Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
Read more
Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
m3-Huwentoxin IV
m3-Huwentoxin IV (m3-HwTx-IV) is a potent inhibitor of sodium channels (NaV), exhibiting half-maximal inhibitory concentrations …
Formula:
C170H271N53O46S6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
3985.69
Ref: TM-T80519
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
Vocacapsaicin hydrochloride
CAS:1931116-92-5
Vocacapsaicin hydrochloride (CA-008 hydrochloride) is a non-opioid TRPV1 agonist, a raw material for capsaicin, and …
Formula:
C26H42ClN3O4
Purity:
98.51% - 99.94%
Color and Shape:
Solid
Molecular weight:
496.08
Ref: TM-T39349
| 1mg | 375.00 € | ||
| 5mg | 915.00 € | ||
| 10mg | 1,217.00 € | ||
| 25mg | 1,839.00 € | ||
| 50mg | 2,471.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
BDS-II
BDS-II, a peptide toxin comprising 43 amino acids, selectively inhibits the Kv3.4 channel [1].
Formula:
C214H301N57O57S6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
4776.42
Ref: TM-T80456
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
ML353
ML353 activates TREK-1/2, binds mGlu5 SAM (Ki=18.2 nM), surpasses 5mpep, may address SAM activity/blocking.
Formula:
C19H15FN2O
Purity:
99.28% - 99.82%
Color and Shape:
Soild
Molecular weight:
306.33
Ref: TM-T67917
| 2mg | 46.00 € | ||
| 5mg | 71.00 € | ||
| 10mg | 103.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 229.00 € | ||
| 100mg | 335.00 € | ||
| 200mg | 454.00 € | ||
| 1mL*10mM (DMSO) | 76.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Fumitremorgin C
CAS:118974-02-0
Fumitremorgin C (12α-Fumitremorgin C) is a mycotoxin and inhibits ABCG2/BRCP.
Formula:
C22H25N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
379.45
Ref: TM-T15355
| 1mg | 1,290.00 € | ||
| 250µg | 503.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Lifastuzumab
CAS:1615697-16-9
Sulfamethoxazole-NO (SMX-NO) is a SMX-NO derivative and is the primary immunogen for sulfonamide hypersensitivity reactions.
Purity:
≥95% (SDS-PAGE/SEC-HPLC) - ≥95% (SDS-PAGE/SEC-HPLC)
Color and Shape:
Liquid
Molecular weight:
145.5 kDa
Ref: TM-T77384
| 1mg | 1,658.00 € | ||
| 5mg | 3,365.00 € | ||
| 10mg | 4,542.00 € | ||
| 25mg | 6,749.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
SLC26A3-IN-2
CAS:950348-60-4
Vilobelimab (CaCP-29) is a human-mouse chimeric IgG antibody targeting human complement component 5a, a C5a …
Formula:
C19H13ClN2O2S
Purity:
100%
Color and Shape:
Liquid
Molecular weight:
368.84
Ref: TM-T74815
| 2mg | 78.00 € | ||
| 5mg | 123.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Chlorahololide C
CAS:1007859-25-7
Chlorahololide C blocks potassium channels, selectively inhibiting I(K) current with an IC50 of 3.6±10.1 µM.
Formula:
C33H36O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
576.63
Ref: TM-TN3636
| 5mg | 668.00 € | ||
| 1mL*10mM (DMSO) | 1,016.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
GS-9191 PM
GS-9191 PM: novel antitumorviral bis-amide prodrug, inhibits MDR1/BCRP, has antiproliferative activity.
Formula:
C11H16N6O
Purity:
99.02%
Color and Shape:
Soild
Molecular weight:
248.28
Ref: TM-T67821
| 1mg | 134.00 € | ||
| 5mg | 316.00 € | ||
| 10mg | 474.00 € | ||
| 25mg | 772.00 € | ||
| 50mg | 1,075.00 € | ||
| 100mg | 1,439.00 € | ||
| 500mg | 2,757.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Apamin acetate
Apamin acetate: Selective Ca2+-activated K+ channel blocker, 18-amino acid bee venom peptide, promotes synapse repair, …
Purity:
96.97%
Color and Shape:
Liquid
Ref: TM-TP1223L
| 1mg | 170.00 € | ||
| 5mg | 387.00 € | ||
| 10mg | 558.00 € | ||
| 25mg | 889.00 € | ||
| 50mg | 1,198.00 € | ||
| 100mg | 1,606.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Lasiodiplodin
CAS:32885-81-7
Lasiodiplodin may have potential anti-inflammatory activity, it shows moderate suppression effects on induced NO production.
Formula:
C17H24O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
292.37
Ref: TM-TN4418
| 5mg | 586.00 € | ||
| 1mL*10mM (DMSO) | 595.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Celivarone
CAS:401925-43-7
Celivarone is a potassium channel blocker used in the study of arrhythmias, atrial flutter and …
Formula:
C34H47NO4
Purity:
99.03%
Color and Shape:
Liquid
Molecular weight:
533.74
Ref: TM-T68038
| 1mg | 178.00 € | ||
| 5mg | 437.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,003.00 € | ||
| 50mg | 1,361.00 € | ||
| 100mg | 1,819.00 € | ||
| 500mg | 3,671.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
TRPA1-IN-2
CAS:2415206-22-1
TRPA1-IN-2 is a potent and orally active TRPA1 inhibitor with an IC50 value of 0.04 …
Formula:
C24H25F3N4O
Purity:
98.05%
Color and Shape:
Soild
Molecular weight:
442.48
Ref: TM-T77511
| 1mg | 124.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 461.00 € | ||
| 25mg | 784.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,475.00 € | ||
| 1mL*10mM (DMSO) | 337.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Lifarizine FA
Lifarizine FA is a sodium channel blocker used in the treatment of neurological disorders and …
Formula:
C30H34N4O2
Purity:
99.87%
Color and Shape:
Liquid
Molecular weight:
482.62
Ref: TM-T27830L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 593.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,700.00 € | ||
| 500mg | 3,416.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
6,7-dimethylisatin
CAS:20205-43-0
6,7-Dimethylisatin (6,7-dimethyl-1H-indole-2,3-dione) inhibits hGAT3 with IC50 of 108 μM. 6,7-Dimethylisatin also inhibits hBGT1, hGAT2.
Formula:
C10H9NO2
Purity:
99.09%
Color and Shape:
Liquid
Molecular weight:
175.18
Ref: TM-T77568
| 1mg | 182.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,699.00 € | ||
| 500mg | 3,428.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Benzocaine hydrochloride
CAS:23239-88-5
Benzocaine hydrochloride (Ethyl 4-aminobenzoate hydrochloride) is a surface anesthetic that acts by preventing transmission of …
Formula:
C9H11NO2·HCl
Purity:
98%
Color and Shape:
Solid
Molecular weight:
201.65
Ref: TM-T6782
| 50mg | 55.00 € | ||
| 100mg | 71.00 € | ||
| 200mg | 115.00 € | ||
| 500mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
3-Hydroxybakuchiol
CAS:178765-54-3
3-Hydroxybakuchiol fights TA3/Ha mammary cancer cells, impairs mitochondria, activates caspase-3, opens MPTP, fragments DNA, and …
Formula:
C18H24O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
272.38
Ref: TM-TN2945
| 5mg | 491.00 € | ||
| 1mL*10mM (DMSO) | 501.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
BMS-394136
CAS:343246-73-1
BMS-394136 (BMS 394136) is a KV1.5 antagonist for the treatment of cardiovascular diseases such as …
Formula:
C24H21Cl2FN4O
Purity:
98.25% - 98.67%
Color and Shape:
Solid
Molecular weight:
471.35
Ref: TM-T30520
| 1mg | 242.00 € | ||
| 5mg | 600.00 € | ||
| 10mg | 853.00 € | ||
| 25mg | 1,290.00 € | ||
| 50mg | 1,727.00 € | ||
| 100mg | 2,311.00 € | ||
| 500mg | 4,579.00 € |
Estimated delivery in United States, on Thursday 2 Jan 2025
Heteropodatoxin-2
CAS:741730-12-1
Heteropodatoxin-2, a 30-amino acid peptide, inhibits the Kv4.2 current in Xenopus laevis oocytes through a …
Formula:
C144H207N39O46S6
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
3412.81
Ref: TM-T80434
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
BmK-M1
BmK-M1, a scorpion-derived toxin, consists of a 64-amino acid polypeptide stabilized by four disulfide bridges.
Formula:
C313H467N91O91S8
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
7217.13
Ref: TM-T80454
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Thursday 2 Jan 2025
