Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(93 products)
- Adiponectin receptor(5 products)
- CFTR(64 products)
- CGRP Receptor(52 products)
- Calcium Channel(496 products)
- Chloride channel(49 products)
- GABA Receptor(337 products)
- Monoamine Transporter(23 products)
- Monocarboxylate transporter(17 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(8 products)
- OAT(27 products)
- OCT(7 products)
- P-gp(53 products)
- Potassium Channel(277 products)
- Proton pump(39 products)
- SGLT(30 products)
- Sodium Channel(202 products)
- TRP/TRPV Channel(93 products)
Show 13 more subcategories
Found 2293 products of "Membrane Transporter/Ion Channel"
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XE991
CAS:<p>XE991 is a Kv7 (KCNQ) channel blocker.XE 991 dihydrochloride inhibits Kv7.1 (KCNQ1) and M-current and can be used in the study of neurological disorders.</p>Formula:C26H20N2OPurity:98.87%Color and Shape:SolidMolecular weight:376.45Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purity:99.90% - 99.99%Color and Shape:SolidMolecular weight:329.48TWIK-1/TREK-1-IN-3
CAS:<p>TWIK-1/TREK-1-IN-3 is a potassium channel TREK-1 inhibitor TWIK-1/TREK-1-IN-3 has antidepressant activity and can be used to study depression.</p>Formula:C19H27F3N2O2Purity:99.04%Color and Shape:SolidMolecular weight:372.43WY-47766
CAS:<p>WY-47766, a proton pump inhibitor, is used potentially for the treatment of postmenopausal osteoporosis.</p>Formula:C14H13N3O2SPurity:97.63% - 99.83%Color and Shape:SolidMolecular weight:287.34VU 0240551
CAS:VU 0240551 is a selective antagonist of neuronal K-Cl cotransporter KCC2 inhibitor with an IC50 of 560 nM. VU 0240551 inhibits L-type calcium channels and hERG.Formula:C16H14N4OS2Purity:99.9%Color and Shape:SolidMolecular weight:342.44DMCM hydrochloride
CAS:<p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>Formula:C17H19ClN2O4Purity:99.56%Color and Shape:SolidMolecular weight:350.8UCCF-853
CAS:<p>UCCF-853 是一种小分子 CFTR 调节剂，可用于研究囊性纤维化。</p>Formula:C14H8ClF3N2OPurity:99.82%Color and Shape:SolidMolecular weight:312.67FR183998 free base
CAS:<p>FR183998 free base is an inhibitor of Na+/Ca2+ Exchanger.</p>Formula:C17H19Cl2N5O2SPurity:99.61%Color and Shape:SolidMolecular weight:428.34NS-2710
CAS:<p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>Formula:C22H20N4OPurity:99.7% - 99.82%Color and Shape:SolidMolecular weight:356.42Sarmazenil
CAS:<p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>Formula:C15H14ClN3O3Purity:99.46%Color and Shape:SolidMolecular weight:319.74R(+)-IAA-94
CAS:<p>R(+)-IAA-94 (Methylindazone) blocks epithelial chloride channels; inhibits Nef-sdAb19 binding.</p>Formula:C17H18Cl2O4Purity:98.95% - 99.17%Color and Shape:SolidMolecular weight:357.23TC-N 1752
CAS:TC-N 1752 is an orally active inhibitor of Nav1.7 channel with IC50 of 0.17 μM. TC-N 1752 shows analgesic activities.Formula:C25H27F3N6O3Purity:99.71%Color and Shape:SolidMolecular weight:516.52Olvanil
CAS:<p>Olvanil (N-Vannilyloleoylamide) is a vanilloid receptor agonist with EC50 of 0.7nM.</p>Formula:C26H43NO3Purity:99.58%Color and Shape:SolidMolecular weight:417.62Ro 25-6981
CAS:<p>Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), useful in Parkinson's research.</p>Formula:C22H29NO2Purity:99.88%Color and Shape:SolidMolecular weight:339.47VRT-532
CAS:<p>VRT-532 (CFpot-532) is an effective modulator of CFTR and is commonly used in studies of cystic fibrosis (CF) caused by CFTR defects.</p>Formula:C16H14N2OPurity:99.88% - 99.93%Color and Shape:SolidMolecular weight:250.3CFTR corrector 8
CAS:<p>CFTR corrector 8: potent for cystic fibrosis research, modulates CFTR protein.</p>Formula:C29H27F2NO7Purity:99.57%Color and Shape:SolidMolecular weight:539.52Mavatrep
CAS:<p>Mavatrep (JNJ-39439335) is a selective antagonist of TRPV1 with Ki of 6.5 nM and can be used for studies about inflammatory pain.</p>Formula:C25H21F3N2OPurity:98.51% - 99.31%Color and Shape:SolidMolecular weight:422.44Dasolampanel
CAS:Dasolampanel (NGX-426) is an ionotropic glutamate receptor AMPA and Kainate receptor antagonist for the study of chronic pain disorders.Formula:C17H20ClN5O3Purity:98.70%Color and Shape:SolidMolecular weight:377.83Saripidem
CAS:<p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>Formula:C19H20ClN3OPurity:99.45%Color and Shape:SolidMolecular weight:341.83Butibufen
CAS:Butibufen (FF-106) is a non-steroidal anti-inflammatory compound and LOX inhibitor with analgesic and antipyretic activity for the study of rheumatic diseases.Formula:C14H20O2Purity:98.11% - 98.91%Color and Shape:SolidMolecular weight:220.31UCL 2077
CAS:<p>UCL 2077 blocks KCNQ channels, related to epilepsy, and selective slow-afterhyperpolarization channels, with 500 nM IC50, sparing Ca2+ channels.</p>Formula:C25H22N2Purity:99.58%Color and Shape:SolidMolecular weight:350.46MSP3
CAS:<p>MSP3 is an agonist of TRPV1 (EC50 = 0.87 μM) and shows antinociceptive and neuroprotective effects.</p>Formula:C16H19NO3SPurity:99.89%Color and Shape:SolidMolecular weight:305.39Nelonemdaz
CAS:Nelonemdaz (Neu2000) is an NMDA receptor antagonist with antioxidant activity that can be used to study cerebral infarction reperfusion injury.Formula:C15H8F7NO3Purity:99.52%Color and Shape:SolidMolecular weight:383.22ELB-139
CAS:<p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>Formula:C14H16ClN3OPurity:>99.99%Color and Shape:SolidMolecular weight:277.75GNE-8324
CAS:<p>GNE-8324 is a GluN2A selective positive allosteric modulator that enhances NMDAR-mediated synaptic responses in inhibitory, but not excitatory, neurons.</p>Formula:C18H18FN3OSPurity:98.68% - 99.34%Color and Shape:SolidMolecular weight:343.42Enecadin
CAS:Enecadin is a neuroprotective agent.Formula:C21H28FN3OPurity:98.53%Color and Shape:SolidMolecular weight:357.46UK 66914
CAS:<p>UK 66914 is a K(+) channel blocker for the study of cardiac arrhythmias.</p>Formula:C18H24N4O3SPurity:99.75%Color and Shape:SolidMolecular weight:376.47Protonstatin-1
CAS:<p>Protonstatin-1: treats hypoglycemia & Alzheimer's, inhibits IGFIR kinase, used in cancer studies.</p>Formula:C8H5NO2S2Purity:99.77%Color and Shape:SolidMolecular weight:211.26FEMA-4809
CAS:<p>FEMA-4809 activates TRPM8, the ion channel for cold sensation, and is used as a cooling agent.</p>Formula:C17H17N3O2SPurity:99.9%Color and Shape:SolidMolecular weight:327.4Transcainide
CAS:Transcainide (R 54718), an oral lidocaine-like antiarrhythmic, blocks BTX-activated Na+ channels in heart/muscle.Formula:C22H35N3O2Purity:99.81%Color and Shape:SolidMolecular weight:373.53Cerebrocrast
CAS:<p>Cerebrocrast (IOS-11212) has anti-inflammatory and hypoglycemic activity, blocks human platelet activation, and is used in the study of diabetes.</p>Formula:C26H35F2NO7Purity:99.71%Color and Shape:SolidMolecular weight:511.56Delucemine Hydrochloride
CAS:<p>Delucemine Hydrochloride (Delucemine) is a polyamine NMDA receptor antagonist used in the study of neurological disorders such as depression.</p>Formula:C16H18ClF2NPurity:98.49% - 99.30%Color and Shape:SolidMolecular weight:297.77Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Formula:C4H7BrN2O2Purity:98.13%Color and Shape:Off-White PowderMolecular weight:195.01Neboglamine hydrochloride
CAS:Neboglamine (CR-2249, XY-2401) hydrochloride boosts NMDA receptor, aids schizophrenia research, and is orally active.Formula:C13H25ClN2O3Purity:99.19%Color and Shape:SolidMolecular weight:292.8Fengabine
CAS:<p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>Formula:C17H17Cl2NOPurity:99%Color and Shape:SolidMolecular weight:322.23HC-070
CAS:HC-070 is a TRPC5 and TRPC4 antagonist (IC50 = 9.3 nM and 46 nM).Formula:C22H20Cl2N4O4Purity:98.48%Color and Shape:SolidMolecular weight:475.32Abeprazan hydrochloride
CAS:<p>Abeprazan hydrochloride (Fexuprazan hydrochloride) is an effective reversible potassium-competitive acid blocker with oral activity, inhibiting H+, K+ -atPase</p>Formula:C19H18ClF3N2O3SPurity:98.57%Color and Shape:SolidMolecular weight:446.87RL648_81
CAS:<p>RL648_81 is a selective activator of KCNQ2/3 channels (EC50 = 190 nM). RL648_81 can be used in studies about neuronal hyperexcitability neurologic disorders.</p>Formula:C17H17F4N3O2Purity:99.82%Color and Shape:SolidMolecular weight:371.33NC-1300-B
CAS:NC-1300-B inhibits H(+)-K(+)-ATPase and is used in the study of gastric ulcers.Formula:C17H19N3OSPurity:99.50%Color and Shape:SolidMolecular weight:313.42Nerisopam
CAS:<p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>Formula:C18H19N3O2Purity:97.07%Color and Shape:SolidMolecular weight:309.36FR-167356
CAS:<p>FR-167356 inhibits a3 isoform H⁺-ATPase (IC50: 170-370 nM), targeting osteoclasts, kidneys, macrophages; reduces B16-F10 bone metastasis.</p>Formula:C19H17Cl2NO3Purity:98.44% - 99.74%Color and Shape:SolidMolecular weight:378.25TASK-1-IN-1
CAS:<p>TASK-1-IN-1: Potent, selective TASK-1 blocker (IC50: 148 nM), weaker on TASK-3 (IC50: 1750 nM), anticancer properties.</p>Formula:C22H20N2O2Purity:99.57%Color and Shape:SoildMolecular weight:344.41Losigamone
CAS:Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about the treatment of partial seizures.Formula:C12H11ClO4Purity:99.98%Color and Shape:SolidMolecular weight:254.67NNC 05-711
CAS:<p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>Formula:C21H23ClN2O3Purity:99.92%Color and Shape:SolidMolecular weight:386.87NaV1.2/1.6 channel blocker-1
CAS:<p>NaV1.2/1.6 channel blocker-1 is a NaV1.2/1.6 channel blocker that inhibits rNaV1.6 and can be used to study generalised epilepsy and movement disorders.</p>Formula:C14H14N2OSPurity:99.54%Color and Shape:SolidMolecular weight:258.34SKF96067
CAS:<p>SKF96067 is a reversible gastric H+/K+-ATPase inhibitor that can induce relaxation of human airway smooth muscle in vitro.</p>Formula:C21H22N2O2Purity:99.89%Color and Shape:SolidMolecular weight:334.41Bamocaftor
CAS:<p>Bamocaftor corrects CFTR in CF, restoring F508del-CFTR function, used with tezacaftor and VX-561 for F508del/MF patients.</p>Formula:C28H32F3N5O4SPurity:99.71%Color and Shape:SolidMolecular weight:591.65Lirequinil
CAS:<p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>Formula:C26H25ClN2O3Purity:98.54%Color and Shape:SolidMolecular weight:448.94Elismetrep
CAS:<p>Elismetrep (MT-8554) is an orally available TRPM8 inhibitor with potential analgesic activity for the study of vasomotor symptoms in postmenopausal women.</p>Formula:C27H21F3N2O5SPurity:99.37% - 99.93%Color and Shape:SolidMolecular weight:542.53Aptiganel
CAS:<p>Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study acute ischemic stroke.</p>Formula:C20H21N3Purity:98.13% - 98.90%Color and Shape:SolidMolecular weight:303.4
