Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(337 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2293 products of "Membrane Transporter/Ion Channel"
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Repaglinide D5
CAS:<p>Repaglinide D5 is deuterium labeled Repaglinide. Repaglinide is an insulin secretagogue for treatment type-2 diabetes mellitus.</p>Formula:C27H36N2O4Purity:98%Color and Shape:SolidMolecular weight:457.62Bumetanide-d5
CAS:Bumetanide D5 is a deuterium-labeled Bumetanide. Bumetanide is a Na+-K+-Cl- (NKCC1) inhibitor (IC50s: 0.68 and 4.0 μM for hNKCC1A and hNKCC2A).Formula:C17H20N2O5SPurity:98%Color and Shape:SolidMolecular weight:369.45Propafenone D7 hydrochloride
CAS:<p>Propafenone D7 hydrochloride is the deuterium labeled Propafenone, and is a classic anti-arrhythmic medication.</p>Formula:C21H28ClNO3Purity:98%Color and Shape:SolidMolecular weight:384.95Nifedipine-d6
CAS:<p>Nifedipine D6 is deuterium labeled nifedipine which is a potent blocker of calcium channel.</p>Formula:C17H18N2O6Purity:98%Color and Shape:SolidMolecular weight:352.37Methocarbamol D5
CAS:<p>Methocarbamol is a central muscle relaxant. Methocarbamol D5 is deuterium labeled Methocarbamol.</p>Formula:C11H15NO5Purity:98%Color and Shape:SolidMolecular weight:246.27MNI-caged-NMDA
CAS:<p>NMDA caged with the photosensitive 4-methoxy-7-nitroindolinyl group</p>Formula:C14H17N3O6Purity:98%Color and Shape:SolidMolecular weight:323.30A-317491 sodium salt hydrate
<p>A-317491 sodium salt hydrate is a non-nucleotide P2X3 and P2X2/3 receptor antagonist, which inhibits calcium flux mediated by the receptors.</p>Formula:C33H29NNaO9Purity:98%Color and Shape:SolidMolecular weight:606.57DL-AP7
CAS:<p>DL-AP7: competitive NMDA antagonist, anticonvulsant, inhibits NMDA convulsions, impairs mice learning.</p>Formula:C7H16NO5PPurity:98%Color and Shape:SolidMolecular weight:225.18N-Acetylglycyl-D-glutamic acid
CAS:<p>Excitatory peptide that induces seizures</p>Formula:C9H14N2O6Purity:98%Color and Shape:SolidMolecular weight:246.22S1647
CAS:S1647 is a dual inhibitor targeting both ASBT and SOAT. It is utilized in research focused on intrahepatic cholestasis, cholestatic pruritus, and constipation.Formula:C19H13Cl2N3O5SMolecular weight:466.30R-(-)-Niguldipine hydrochloride
CAS:<p>R-(-)-Niguldipine HCl: L-type Ca2+ blocker, K+ agonist, α1A antagonist; lowers blood pressure; weaker enantiomer.</p>Formula:C36H40ClN3O6Color and Shape:SolidMolecular weight:646.17Pradigastat
CAS:Pradigastat (LCQ-908) is a diacylglycerol acyltransferase 1 (DGAT1) inhibitor for the treatment of constipation and can be used in the study of obesityFormula:C25H24F3N3O2Purity:95.21% - 95.21%Color and Shape:SolidMolecular weight:455.47LY 303511
CAS:<p>LY303511, an inactive analogue of LY294002, is a mTOR inhibitor and no inhibition for PI3-K.</p>Formula:C19H18N2O2Purity:98%Color and Shape:SolidMolecular weight:306.36Tetradifon
CAS:<p>Tetradifon is a broad-spectrum organochlorine acaricide that inhibits mitochondrial OSCP, blocking energy production (IC50=4.5-27nmoL/mg) with oligomycin-like effects.</p>Formula:C12H6Cl4O2SPurity:99.84%Color and Shape:Yellowish Odorless OilMolecular weight:356.058-Pcpt-cGMP sodium
CAS:<p>8-Pcpt-cGMP sodium, with an EC50 of 0.5 μM, acts as an agonist for cyclic nucleotide-gated (CNG) channels and demonstrates effective membrane permeability. This compound is utilized in research focused on the role of CNG channels in visual and olfactory signal transduction.</p>Formula:C16H14ClN5NaO7PSColor and Shape:SolidMolecular weight:509.79ORM-10103
CAS:ORM-10103 is a novel potent and selective inhibitor of the Na+/Ca2+ exchanger (NCX).ORM-10103 inhibited NCX currents with estimated IC50 values of 55 and 67 nMFormula:C20H16N2O4Purity:99.9%Color and Shape:SolidMolecular weight:348.35FFN 511 hydrochloride
CAS:<p>FFN 511 hydrochloride is a fluorescent pseudo-neurotransmitter (FFNs) targeting VMA T2 that can be used to label baraminergic nerve endings.</p>Formula:C17H21ClN2O2Purity:99.83%Color and Shape:SoildMolecular weight:320.81Diphenidol
CAS:<p>Diphenidol, a muscarinic antagonist, is employed as an antivertigo and antiemetic agent.</p>Formula:C21H27NOColor and Shape:Needles From Petroleum Ether SolidMolecular weight:309.45IEM 1754 2HBr
CAS:<p>IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.</p>Formula:C16H30N2·2HBrPurity:99.71% - 99.72%Color and Shape:SolidMolecular weight:412.25Verapamil
CAS:<p>Verapamil (CP-16533-1), an oral calcium channel blocker, inhibits P-gp and CYP3A4, used for hypertension, arrhythmias, and angina research.</p>Formula:C27H38N2O4Purity:99.61% - 99.93%Color and Shape:OilMolecular weight:454.6Clopamide
CAS:<p>Clopamide (Brinaldix) is a piperidine and sulfamoylbenzamide-based diuretic with thiazide-like diuretic activity.</p>Formula:C14H20ClN3O3SPurity:99.71%Color and Shape:White To Yellowish Crystalline PowderMolecular weight:345.84Aprikalim
CAS:<p>Aprikalim opens KATP channels, protects the heart, and at high doses, dilates blood vessels.</p>Formula:C12H16N2OS2Purity:99.42% - 99.90%Color and Shape:SolidMolecular weight:268.4SCH 50911 hydrochloride
CAS:<p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>Formula:C8H16ClNO3Purity:98%Color and Shape:SolidMolecular weight:209.67PPNDS
CAS:<p>P2X1 receptor antagonist</p>Formula:C18H15N4NaO14PS2Purity:98%Color and Shape:SolidMolecular weight:629.42NO 711
CAS:<p>NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.</p>Formula:C21H22N2O3Purity:99.70%Color and Shape:SolidMolecular weight:350.41(±)-Homoproline Hydrochloride
CAS:<p>(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can Trust</p>Formula:C6H12ClNO2Purity:99.69%Color and Shape:SolidMolecular weight:165.62VU0405601
CAS:<p>VU0405601 is a hERG channel activator that protects against drug-induced cardiac arrhythmias.</p>Formula:C17H13BrN2O2Purity:99.16%Color and Shape:SolidMolecular weight:357.2JTV-519 hemifumarate
CAS:<p>JTV-519 hemifumarate: Ca2+ blocker, SERCA inhibitor, ryanodine receptor partial agonist; antiarrhythmic, cardioprotective.</p>Formula:C54H68N4O8S2Purity:98%Color and Shape:SolidMolecular weight:965.28HN37
CAS:<p>HN37, KCNQ2 activator (EC50=37 nM). Affordable Excellence: Reliable Quality You Can Trust</p>Formula:C20H21FN2O2Purity:99.27%Color and Shape:SolidMolecular weight:340.39ICA
CAS:ICA (N-[4-(2-Pyridinyl)-2-thiazolyl]-2-pyridinamine) is a SK channel inhibitor and exhibits antileishmanial activity (IC50: 2.1 µM).Formula:C13H10N4SPurity:99.68%Color and Shape:SolidMolecular weight:254.31Benzamil hydrochloride
CAS:<p>Benzamil hydrochloride is a specific and potent sodium channel (ENaC) blocker.</p>Formula:C13H15Cl2N7OPurity:98%Color and Shape:SolidMolecular weight:356.21V-9302
CAS:<p>V-9302 (V9302) is a competitive antagonist of transmembrane glutamine flux that selectively and potently targets the amino acid transporter ASCT2 (IC50: 9.6 uM</p>Formula:C34H38N2O4Purity:98% - 99.54%Color and Shape:SolidMolecular weight:538.68Nifekalant hydrochloride
CAS:Nifekalant hydrochloride is an IKr potassium channel blocker with an IC50 of 10 µM.Formula:C19H28ClN5O5Purity:99.91%Color and Shape:SolidMolecular weight:441.91CFTR corrector 9
CAS:<p>CFTR corrector 9 is a CF modulator used to research cystic fibrosis and related disorders.</p>Formula:C16H14N2O4Purity:98.24%Color and Shape:SolidMolecular weight:298.29L-4FPG
CAS:<p>L-4FPG is a Glycine derivative, inhibits the neutral amino acid transporters ASCT1 and ASCT2.</p>Formula:C8H8FNO2Purity:99.26%Color and Shape:SolidMolecular weight:169.15TRPC6-PAM-C20
CAS:<p>TRPC6-PAM-C20, a selective enhancer for TRPC6, boosts calcium in HEK cells and OAG-related platelet clumping, EC50: 2.37μM.</p>Formula:C22H21NO4Purity:98.16%Color and Shape:SolidMolecular weight:363.41CP-100356 hydrochloride
CAS:<p>CP-100356 hydrochloride is an MDR1 (P-gp) and BCRP inhibitor, a nucleotide-derived substrate analog that induces stomatal opening in the dark.</p>Formula:C31H37ClN4O6Purity:99.19%Color and Shape:SolidMolecular weight:597.1Nav1.7 inhibitor
CAS:<p>Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.</p>Formula:C15H11Cl3FNO4SPurity:97.52%Color and Shape:SolidMolecular weight:426.68CP-457920
CAS:<p>CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.</p>Formula:C18H17N3O3Purity:99.06% - 99.74%Color and Shape:SolidMolecular weight:323.35FSBA hydrochloride
CAS:<p>FSBA hydrochloride(5'-p-Fluorosulfonylbenzoyladenosine) is an ATP analogue serving as an affinity probe for the ATP site of Na/K-ATPase.</p>Formula:C17H17ClFN5O7SPurity:97.96%Color and Shape:SolidMolecular weight:489.86Sodium Channel inhibitor 2
CAS:<p>Sodium Channel inhibitor 2 is a blocker of sodium channel.</p>Formula:C26H25Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:466.4Cilobradine hydrochloride
CAS:<p>Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of neuronal Ih and related cardiac If channels.</p>Formula:C28H39ClN2O5Purity:98.40%Color and Shape:SolidMolecular weight:519.07TC-AQP1-1
CAS:TC-AQP1-1 blocks aquaporin 1; found via virtual screening; hinders water flux in Xenopus oocytes at low µM.Formula:C12H10O4Purity:97.59%Color and Shape:SolidMolecular weight:218.21Bamaluzole
CAS:<p>Bamaluzole is an agonist of GABA receptor.</p>Formula:C14H12ClN3OPurity:98%Color and Shape:SolidMolecular weight:273.72BK 129
CAS:BK 129 is a local anesthetic with relaxant properties. BK 129 inhibits Ca2+ entry into the smooth muscle cell and Ca2+ release from sarcoplasmic reticulum.Formula:C22H36N2O4Purity:98%Color and Shape:SolidMolecular weight:392.53Almokalant
CAS:<p>Almokalant: Class III antiarrhythmic, K+ channel blocker, inhibits Ikr current.</p>Formula:C18H28N2O3SPurity:98%Color and Shape:SolidMolecular weight:352.49V116517
CAS:<p>V-116517, a TRPV1 antagonist, is used potentially for the treatment of severe pain due to osteoarthritis and chronic pain due postherpetic neuralgia (PHN).</p>Formula:C19H18ClF3N4O3Color and Shape:SolidMolecular weight:442.82AMG8788
CAS:<p>AMG8788 is a selective, potent and orally active TRPM8 antagonist (IC50: 63.2 nM).</p>Formula:C23H18F4N2OColor and Shape:SolidMolecular weight:414.4JTV-519 fumarate
CAS:Ryanodine receptor (RyR) inhibitor; stabilizes RyR2 in a closed conformation. Exhibits antiarrhythmic and cardioprotective properties in vivo.Formula:C29H36N2O6SColor and Shape:SolidMolecular weight:540.67PD 122860
CAS:<p>PD 122860 is a dihydropyridine enhancing heart contractility, altering ECG, and relaxing aortic rings.</p>Formula:C23H20F3N3O4SPurity:98%Color and Shape:SolidMolecular weight:491.48
