Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
Tertiapin-RQ
Tertiapin-RQ, an inward rectifier potassium (K+) channel-blocking peptide, exhibits antidepressant effects [1].
Formula:
C106H175N37O25S4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
2496.02
Ref: TM-T80510
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
E 0747 FA
E 0747 FA is an antiarrhythmic compound that inhibits the voltage of action potential Vmax …
Formula:
C22H30ClN3O6
Purity:
98.54%
Color and Shape:
Liquid
Molecular weight:
467.94
Ref: TM-T24021L
| 1mg | 198.00 € | ||
| 5mg | 489.00 € | ||
| 10mg | 686.00 € | ||
| 25mg | 1,070.00 € | ||
| 50mg | 1,476.00 € | ||
| 100mg | 1,890.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
(S)-ABT 102
CAS:808756-70-9
N-[(1S)-1H-inden-1-yl]-N'-indazol-4-ylurea is a strong TRPV1 blocker with a 123 nM IC50 against capsaicin.
Formula:
C21H24N4O
Purity:
99.41% - 99.78%
Color and Shape:
Soild
Molecular weight:
348.44
Ref: TM-T29522L
| 1mg | 78.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 340.00 € | ||
| 50mg | 476.00 € | ||
| 100mg | 649.00 € | ||
| 200mg | 873.00 € | ||
| 1mL*10mM (DMSO) | 164.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
RN-1665
CAS:1803003-65-7
RN-1665 is a potent and selective TRPV4 receptor antagonist.
Formula:
C20H24F5N3O3S2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
513.54
Ref: TM-T77723
| 1mg | 152.00 € | ||
| 5mg | 364.00 € | ||
| 10mg | 503.00 € | ||
| 25mg | 831.00 € | ||
| 50mg | 1,104.00 € | ||
| 100mg | 1,512.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
JC-229
CAS:3026716-22-0
JC-229 is a potent and selective TbRPA1 inhibitor that can inhibit RPA1 in Trypanosoma brucei. …
Formula:
C20H14Cl4N2O3S
Purity:
97.14%
Color and Shape:
Liquid
Molecular weight:
504.21
Ref: TM-T77645
| 10mg | 43.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 90.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Goniothalamin
CAS:17303-67-2
Goniothalamin induces apoptosis in various cancer cell lines and has gastroprotective activity.
Formula:
C13H12O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
200.23
Ref: TM-TN4160
| 1mg | 349.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Pinacidil monohydrate
CAS:85371-64-8
Pinacidil monohydrate is a potassium channel activator, antihypertensive drug.
Formula:
C13H21N5O
Purity:
99.94% - 99.96%
Color and Shape:
Powder
Molecular weight:
263.34
Ref: TM-T12478
| 10mg | 34.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 82.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Tap1a
Theraphotoxin-Tap1a (Tap1a) is a spider venom-derived peptide that acts as an inhibitor of sodium channels, …
Formula:
C174H258N52O55S7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
4182.68
Ref: TM-T80494
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
Dendrotoxin-I
CAS:107950-33-4
Dendrotoxin-I, a neurotoxin from Dendroaspis snake venom, potently blocks K⁺ channels, specifically targeting voltage-gated potassium …
Formula:
C312H491N99O83S6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
7149.24
Ref: TM-T80064
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
Oleoyl Serotonin
CAS:1002100-44-8
Oleoyl Serotonin is an antagonist of hTRPV1 with an IC50 of 2.57 μM.
Formula:
C28H44N2O2
Purity:
100.00%
Color and Shape:
Solid
Molecular weight:
440.66
Ref: TM-T22124
| 5mg | 64.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 181.00 € | ||
| 50mg | 309.00 € | ||
| 100mg | 536.00 € | ||
| 500mg | 1,170.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Cycloartane-3,24,25-triol
CAS:57576-29-1
Cycloartane-3,24,25-triol has potential for development as an anti-cancer agent against prostate cancer.
Formula:
C30H52O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
460.743
Ref: TM-TN3737
| 5mg | 586.00 € | ||
| 1mL*10mM (DMSO) | 595.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
AmmTX3 TFA
AmmTX3 TFA, a peptide toxin derived from Androctonus mauretanicus scorpion venom, functions as a selective …
Formula:
C158H262N50O48S6·xC2HF3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
3822.47 (free acid)
Ref: TM-T80036
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
Spinoxin
CAS:752984-66-0
Spinoxin, a 34-residue peptide neurotoxin extracted from the venom of Heterometrus spinifer, is characterized by …
Formula:
C147H236N48O46S9
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
3700.33
Ref: TM-T80530
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
BDS-I
CAS:207621-38-3
BDS-I, a marine toxin derived from Anemonia sulcata, functions as a selective inhibitor of the …
Formula:
C210H297N57O56S6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
4708.34
Ref: TM-T80173
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
Epaminurad HCl
CAS:1198153-46-6
Epaminurad HCl is a URAT1 inhibitor with partial inhibition of OAT1 and OAT3 (organic anion …
Formula:
C14H11Br2ClN2O3
Purity:
100% - 99.01%
Color and Shape:
Soild
Molecular weight:
450.51
Ref: TM-T27275L
| 1mg | 121.00 € | ||
| 5mg | 291.00 € | ||
| 10mg | 476.00 € | ||
| 25mg | 760.00 € | ||
| 50mg | 1,002.00 € | ||
| 100mg | 1,382.00 € | ||
| 1mL*10mM (DMSO) | 323.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Pterinotoxin-1
Pterinotoxin-1 is a peptide toxin that functions as an inhibitor of sodium channels [1].
Formula:
C163H251N49O53S7
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
3969.49
Ref: TM-T80534
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
Iberiotoxin TFA
Iberiotoxin (TFA) is a selective inhibitor of high conductance Ca2+-activated K+ channels, exhibiting a dissociation …
Formula:
C179H274N50O55S7·xC2HF3O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
4230.85 (free base)
Ref: TM-T80028
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
Caloxin 2A1 acetate
Caloxin 2A1 acetate is an inhibitor of extracellular plasma membrane Ca2+-ATPase (PMCA) peptide.
Formula:
C66H95N19O24
Purity:
98.2%
Color and Shape:
Liquid
Molecular weight:
1538.57
Ref: TM-T40437L
| 1mg | 56.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 316.00 € | ||
| 50mg | 471.00 € | ||
| 100mg | 687.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
4-Hydroxytolbutamide
CAS:5719-85-7
4-Hydroxytolbutamide, a metabolite of the sulfonylurea antidiabetic Tolbutamide, is processed by CYP2C8 and CYP2C9.
Formula:
C12H18N2O4S
Purity:
98%
Color and Shape:
White To Off-White
Molecular weight:
286.35
Ref: TM-T14040
| 1mg | 97.00 € | ||
| 5mg | 364.00 € | ||
| 10mg | 679.00 € | ||
| 25mg | 1,565.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
ASG-5ME
ASG-5ME is a drug-antibody coupling targeting SLC44A4 that shows anti-tumor activity in xenograft models and …
Color and Shape:
Liquid
Molecular weight:
145.5 kDa
Ref: TM-T77382
| 1mg | 203.00 € | ||
| 5mg | 493.00 € | ||
| 10mg | 706.00 € | ||
| 25mg | 1,101.00 € | ||
| 50mg | 1,519.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
