Transferase
Transferases are a large class of enzymes that catalyze the transfer of functional groups, such as methyl, glycosyl, and phosphate groups, from one molecule to another. Inhibitors of transferases are used to study a wide range of biological processes, including signal transduction, metabolism, and gene expression. These inhibitors are essential tools in research areas such as cancer, metabolic diseases, and epigenetics, where dysregulation of transferase activity is implicated. At CymitQuimica, we offer a comprehensive selection of transferase inhibitors to support your research in enzymology, cell signaling, and disease mechanisms.
Found 42 products for "Transferase".
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CP-609754
CAS:CP-609754 shows selective inhibition of farnesyltransferase.Formula:C29H22ClN3O2Purity:99.86% - 99.87%Color and Shape:SolidMolecular weight:479.957Tipifarnib
CAS:Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.Formula:C27H22Cl2N4OPurity:97.1% - 99.94%Color and Shape:Off-White To Pale Beige SolidMolecular weight:489.3963-O-Methyltolcapone
CAS:3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.Formula:C15H13NO5Purity:98%Color and Shape:SolidMolecular weight:287.2674FUT8-IN-1
FUT8-IN-1 (Compound 37) is an inhibitor of α-1,6-fucosyltransferase (FUT8), with a dissociation constant (KD) of 49 nM and an IC50 around 50 µM. In the presence of FUT8, FUT8-IN-1 forms a highly active naphthoquinone imine intermediate, thereby inhibiting FUT8's enzymatic activity.Formula:C23H25ClN2OColor and Shape:SolidMolecular weight:380.91Lith-O-Asp
CAS:Lith-O-Asp is a sialyltransferase inhibitor; Ki=1.3 μM; reduces sialylation; inhibits cancer cell invasion; metastasis research.Formula:C28H45NO6Color and Shape:White SolidMolecular weight:491.66Lucerastat
CAS:Lucerastat（NBDGJ） is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.Formula:C10H21NO4Purity:98%Color and Shape:White SolidMolecular weight:219.278P-3FAX-Neu5Ac
CAS:P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.Formula:C22H30FNO14Purity:97.08%Color and Shape:White SolidMolecular weight:551.47Prenyl-IN-1
CAS:Prenyl-IN-1 inhibits prenylation selectively, counters oxidative stress in Parkinson's.Formula:C28H24ClN5O2Purity:>99.99%Color and Shape:SolidMolecular weight:497.98PDMP hydrochloride
CAS:PDMP, a glucosylceramide synthase inhibitor with 4 stereoisomers, acts at 0.8μM; D-threo enantiomer also blocks lactosylceramide synthesis.Formula:C23H39ClN2O3Color and Shape:SolidMolecular weight:427.03DGAT1-IN-3
CAS:DGAT1-IN-3 is an orally active DGAT-1 inhibitor (IC₅₀: 38 nM human, 120 nM rat) for obesity and metabolic syndrome research.Formula:C20H19F3N4O3Purity:99.83%Color and Shape:SolidMolecular weight:420.3851EBU-141
EBU-141 is a human monoclonal antibody (mAb) targeting CD75/ST6GAL1, suitable for research in B-cell lymphoma and multiple myeloma.Ibiglustat (L-Malic acid)
CAS:Ibiglustat (L-Malic acid) (Ibiglustat L-Malic acid) is a selective, brain-penetrant, and allosteric inhibitor of glucosylceramide synthase.Formula:C24H30FN3O7SPurity:99.54%Color and Shape:SolidMolecular weight:523.574FGTI-2734
CAS:FGTI-2734, a dual FT/GGT-1 inhibitor (IC50: 250/520 nM), blocks KRAS membrane binding and curbs KRAS-driven pancreatic cancer.Formula:C26H31FN6O2SPurity:99.69%Color and Shape:SolidMolecular weight:510.627Pactimibe sulfate
CAS:Pactimibe sulfate (CS-505) is a dual ACAT1/2 inhibitor for cholesterol metabolism and atherosclerosis research.Formula:C50H82N4O10SPurity:99.08%Color and Shape:SolidMolecular weight:931.27Miglustat hydrochloride
CAS:Miglustat hydrochloride (N-Butyldeoxynojirimycin hydrochloride) is an inhibitor of glucosylceramide synthase and can be used for studies about Type I GaucherFormula:C10H22ClNO4Purity:99.85%Color and Shape:SolidMolecular weight:255.74OSMI-1
CAS:OSMI-1: cell-permeable OGT inhibitor, blocks O-GlcNAcylation (IC50: 2.7 μM), no effect on other cell glycans.Formula:C28H25N3O6S2Purity:96.79% - 99.66%Color and Shape:White SolidMolecular weight:563.645Darlifarnib
CAS:Darlifarnib (Compound (S)-058) is an inhibitor of farnesyl transferase and geranylgeranyltransferase, with IC50 values of ≤ 10 nM and > 1000 nM, respectively. It exhibits high metabolic stability in human and mouse liver microsomes, with a half-life of over 100 minutes.Formula:C29H20N6OColor and Shape:SolidMolecular weight:468.509Glucosylceramide synthase-IN-4
CAS:Glucosylceramide Synthase-IN-4 (compound 12) serves as a potent inhibitor of glucosylceramide synthase (GCS), exhibiting an IC50 of 6.8 nM. It demonstrates superior pharmacokinetic properties and robust stability in human hepatocytes. Additionally, this compound is noted for its effective CNS penetration and acceptable PXR selectivity [1].Formula:C22H18F5N3O3Color and Shape:SolidMolecular weight:467.39ICMT-IN-55
CAS:ICMT-IN-55 (compound 31) acts as an ICMT inhibitor, exhibiting an IC50 value of 90 nM [1].Formula:C22H26F3NO2Color and Shape:SolidMolecular weight:393.44PF-07202954
CAS:PF-07202954 is a DGAT2 inhibitor with a long half-life. reduce the triglyceride content in the liver of rats fed with a Western diet, NASH.Formula:C22H23FN6O3Purity:98.99%Color and Shape:Yellow SolidMolecular weight:438.45
