Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(100 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(54 products)
- Calcium Channel(545 products)
- Chloride channel(53 products)
- GABA Receptor(369 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(283 products)
- Proton pump(41 products)
- SGLT(31 products)
- Sodium Channel(219 products)
- TRP/TRPV Channel(96 products)
Show 13 more subcategories
Found 2586 products of "Membrane Transporter/Ion Channel"
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Cavα2δ1&NET-IN-2
CAS:Cavα2δ1&NET-IN-2 .Formula:C22H26N6O2SColor and Shape:SolidMolecular weight:438.55Bliretrigine
CAS:Bliretrigine, a sodium channel blocker, effectively relieves pain [1] [2] [3].Formula:C20H24N4O2Color and Shape:SolidMolecular weight:352.43AJG-049 HCl
CAS:AJG-049 HCl is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).Formula:C27H31ClN2O2Color and Shape:SolidMolecular weight:451.01NNC052090
CAS:NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).Formula:C27H30N2O2Color and Shape:SolidMolecular weight:414.54A 784168
CAS:A-784168: potent, oral TRPV1 inhibitor with good CNS penetration.Formula:C19H15F6N3O3SColor and Shape:SolidMolecular weight:479.4Arachidonyl serotonin
CAS:Dual FAAH inhibitor/TRPV1 antagonistFormula:C30H42N2O2Purity:98%Color and Shape:SolidMolecular weight:462.67P-CAB agent 1
CAS:Compound B19, a P-CAB, inhibits H+/K+-ATPase with IC50 of 60.50 nM, useful in ARD research.Formula:C26H23FN4OColor and Shape:SolidMolecular weight:426.49UR-MB108
CAS:UR-MB108 is a potent and selective inhibitor of ABCG2 (BCRP), displaying an IC50 value of 79 nM, and exhibits stability in blood plasma.Formula:C40H38N6O4Color and Shape:SolidMolecular weight:666.77Cariporide Mesylate
CAS:Cariporide Mesylate is a selective inhibitor of the Na+/H+ exchanger isoform 1.Formula:C13H21N3O6S2Color and Shape:SolidMolecular weight:379.45U89232
CAS:U-89232 is an opener of the cardioselective KATP channel.Formula:C19H25N5O2Purity:98%Color and Shape:SolidMolecular weight:355.43TC-P 262
CAS:P2X3 and P2X2/3 receptor antagonistFormula:C14H18N4OPurity:98%Color and Shape:SolidMolecular weight:258.32Azimilide
CAS:class III anti-arrhythmic drugFormula:C23H28ClN5O3Purity:98%Color and Shape:SolidMolecular weight:457.95DDO-02001
CAS:DDO-02001 can be used in anti-arrhythmia research. DDO-02001 is a moderately potent inhibitor of Kv1.5 potassium channel with an IC50 value of 17.7 μM [1].Formula:C20H24N2O2Color and Shape:SolidMolecular weight:324.42ASIC-IN-1
CAS:ASIC-IN-1 is a potent inhibitor of acid-sensing ion channels, demonstrating an IC 50 value of less than 10 μM.Formula:C23H25N3O2Color and Shape:SolidMolecular weight:375.46Becampanel
CAS:Becampanel (AMP397) is the first competitive AMPA antagonist. Becampanel (AMP397) also is an antiepileptic agent.Formula:C10H11N4O7PPurity:98%Color and Shape:SolidMolecular weight:330.19MRK-623
CAS:MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.Formula:C20H17FN4OColor and Shape:SolidMolecular weight:348.37CAY10608
CAS:CAY10608 selectively blocks NR2B NMDA receptors (IC50 = 50 nM), is neuroprotective, and reduces brain infarct size in ischemia.Formula:C18H22Cl2N2O4SColor and Shape:SolidMolecular weight:433.356'-Iodoresiniferatoxin
CAS:TRPV1 (VR1) vanilloid receptor partial agonistFormula:C37H39IO9Purity:98%Color and Shape:SolidMolecular weight:754.6LUF7244
CAS:LUF7244 is a K v 11.1 channel modulator with anti-arrhythmia research potential, curbing early afterdepolarizations.Formula:C20H15ClN2O3Color and Shape:SolidMolecular weight:366.8PMPA (NMDA antagonist)
CAS:PMPA (NMDA antagonist) is a Competitive NMDA receptor antagonist.Formula:C6H13N2O5PPurity:98%Color and Shape:SolidMolecular weight:224.15piCRAC-1
CAS:piCRAC-1 is a powerful inhibitor of the photoinducible Ca2+ release-activated Ca2+ (CRAC) channel.Formula:C17H10F6N4Color and Shape:SolidMolecular weight:384.28RyRs activator 3
CAS:RyRs activator 3 (compound A4) serves as an insecticide highly effective against both the diamondback moths, M.Formula:C23H19BrCl2N6O3Purity:98%Color and Shape:SolidMolecular weight:578.25Ned-K
CAS:Ned-K blocks NAADP, reduces heart ischemia-reperfusion calcium waves.Formula:C31H31N5O3Color and Shape:SolidMolecular weight:521.61Relutrigine
CAS:Relutrigine, Oral sodium current inhibitor, suppresses sustained INa (SCN8A mutations), reduces neuronal excitability, for anticonvulsant therapy.Formula:C15H11F6N5O2Purity:99.68%Color and Shape:SolidMolecular weight:407.27Ref: TM-T69652
1mg260.00€5mg650.00€10mg1,009.00€25mg1,504.00€50mg1,963.00€100mg2,520.00€1mL*10mM (DMSO)583.00€(R)-(+)-HA-966
CAS:(R)-(+)-HA-966 ((+)-HA-966) is a partial agonist/antagonist of glycine site of the N-methyl-D-aspartate (NMDA) receptor complex. (R)-(+)-HA-966 selectively blocks the activation of the mesolimbic dopamine system by amphetamine, has the potential for neuroFormula:C4H8N2O2Color and Shape:White SolidMolecular weight:116.12Otaplimastat
CAS:SP-8203 is a reactive oxygen species inhibitor and superoxide dismutase stimulant.Formula:C28H34N6O5Purity:98%Color and Shape:SolidMolecular weight:534.61DL-AP5 Sodium salt
CAS:DL-AP5 Sodium salt is a NMDA receptor antagonist.Formula:C5H12NNaO5PPurity:98%Color and Shape:SolidMolecular weight:220.12Linopirdine dihydrochloride
CAS:KV7 (KCNQ) voltage-gated potassium channels blockerFormula:C26H22ClN3OPurity:98%Color and Shape:SolidMolecular weight:427.93TDN345
CAS:TDN345 is a antagonist of Ca2+, for the treatment of vascular and senile dementia including Alzheimer's disease.Formula:C28H34F2N2O2Purity:98%Color and Shape:SolidMolecular weight:468.58PK-THPP
CAS:PK-THPP is a channel blocker of TASK-3.Formula:C29H32N4O2Color and Shape:SolidMolecular weight:468.59MPX-007
CAS:MPX-007, a potent NMDA inhibitor, inhibits GluN2A-containing NMDA receptors expressed in HEK cells with IC50s of 27 nM.Formula:C18H17F2N5O3S2Color and Shape:SolidMolecular weight:453.49NS5818
CAS:NS5818 inhibits ClC.Formula:C23H19Cl2N7O2Purity:98%Color and Shape:SolidMolecular weight:496.35P-CAB agent 2
CAS:Potent P-CAB agent 2 blocks gastric acid secretion; H+/K+-ATPase IC50 <100 nM, hERG IC50 18.69 μM; non-toxic.Formula:C22H25FN2O4SColor and Shape:SolidMolecular weight:432.51RS 029
CAS:RS 029 is a nitroimidazole that has been exhibited to significantly inhibit (Na+K+) ATP-ase activity.Formula:C13H16N6O6Purity:98%Color and Shape:SolidMolecular weight:352.3CP 339818 hydrochloride
CAS:KV1.3 channel antagonistFormula:C21H25ClN2Purity:98%Color and Shape:SolidMolecular weight:340.89Vincanol
CAS:Vincanol is a potent voltage-gated Na+ channels blocker.Formula:C19H24N2OPurity:98%Color and Shape:SolidMolecular weight:296.41NS004
CAS:NS004 is a large-conductance K+ channel opener, it inhibits mitochondrial function in glioma cells.Formula:C14H8ClF3N2O2Purity:98%Color and Shape:SolidMolecular weight:328.67KCa2 channel modulator 1
CAS:Compound 2o, a selective K/Ca2 channel enhancer, boosts rat K Ca 2.2 (EC50: 0.99 μM) and human K Ca 2.3 (EC50: 0.19 μM).Formula:C16H15ClFN5Color and Shape:SolidMolecular weight:331.78Leconotide
CAS:Leconotide is a calcium channel blocker and antihyperalgesia agent; isolated from the venom of the cone snail, Conus catus.Formula:C107H179N35O36S7Color and Shape:SolidMolecular weight:2756.23TTA-P2
CAS:TTA-P2: potent CNS-penetrating T-type Ca2+ channel blocker; eliminates Cav3.1 window currents.Formula:C21H29Cl2FN2O2Color and Shape:SolidMolecular weight:431.37NAV26
CAS:NAV26 is a selective blocker of the Nav1.7 channel.Formula:C22H21F3N2O4Purity:98%Color and Shape:SolidMolecular weight:434.41GABAA receptor modulator-2
CAS:Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.Formula:C22H22FN3O5SColor and Shape:SolidMolecular weight:459.49ANO1-IN-2
CAS:ANO1-IN-2: potent ANO1 blocker (IC50: 1.75 μM), less effective on ANO2 (IC50: 7.43 μM), inhibits glioblastoma cell growth.Formula:C16H14ClN3O2S2Color and Shape:SolidMolecular weight:379.88BMS-284640
CAS:BMS-284640 is a NHE inhibitor that protects against MI in animal studies.Formula:C15H19N3O2Color and Shape:SolidMolecular weight:273.33Lanicemine
CAS:Lanicemine is a low-trapping NMDA channel blocker. It also has a binding (Ki: 0.56-2.1 μM).Formula:C13H14N2Purity:98%Color and Shape:SolidMolecular weight:198.26P2X2/3 modulator-1
CAS:Compound 46, a P2X2/3 modulator, could aid in research of pain, CNS disorders, and inflammation.Formula:C26H21N5OColor and Shape:SolidMolecular weight:419.48UTA1inh-C1
CAS:UTA1inh-C1 is a novel inhibitor of kidney urea transporter UT-A1.Formula:C22H24N6O4S2Color and Shape:SolidMolecular weight:500.59TRPC6-IN-3
CAS:TRPC6-IN-3 is an oral TRPC6 ion channel inhibitor, regulating calcium levels and membrane potential.Formula:C22H22FN5O3Color and Shape:SolidMolecular weight:423.44KR-30450
CAS:KR-30450, a potassium channel agonist, is used potentially for the treatment of hypertension.Formula:C17H18N2O6Color and Shape:SolidMolecular weight:346.33Taquidil
CAS:Tocainide hydrochloride: oral antiarrhythmic, sodium channel blocker, akin to lidocaine.Formula:C11H17ClN2OColor and Shape:SolidMolecular weight:228.718
