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Membrane Transporter/Ion Channel

Membrane Transporter/Ion Channel

Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.

Subcategories of "Membrane Transporter/Ion Channel"

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Found 2293 products of "Membrane Transporter/Ion Channel"

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  • Nav1.8-IN-1

    CAS:
    <p>Nav1.8-IN-1 (CHEMBL1270208) is an inhibitor of human NaV1.8</p>
    Formula:C20H15ClF3N3O2
    Purity:97.59%
    Color and Shape:Solid
    Molecular weight:421.8
  • SG-209

    CAS:
    <p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>
    Formula:C10H12N2O3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:208.21
  • 6-(4-Methoxyphenyl)-3-pyridazinamine

    CAS:
    <p>6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonist</p>
    Formula:C11H11N3O
    Purity:99.03%
    Color and Shape:Solid
    Molecular weight:201.22
  • Tulrampator

    CAS:
    Tulrampator (S-47445) is an orally bioavailable positive AMPAR with antidepressant effects.
    Formula:C20H17FN4O3
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:380.37
  • Acetoxyvalerensre

    CAS:
    <p>Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.</p>
    Formula:C17H24O4
    Purity:98.22%
    Color and Shape:Solid
    Molecular weight:292.37
  • Argireline

    CAS:
    <p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>
    Formula:C34H60N14O12S
    Purity:96.79% - 99.65%
    Color and Shape:White Powder
    Molecular weight:888.99
  • Vonoprazan fumarate

    CAS:
    <p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>
    Formula:C17H16FN3O2S·C4H4O4
    Purity:99.16% - 99.98%
    Color and Shape:Solid
    Molecular weight:461.46
  • (R)-baclofen

    CAS:
    <p>(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.</p>
    Formula:C10H12ClNO2
    Purity:97.20% - 98.94%
    Color and Shape:Solid
    Molecular weight:213.66
  • CL 218872

    CAS:
    <p>CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.</p>
    Formula:C13H9F3N4
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:278.23
  • AZ194

    CAS:
    <p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>
    Formula:C34H31F2N3O3
    Purity:99.61%
    Color and Shape:Solid
    Molecular weight:567.62
  • Revaprazan

    CAS:
    <p>Revaprazan: novel, K⁺-competitive acid blocker; reversibly halts gastric H⁺/K⁺-ATPase; rivals PPIs in acid reduction.</p>
    Formula:C22H23FN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.44
  • TGN-020

    CAS:
    <p>TGN-020 is an inhibitor of Aquaporin 4 (AQP4, IC50: 3.1 μM), the most abundant water channel in the brain.</p>
    Formula:C8H6N4OS
    Purity:99.54% - 99.99%
    Color and Shape:Solid
    Molecular weight:206.22
  • Ko 143

    CAS:
    <p>Ko 143 is a selective inhibitor of ATP-binding cassette sub-family G member 2 (ABCG2; BCRP).</p>
    Formula:C26H35N3O5
    Purity:99.01% - 99.89%
    Color and Shape:Solid
    Molecular weight:469.57
  • DHQ

    CAS:
    <p>DHQ (2,3-dihydroxy-quinoxalin) is an inducer of ATPase activity that of Herpes Simplex Virus thymidine kinase.</p>
    Formula:C8H6N2O2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:162.15
  • M8-B Hydrochloride

    CAS:
    <p>M8-B Hydrochloride is a selective transient receptor potential melastatin-8 (TRPM8) channel antagonist.</p>
    Formula:C22H25ClN2O3S
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:432.96
  • Rufinamide

    CAS:
    <p>Rufinamide (E 2080), a triazole derivative, is used as voltage-gated sodium channel blocker for the treatment of seizure disorders.</p>
    Formula:C10H8F2N4O
    Purity:99.77% - >99.99%
    Color and Shape:White Powder
    Molecular weight:238.19
  • Chloroprocaine hydrochloride

    CAS:
    Chloroprocaine hydrochloride (Chloroprocaine HCl) is a local anesthetic during surgical procedures.
    Formula:C13H20Cl2N2O2
    Purity:99.65%
    Color and Shape:White Crystalline Powder
    Molecular weight:307.22
  • AZD7325

    CAS:
    <p>AZD7325 (AZD-7325) is a GABA-Aα2,3 -selective receptor modulator.</p>
    Formula:C19H19FN4O2
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:354.38
  • DS-1971a

    CAS:
    <p>DS-1971a is a highly potent and selective NaV1.7 inhibitor. DS-1971a exhibits a favorable toxicological profile and analgesic effects.</p>
    Formula:C20H21ClFN5O3S
    Purity:99.66%
    Color and Shape:Solid
    Molecular weight:465.93
  • O4I2

    CAS:
    <p>O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.</p>
    Formula:C12H11ClN2O2S
    Purity:97.97% - 99.84%
    Color and Shape:Solid
    Molecular weight:282.75