and has anti-cancer properties.</p>Formula:C160H250F3N53O49S11Color and Shape:SolidMolecular weight:4109.74APETx2 TFA
<p>APETx2 TFA from sea anemone is a selective ASIC3 inhibitor with a 63 nM IC50, reversing acid and inflammatory pain.</p>Formula:C198H281F3N54O62S6Color and Shape:SolidMolecular weight:4675.02sFTX-3.3
CAS:<p>sFTX-3.3 is a calcium ion channel antagonist, exhibiting IC50 values of approximately 0.24 mM and 0.70 mM against P-type and N-type channels respectively.</p>Formula:C12H29N7OColor and Shape:SolidMolecular weight:287.412NMDA receptor antagonist 2
CAS:<p>Potent, oral NR2B-selective NMDA receptor antagonist; IC50 of 1.0 nM, Ki of 0.88 nM; used for neuropathic pain and Parkinson's research.</p>Formula:C20H21N7OColor and Shape:SolidMolecular weight:375.436Lyso-Globotriaosylceramide (d18:1)
CAS:<p>Lyso-Gb3, lacking fatty acyl, binds Stx1 with cholesterol and phosphatidylcholine, not Stx2; lowers neutrophil viability; accumulates in Fabry disease.</p>Formula:C36H67NO17Color and Shape:SolidMolecular weight:785.922Lesogaberan napadisylate
CAS:<p>Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.</p>Formula:C13H17FNO5PSColor and Shape:SolidMolecular weight:349.31(Rac)-Tezacaftor
CAS:<p>(Rac)-Tezacaftor, a racemate, corrects F508del CFTR for cystic fibrosis research.</p>Formula:C26H27F3N2O6Color and Shape:SolidMolecular weight:520.5Mesoridazine free base
CAS:<p>Mesoridazine (thioridazine EP impurity B) is a phenothiazine antipsychotic with effects similar to chlorpromazine.</p>Formula:C21H26N2OS2Color and Shape:SolidMolecular weight:386.57NSC799462
<p>NSC799462, a triazole inhibitor, specifically targets p97 ATPase, exerting its effect by binding to a designated site on the p97 enzyme. This interaction induces localized structural alterations in p97, effectively inhibiting its ATPase activity with an IC 50 value of 15 nM.</p>Formula:C30H32F2N6O3SColor and Shape:SolidMolecular weight:594.68Aglafoline
CAS:Aglafoline inhibits in a concentration-dependent manner the aggregation and ATP release reaction induced in washed rabbit platelets by PAF (platelet-activatingFormula:C28H28O8Color and Shape:SolidMolecular weight:492.52Bendroflumethiazide
CAS:<p>Bendroflumethiazide (Naturetin) is a thiazide diuretic with actions and uses similar to those of HYDROCHLOROTHIAZIDE. It has been used in the treatment of familial hyperkalemia, hypertension, edema, and urinary tract disorders. (From Martindale, The Extra Pharmacopoeia, 30th ed, p810)</p>Formula:C15H14F3N3O4S2Purity:98% - >99.99%Color and Shape:Crystals From Dioxane SolidMolecular weight:421.41Venturicidin A
CAS:<p>Venturicidin A is a macrolide antibiotic.</p>Formula:C41H67NO11Purity:98%Color and Shape:SolidMolecular weight:749.97CALP3
CAS:<p>Cell-permeable CaM agonist, binds EF-hand, activates phosphodiesterase without Ca2+, inhibits Ca2+ toxicity, IC50=33μM.</p>Formula:C44H68N10O9Purity:98%Color and Shape:SolidMolecular weight:881.0812,14-Dichlorodehydroabietic acid
CAS:<p>12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.</p>Formula:C20H26Cl2O2Color and Shape:SolidMolecular weight:369.33
