Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(100 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(54 products)
- Calcium Channel(545 products)
- Chloride channel(53 products)
- GABA Receptor(369 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(283 products)
- Proton pump(41 products)
- SGLT(31 products)
- Sodium Channel(219 products)
- TRP/TRPV Channel(96 products)
Show 13 more subcategories
Found 2586 products of "Membrane Transporter/Ion Channel"
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P-gp inhibitor 4
CAS:P-gp inhibitor 4 is a selective P-glycoprotein modulator with an EC 50 of 94 nM.Formula:C38H38N2O8S2Color and Shape:SolidMolecular weight:714.85NMDA-IN-2
CAS:NMDA-IN-2 (compound 6b) is a Procaine derivative that is an inhibitor of NMDA receptor 2B subtype [1].Formula:C15H22N2O3Color and Shape:SolidMolecular weight:278.35PD-307243
CAS:PD-307243 is an activator of hERG channel.Formula:C20H15Cl2N3O2Color and Shape:SolidMolecular weight:400.26RQ-00311651
CAS:RQ-00311651 is a novel T-type Ca2+ channel blocker. RQ-00311651 also inhibited high K-induced Ca signaling in those cells.Formula:C19H18F3N5O2Color and Shape:SolidMolecular weight:405.37DDO-02005
CAS:DDO-02005, a Kv1.5 inhibitor (IC50: 0.72 μM), counters fibrillation and arrhythmias in rats.Formula:C21H27Cl2N3O2Color and Shape:SolidMolecular weight:424.37(±)-C3001a
CAS:(RS)-C3001a is the racemic mixture of C3001a (CAS: 2415154-29-7). C3001a is a selective activator of the TREK channel.Formula:C21H20N2O3SPurity:99.13%Color and Shape:SolidMolecular weight:380.46TRPC3/6-IN-1
CAS:TRPC3/6-IN-1 selectively inhibits hTRPC3/6 with IC50 of 1260/500 nM, useful in heart failure research.Formula:C20H19N3O2SColor and Shape:SolidMolecular weight:365.45Ivacaftor-D9
CAS:CTP-656, a cystic fibrosis transmembrane conductance regulator (CFTR) channel activator, is used potentially for the treatment of cystic fibrosis.Formula:C24H19D9N2O3Color and Shape:SolidMolecular weight:401.55RG100204
CAS:RG100204 is an orally active AQP9 inhibitor with anti-inflammatory properties. It alleviates cardiac dysfunction (systolic and diastolic) induced by sepsis, improves renal dysfunction, and reduces the elevation of the cellular damage marker LDH.Formula:C20H26N6O2S2Color and Shape:SolidMolecular weight:446.59P-gp inhibitor 17
CAS:P-gp Inhibitor 17 (compound 2g), a potent inhibitor, directly interacts with the transmembrane domain of P-gp. This compound is useful for studying P-gp-mediated multidrug resistance in tumor cells [1].Formula:C36H49N3O3Color and Shape:SolidMolecular weight:571.79CW0134
CAS:CW0134 (Compound 12) serves as a modulator for exportin1 (XPO1), disrupting chromatin binding and inhibiting NFAT transcription factors and T cell activation [1].Formula:C11H7ClF3N3O2Color and Shape:SolidMolecular weight:305.64DPI 201-106
CAS:DPI 201-106: cardioselective h1 Na channel inhibitor, enhances heart contraction, blocks potassium and calcium currents.Formula:C29H30N4O2Purity:99.94%Color and Shape:SolidMolecular weight:466.57(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Formula:C6H11NO2Purity:99.38%Color and Shape:SolidMolecular weight:129.16Anxiolytic/nonsedative agent-1
CAS:TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.Formula:C18H15N3O4Purity:98.61%Color and Shape:SolidMolecular weight:337.33Ref: TM-T23445
1mg64.00€2mg96.00€5mg115.00€10mg150.00€25mg330.00€50mg472.00€100mg655.00€500mg1,293.00€(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Formula:C30H35NO6Purity:98.20%Color and Shape:SolidMolecular weight:505.6Ref: TM-T16831
5mg52.00€10mg78.00€25mg160.00€50mg225.00€100mg325.00€200mg445.00€1mL*10mM (DMSO)51.00€Psora 4
CAS:Psora 4 (5-(4-Phenylbutoxy)psoralen) is a Kv1.3 blocker and a caloric restriction mimetic.Formula:C21H18O4Color and Shape:SolidMolecular weight:334.373α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Formula:C21H34O3Purity:98.00%Color and Shape:SolidMolecular weight:334.49AVE-0118
CAS:AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.Formula:C30H29N3O3Purity:97.04% - 98.93%Color and Shape:SolidMolecular weight:479.57Ref: TM-T26689
1mg70.00€5mg132.00€10mg173.00€25mg304.00€50mg449.00€100mg652.00€500mg1,369.00€1mL*10mM (DMSO)159.00€L589-420
CAS:L589-420 is a sodium pump inhibitor in human erythrocytes.Formula:C14H14Cl2O4Purity:98%Color and Shape:SolidMolecular weight:317.16YM928
CAS:YM928 is an orally active antagonist of the AMPA receptor.Formula:C14H10ClN3OSPurity:98%Color and Shape:SolidMolecular weight:303.77CCMQ
CAS:inhibits [3H]-homoquinolinic acid binding to non-NMDA sensitive sitesFormula:C12H9NO4Purity:98%Color and Shape:SolidMolecular weight:231.2Bms 188107
CAS:Bms 188107 is a calcium antagonist, it has cardioprotective effects.Formula:C25H26N2O4Purity:98%Color and Shape:SolidMolecular weight:418.48Caramiphen
CAS:Caramiphen is an antimuscarinic and anticholinergic agent that acts as an antagonist of the NMDA receptor.Formula:C18H27NO2Purity:98%Color and Shape:SolidMolecular weight:289.41Viquidil
CAS:Viquidil is an agent with the activity of a vasodilator.Formula:C20H24N2O2Purity:98%Color and Shape:SolidMolecular weight:324.42(R)-Licarbazepine Acetate
CAS:(R)-Licarbazepine Acetate is a hopeful antiepileptic drug structurally related to Carbamazepine and Oxcarbazepine.Formula:C17H16N2O3Color and Shape:SolidMolecular weight:296.32COR628
CAS:COR628 is the GABA(B) receptor positive allosteric modulator.Formula:C16H23NO3SColor and Shape:SolidMolecular weight:309.42AZD 2066
CAS:AZD 2066 is a selective, orally active, and brain-penetrant mGluR5 antagonist with analgesic activity.Formula:C19H16ClN5O2Purity:98%Color and Shape:SolidMolecular weight:381.82BBR 2160
CAS:BBR 2160: a calcium-antagonist dihydropyridine derivative, reduces heart tissue contractility and shortens action potentials.Formula:C21H25N3O7SColor and Shape:SolidMolecular weight:463.5LY-395153
CAS:LY-395153 is a novel potentiator of AMPA receptor.Formula:C19H24N2O3SColor and Shape:SolidMolecular weight:360.47Tolperisone free base
CAS:Tolperisone free base, a centrally acting muscle relaxant, has been used for the symptomatic treatment of spasticity and muscle spasm.Formula:C16H23NOPurity:98%Color and Shape:SolidMolecular weight:245.36Lercanidipine, (S)-
CAS:(S)-Lercanidipine: a dihydropyridine calcium blocker with prolonged antihypertensive and kidney-protective properties.Formula:C36H41N3O6Purity:98%Color and Shape:SolidMolecular weight:611.73Ensaculin HCl
CAS:Ensaculin: NMDA antagonist, 5HT1A agonist, may treat Alzheimer's, enhances memory, neuroprotective, binds multiple receptors.Formula:C26H33ClN2O5Purity:98%Color and Shape:SolidMolecular weight:489Naftazone
CAS:Naftazone: vasoprotectant for hemostasis; boosts vein cell growth in vitro without affecting clotting.Formula:C11H9N3O2Purity:98%Color and Shape:SolidMolecular weight:215.21Tiropramide
CAS:Tiropramide is an antispasmodic drug. It also useful to inhibit the contractile response of the urinary bladder and in managing abdominal pain in IBS.Formula:C28H41N3O3Purity:98%Color and Shape:SolidMolecular weight:467.64Riodipine
CAS:Riodipine, a calcium channel blocker, is used as cardiovascular drugs.Formula:C18H19F2NO5Purity:98%Color and Shape:SolidMolecular weight:367.34DS28120313
CAS:DS28120313 is an oral inhibitor of hepcidin production (IC50: 0.093 μM).Formula:C16H17N5O2Color and Shape:SolidMolecular weight:311.34CPP-115
CAS:CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.Formula:C7H9F2NO2Color and Shape:SolidMolecular weight:177.15Ethopropazine Hydrochloride
CAS:Ethopropazine Hydrochloride is the salt form of Profenamine，anticholinergic, antihistamine, and anti-adrenergic，Parkinson's disease,an AChE inhibitorFormula:C19H25ClN2SPurity:98.25%Color and Shape:SolidMolecular weight:348.93DHP-218
CAS:DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) & 66 nmol/L (phenylephrine).Formula:C18H21N2O7PPurity:98%Color and Shape:SolidMolecular weight:408.34BCTP
CAS:BCTP is a polymodal inhibitor of TRPV1. It has a reduced liability for hyperthermia.Formula:C17H16ClN3OSPurity:98%Color and Shape:SolidMolecular weight:345.85Chlormethiazole edisylate
CAS:Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.Formula:C8H14ClNO6S3Purity:98%Color and Shape:SolidMolecular weight:351.85Talopram hydrochloride
CAS:noradrenalin transporter (NET) inhibitorFormula:C20H26ClNOPurity:98%Color and Shape:SolidMolecular weight:331.88IAA-94
CAS:IAA-94 is an inhibitor of chloride channels, it binds channels in bovine kidney cortex microsomes with a Ki value of 1 µM.Formula:C17H18Cl2O4Color and Shape:SolidMolecular weight:357.23A 39355
CAS:A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.Formula:C28H39Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:504.54UBP512
CAS:UBP512 is a NMDA receptor modulator.Formula:C15H9IO2Purity:98%Color and Shape:SolidMolecular weight:348.14Ronipamil
CAS:Ronipamil is an analogue of verapamil that used as a calcium entry blocker.Formula:C32H48N2Color and Shape:SolidMolecular weight:460.74L 644711
CAS:L 644711 is an antagonist of HCO3(-)/Cl(-) antiporter.Formula:C18H18Cl2O4Color and Shape:SolidMolecular weight:369.24N12N
CAS:N12N is a polyamine inverse NMDA receptor agonist.Formula:C12H28N2Purity:98%Color and Shape:White SolidMolecular weight:200.36Bromotetrandrine
CAS:Bromotetrandrine enhances chemo by inhibiting P-glycoprotein, countering efflux pumps.Formula:C38H41BrN2O6Color and Shape:SolidMolecular weight:701.65Tedisamil
CAS:Tedisamil blocks cardiac K+ currents, slows heart rate, is a class III antiarrhythmic, and treats angina.Formula:C19H32N2Purity:98%Color and Shape:SolidMolecular weight:288.47
