Membrane Transporter/Ion Channel
Membrane transporter and ion channel inhibitors are compounds that block the function of proteins responsible for the transport of ions, nutrients, and other molecules across cell membranes. These inhibitors are crucial for studying the regulation of cellular homeostasis, signal transduction, and neurotransmission. Membrane transporter and ion channel inhibitors are also important in developing treatments for disorders such as epilepsy, cardiovascular diseases, and metabolic syndromes. At CymitQuimica, we provide a diverse selection of high-quality membrane transporter and ion channel inhibitors to support your research in physiology, neuroscience, and pharmacology.
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Subcategories of "Membrane Transporter/Ion Channel"
ABC
ATPase
Adiponectin receptor
CFTR
CGRP Receptor
Calcium Channel
Chloride channel
GABA Receptor
Monoamine Transporter
Monocarboxylate transporter
NKCC
NPC1L1
Na-K-Cl cotransporter
OAT
OCT
P-gp
Potassium Channel
Proton pump
SGLT
Sodium Channel
TRP/TRPV Channel
Show 13 more subcategories
Products of "Membrane Transporter/Ion Channel"
AVE-0118
CAS:498577-53-0
AVE-0118 is a potassium channel blocker and suppresses persistent atrial fibrillation.
Formula:
C30H29N3O3
Purity:
98.89% - 99.52%
Color and Shape:
Solid
Molecular weight:
479.57
Ref: TM-T26689
| 1mg | 74.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 320.00 € | ||
| 50mg | 473.00 € | ||
| 100mg | 688.00 € | ||
| 500mg | 1,412.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
JNJ-26489112
CAS:871824-55-4
JNJ-26489112 is a CNS-active agent and an inhibitor of voltage-gated Na+ channels and N-type Ca2+ …
Formula:
C9H11ClN2O4S
Purity:
99.31%
Color and Shape:
Solid
Molecular weight:
278.71
Ref: TM-T27672
| 1mg | 187.00 € | ||
| 5mg | 462.00 € | ||
| 10mg | 662.00 € | ||
| 25mg | 1,033.00 € | ||
| 50mg | 1,425.00 € | ||
| 100mg | 1,885.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Nisoxetine hydrochloride
CAS:57754-86-6
Nisoxetine hydrochloride is a noradrenaline transporter (NET) inhibitor
Formula:
C17H21NO2·HCl
Purity:
98.52%
Color and Shape:
White Solid
Molecular weight:
307.82
Ref: TM-T23070
| 5mg | 69.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 171.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 426.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Dicirenone
CAS:41020-79-5
Dicirenone (SC26304) inhibits the Mineralocorticoid receptor (MR), aldosterone regulation of the urinary K+:Na+ ratio, and …
Formula:
C26H36O5
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
428.56
Ref: TM-T13881
| 1mg | 650.00 € | ||
| 5mg | 1,672.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
GSK1702934A
CAS:924377-85-5
GSK1702934A is a TRPC3 agonist with pro-arrhythmic and positive inotropic effects and is used in …
Formula:
C22H25N3O2S
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
395.52
Ref: TM-T15425
| 1mg | 77.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
GS 39783
CAS:39069-52-8
GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties …
Formula:
C15H23N5O2S
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
337.44
Ref: TM-T22813
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 399.00 € | ||
| 100mg | 579.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
SM-6586
CAS:103898-38-0
SM-6586 is a potent calcium channel antagonist with inhibitory effects on Na+/H+ and Na+/Ca2+ exchange …
Formula:
C26H27N5O5
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
489.52
Ref: TM-T16897
| 1mg | 652.00 € | ||
| 5mg | 1,677.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
(5R)-BW-4030W92
CAS:189013-61-4
(5R)-BW-4030W92 is the R-type of BW-4030W92, the active enantiomer.
Formula:
C11H9Cl2FN4
Purity:
98.27%
Color and Shape:
Solid
Molecular weight:
287.12
Ref: TM-T13428
| 1mg | 650.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Dimethindene
CAS:5636-83-9
Dimethindene (Dimetindeno) is a selective antagonist of H1 receptor and blocks K+ current. Dimethindene exhibits …
Formula:
C20H24N2
Purity:
99% - 99.44%
Color and Shape:
Solid
Molecular weight:
292.42
Ref: TM-T31488
| 1mg | 78.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 227.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
AM12
CAS:2387510-84-9
AM12 inhibits Lanthanide-evoked TRPC5 activity (IC50: 0.28 μM).
Formula:
C15H9BrO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
349.13
Ref: TM-T13546
| 10mg | 448.00 € | ||
| 50mg | 1,874.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Rilmakalim
CAS:132014-21-2
Rilmakalim is a potassium channel opener. Rilmakalim shows antivasoconstrictor effect.
Formula:
C21H23NO5S
Purity:
100% - 99.63%
Color and Shape:
Liquid
Molecular weight:
401.48
Ref: TM-T26086
| 1mg | 126.00 € | ||
| 5mg | 299.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 735.00 € | ||
| 50mg | 1,009.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Losigamone
CAS:112856-44-7
Losigamone (AO-33) is an agonist of GABA receptor and can be used in studies about …
Formula:
C12H11ClO4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
254.67
Ref: TM-T27845
| 1mg | 81.00 € | ||
| 5mg | 168.00 € | ||
| 10mg | 253.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 631.00 € | ||
| 100mg | 920.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Panadiplon
CAS:124423-84-3
Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, …
Formula:
C18H17N5O2
Purity:
100% - 99.75%
Color and Shape:
Solid
Molecular weight:
335.36
Ref: TM-T28294
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,477.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
ML402
CAS:298684-44-3
ML402 (ZINC3671497) is an activator of TREK-1 and TREK-2 with EC50s of 13.7 μM and …
Formula:
C14H14ClNO2S
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
295.78
Ref: TM-T16109
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 232.00 € | ||
| 50mg | 373.00 € | ||
| 100mg | 553.00 € | ||
| 500mg | 1,188.00 € | ||
| 1mL*10mM (DMSO) | 86.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
ABT 102
CAS:808756-71-0
ABT 102 (CHEMBL398338) is a selective antagonist of transient receptor potential vanilloid 1 (TRPV1) receptor.
Formula:
C21H24N4O
Purity:
98.38% - 99.72%
Color and Shape:
Solid
Molecular weight:
348.44
Ref: TM-T29522
| 1mg | 112.00 € | ||
| 5mg | 242.00 € | ||
| 10mg | 359.00 € | ||
| 25mg | 547.00 € | ||
| 50mg | 765.00 € | ||
| 100mg | 1,026.00 € | ||
| 200mg | 1,367.00 € | ||
| 1mL*10mM (DMSO) | 252.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Bifenazate
CAS:149877-41-8
Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls …
Formula:
C17H20N2O3
Purity:
99.44%
Color and Shape:
Solid Crystalline
Molecular weight:
300.35
Ref: TM-T14571
| 25mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
BMS-919373
CAS:1272353-82-8
BMS-919373 is a potassium channel Kv1.5 (KCNA5) inhibitor for atrial fibrillation and acute coronary syndrome.
Formula:
C25H20N6O2S
Purity:
98.51%
Color and Shape:
Solid
Molecular weight:
468.53
Ref: TM-T30544
| 1mg | 237.00 € | ||
| 5mg | 581.00 € | ||
| 10mg | 817.00 € | ||
| 25mg | 1,207.00 € | ||
| 50mg | 1,628.00 € | ||
| 100mg | 2,185.00 € | ||
| 1mL*10mM (DMSO) | 632.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Sipatrigine
CAS:130800-90-7
Sipatrigine (619C89) is an inhibitor of glutamate release, TREK ion channels, TRESK channels, sodium channels, …
Formula:
C15H16Cl3N5
Purity:
100% - 99.49%
Color and Shape:
Solid
Molecular weight:
372.68
Ref: TM-T16887
| 1mg | 96.00 € | ||
| 2mg | 124.00 € | ||
| 5mg | 201.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 503.00 € | ||
| 1mL*10mM (DMSO) | 222.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
(R)-Baclofen hydrochloride
CAS:63701-55-3
Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.
Formula:
C10H13Cl2NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
250.12
Ref: TM-T17306
| 10mg | 87.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 328.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Vernakalant
CAS:794466-70-9
Vernakalant (RSD-1235) is a mixed ion channel blocker.
Formula:
C20H31NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
349.46
Ref: TM-TQ0307
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
