Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
NHE3-IN-1
CAS:632355-68-1
NHE3-IN-1 is a inhibitor of Na+/H+-exchanger 3 (NHE-3).
Formula:
C12H10ClN3S
Purity:
97.44%
Color and Shape:
Solid
Molecular weight:
263.75
Ref: TM-T12219
| 25mg | 57.00 € | ||
| 50mg | 94.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
OR-1896
CAS:220246-81-1
OR-1896 is a PDE III inhibitor, a vasodilator with partial anti-inflammatory properties, and can be …
Formula:
C13H15N3O2
Purity:
99.51%
Color and Shape:
Solid
Molecular weight:
245.28
Ref: TM-T12315
| 1mg | 91.00 € | ||
| 2mg | 134.00 € | ||
| 5mg | 215.00 € | ||
| 10mg | 390.00 € | ||
| 25mg | 841.00 € | ||
| 50mg | 1,151.00 € | ||
| 100mg | 1,556.00 € | ||
| 1mL*10mM (DMSO) | 239.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
L-838417
CAS:286456-42-6
L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in …
Formula:
C19H19F2N7O
Purity:
98.12% - 99.82%
Color and Shape:
Solid
Molecular weight:
399.4
Ref: TM-T19702
| 1mg | 55.00 € | ||
| 5mg | 207.00 € | ||
| 10mg | 330.00 € | ||
| 25mg | 721.00 € | ||
| 50mg | 1,151.00 € | ||
| 100mg | 1,841.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Cirsimaritin
CAS:6601-62-3
Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.
Formula:
C17H14O6
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
314.29
Ref: TM-TQ0119
| 1mg | 56.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TRPC6-PAM-C20
CAS:667427-75-0
TRPC6-PAM-C20, a selective enhancer for TRPC6, boosts calcium in HEK cells and OAG-related platelet clumping, …
Formula:
C22H21NO4
Purity:
90%
Color and Shape:
Liquid
Molecular weight:
363.41
Ref: TM-T37428
| 1mg | 171.00 € | ||
| 5mg | 424.00 € | ||
| 10mg | 628.00 € | ||
| 25mg | 988.00 € | ||
| 50mg | 1,327.00 € | ||
| 1mL*10mM (DMSO) | 461.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Pipequaline
CAS:77472-98-1
Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that …
Formula:
C22H24N2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
316.44
Ref: TM-T4655
| 5mg | 49.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 379.00 € | ||
| 1ml*10 (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
CP-100356 hydrochloride
CAS:142715-48-8
CP-100356 hydrochloride is an MDR1 (P-gp) and BCRP inhibitor, a nucleotide-derived substrate analog that induces …
Formula:
C31H37ClN4O6
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
597.1
Ref: TM-T22680
| 1mg | 74.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Nav1.7 inhibitor
CAS:1355631-24-1
Nav1.7 inhibitor is a Nav1.7 inhibitor for research in the field of pain and anesthesia.
Formula:
C15H11Cl3FNO4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
426.68
Ref: TM-T12184
| 1mg | 135.00 € | ||
| 2mg | 186.00 € | ||
| 5mg | 325.00 € | ||
| 25mg | 1,058.00 € | ||
| 50mg | 1,411.00 € | ||
| 100mg | 1,849.00 € | ||
| 1mL*10mM (DMSO) | 361.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Sulcardine sulfate
CAS:343935-61-5
Sulcardine sulfate (B-87823) is a multi-ion channel blocker with antiarrhythmic activity that inhibits Na+, K+, …
Formula:
C24H35N3O8S2
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
557.68
Ref: TM-T28879
| 25mg | 1,435.00 € | ||
| 50mg | 1,869.00 € | ||
| 100mg | 2,359.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Pyr3
CAS:1160514-60-2
Pyr3 selectively blocks TRPC3 channels, reducing Ca2+ influx; it's effective at 700 nM.
Formula:
C16H11Cl3F3N3O3
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
456.63
Ref: TM-T16687
| 1mg | 35.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 76.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 505.00 € | ||
| 200mg | 729.00 € | ||
| 500mg | 1,096.00 € | ||
| 1mL*10mM (DMSO) | 85.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Bisaramil hydrochloride
CAS:96480-44-3
Bisaramil hydrochloride (Bisaramil) is an antiarrhythmic compound that inhibits free radical production.
Formula:
C17H24Cl2N2O2
Purity:
98.90% - 99.64%
Color and Shape:
Solid
Molecular weight:
359.29
Ref: TM-T26822
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € | ||
| 100mg | 2,357.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Sodium Channel inhibitor 2
CAS:653573-60-5
Sodium Channel inhibitor 2 is a blocker of sodium channel.
Formula:
C26H25Cl2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
466.4
Ref: TM-T12951
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
GABAB receptor antagonist 1
CAS:797-17-1
(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB …
Formula:
C18H24O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11350
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
RWJ-51204
CAS:205701-85-5
RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:
C21H19F2N3O3
Purity:
100% - 99.57%
Color and Shape:
Solid
Molecular weight:
399.39
Ref: TM-T16811
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,549.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Cilobradine hydrochloride
CAS:186097-54-1
Cilobradine hydrochloride (DK-AH 269) is an HCN Channel blocker and an open channel blocker of …
Formula:
C28H39ClN2O5
Purity:
97.46%
Color and Shape:
Solid
Molecular weight:
519.07
Ref: TM-T10813
| 1mg | 63.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 331.00 € | ||
| 50mg | 463.00 € | ||
| 100mg | 631.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
SET 2
CAS:2313525-20-9
SET 2 is an antagonist of transient receptor potential vanilloid type 2(TRPV2) with an IC50 …
Formula:
C17H21F3N4O2S
Purity:
98.43%
Color and Shape:
Liquid
Molecular weight:
402.43
Ref: TM-T37097
| 5mg | 57.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 294.00 € | ||
| 100mg | 429.00 € | ||
| 500mg | To inquire | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
TC-AQP1-1
CAS:37710-81-9
TC-AQP1-1 blocks aquaporin 1; found via virtual screening; hinders water flux in Xenopus oocytes at …
Formula:
C12H10O4
Purity:
97.26%
Color and Shape:
Solid
Molecular weight:
218.21
Ref: TM-T24859
| 5mg | 41.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 174.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 388.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Saviprazole
CAS:121617-11-6
Saviprazole (Hoe-731), a proton pump inhibitor, is used potentially for treatment of gastric ulcer.
Formula:
C15H10F7N3O2S2
Purity:
97.73% - 99.20%
Color and Shape:
Solid
Molecular weight:
461.38
Ref: TM-T28665
| 1mg | 139.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 496.00 € | ||
| 25mg | 803.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Bamaluzole
CAS:87034-87-5
Bamaluzole is an agonist of GABA receptor.
Formula:
C14H12ClN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
273.72
Ref: TM-T10456
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
SKA-111
CAS:1369170-24-0
SKA-111 activates KCa3.1 potassium channels, modulates membrane potential in endothelial cells, and dilates rat coronary …
Formula:
C12H10N2S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
214.29
Ref: TM-T24799
| 1mg | 69.00 € | ||
| 5mg | 149.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 496.00 € | ||
| 50mg | 711.00 € | ||
| 100mg | 993.00 € | ||
| 500mg | 1,997.00 € | ||
| 1mL*10mM (DMSO) | 166.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
