CymitQuimica logo
Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

Show 13 more subcategories

Found 2290 products of "Membrane Transporter/Ion Channel"

Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • Cavα2δ-IN-1
    Targetmol
    + Info

    Cavα2δ-IN-1

    CAS:
    <p>Cavα2δ-IN-1 demonstrates exceptional specificity for voltage-gated calcium channels Cavα2δ-1 (with a Ki value of 6 nM), in comparison to Cavα2δ-2 (with a Ki</p>
    Formula:C18H27N5O
    Color and Shape:Solid
    Molecular weight:329.448

    Ref: TM-T40071

  • Pinacidil monohydrate
    Targetmol
    + Info

    Pinacidil monohydrate

    CAS:
    <p>Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.</p>
    Formula:C13H21N5O
    Purity:99.94% - 99.98%
    Color and Shape:Powder
    Molecular weight:263.34

    Ref: TM-T12478

  • CymitQuimica logo
    Targetmol
    + Info

    EVT-401

    <p>EVT-401 (P2X7 receptor antagonist-1), a purinergic P2X7 receptor antagonist, demonstrates efficacy in combating neuroinflammation [1].</p>
    Formula:C22H20F4N2O3
    Color and Shape:Solid
    Molecular weight:436.4

    Ref: TM-T74409

  • Emamectin B1a
    Targetmol
    + Info

    Emamectin B1a

    CAS:
    <p>Emamectin B1a can be used in relevant research in the life sciences. Its product number is T37663 and CAS number is 121124-29-6.</p>
    Formula:C49H75NO13
    Color and Shape:Solid
    Molecular weight:886.133

    Ref: TM-T37663

  • BeKm-1
    Targetmol
    + Info

    BeKm-1

    CAS:
    <p>Potent, selective hERG (KV11.1) blocker; doesn't affect 14 other K+ channels; extends QTc in rabbit heart dose-dependently.</p>
    Formula:C174H261N51O52S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:4091.65

    Ref: TM-TP2072

  • Carbonic anhydrase inhibitor 32
    Targetmol
    + Info

    Carbonic anhydrase inhibitor 32

    <p>Carbonic anhydrase inhibitor32 (compound 5B) is an orally active, selective inhibitor of hCA (carbonic anhydrase) II/VII, with Ki values of 6.3 nM for hCA II, 10.1 nM for hCA VII, and 681 nM for hCA I. It shows potential for neuroprotection and anticonvulsant effects by reducing mTOR activation and increasing hippocampal KCC2 levels.</p>
    Formula:C17H16N6O3S
    Color and Shape:Solid
    Molecular weight:384.41

    Ref: TM-T207684

  • CymitQuimica logo
    Targetmol
    + Info

    Huwentoxin I

    CAS:
    <p>Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.</p>
    Formula:C161H246N48O44S6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:3750.36

    Ref: TM-T80185

  • Conantokin G
    Targetmol
    + Info

    Conantokin G

    CAS:
    GluN2B-specific NMDA receptor blocker; IC50=480 nM in neurons, ~300 nM in oocytes; neuroprotective.
    Formula:C88H138N26O44
    Purity:98%
    Color and Shape:White Lyophilised Solid
    Molecular weight:2264.21

    Ref: TM-TP2060

  • CP-628006
    Targetmol
    + Info

    CP-628006

    CAS:
    <p>CP-628006 is a small molecule CFTR potentiator that effectively restores ATP-dependent channel gating to G551D-CFTR, the mutant form found in cystic fibrosis.</p>
    Formula:C32H35F3N2O2
    Color and Shape:Solid
    Molecular weight:536.639

    Ref: TM-T40386

  • FD 12-9
    Targetmol
    + Info

    FD 12-9

    CAS:
    FD 12-9, Anti-glioblastoma activity. is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively.
    Formula:C51H47N3O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:877.93

    Ref: TM-T11268

  • UK-59811 hydrochloride
    Targetmol
    + Info

    UK-59811 hydrochloride

    CAS:
    <p>UK-59811 hydrochloride, Br-dihydropyridine derivative, blocks Ca V Ab channels in bacteria, IC50: 194 nM.</p>
    Formula:C22H30BrClN2O5
    Color and Shape:Solid
    Molecular weight:517.85

    Ref: TM-T39770

  • NAADP tetrasodium salt
    Targetmol
    + Info

    NAADP tetrasodium salt

    CAS:
    <p>Ca2+ mobilizing agent</p>
    Formula:C21H27N6O18P3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:744.39

    Ref: TM-T23049

  • Chlorocresol
    Targetmol
    + Info

    Chlorocresol

    CAS:
    <p>Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.</p>
    Formula:C7H7ClO
    Color and Shape:Solid
    Molecular weight:142.58

    Ref: TM-T75311

  • L-R4W2
    Targetmol
    + Info

    L-R4W2

    CAS:
    <p>Vanilloid TRPV1 (VR1) receptor antagonist peptide (IC50 ~ 0.1 μM); blocks Ca2+ currents in dorsal root ganglion neurons. Analgesic in vivo.</p>
    Formula:C46H71N21O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1014.2

    Ref: TM-TP1934

  • CymitQuimica logo
    Targetmol
    + Info

    SLC6A8 corrector 1

    <p>SLC6A8 Corrector 1 is an orally active corrector for mutant SLC6A8 variants, capable of crossing the blood-brain barrier. It is utilized in the study of creatine transporter deficiency (CTD).</p>
    Formula:C21H25N3O2
    Color and Shape:Solid
    Molecular weight:351.44

    Ref: TM-T201220

  • Dofetilide N-oxide
    Targetmol
    + Info

    Dofetilide N-oxide

    CAS:
    Dofetilide N-oxide (UK-116856) is a metabolite of dofetilide. Dofetilide can block potassium channels and is a tertiary antiarrhythmic drug.
    Formula:C19H27N3O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:457.56

    Ref: TM-T11073

  • (±)17-HETE
    Targetmol
    + Info

    (±)17-HETE

    CAS:
    <p>Electrolyte and fluid transport in the kidney are regulated in part by arachidonic acid and its metabolites.</p>
    Formula:C20H32O3
    Color and Shape:Solid
    Molecular weight:320.473

    Ref: TM-T35523

  • CymitQuimica logo
    Targetmol
    + Info

    AQP4 (205-215) TFA

    <p>AQP4 (205-215) TFA is a fragment of the water channel protein-4 (AQP4). AQP4 acts as an autoimmune antigen in neuromyelitis optica, upregulating and presenting in B cells upon binding with CD40. AQP4 is associated with neuromyelitis optica (NMO), an autoimmune inflammatory disease of the central nervous system (CNS).</p>
    Color and Shape:Odour Solid

    Ref: TM-TP3237

  • N-hydroxy Riluzole
    Targetmol
    + Info

    N-hydroxy Riluzole

    CAS:
    <p>N-hydroxy Riluzole, a metabolite of riluzole, is mainly produced by CYP1A2 in human liver.</p>
    Formula:C8H5F3N2O2S
    Color and Shape:Solid
    Molecular weight:250.20

    Ref: TM-T35919

  • 8-Azido-ATP
    Targetmol
    + Info

    8-Azido-ATP

    CAS:
    <p>8-Azido-ATP is a nucleotide analog that demonstrates photo-reactivity properties.</p>
    Formula:C10H15N8O13P3
    Color and Shape:Solid
    Molecular weight:548.19

    Ref: TM-T40616