Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(337 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2293 products of "Membrane Transporter/Ion Channel"
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S107
CAS:<p>S107 stabilizes RyR2 by improving calstabin2 binding to mutant/PKA-phosphorylated channels.</p>Formula:C11H15NOSPurity:99.90%Color and Shape:SolidMolecular weight:209.31Flupirtine
CAS:<p>Flupirtine(D 9998) is a selective neuronal potassium channel opener as well as shows properties of NMDA receptor antagonist.</p>Formula:C15H17FN4O2Color and Shape:SolidMolecular weight:304.32Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:<p>Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and dogs.</p>Formula:C24H32NO6ClPurity:99.9%Color and Shape:SolidMolecular weight:465.97Levamlodipine hydrochloride
CAS:<p>Levamlodipine hydrochloride is a medication used to lower blood pressure and prevent chest pain.</p>Formula:C20H26Cl2N2O5Color and Shape:SolidMolecular weight:445.34Cis-ACBD
CAS:<p>Cis-ACBD (cis-1-aminocyclobutane-1,3-dicarboxylic acid) is a potent and selective N-methyl-D-aspartate receptor agonist.</p>Formula:C6H9NO4Purity:99.77%Color and Shape:SolidMolecular weight:159.14A2793
CAS:<p>A2793 is a dual inhibitor of TWIK-associated acid-sensitive K+ channel 1 (TASK-1)/TRESK, with an IC50 for mTRESK of 6.8 μM.</p>Formula:C13H12ClNO3Purity:98.54%Color and Shape:SolidMolecular weight:265.69HC067047 Hydrochloride(883031-03-6 free base)
CAS:HC-067047 hydrochloride, a TRPV4 antagonist, selectively inhibits human, rat, and mouse currents with IC50s: 486 nM, 133 nM, and 17 nM.Formula:C26H29ClF3N3O2Purity:99.95%Color and Shape:SolidMolecular weight:507.98Esomeprazole
CAS:Esomeprazole is the S-isomer of omeprazole, inhibits the lysosomal cysteine protease legumain to prevent cancer metastasis.Formula:C17H19N3O3SPurity:97.3%Color and Shape:SolidMolecular weight:345.42Eperisone hydrochloride
CAS:<p>Eperisone is a skeletal muscle relaxant and a spasmolytic agent related structurally to Tolperisone.</p>Formula:C17H26ClNOPurity:99.80%Color and Shape:White Or Similar To White Crystalline Powder With Peculiar Smell And Bitter TasteMolecular weight:295.85Epaminurad
CAS:<p>Epaminurad (UR-1102) is an oral URAT1 inhibitor for gout research with a Ki of 0.057 μM, modestly affects OAT1/3.</p>Formula:C14H10Br2N2O3Color and Shape:SolidMolecular weight:414.05ML335
CAS:<p>ML335 is a selective activator of TREK-1 and TREK-2.</p>Formula:C15H14Cl2N2O3SPurity:99.73% - 99.79%Color and Shape:SolidMolecular weight:373.25HC-030031
CAS:<p>HC-030031 (TOSLAB 829227) is a potent TRPA1 inhibitor, which antagonizes AITC- and formalin-evoked calcium influx with IC50s of 6.2 and 5.3 μM, respectively.</p>Formula:C18H21N5O3Purity:99.69% - ≥95%Color and Shape:SolidMolecular weight:355.39JNJ-26990990
CAS:"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."Formula:C9H10N2O2S2Purity:97.37%Color and Shape:SolidMolecular weight:242.32Mitiglinide calcium hydrate
CAS:<p>Mitiglinide calcium hydrate (S-21403 calcium hydrate) is a drug for the treatment of type 2 diabetes.</p>Formula:C38H52CaN2O8Purity:98.97% - 99.96%Color and Shape:White SolidMolecular weight:704.91Ipidacrine
CAS:Ipidacrine (NIK‐247) (NIK‐247) is an Antidementia AgentFormula:C12H16N2Purity:97.73% - 99.99%Color and Shape:SolidMolecular weight:188.27AZD-6280
CAS:<p>AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.</p>Formula:C20H22N4O3Purity:98.99%Color and Shape:SolidMolecular weight:366.41Licarbazepine
CAS:<p>Licarbazepine (10,11-hydroxy-10,11 Dihydrocarbamezer) is the pharmacologically active metabolite of oxcarbazepine, a drug indicated for the treatment of partial</p>Formula:C15H14N2O2Purity:99.11%Color and Shape:SolidMolecular weight:254.28Bicuculline
CAS:<p>Bicuculline, a plant-derived GABAA receptor antagonist, identified in 1932, reacts to light.</p>Formula:C20H17NO6Purity:98% - 99.99%Color and Shape:Light Yellow PowderMolecular weight:367.35Enflurane
CAS:Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.Formula:C3H2ClF5OPurity:99.64%Color and Shape:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As AnMolecular weight:184.49TRPM8 antagonist 2
CAS:<p>TRPM8 antagonist 2 is a potent and selective TRPM8 antagonist with an IC50 of 0.2 nM. TRPM8 antagonist 2 is used in the research of neuropathic pain syndromes.</p>Formula:C26H26N2O2Purity:98.1%Color and Shape:SolidMolecular weight:398.5N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride
CAS:<p>N4-benzyl-N2-methylquinazoline-2,4-diamine hydrochloride is an inhibitor of TRPC4.</p>Formula:C16H17ClN4Purity:99.25%Color and Shape:SolidMolecular weight:300.79Aptiganel hydrochloride
CAS:<p>Aptiganel hydrochloride（Cerestat） is the salt form of Aptiganel.Aptiganel is a non-competitive NMDA antagonist with neuroprotective effects used in the treatment of stroke and focal cerebral ischemia.</p>Formula:C20H22ClN3Purity:99.89%Color and Shape:SolidMolecular weight:339.86UBP710
CAS:<p>UBP710 is an effective and selective NMDA receptor modulator.</p>Formula:C18H14O2Purity:98.05%Color and Shape:SolidMolecular weight:262.3Tiagabine hydrochloride hydrate
CAS:<p>Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.</p>Formula:C20H28ClNO3S2Color and Shape:SolidMolecular weight:430.02SKF89976A hydrochloride
CAS:<p>SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) and</p>Formula:C22H26ClNO2Purity:98.02%Color and Shape:SolidMolecular weight:371.9DAAO inhibitor-1
CAS:<p>DAAO inhibitor-1 is a potent D-amino acid oxidase (DAAO) inhibitor (IC50: 0.12 μM).</p>Formula:C7H5FN2OPurity:97.84%Color and Shape:SolidMolecular weight:152.13Pipequaline hydrochloride
CAS:<p>Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.</p>Formula:C22H25ClN2Purity:99.46%Color and Shape:SolidMolecular weight:352.9Tezacaftor
CAS:<p>Tezacaftor (VX661) is a small molecule that can be used as a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR) gene function.</p>Formula:C26H27F3N2O6Purity:98.84% - >99.99%Color and Shape:SolidMolecular weight:520.5Memantine
CAS:Memantine treats moderate to severe Alzheimer's; it's an amantadine derivative blocking NMDA receptors.Formula:C12H21NPurity:≥98%Color and Shape:White PowderMolecular weight:179.3Trans-ACBD
CAS:<p>Trans-ACBD (Trans-1-aminocyclobutane-1,3-dicarboxylic acid) is an effective and specific N-methyl-D-aspartate receptor agonist.</p>Formula:C6H9NO4Purity:99.47%Color and Shape:SolidMolecular weight:159.14AZ194
CAS:<p>CRMP2-Ubc9-NaV1.7 inhibitor 194, is a CRMP2-Ubc9-NaV1.7 inhibitor.</p>Formula:C34H31F2N3O3Purity:99.61%Color and Shape:SolidMolecular weight:567.62AM92016
CAS:<p>AM92016 is a specific blocker of the time dependent delayed rectifier potassium current. AM92016 does not show any β-adrenoceptor blocking activity.</p>Formula:C26H30Cl2N2O6SColor and Shape:SolidMolecular weight:569.49SG-209
CAS:<p>SG 209 is an analog of nicorandil and acts as a K+ channel opener and nitrate-free coronary vasodilator.</p>Formula:C10H12N2O3Purity:99.84%Color and Shape:SolidMolecular weight:208.21Dotinurad
CAS:Dotinurad ((3,5-dichloro-4-hydroxyphenyl)(1,1-dioxidobenzo[d]thiazol-3(2H)-yl)methanone) is a potent agent of uricosuric (IC50: 3.6 μM for uric acid).Formula:C14H9Cl2NO4SPurity:97.43% - 98.04%Color and Shape:SolidMolecular weight:358.2(S)-(-)-5-Fluorowillardiine hydrochloride
CAS:<p>(S)-(-)-5-Fluorowillardiine hydrochloride is a potent and specific agonist of AMPAR.</p>Formula:C7H9ClFN3O4Color and Shape:SolidMolecular weight:253.62ML213
CAS:<p>ML213 (CID-3111211) is a selective activator of Kv7.2 (KCNQ2) and Kv7.4 (KCNQ4) channels, enhances Kv7.2 and Kv7.4 channels with EC50s of 230 and 510 nM,</p>Formula:C17H23NOPurity:>99.99%Color and Shape:SolidMolecular weight:257.37GNE-131
CAS:<p>GNE-131 is a potent and specific inhibitor of human sodium channel NaV1.7 (IC50: 3 nM).</p>Formula:C23H30N4O3SPurity:98.54% - 99.59%Color and Shape:SolidMolecular weight:442.57XEN907
CAS:<p>XEN907 is a novel spiro oxindole NaV1.7 blocker. XEN907 also inhibits hNaV1.7 (IC50: 3 nM).</p>Formula:C21H21NO4Purity:99.92%Color and Shape:SolidMolecular weight:351.4Trofinetide
CAS:Trofinetide (NNZ-2566) is a synthetic analog of the endogenous N-terminus tripeptide. It has been shown to be neuroprotective in animal models of brain injury.Formula:C13H21N3O6Purity:98.70% - 99.50%Color and Shape:SolidMolecular weight:315.32Esomeprazole magnesium salt
CAS:<p>Esomeprazole magnesium, an oral proton pump inhibitor, curbs gastric acid by blocking H+, K+-ATPase; used in treating GERD.</p>Formula:C17H21MgN3O3SColor and Shape:SolidMolecular weight:371.74Propafenone hydrochloride
CAS:<p>Propafenone hydrochloride (Arythmol8) is a classic anti-arrhythmic medication, which treats illnesses associated with rapid heartbeats such as atrial.</p>Formula:C21H27NO3·HClPurity:99.67%Color and Shape:White SolidMolecular weight:377.9Argireline
CAS:<p>Argireline (Acetyl hexapeptide-3) is a peptide that inhibits neurotransmitter release, reducing wrinkles.</p>Formula:C34H60N14O12SPurity:96.79% - 99.65%Color and Shape:White PowderMolecular weight:888.99ASP7663
CAS:ASP7663 is a TRPA1 Receptor Agonist and exhibiting an abdominal analgesic effect in vivo.Formula:C14H14FNO3Purity:98.61%Color and Shape:SolidMolecular weight:263.26KCNQ2/3 activator-1
CAS:<p>KCNQ2/3 activator-1 is a Kv7.2/Kv7.3 (KCNQ2/3) potassium channel activator.</p>Formula:C23H29FN2OPurity:99.16% - 99.47%Color and Shape:SolidMolecular weight:368.49PF 05089771
CAS:<p>PF 05089771 is a Selective inhibitor of Nav1.7 (IC50 = 11 nM) that interacts with the voltage-sensor domain of domain IV.</p>Formula:C18H12Cl2FN5O3S2Purity:99.03% - 99.42%Color and Shape:SolidMolecular weight:500.35Cinacalcet metabolite M4
CAS:<p>Cinacalcet metabolite M4 (Rarechem AL BW 1078) is a metabolite of Cinacalcet. Cinacalcet is an allosteric agonist of Ca receptor.</p>Formula:C10H12F3NPurity:97.13%Color and Shape:SolidMolecular weight:203.2Acecainide hydrochloride
CAS:<p>Acecainide hydrochloride (NAPA) is the major hepatic metabolite of procainamide.Cost-effective and quality-assured.</p>Formula:C15H24ClN3O2Purity:98.023% - 99.81%Color and Shape:SolidMolecular weight:313.83Tegoprazan
CAS:<p>Tegoprazan is an orally active, highly selective gastric H+/K+-ATPase inhibitor.Cost-effective and quality-assured.</p>Formula:C20H19F2N3O3Purity:98.22%Color and Shape:SolidMolecular weight:387.38Bisaramil
CAS:<p>Bisaramil is a new class I antiarrhythmic agent.</p>Formula:C17H23ClN2O2Color and Shape:SolidMolecular weight:322.83ML277
CAS:<p>ML277 (CID-53347902) was identified as a potent activator of KCNQ1 channels (EC(50)=260 nM).</p>Formula:C23H25N3O4S2Purity:99.35%Color and Shape:SolidMolecular weight:471.59
