Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(337 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2293 products of "Membrane Transporter/Ion Channel"
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HC067047 Hydrochloride(883031-03-6 free base)
CAS:HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.Formula:C26H29ClF3N3O2Purity:99.95%Color and Shape:SolidMolecular weight:507.98O4I2
CAS:<p>O4I2 is an effective Oct3/4 inducer in various human cell lines including human fibroblasts.</p>Formula:C12H11ClN2O2SPurity:97.97% - 99.84%Color and Shape:SolidMolecular weight:282.75A2793
CAS:<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Formula:C13H12ClNO3Purity:98.54%Color and Shape:SolidMolecular weight:265.69Dotinurad
CAS:Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).Formula:C14H9Cl2NO4SPurity:97.43% - 98.04%Color and Shape:SolidMolecular weight:358.2Lorediplon
CAS:<p>Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.</p>Formula:C20H15FN4O2SPurity:99.12% - 99.19%Color and Shape:SolidMolecular weight:394.42Parimifasor
CAS:<p>Parimifasor (LYC30937) is an immunomodulator, with anti-inflammatory activity.</p>Formula:C18H11Cl2F4N5OPurity:96.77% - 98.97%Color and Shape:SolidMolecular weight:460.21DL-Willardiine
CAS:<p>DL-Willardiine (2-amino-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)propanoic acid) is an unnatural amino acid, a derivative of glutamate.</p>Formula:C7H9N3O4Purity:99.83%Color and Shape:SolidMolecular weight:199.16Tirofiban hydrochloride monohydrate
CAS:<p>Tirofiban（MK383） hydrochloride monohydrate is a non-peptide glycoprotein IIb/IIIa antagonist. Cost-effective and quality-assured.</p>Formula:C22H39ClN2O6SPurity:98.81% - >99.99%Color and Shape:White SolidMolecular weight:495.07Vanillyl butyl ether
CAS:<p>Vanillyl butyl ether (Butyl vanillyl ether) (VBE)is a capsaicin analogue,induce sensory irritation in humans,Vanillyl butyl ether is an alkoxy-substituted</p>Formula:C12H18O3Purity:99.57%Color and Shape:Yellowish Liquid LiquidMolecular weight:210.27HC-056456
CAS:<p>HC-056456 (3,4-Bis(2-thienoyl)-1,2,5-oxadiazole-N-oxide) is a CatSper channel modulator.</p>Formula:C12H6N2O4S2Purity:99.62% - 99.65%Color and Shape:SolidMolecular weight:306.32Vonoprazan fumarate
CAS:<p>Vonoprazan fumarate (TAK-438) is a novel P-CAB (potassium-competitive acid blocker) that reversibly inhibits H+/K+, ATPase.</p>Formula:C17H16FN3O2S·C4H4O4Purity:99.16% - 99.98%Color and Shape:SolidMolecular weight:461.46Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Formula:C6H9NO4Purity:99.77%Color and Shape:SolidMolecular weight:159.14Azimilide Dihydrochloride
CAS:Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.Formula:C23H30Cl3N5O3Purity:97.59% - ≥95%Color and Shape:SolidMolecular weight:530.88Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Formula:C24H32NO6ClPurity:99.9%Color and Shape:SolidMolecular weight:465.97S107
CAS:<p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Formula:C11H15NOSPurity:99.90%Color and Shape:SolidMolecular weight:209.31L-Phenylalanine-15N
CAS:L-Phenylalanine-15N, essential amino acid, Ca+ channel and NMDARs antagonist, used in food flavors and pharmaceuticals.Formula:C9H11NO2Purity:98.98%Color and Shape:SolidMolecular weight:166.18QX-222 chloride
CAS:<p>QX-222 chloride (Lidocaine N-Methyl Hydrochloride) is a sodium channel blocker.</p>Formula:C13H21ClN2OPurity:97.37%Color and Shape:SolidMolecular weight:256.77SB-705498
CAS:<p>SB705498 is a TRPV1 antagonist for hTRPV1. SB-705498 has been investigated for the treatment of Rhinitis, Chronic Cough, and Non-allergic Rhinitis.</p>Formula:C17H16BrF3N4OPurity:99.57% - ≥95%Color and Shape:SolidMolecular weight:429.23Quadrol
CAS:<p>Quadrol (EDTP) is an immunostimulant, accelerated wound healing.</p>Formula:C14H32N2O4Purity:99.91% - 99.92%Color and Shape:Viscous Liquid Liquid ViscousMolecular weight:292.41(E)-KPT330
CAS:<p>(E)-RN (KPT 330) is a CRM1-selective inhibitor of nuclear export. (E)-RN inhibits protein trafficking from the nucleus and induces cell cycle arrest.</p>Formula:C17H11F6N7OPurity:98.69% - 99.49%Color and Shape:SolidMolecular weight:443.31L-DABA
CAS:<p>L-DABA (L-2,4-Diaminobutyric acid) is an inhibitor of GABA transaminase (IC50 > 500 μM).</p>Formula:C4H10N2O2Purity:99.32%Color and Shape:SolidMolecular weight:118.13AMG9810
CAS:<p>AMG 9810 blocks capsaicin's action on TRPV1; human IC50=24.5 nM, rat IC50=85.6 nM.</p>Formula:C21H23NO3Purity:99.79% - 99.95%Color and Shape:SolidMolecular weight:337.41Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Formula:C17H26ClNOPurity:99.80%Color and Shape:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TasteMolecular weight:295.85Mitiglinide calcium hydrate
CAS:<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Formula:C38H52CaN2O8Purity:98.97% - 99.96%Color and Shape:White SolidMolecular weight:704.91TCN 213
CAS:<p>TCN 213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over NR1/NR2B</p>Formula:C18H24N4OS2Purity:99.68%Color and Shape:SolidMolecular weight:376.54Flecainide acetate
CAS:<p>Flecainide acetate (R-818) is a class Ic antiarrhythmic agent used to prevent and treat tachyarrhythmias (abnormal fast rhythms of the heart).</p>Formula:C19H24F6N2O5Purity:99.42%Color and Shape:SolidMolecular weight:474.39Selamectin
CAS:<p>Selamectin (UK-124114) is a macrocyclic lactone derivative of ivermectin, an anthelmintic that potentiates glutamate- and GABA-gated chloride channel opening in</p>Formula:C43H63NO11Purity:99.84%Color and Shape:SolidMolecular weight:769.96DAAO inhibitor-1
CAS:<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Formula:C7H5FN2OPurity:97.84%Color and Shape:SolidMolecular weight:152.13Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formula:C34H60N14O12SPurity:96.79% - 99.65%Color and Shape:White PowderMolecular weight:888.99VK-II-36
CAS:<p>VK-II-36, a carvedilol analog, suppresses sarcoplasmic reticulum (SR) Ca(2+) release but does not block the β-receptor.</p>Formula:C26H26N2O5Purity:99.12%Color and Shape:SolidMolecular weight:446.49ICA-069673
CAS:<p>ICA-069673 is an activator of KCNQ2/Q3 potassium channel (IC50: 0.69 μM).</p>Formula:C11H6ClF2N3OPurity:99.04% - 99.68%Color and Shape:SolidMolecular weight:269.63ML133 hydrochloride
CAS:<p>ML133 hydrochloride (ML133 HCl) is a selective potassium channel inhibitor for Kir2.1, has no effect on Kir1.1 and weak activity for Kir4.1 and Kir7.1.</p>Formula:C19H19NO·HClPurity:99.48%Color and Shape:SolidMolecular weight:313.82TKIM
CAS:<p>TKIM is a TWIK-related potassium channel 1 (TREK-1) inhibitor, binding to the pocket of the intermediate (IM) state of TREK-1.</p>Formula:C18H14ClN3O2SPurity:99.47%Color and Shape:SolidMolecular weight:371.84SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Formula:C10H12N2O3Purity:99.84%Color and Shape:SolidMolecular weight:208.21Budipine
CAS:Budipine is a low affinity, N-methyl-D-aspartate receptor antagonist,is an antiparkinsonian agent.Formula:C21H27NPurity:99.64%Color and Shape:SolidMolecular weight:293.452'-O-Methylisoliquiritigenin
CAS:<p>2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-</p>Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28AER-271
CAS:<p>AER-271 is an inhibitor of aquaporin-4.</p>Formula:C15H9ClF6NO5PPurity:97.45%Color and Shape:SolidMolecular weight:463.65AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Formula:C34H31F2N3O3Purity:99.61%Color and Shape:SolidMolecular weight:567.62Ilaprazole sodium
CAS:<p>Ilaprazole sodium (IY-81149 sodium) , a substituted benzimidazole prodrug, is a selective and irreversible proton pump inhibitor.</p>Formula:C19H17N4NaO2SPurity:99.06%Color and Shape:SolidMolecular weight:388.42Tariquidar dihydrochloride
CAS:Tariquidar dihydrochloride, also known as XR9576 dihydrochloride, is a potent, specific P-glycoprotein (P-gp) inhibitor exhibiting high affinity (Kd = 5.1 nM).Formula:C38H40Cl2N4O6Color and Shape:SolidMolecular weight:719.65Trofinetide
CAS:Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.Formula:C13H21N3O6Purity:98.70% - 99.50%Color and Shape:SolidMolecular weight:315.32YHO-13351
CAS:YHO-13351 is an ABCG2 inhibitor that induces sensitization of cancer stem cells/initiating-like side population cells to irinotecan.Formula:C27H37N3O7S2Purity:97.88%Color and Shape:SolidMolecular weight:579.73Rimeporide hydrochloride
CAS:<p>Rimeporide hydrochloride (EMD-87580 hydrochloride) is a potent and selective Sodium hydrogen exchange 1 (NHE-1) inhibitor.</p>Formula:C11H16ClN3O5S2Purity:99.82%Color and Shape:SolidMolecular weight:369.84Verinurad
CAS:<p>Verinurad (RDEA3170) (RDEA3170) is an organic anion transporter URAT1 (SLC22A12) inhibitor for the treatment of gout and hyperuricemia.</p>Formula:C20H16N2O2SPurity:97.36% - 99.22%Color and Shape:SolidMolecular weight:348.42SN 2
CAS:<p>SN 2 is a novel and potent TRPML3 ion channel activator(EC50 = 1.13 μM). SN 2 also shares a similar antiviral effect against DENV2 and ZIKV.</p>Formula:C17H21NOPurity:99.86%Color and Shape:SolidMolecular weight:255.35Ocinaplon
CAS:<p>Ocinaplon (DOV 273547) is a GABAA receptors modulator.</p>Formula:C17H11N5OPurity:99.81%Color and Shape:SolidMolecular weight:301.3(-)-Blebbistatin
CAS:<p>(-)-Blebbistatin ((S)-(-)-Blebbistatin) is an S enantiomer of blebbistatin. It is a potent and selective myosin II inhibitor with IC50 ranging from 0.5 to 5 μM.</p>Formula:C18H16N2O2Purity:99.38% - 99.61%Color and Shape:SolidMolecular weight:292.33Metaflumizone
CAS:<p>Metaflumizone (BAS-320I) is a sodium channel blocker insecticide.</p>Formula:C24H16F6N4O2Purity:98.73%Color and Shape:SolidMolecular weight:506.40LY 303511 hydrochloride
CAS:<p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>Formula:C19H19ClN2O2Purity:98.47%Color and Shape:SolidMolecular weight:342.82NBI-98782
CAS:<p>NBI-98782 ((+)-α-DHTBZ) is an inhibtior of vesicular monoamine transporter (VMAT2) (Ki: 0.97 nM)</p>Formula:C19H29NO3Purity:99.29%Color and Shape:SolidMolecular weight:319.44
