GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 363 products for "GABA Receptor".
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CGP 36742
CAS:CGP 36742 blocks GABAB receptor, crosses blood-brain barrier, aids depression treatment (IC50: 32 μM).Formula:C7H18NO2PColor and Shape:SolidMolecular weight:179.2Vigabatrin Hydrochloride
CAS:Vigabatrin Hydrochloride (γ-Vinyl-GABA hydrochloride) is a structural analog of the GABA, irreversibly inhibiting the catabolism of GABA by GABA transaminase.Formula:C6H11NO2·HClPurity:98%Color and Shape:SolidMolecular weight:165.62Valnoctamide
CAS:Valnoctamide (Valmethamide) has antiepileptic and anticonvulsant activity and may be used in the study of neurological disorders.Formula:C8H17NOPurity:98%Color and Shape:SolidMolecular weight:143.23DL-Menthol
CAS:DL-Menthol ((±)-Menthol) is a racemic mixture of the monoterpene alcohols (–)-menthol and (+)-menthod, which have been found in Cannabis.Formula:C10H20OPurity:99.16% - 99.74%Color and Shape:White Crystals /89-78-1/ Physical Description White Crystalline Solid With A Peppermint Odor And Taste (Ntp 1992)Molecular weight:156.27Neurotensin TFA
Neurotensin TFA (39379-15-2) is a 13-amino acid neuropeptide with opioid-independent pain relief, acting in the CNS and gut, linked to numerous disorders.Formula:C80H122F3N21O22Purity:99.41%Color and Shape:White SolidMolecular weight:1786.98Ocinaplon
CAS:Ocinaplon (DOV 273547) is a GABAA receptors modulator.Formula:C17H11N5OPurity:99.81%Color and Shape:SolidMolecular weight:301.3Gabazine free base
CAS:Gabazine free base is a specific antagonist of the GABA receptor. It does not affect GABA-transaminase or glutamate-decarboxylase activities.Formula:C15H17N3O3Color and Shape:SolidMolecular weight:287.31Ginkgolide A
CAS:Ginkgolide A (BN-52020), from Ginkgo biloba leaves, is an active PAF antagonist with potential in treating inflammation and immune disorders.Formula:C20H24O9Purity:98.76% - 99.81%Color and Shape:White SolidMolecular weight:408.406-Methylflavone
CAS:6-Methylflavone is an activator of α1β2γ2L and α1β2 GABAA receptors.Formula:C16H12O2Purity:99.69%Color and Shape:White SolidMolecular weight:236.27Saclofen
CAS:Saclofen is a GABA analog and GABAB receptor antagonist, useful for studying inhibitory brain signals. IC50: 7.8 μM.Formula:C9H12ClNO3SPurity:99.17%Color and Shape:SolidMolecular weight:249.71Ref: TM-T4440
1mg52.00€1mL*10mM (DMSO)108.00€5mg113.00€10mg177.00€25mg340.00€50mg550.00€100mg860.00€200mg1,161.00€Baclofen hydrochloride
CAS:Baclofen HCL, a GABA-B agonist, treats muscle spasticity by reducing excitatory transmission.Formula:C10H13Cl2NO2Purity:99.55%Color and Shape:SolidMolecular weight:250.122γ-Acetylenic GABA
CAS:γ-Acetylenic GABA (4-Aminohex-5-ynoic acid) is a potent, irreversible inhibitor of GABA-transaminase.Formula:C6H9NO2Color and Shape:SolidMolecular weight:127.143(+)-Kavain
CAS:(+)-Kavain ((R)-KAWAIN) is one of the six major kavalactones found in the Piper methysticum (kava) plant; reversible inhibitor of MAO-B.Formula:C14H14O3Purity:97% - ≥95%Color and Shape:White Fine PowderMolecular weight:230.26Phenibut (hydrochloride)
CAS:Phenibut hydrochloride (3-Amino-4-phenylbutyric acid hydrochloride) is a GABA mimetic that acts as an agonist at GABAB receptors.Formula:C10H14ClNO2Purity:99.93%Color and Shape:White SolidMolecular weight:215.68Thiocolchicoside
CAS:Thiocolchicoside, a muscle relaxant, has anti-inflammatory and analgesic properties; not for seizure-prone people.Formula:C27H33NO10SPurity:99.11% - 99.39%Color and Shape:SolidMolecular weight:563.62(-)-Securinine
CAS:(-)-Securinine (Securinine) is plant-derived alkaloid and also a GABAA receptor antagonist.Formula:C13H15NO2Purity:99.58% - 99.87%Color and Shape:Yellow SolidMolecular weight:217.26Imepitoin
CAS:Imepitoin (AWD 131-138), a new low-affinity partial benzodiazepine receptor agonist, shows potent anticonvulsant and anxiolytic properties in rodent models.Formula:C13H14ClN3O2Purity:99.82%Color and Shape:SolidMolecular weight:279.72Tiagabine hydrochloride
CAS:Tiagabine hydrochloride, a nipecotic acid derivative, is an anticonvulsant and selective GABA reuptake inhibitor.Formula:C20H25NO2S2·HClPurity:99.09% - 99.77%Color and Shape:SolidMolecular weight:412.016-(4-Methoxyphenyl)-3-pyridazinamine
CAS:6-(4-Methoxyphenyl)-3-pyridazinamine is a GABAA receptor antagonistFormula:C11H11N3OPurity:99.03%Color and Shape:Yellow SolidMolecular weight:201.22L-838417-D9
CAS:L-838417 D9 (C-21191) is a novel deuterated subtype-selective GABAA positive allosteric modulator, acting as a partial agonist at α2, α3 and α5 subtypes[1].Formula:C19H10D9F2N7OPurity:99.65%Color and Shape:SolidMolecular weight:408.45(R)-baclofen
CAS:(R)-baclofen (STX209), a derivative of gamma-aminobutyric acid, is commonly utilized for the treatment of spasticity.Formula:C10H12ClNO2Purity:97.20% - 98.94%Color and Shape:White SolidMolecular weight:213.66Arecaidine hydrochloride
CAS:Arecaidine hydrochloride may have carcinogenesis.Formula:C7H12ClNO2Purity:99.69% - ≥95%Color and Shape:White SolidMolecular weight:177.63Ref: TM-T5799
2mg34.00€5mg48.00€1mL*10mM (DMSO)49.00€10mg67.00€25mg100.00€50mg149.00€100mg213.00€200mg316.00€Temgicoluril
CAS:Temgicoluril (mebikar) acts on GABA Receptor.Formula:C8H14N4O2Purity:99.8%Color and Shape:SolidMolecular weight:198.22SKF89976A HCl
CAS:SKF89976A: GABA uptake inhibitor, selective for GAT-1, passes blood-brain barrier, active in vivo (IC50: 0.13 μM hGAT-1).Formula:C22H25NO2Color and Shape:SolidMolecular weight:335.44Gaboxadol hydrochloride
CAS:Gaboxadol (hydrochloride) is a GABAA receptor agonist.Formula:C6H9ClN2O2Purity:98.43% - 99.39%Color and Shape:White SolidMolecular weight:176.601Lorediplon
CAS:Lorediplon is a novel hypnotic drug acting as a GABAA receptor modulator, differentially active at the α1-subunit, associated with promoting sleep.Formula:C20H15FN4O2SPurity:99.12% - 99.19%Color and Shape:SolidMolecular weight:394.42Gabazine
CAS:Gabazine (SR95531) is an antagonist of GABAA receptors (Ki : 74-150 nM)Formula:C15H18BrN3O3Purity:98.51% - 99.24%Color and Shape:White SolidMolecular weight:368.23Pipequaline hydrochloride
CAS:Pipequaline hydrochloride (PK-8165 hydrochloride) is an anticonflict & anticonvulsant quinoline derivative.Formula:C22H25ClN2Purity:99.78%Color and Shape:Yellow SolidMolecular weight:352.9(2S)-6-Prenylnaringenin
CAS:(2S)-6-Prenylnaringenin (6-Prenylnaringenin) is an isomer of the potent phytoestrogen, 8-prenylnaringenin.Formula:C20H20O5Purity:99.47%Color and Shape:SolidMolecular weight:340.37α-Thujone
CAS:α-Thujone is an inhibitor of ACh with an IC50 value of 24.7μM.Formula:C10H16OPurity:97.02% - 98.41%Color and Shape:Transparent OilMolecular weight:152.23Piperazine citrate
CAS:Piperazine citrate, an organic compound, consists of a six-membered ring, containing two nitrogen atoms at opposite positions in the ring.Formula:C24H46N6O14Purity:99.8%Color and Shape:Crystals IndicationMolecular weight:642.652'-O-Methylisoliquiritigenin
CAS:2'-O-Methylisoliquiritigenin, a compound synthesized by enzymes specifically induced in NR.2'-O-Methylisoliquiritigenin, isolated from the Arachis species, up-Formula:C16H14O4Purity:98.75%Color and Shape:SolidMolecular weight:270.28U93631
CAS:GABAA antagonist; binds picrotoxin site, stabilizes inactive channel. Speeds GABA-induced Cl- decay, minor peak effect. Inhibits 5-HT3A receptors.Formula:C17H21N3O2Purity:99.65% - 99.76%Color and Shape:SolidMolecular weight:299.37Ginsenoside Rc
CAS:Ginsenoside Rc (Panaxoside Rc) is one of the ginsenosides from Panax ginseng, inhibits the expression of TNF-α and IL-1β.Formula:C53H90O22Purity:98.83% - 99.86%Color and Shape:White SolidMolecular weight:1079.27Cholesterol myristate
CAS:Cholesterol myristate, a natural steroid in Chinese medicine, affects GABAA, nicotinic receptors, and potassium channels.Formula:C41H72O2Purity:99.65%Color and Shape:White SolidMolecular weight:597.01Tiagabine
CAS:Tiagabine (NO050328) is an Anti-epileptic Agent.Formula:C20H25NO2S2Purity:99.25% - 99.67%Color and Shape:White To Off-White Crystalline SolidMolecular weight:375.55Acetoxyvalerensre
CAS:Acetoxyvalerensre (acetylvalerenolic acid) (acetylvalerenolic acid) is a derivative of valerenic acid, which is a a GABAA receptor modulator.Formula:C17H24O4Purity:98.22%Color and Shape:SolidMolecular weight:292.37Fipronil
CAS:Controlled ProductFipronil (Fluocyanobenpyrazole) is a broad-use insecticide that belongs to the phenylpyrazole chemical family.Formula:C12H4Cl2F6N4OSPurity:97.21%Color and Shape:White SolidMolecular weight:437.15SKF89976A hydrochloride
CAS:SKF89976A hydrochloride (d,l-SKF89976A hydrochloride) is a selective inhibitor GABA transporter such as GAT-1 (IC50s = 0.28 μM), GAT-2 (IC50s = 137.34 μM) andFormula:C22H26ClNO2Purity:98.02%Color and Shape:SolidMolecular weight:371.9Ref: TM-T12930
1mg34.00€5mg65.00€1mL*10mM (DMSO)71.00€10mg89.00€25mg167.00€50mg264.00€100mg409.00€200mg590.00€α-Asarone
CAS:alpha-Asarone (trans-Asarone) is a psychoactive compound with antidepressant-like activity in mice.Formula:C12H16O3Purity:99.64% - 99.64%Color and Shape:SolidMolecular weight:208.25Miltirone
CAS:Miltirone is a CYPs inhibitor, it has been characterized as a low-affinity ligand for central benzodiazepine receptors.Formula:C19H22O2Purity:99.22% - 99.66%Color and Shape:SolidMolecular weight:282.38Amentoflavone
CAS:Amentoflavone (3',8''-Biapigenin), as a potent inhibitor of CYP3A4 and CYP2C9, can interact with many other medications.Formula:C30H18O10Purity:98.81% - 99.78%Color and Shape:Yellow SolidMolecular weight:538.46Ref: TM-T3417
2mg34.00€5mg50.00€1mL*10mM (DMSO)59.00€10mg80.00€25mg126.00€50mg215.00€100mg349.00€200mg512.00€AZD-6280
CAS:AZD6280 is a novel, subtype-selective GABAAα2/3 receptor positive modulators, used for treatment of generalized anxiety disorder.Formula:C20H22N4O3Purity:98.99%Color and Shape:White SolidMolecular weight:366.41Ref: TM-T7136
1mg215.00€5mg439.00€1mL*10mM (DMSO)484.00€10mg640.00€25mg1,018.00€50mg1,423.00€100mg1,935.00€Songorine
CAS:Songorine (Napellonine) shows anti-tumor activity in preliminary pharmacological verification trials including cell proliferation and molecular docking assays.Formula:C22H31NO3Purity:98% - 99.92%Color and Shape:SolidMolecular weight:357.49CL 218872
CAS:CL 218872: selective α1 GABAA receptor agonist, anxiolytic, and anticonvulsant; Ki=130 nM for α1, less potent for α2-α6.Formula:C13H9F3N4Purity:99.92%Color and Shape:SolidMolecular weight:278.23Kavain
CAS:Kavain, a compound extracted from the Kava plant, Piper methysticum, is found to be involved in TNF-α expression in human and mouse cells via regulation ofFormula:C14H14O3Purity:99.93% - ≥95%Color and Shape:SolidMolecular weight:230.26SSD114 HCl
CAS:SSD114 is a novel GABAB receptor positive allosteric modulator.Formula:C18H21ClF3N3OPurity:99.03% - 99.95%Color and Shape:White SolidMolecular weight:387.83Ref: TM-T4522
2mg34.00€1mL*10mM (DMSO)46.00€5mg50.00€10mg75.00€25mg111.00€50mg172.00€100mg290.00€200mg419.00€2'MeO6MF
CAS:2'MeO6MF is a brain-penetrant positive allosteric modulator at α2β1γ2L and all α1-containing GABAA receptors.It offers neuroprotection and improved functionalFormula:C17H14O3Purity:99.28% - 99.63%Color and Shape:SolidMolecular weight:266.29Ref: TM-T8887
1mg49.00€1mL*10mM (DMSO)96.00€5mg102.00€10mg152.00€25mg243.00€50mg340.00€100mg460.00€200mg627.00€Tiagabine hydrochloride hydrate
CAS:Tiagabine HCl hydrate, IC50: 67-446 nM, selectively inhibits GABA uptake, acts as an anticonvulsant.Formula:C20H28ClNO3S2Color and Shape:SolidMolecular weight:430.02rac-BHFF
CAS:rac-BHFF, a GABA B receptor modulator, boosts GABA potency >15x, efficacy >149%, has anxiolytic effects, and is orally active.Formula:C17H21F3O3Purity:99.69% - >99.99%Color and Shape:SolidMolecular weight:330.34Ref: TM-T4176
2mg40.00€5mg57.00€1mL*10mM (DMSO)67.00€10mg90.00€25mg177.00€50mg295.00€100mg447.00€200mg622.00€
