PPAR
Peroxisome Proliferator-Activated Receptors (PPARs) are a group of nuclear receptor proteins that function as transcription factors regulating the expression of genes involved in metabolism, particularly fatty acid storage and glucose metabolism. PPAR inhibitors are important tools for studying metabolic disorders such as diabetes, obesity, and cardiovascular diseases. These inhibitors can modulate lipid metabolism, insulin sensitivity, and inflammation, making them valuable in therapeutic research. At CymitQuimica, we offer a range of PPAR inhibitors to support your research in metabolic diseases, endocrinology, and drug development.
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OPHIOPOGONIN D
CAS:945619-74-9
Ophiopogonin D is a natural product,and is a CYP2J3 inducer that significantly inhibits Ang II …
Formula:
C44H70O16
Purity:
99.46% - ≥95%
Color and Shape:
Solid
Molecular weight:
855.02
Ref: TM-T5701
| 1mg | 69.00 € | ||
| 5mg | 152.00 € | ||
| 10mg | 198.00 € | ||
| 25mg | 334.00 € | ||
| 50mg | 487.00 € | ||
| 100mg | 693.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
BMS-687453
CAS:1000998-59-3
BMS-687453 is a potent and selective PPAR alpha agonist, with an EC(50) of 10 nM …
Formula:
C22H21ClN2O6
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
444.86
Ref: TM-T5532
| 1mg | 46.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 427.00 € | ||
| 100mg | 647.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Furegrelate
CAS:85666-24-6
FUREGRELATE, a thromboxane A2 (TxA2) synthase inhibitor, blunts the development of pulmonary arterial hypertension in …
Formula:
C15H11NO3
Purity:
100%
Color and Shape:
Odour Color
Molecular weight:
253.25
Ref: TM-T11339L
| 1mg | 111.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 355.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 1,016.00 € | ||
| 200mg | 1,354.00 € | ||
| 1mL*10mM (DMSO) | 218.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Licarin B
CAS:51020-87-2
1.(-)-Licarin B (Licarine B) has anti-mycobacterial activity.
Formula:
C20H20O4
Purity:
100% - ≥95%
Color and Shape:
Solid
Molecular weight:
324.37
Ref: TM-T4S1545
| 1mg | 39.00 € | ||
| 5mg | 75.00 € | ||
| 10mg | 106.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 252.00 € | ||
| 100mg | 379.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Eupatilin
CAS:22368-21-4
Eupatilin (NSC-122413), a flavone derived from Artemisia princepsPampanini, is a PPARα agonist, with pharmacological activity.
Formula:
C18H16O7
Purity:
98.42% - 99%
Color and Shape:
Solid
Molecular weight:
344.32
Ref: TM-T3362
| 1mg | 36.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 202.00 € | ||
| 50mg | 357.00 € | ||
| 100mg | 522.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
GW9662
CAS:22978-25-2
GW9662 (TIMTEC-BB SBB006523) is a specific PPARγ antagonist, with 100 to 1000-fold functional selectivity for …
Formula:
C13H9ClN2O3
Purity:
98% - 99.94%
Color and Shape:
Off-White Solid
Molecular weight:
276.68
Ref: TM-T2260
| 5mg | 51.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 202.00 € | ||
| 500mg | 504.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
SR1664
CAS:1338259-05-4
SR1664 is a potent and selective PPARγ inhibitor with potential antidiabetic activity.
Formula:
C33H29N3O5
Purity:
98.02%
Color and Shape:
Solid
Molecular weight:
547.6
Ref: TM-T23389
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 300.00 € | ||
| 50mg | 533.00 € | ||
| 100mg | 766.00 € | ||
| 500mg | 1,574.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Lonazolac
CAS:53808-88-1
Lonazolac is a nonsteroidal anti-inflammatory drug[1].
Formula:
C17H13ClN2O2
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
312.75
Ref: TM-T50025
| 5mg | 57.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 128.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 277.00 € | ||
| 200mg | 417.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
FH535
CAS:108409-83-2
FH535, a Wnt/β-catenin signaling and PPAR inhibitor, exhibits anti-tumor activities.
Formula:
C13H10Cl2N2O4S
Purity:
98.25% - 99.5%
Color and Shape:
Solid
Molecular weight:
361.2
Ref: TM-T2413
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 92.00 € | ||
| 50mg | 161.00 € | ||
| 100mg | 270.00 € | ||
| 200mg | 397.00 € | ||
| 500mg | 642.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Icariin
CAS:489-32-7
Icariin (Ieariline) is a flavonol glycoside that inhibits PDE5 and PDE4 activity and is a …
Formula:
C33H40O15
Purity:
97.64% - 98.49%
Color and Shape:
Solid
Molecular weight:
676.66
Ref: TM-T2855
| 50mg | 44.00 € | ||
| 100mg | 56.00 € | ||
| 200mg | 77.00 € | ||
| 500mg | 103.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Glabrone
CAS:60008-02-8
Glabrone shows antiviral activity against influenza virus.
Formula:
C20H16O5
Purity:
99.08% - 99.55%
Color and Shape:
Solid
Molecular weight:
336.34
Ref: TM-TN1693
| 1mg | 113.00 € | ||
| 5mg | 278.00 € | ||
| 10mg | 403.00 € | ||
| 25mg | 669.00 € | ||
| 50mg | 921.00 € | ||
| 100mg | 1,278.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
GW6471
CAS:880635-03-0
GW6471 is an antagonist of PPARα. GW6471 enhances the binding affinity of the PPAR α …
Formula:
C35H36F3N3O4
Purity:
98.38% - 99.88%
Color and Shape:
Solid
Molecular weight:
619.67
Ref: TM-T8486
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 104.00 € | ||
| 25mg | 211.00 € | ||
| 50mg | 420.00 € | ||
| 100mg | 609.00 € | ||
| 500mg | 1,263.00 € | ||
| 1mL*10mM (DMSO) | 121.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Palmitelaidic Acid
CAS:10030-73-6
Palmitelaidic Acid (trans-Palmitoleic acid) is one of the most abundant fatty acids in serum and …
Formula:
C16H30O2
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
254.41
Ref: TM-T19500
| 10mg | 86.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
NSC-87877 disodium
CAS:56932-43-5
NSC-87877 disodium (NSC87877) is a cell-permeable inhibitor of both SHP-1 and SHP-2. NSC-87877 also inhibits …
Formula:
C19H13N3O7S2·2Na
Purity:
97.89%
Color and Shape:
Solid
Molecular weight:
503.42
Ref: TM-T6911
| 5mg | 45.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 268.00 € | ||
| 200mg | 382.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
SR 16832
CAS:2088135-12-8
SR 16832: Dual-site PPARγ inhibitor; outperforms GW 9662, T 0070907 in ligand binding, transcription inhibition.
Formula:
C17H12ClN3O4
Purity:
99.60%
Color and Shape:
Solid
Molecular weight:
357.75
Ref: TM-T24827
| 5mg | 45.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 300.00 € | ||
| 200mg | 434.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
GW0742
CAS:317318-84-6
GW0742 (GW610742) is an effective and specific PPARδ agonist (EC50: 1 nM/1.1 μM/2 μM, for …
Formula:
C21H17F4NO3S2
Purity:
99.83% - 99.85%
Color and Shape:
Solid
Molecular weight:
471.49
Ref: TM-T6524
| 5mg | 50.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 215.00 € | ||
| 100mg | 373.00 € | ||
| 500mg | 886.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
CDDO-Im
CAS:443104-02-7
CDDO-Im (TP-235) is an activator of Nrf2 and PPAR (Kis: 232/344 nM for PPARα/PPARγ).
Formula:
C34H43N3O3
Purity:
100% - 98.3%
Color and Shape:
Solid
Molecular weight:
541.72
Ref: TM-TQ0120
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 331.00 € | ||
| 100mg | 500.00 € | ||
| 500mg | 1,068.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
SC-236
CAS:170569-86-5
SC-236 (Sc 236) is an orally active and selective inhibitor of COX-2 (IC50 of 0.005 …
Formula:
C16H11ClF3N3O2S
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
401.79
Ref: TM-T8505
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 195.00 € | ||
| 50mg | 347.00 € | ||
| 100mg | 515.00 € | ||
| 1mL*10mM (DMSO) | 84.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Raspberry ketone
CAS:5471-51-2
1.
Formula:
C10H12O2
Purity:
99.89%
Color and Shape:
White Solid Crystalline
Molecular weight:
164.2
Ref: TM-T2S0633
| 100mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
Fisetin
CAS:528-48-3
Fisetin belongs to a group of natural flavonols with anti-inflammatory, antioxidant, anti-tumor, anti-aging and neuroprotective …
Formula:
C15H10O6
Purity:
94.14% - 98.31%
Color and Shape:
Yellow To Brown Crystalline Powder
Molecular weight:
286.24
Ref: TM-T2879
| 100mg | 53.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 18 Dec 2024
