Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Lubeluzole dihydrochloride
CAS:144665-09-8
Lubeluzole (dihydrochloride) acts as a neuroprotective agent by blocking neuronal voltage-gated sodium channels and also …
Formula:
C22H27Cl2F2N3O2S
Color and Shape:
Liquid
Molecular weight:
506.44
Ref: TM-T200178
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Picrotoxinin
CAS:17617-45-7
Picrotoxinin blocks chloride channels, antagonizes GABAA noncompetitively (IC50: 1.15 μM, α1β2γ2L), and induces convulsions.
Formula:
C15H16O6
Purity:
98.07%
Color and Shape:
Solid
Molecular weight:
292.28
Ref: TM-T16535
| 10mg | 47.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 133.00 € | ||
| 500mg | 314.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
V-ATPase-IN-1
CAS:1243603-61-3
V-ATPase-IN-1 (Compound 3b-03) is an inhibitor of Vacuolar-type H+-ATPases (V-ATPase), exhibiting an inhibition constant (IC50) …
Formula:
C21H20ClNO2
Color and Shape:
Liquid
Molecular weight:
353.84
Ref: TM-T200467
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 9 Apr 2025
TP003
CAS:628690-75-5
TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, …
Formula:
C23H16F3N3O
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
407.39
Ref: TM-T23466
| 2mg | 40.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 368.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Kv7.2/Kv7.3 activator-1
CAS:2376398-43-3
Kv7.2/Kv7.3 Activator-1 (compound 517) serves as a powerful activator of the Kv7.2/Kv7.3 channels, exhibiting an …
Formula:
C19H22F2N4O
Color and Shape:
Liquid
Molecular weight:
360.4
Ref: TM-T89880
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 9 Apr 2025
PF-05661014
CAS:2153474-85-0
PF-05661014, a demethylated analogue of PF-06526290, selectively inhibits Nav1.3 and Nav1.7 currents by stabilizing the …
Formula:
C17H16N4O3S2
Color and Shape:
Liquid
Molecular weight:
388.46
Ref: TM-T89885
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 9 Apr 2025
CFTR corrector 16
CAS:1210305-23-9
CFTRcorrector 16 (Compound 39) is a corrector of the cystic fibrosis transmembrane conductance regulator (CFTR), …
Formula:
C27H26ClN5O2S
Color and Shape:
Liquid
Molecular weight:
520.05
Ref: TM-T200113
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 9 Apr 2025
SP100030 analogue 1
CAS:154934-68-6
SP100030 analogue 1 (compound 11) is a selective transcription activation (SITA) inhibitor within the SP100030 …
Formula:
C13H5ClF7N3O
Color and Shape:
Liquid
Molecular weight:
387.64
Ref: TM-T89990
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 9 Apr 2025
SYM2206
CAS:173952-44-8
SYM2206 is a low affinity non-competitive AMPA receptor antagonist with an IC50 value of 1.6 …
Formula:
C20H22N4O3
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
366.41
Ref: TM-T16964
| 1mg | 41.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 256.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
TRPA1 Antagonist 1
CAS:1984825-08-2
TRPA1 Antagonist 1 is an antagonist of TRPA1(IC50: 8 nM) and is a methylene phosphate …
Formula:
C24H22F6N5Na2O7PS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
715.47
Ref: TM-T13212
| 25mg | 3,079.00 € | ||
| 50mg | 4,094.00 € | ||
| 100mg | 5,701.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Valbenazine tosylate
CAS:1639208-54-0
Valbenazine tosylate, the tosylate salt of valbenazine, is a vesicular monoamine transporter 2 (VMAT2) inhibitor …
Formula:
C38H54N2O10S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
762.97
Ref: TM-T22452
| 25mg | 2,662.00 € | ||
| 50mg | 3,533.00 € | ||
| 100mg | 4,860.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
GSK2798745
CAS:1419609-94-1
GSK2798745 is an orally active transient receptor potential vanilloid 4 (TRPV4) ion channel blocker (IC50s: …
Formula:
C25H28N6O3
Color and Shape:
Solid
Molecular weight:
460.53
Ref: TM-T15434
| 25mg | 2,106.00 € | ||
| 50mg | 2,789.00 € | ||
| 100mg | 3,744.00 € |
Estimated delivery in United States, on Wednesday 9 Apr 2025
Indiplon
CAS:325715-02-4
Indiplon is a short-acting hypnotic with high-affinity allosteric potentiator of GABAA responses that demonstrates preference …
Formula:
C20H16N4O2S
Purity:
98.45%
Color and Shape:
Liquid
Molecular weight:
376.43
Ref: TM-T21362
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
N-Arachidonyl-GABA
CAS:128201-89-8
N-Arachidonyl-GABA (NA-GABA) is a novel active fatty amino acid related to anandamide (ANA) found in …
Formula:
C24H39NO3
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
389.57
Ref: TM-T23039
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Lopirazepam
CAS:42863-81-0
Lopirazepam is a potent small molecule GABAA receptor agonist, which can be used to treat …
Formula:
C14H9Cl2N3O2
Purity:
99.30% - 99.51%
Color and Shape:
Solid
Molecular weight:
322.15
Ref: TM-T32872
| 5mg | Discontinued | Request information |
Pagoclone
CAS:133737-32-3
Pagoclone (IP456) is a GABA receptor agonist and can be used for studies on the …
Formula:
C23H22ClN3O2
Purity:
99.45%
Color and Shape:
Solid
Molecular weight:
407.89
Ref: TM-T7822
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
4-Aminopyridine
CAS:504-24-5
4-Aminopyridine (Dalfampridine) is a nonselective potassium (K+) channel blocker that binds to the cytoplasmic side …
Formula:
C5H6N2
Purity:
90%
Color and Shape:
Liquid
Molecular weight:
94.11
Ref: TM-T0817
| 50mg | Discontinued | Request information |
MitTx-α
MitTx-alpha, a component of the complex MitTx, acts as a powerful and enduring agonist specifically …
Formula:
C317H440N86O89S7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
7103.94
Ref: TM-T80181
| Undefined size | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information |
T-2000
CAS:97846-21-4
T-2000 (DMMDPB) is a GABA receptor agonist that can be used to study myoclonus and …
Formula:
C20H20N2O5
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
368.38
Ref: TM-T28900
| 1mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 500mg | Discontinued | Request information |
MitTx
MitTx, a complex consisting of MitTx-α and MitTx-β, serves as an ASIC1 channel activator, demonstrating …
Formula:
C899H1331N259O271S23
Purity:
98%
Color and Shape:
Solid
Molecular weight:
20840.26
Ref: TM-T80182
| Undefined size | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information |
