Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Subcategories of "Membrane Transporter/Ion Channel"
- ABC(3 products)
- ATPase(98 products)
- Adiponectin receptor(5 products)
- CFTR(66 products)
- CGRP Receptor(52 products)
- Calcium Channel(556 products)
- Chloride channel(54 products)
- GABA Receptor(369 products)
- Monoamine Transporter(30 products)
- Monocarboxylate transporter(18 products)
- NKCC(2 products)
- NPC1L1(3 products)
- Na-K-Cl cotransporter(10 products)
- OAT(32 products)
- OCT(7 products)
- P-gp(55 products)
- Potassium Channel(290 products)
- Proton pump(42 products)
- SGLT(31 products)
- Sodium Channel(233 products)
- TRP/TRPV Channel(96 products)
Show 13 more subcategories
Found 2654 products of "Membrane Transporter/Ion Channel"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
α,β-Methylene-ATP dilithium
CAS:α,β-Methylene ATP dilithium, a phosphonic analog of ATP, serves as a ligand for P2X3 and P2X7 receptors.Formula:C11H16Li2N5O12P3Color and Shape:SolidMolecular weight:517.07MMK 1
CAS:Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.Formula:C75H123N19O18SPurity:98%Color and Shape:SolidMolecular weight:1610.97Conantokin-R
CAS:Conantokin-R is an NMDA receptor peptide antagonist (IC50=93 nM); Conantokin-R exhibits anticonvulsant activity; Conantokin-R binds Zn2+ and Mg2+ (Kds 0.15 μM
Formula:C127H201N35O49S3Color and Shape:SolidMolecular weight:3098.38LY-466195
CAS:LY-466195 is a competitive antagonist of GLUK5 receptor.Formula:C16H24F2N2O4Color and Shape:SolidMolecular weight:346.37Venturicidin A
CAS:Venturicidin A is a macrolide antibiotic.Formula:C41H67NO11Purity:98%Color and Shape:SolidMolecular weight:749.97SC 4453
CAS:SC 4453 is a digoxin analog and a cardiac glycoside derivative.Formula:C41H64N2O12Color and Shape:SolidMolecular weight:776.9656-FAM-AEEAC-SHK TFA
6-FAM-AEEAC-SHK TFA, a peptide neurotoxin derived from Stichodactyla helianthus and conjugated with a fluorescent marker, selectively blocks voltage-gated potassium channels (kv1.1 and kv1.2). By prolonging action potentials, it interferes with neural signal conduction, making it valuable in neuroscience research.Formula:C196H295N55O57S7·xCHF3O2Color and Shape:SolidMolecular weight:4558.23 (free acid)AChE/Aβ-IN-1
AChE/Aβ-IN-1 (compound 32) is a potent, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 86 nM and an NMDA receptor antagonist targeting theFormula:C20H25BrN4Color and Shape:SolidMolecular weight:401.34G-Glu-Ser
CAS:G-Glu-Ser is a calcium receptor activator and Flavor-enriching agent.Formula:C8H14N2O6Color and Shape:SolidMolecular weight:234.21AmmTX3
KV4 channel blocker that inhibits A-type K+ current in mouse neurons; requires DPP6 and DPP10 for effect.Formula:C158H262N50O48S6Purity:98%Color and Shape:SolidMolecular weight:3822.47Apamin acetate
Apamin acetate: Selective Ca2+-activated K+ channel blocker, 18-amino acid bee venom peptide, promotes synapse repair, anti-inflammatory.Purity:96.97%Color and Shape:SolidAP14145 hydrochloride
CAS:AP14145 hydrochloride inhibits KCa2.2 and KCa2.3 channels with 1.1 μM IC50, affecting AERP and antiarrhythmic in AF models.Formula:C18H18ClF3N4OColor and Shape:SolidMolecular weight:398.81Elgodipine
CAS:Elgodipine decreases angina severity, inhibits muscle growth, and is voltage-sensitive, showing promise for angina treatment.Formula:C29H33FN2O6Purity:99.84% - 99.98%Color and Shape:SolidMolecular weight:524.58Urease-IN-19
Urease-IN-19 (Compound 3c) is a potent inhibitor of urease, demonstrating an IC50 value of 2.7 µM. It shows potential for use in research related to kidney stones and gastric ulcers.
Formula:C17H16FN3SColor and Shape:SolidMolecular weight:313.39D-myo-Inositol-1,3,4,5-tetraphosphate (sodium salt)
CAS:Ins(1,3,4,5)-P4, made via Ins(1,4,5)P3 phosphorylation, boosts calcium by opening ER and plasma membrane channels.Formula:C6H8Na8O18P4Color and Shape:SolidMolecular weight:675.93Flufiprole
CAS:Flufiprole is used as a phenylpyrazole pesticide. It has enantioselective metabolism in human and rat liver microsomes.Formula:C16H10Cl2F6N4OSColor and Shape:SolidMolecular weight:491.24CP-628006
CAS:CP-628006 is a small molecule CFTR potentiator that effectively restores ATP-dependent channel gating to G551D-CFTR, the mutant form found in cystic fibrosis.Formula:C32H35F3N2O2Color and Shape:SolidMolecular weight:536.639GSK2332255B
CAS:GSK2332255B: potent TRPC3/6 antagonist; IC50 5 nM (TRPC3), 4 nM (TRPC6); over 100-fold selectivity vs other Ca2+ channels.Formula:C18H19ClFN3O3SColor and Shape:SolidMolecular weight:411.88AChE/Aβ-IN-2
AChE/Aβ-IN-2 (compound 33) is a powerful, orally active acetylcholinesterase (AChE) inhibitor with an IC50 of 135 nM.Formula:C20H25ClN4Color and Shape:SolidMolecular weight:356.89Eltanexor
CAS:Eltanexor, an oral XPO1 inhibitor, induces apoptosis in leukemia cells; EC50=60.9 nM.Formula:C17H10F6N6OPurity:99.68% - ≥98%Color and Shape:SolidMolecular weight:428.29Ref: TM-T11766L
1mg63.00€5mg213.00€10mg250.00€25mg404.00€50mg595.00€100mg863.00€200mg1,161.00€1mL*10mM (DMSO)200.00€
