GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 363 products for "GABA Receptor".
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Nikethamide
CAS:Nikethamide is a stimulant which mainly influences the respiratory cycle. Widely known by its former sales name of Coramine, it was used in the mid-twentieth century as a medical countermeasure against tranquilizer overtreatments, before the advent of endFormula:C10H14N2OPurity:99.42%Color and Shape:SolidMolecular weight:178.23Baclofen
CAS:Baclofen (Lioresal), a chlorophenyl-butanoic acid derivative, treats spasms from spinal cord injury and MS by mimicking GABA at GABA-B receptors.Formula:C10H12ClNO2Purity:98% - 99.94%Color and Shape:1992)Molecular weight:213.66Isoguvacine hydrochloride
CAS:Isoguvacine hydrochloride (1,2,3,6-tetrahydro-4-pyridinecarboxylic acid hydrochloride) is a GABA receptor agonist.Formula:C6H10ClNO2Purity:99.59%Color and Shape:SolidMolecular weight:163.6Bemegride
CAS:Bemegride (3-Ethyl-3-methylglutarimide), a central nervous system stimulant, serves as an antidote for barbiturate poisoning.Formula:C8H13NO2Purity:99.89%Color and Shape:SolidMolecular weight:155.19Etifoxine hydrochloride
CAS:Etifoxine hydrochloride (HOE 36-801 hydrochloride) is an anxiolytic and anticonvulsant drug.Formula:C17H18Cl2N2OPurity:99.36%Color and Shape:SolidMolecular weight:337.24Fluxametamide
CAS:Fluxametamide, an isoxazoline insecticide, targets insect chloride channels with IC50s of 1.95 nM (GABA) and 225 nM (glutamate).Formula:C20H16Cl2F3N3O3Purity:99.49%Color and Shape:SolidMolecular weight:474.26Lotilaner
CAS:Lotilaner is a parasiticide.Formula:C20H14Cl3F6N3O3SPurity:99.56%Color and Shape:SolidMolecular weight:596.76Ref: TM-T15775
1mg42.00€2mg55.00€5mg89.00€1mL*10mM (DMSO)105.00€10mg137.00€25mg318.00€50mg522.00€100mg835.00€200mg1,125.00€FG 7142
CAS:FG 7142 (LSU-65), a benzodiazepine inverse agonist, targets α1 subunit GABAA receptors (EC50=137 nM, Ki=91 nM) and upregulates β-adrenoceptors.Formula:C13H11N3OPurity:98.75%Color and Shape:White SolidMolecular weight:225.25Ref: TM-T11277
2mg33.00€1mL*10mM (DMSO)39.00€5mg60.00€10mg92.00€25mg149.00€50mg213.00€100mg318.00€200mg442.00€3,4,5-Trimethoxycinnamic acid
CAS:3,4,5-Trimethoxycinnamic acid (O-Methylsinapic acid) (TMCA) is one of the constituents of Polygalae Radix and may exert anti-seizure activity by acting at theFormula:C12H14O5Purity:98.91%Color and Shape:SolidMolecular weight:238.24Furosemide sodium
CAS:Furosemide sodium: potent NKCC inhibitor, loop diuretic, treats heart failure, hypertension, edema, selective GABAA antagonist.Formula:C12H10ClN2NaO5SPurity:99.52% - >99.99%Color and Shape:SolidMolecular weight:352.73GET73
CAS:GET73 (Gamma hydroxybutyric acid analogue) is an negative allosteric modulator of mGluR5.Formula:C13H16F3NO2Purity:99.54%Color and Shape:SolidMolecular weight:275.27Ref: TM-T11393
5mg39.00€1mL*10mM (DMSO)44.00€10mg56.00€25mg104.00€50mg158.00€100mg230.00€200mg340.00€γ-Aminobutyric acid
CAS:γ-Aminobutyric acid (4-Aminobutyric acid) is the most common inhibitory neurotransmitter in the central nervous system.Formula:C4H9NO2Purity:99.95%Color and Shape:White SolidMolecular weight:103.12Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formula:C14H18N2O2Purity:97.37%Color and Shape:SolidMolecular weight:246.3Oxiracetam
CAS:Oxiracetam (ISF2522), a cyclic derivative of gamma-aminobutyric acid (GABA), is utilized for the treatment of cognitive impairments.Formula:C6H10N2O3Purity:99.67%Color and Shape:White Crystalline PowderMolecular weight:158.16L-Cycloserine
CAS:L-Cycloserine irreversibly inhibits E. coli GABA aminotransferase, raising GABA levels, an inhibitory neurotransmitter.Formula:C3H6N2O2Purity:99.92% - 99.99%Color and Shape:White SolidMolecular weight:102.09UK-124114
CAS:Selamectin, a derivative of ivermectin, is a macrocyclic lactone that enhances chloride channels in nematodes, inhibiting H. contortus larval growth.Formula:C43H63NO11Purity:99.64%Color and Shape:White SolidMolecular weight:769.96Phenibut
CAS:Phenibut (Aminophenylbutyric acid) is a central depressant and derivative of the naturally occurring inhibitory neurotransmitter γ-aminobutyric acid (GABA).Formula:C10H13NO2Purity:99.55%Color and Shape:SolidMolecular weight:179.22Chlormezanone
CAS:Chlormezanone (Trancopal) is a non-benzodiazepine that is used in the management of anxiety. It has been suggested for use in the treatment of muscle spasm.Formula:C11H12ClNO3SPurity:99.86% - >99.99%Color and Shape:Crystals SolidMolecular weight:273.74Broflanilide
CAS:Broflanilide metabolite desmethyl-broflanilide blocks GABA receptor in dieldrin-resistant insects, inhibiting S. litura at IC50 1.3 nM.Formula:C25H14BrF11N2O2Purity:99.82%Color and Shape:SolidMolecular weight:663.29Ref: TM-T10618
1mg50.00€2mg71.00€5mg105.00€1mL*10mM (DMSO)124.00€10mg170.00€25mg339.00€50mg557.00€100mg792.00€Pentetrazol
CAS:Pentylenetetrazol is a GABA(A) receptor antagonist, that displays activity as a central nervous system and respiratory stimulant.Formula:C6H10N4Purity:99.67% - 99.90%Color and Shape:SolidMolecular weight:138.17NEO 376
CAS:NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.Formula:C20H24ClN3OPurity:99.56%Color and Shape:SolidMolecular weight:357.88Ref: TM-T12207
1mg71.00€5mg133.00€1mL*10mM (DMSO)147.00€10mg205.00€25mg353.00€50mg495.00€100mg665.00€200mg893.00€Pivagabine
CAS:Pivagabine (CXB-722), a 4-aminobutyric acid derivative, modulates GABA, CRF, and crosses the rat blood-brain barrier.Formula:C9H17NO3Purity:99.87%Color and Shape:White SolidMolecular weight:187.24Topiramate
CAS:Topiramate (RWJ 17021) is a unique antiseizure medication that is used in the treatment of partial and generalized seizures.Formula:C12H21NO8SPurity:99.79% - 99.92%Color and Shape:White To Off-White Crystalline PowderMolecular weight:339.36GABAA receptor agent 1
CAS:GABAA receptor agent 1 has strong anticonvulsant activity and is a high affinity ligand of GABAA receptor.Formula:C13H8ClN3O2Purity:99.31%Color and Shape:SolidMolecular weight:273.67Ref: TM-T11349
1mg35.00€5mg79.00€1mL*10mM (DMSO)86.00€10mg111.00€25mg215.00€50mg323.00€100mg469.00€200mg647.00€Emamectin Benzoate
CAS:Emamectin Benzoate (MK-244), by binding gamma-aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropodsFormula:C56H81NO15Purity:98.68%Color and Shape:SolidMolecular weight:1008.256Clomethiazole
CAS:Clomethiazole (Distraneurin) is an orally active GABAA agonist and it is an anticonvulsant agent. It has potential for treating convulsive status epilepticus.Formula:C6H8ClNSPurity:99.06%Color and Shape:SolidMolecular weight:161.65LAU159
CAS:LAU159 is a functionally selective positive α1β3 GABA(A) receptor modulator(EC50 : 2.2 μM).Formula:C17H12ClN3O2Purity:98.7% - 99.38%Color and Shape:Yellow SolidMolecular weight:325.75Ref: TM-T11822
1mg110.00€2mg160.00€5mg219.00€10mg395.00€25mg653.00€50mg888.00€100mg1,243.00€500mg2,493.00€Phenelzine sulfate
CAS:Phenelzine sulfate is a non-selective and irreversible inhibitor of monoamine oxidase (MAOI), and with antidepressant and anxiolytic.Formula:C8H14N2O4SPurity:98.38% - 99.83%Color and Shape:SolidMolecular weight:234.27Domperidone EP Impurity A
CAS:Domperidone EP Impurity A is used as pharmaceutical intermediates.Formula:C12H14ClN3OPurity:99.97%Color and Shape:White SolidMolecular weight:251.71Flumazenil
CAS:Flumazenil (Ro 15-1788) antagonizes the benzodiazepine binding site of the gamma-aminobutyric acid (GABA)/benzodiazepine receptor complex in the central nervousFormula:C15H14FN3O3Purity:99.72% - 99.98%Color and Shape:Less Crystals Colourless CrystalsMolecular weight:303.29Afoxolaner
CAS:Afoxolaner is an isoxazoline insecticide/acaricide against Ixodes scapularis in dogs.Formula:C26H17ClF9N3O3Purity:99.1% - 99.38%Color and Shape:SolidMolecular weight:625.87α5-GABAA receptor modulator 1
α5-GABAA receptor modulator 1 (Compound A-4) is a selective silent allosteric modulator (SAM) targeting the α5 subunit of GABAA receptors, useful for research into central nervous system (CNS) disorders.Formula:C21H20FN3O4Color and Shape:SolidMolecular weight:397.4α-Casozepine
CAS:α-Casozepine,Bioactive peptide from milk α-S1 casein. Binds GABA receptors. Anti-anxiety effects.Formula:C60H94N14O16Purity:99.81%Color and Shape:SolidMolecular weight:1267.47RuBi-GABA
CAS:Ruthenium-bipyridine-triphenylphosphine caged GABAFormula:C42H39F6N5O2P2RuPurity:98%Color and Shape:SolidMolecular weight:922.8Emamectin B1a
CAS:Emamectin B1a can be used in relevant research in the life sciences. Its product number is T37663 and CAS number is 121124-29-6.Formula:C49H75NO13Color and Shape:SolidMolecular weight:886.133DAA-1106
CAS:DAA-1106 is a potent and selective ligand for PBR, acting as a potent and selective agonist at the peripheral benzodiazepine receptor.Formula:C23H22FNO4Purity:99.54%Color and Shape:SolidMolecular weight:395.42Nipecotic acid
CAS:Nipecotic acid ,with CAS No. 498-95-3, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Nipecotic acid provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.Formula:C6H11NO2Color and Shape:Off-White To Pale Yellow-Beige PowderMolecular weight:129.16AHN-683
CAS:AHN-683 is a fluorescent ligand. It was used for peripheral-type benzodiazepine receptors.Formula:C42H32FN3O7Purity:98%Color and Shape:SolidMolecular weight:709.72Chrodrimanin B
CAS:Chrodrimanin B is a useful organic compound for research related to life sciences. The catalog number is T126052 and the CAS number is 132196-54-4.Formula:C27H32O8Color and Shape:SolidMolecular weight:484.545Anticonvulsant agent 8
Anticonvulsant agent 8 (compound D4) is a chemical used in treating epilepsy by inhibiting GABAA currents. In mouse models, its ED50 values are 2.23 mg/kg for the maximal electroshock (MES) test and 24.60 mg/kg for the pentylenetetrazol (PTZ) test.Formula:C15H11N5OColor and Shape:SolidMolecular weight:277.28(Iso)-Atagabalin HCl
CAS:(Iso)-Atagabalin HCl(isomer-Atagabalin HCl) is an alpha -2- delta ligand that can be used to treat non-restorative sleep.Formula:C10H20ClNO2Purity:99.88% - >99.99%Color and Shape:SoildMolecular weight:221.72Azocarnil
Azocarnil is a GABAergic agonist-enhancer used in neurological system research.Color and Shape:Odour SolidLesogaberan napadisylate
CAS:Lesogaberan (AZD-3355) is a selective GABAB agonist with EC50 of 8.6 nM, Ki of 5.1 nM in rats, and acts peripherally on the esophageal sphincter.Formula:C13H17FNO5PSColor and Shape:SolidMolecular weight:349.3112,14-Dichlorodehydroabietic acid
CAS:12,14-Dichlorodehydroabietic acid activates BK channels, blocks GABA A receptors, and increases calcium and neurotransmitter release.Formula:C20H26Cl2O2Color and Shape:SolidMolecular weight:369.33Antidepressant agent 4
Antidepressant agent 4: orally active, has antidepressant, anxiolytic, and nootropic effects.Formula:C19H38ClN5O2SColor and Shape:SolidMolecular weight:436.06epi-Aszonalenin A
CAS:epi-Aszonalenin A: a psychoactive benzodiazepine from Aspergillus novofumigatus.Formula:C25H25N3O3Color and Shape:SolidMolecular weight:415.48Neurotransmitter Receptor Compound Library
A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；
Color and Shape:Odour SolidIon Channel Targeted Library
A unique collection of 931 compounds targeting ion channels for research in ion channels-related diseases and ion channel drug discovery;Color and Shape:Odour SolidRef: TM-L2300
1mgTo inquire30μL*10mM (DMSO)To inquire50μL*10mM (DMSO)To inquire100μL*10mM (DMSO)To inquire250μL*10mM (DMSO)To inquireCGP 35348
CAS:CGP 35348 是 GABAB 受体的选择性拮抗剂 (EC50 = 34 μM)。 CGP 35348 可用于研究白化新生小鼠脑损伤后的神经肌肉协调和空间学习。Formula:C8H20NO4PPurity:99.92%Color and Shape:Yellow SolidMolecular weight:225.22Fipronil sulfone
CAS:Fipronil sulfone is an insecticide fipronil. Its metabolite fipronil sulphone is an inhibitor of rat ɑ1β2γ2L GABA(A) receptor.Formula:C12H4Cl2F6N4O2SPurity:98%Color and Shape:SolidMolecular weight:453.14
