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5-HT Receptor

5-HT Receptor

5-HT receptors, also known as serotonin receptors, are a group of G protein-coupled receptors (GPCRs) that mediate the effects of serotonin, a neurotransmitter involved in mood regulation, anxiety, sleep, appetite, and other physiological processes. These receptors are divided into several subtypes, each with distinct functions and pharmacological properties. 5-HT receptor modulators are widely studied for their roles in treating depression, anxiety disorders, and other neuropsychiatric conditions. At CymitQuimica, we offer a range of high-quality 5-HT receptor modulators to support your research in neuropharmacology, mood disorders, and GPCR signaling.

Found 940 products of "5-HT Receptor"

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  • Cisapride hydrate

    CAS:
    <p>Cisapride acts directly as a selective agonist of serotonin 5-HT4 receptor with IC50 value of 0.483 μM. And It also acts indirectly as a parasympathomimetic.</p>
    Formula:C23H31ClFN3O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:483.96
  • Cinanserin hydrochloride

    CAS:
    <p>Cinanserin hydrochloride (SQ 10643) is a 5-HT2 receptor blocker (Ki: 41 nM) and SARS-CoV 3C-like protease inhibitor.</p>
    Formula:C20H25ClN2OS
    Purity:99.57%
    Color and Shape:Solid
    Molecular weight:376.94
  • pCPA methyl ester hydrochloride

    CAS:
    <p>pCPA methyl ester HCl inhibits tryptophan hydroxylase, 5-HT synthesis, crosses blood-brain barrier, lowers central 5-HT.</p>
    Formula:C10H13Cl2NO2
    Purity:99.73% - 99.88%
    Color and Shape:Solid
    Molecular weight:250.12
  • Galanin (1-15) (porcine, rat)

    CAS:
    <p>N-terminal galanin fragment used to mediate central cardiovascular effects</p>
    Formula:C72H105N19O20
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1556.72
  • Oxatomide

    CAS:
    <p>Oxatomide: Dual H1/P2X7 antagonist, antihistamine, anti-allergic, treats immune diseases, IC50: 0.95 μM (P2X7), 0.43 μM (5-HT).</p>
    Formula:C27H30N4O
    Purity:98.82% - 99.72%
    Color and Shape:White Powder
    Molecular weight:426.55
  • SC-53116

    CAS:
    <p>SC-53116 HCl can increase the production of serotonin in central nervous system tissues and is a psychoactive agent.</p>
    Formula:C16H22ClN3O2
    Color and Shape:Solid
    Molecular weight:323.82
  • Minaprine

    CAS:
    <p>Minaprine is a reversible inhibitor of MAO-A, used in the treatment of various depressive states.</p>
    Formula:C17H22N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:298.38
  • 4-fluoro MBZP

    CAS:
    <p>4-fluoro MBZP is a novel psychoactive substance in the phenylpiperazine class, utilized for studies on the 5-HT2 receptors in the central nervous system.</p>
    Formula:C12H17FN2
    Color and Shape:Solid
    Molecular weight:208.28
  • FFN246

    CAS:
    <p>FFN246, a fluorescent probe, concurrently targets the serotonin transporter (SERT) and vesicular monoamine transporter 2 (VMAT2), exhibiting excitation and</p>
    Formula:C15H13FN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:256.27
  • Antipsychotic agent-2


    <p>Compound 11: potent antipsychotic, binds 5-HT1A/2A/2C, D2, H1 receptors; K is 56.6-1140 nM, BBB permeable.</p>
    Formula:C22H26FN5O
    Color and Shape:Solid
    Molecular weight:395.47
  • Tiaspirone hydrochloride

    CAS:
    <p>Tiaspirone hydrochloride (BMY-13859 hydrochloride) exhibits antipsychotic activity and influences the electrophysiological activity of dopaminergic neurons.</p>
    Formula:C24H33ClN4O2S
    Purity:99.87%
    Color and Shape:Soild
    Molecular weight:477.06
  • Ro60-0175

    CAS:
    <p>Ro60-0175 is a selective 5-HT2B and 5-HT2C serotonin receptor agonist, often used as fumarate.</p>
    Formula:C11H12ClFN2
    Purity:97.09%
    Color and Shape:Solid
    Molecular weight:226.68
  • AL 34662

    CAS:
    <p>AL 34662 is a selective and potent 5-HT2A receptor agonist with IC50s of 0.77 nM and 1.5 nM for rat and human 5-HT2 receptors, respectively.AL 34662 is also a</p>
    Formula:C10H13N3O
    Purity:99.77%
    Color and Shape:Solid
    Molecular weight:191.23
  • Xaliproden

    CAS:
    <p>Xaliproden is a biochemical.</p>
    Formula:C24H22F3N
    Color and Shape:Solid
    Molecular weight:381.43
  • Mesoridazine Besylate

    CAS:
    <p>Mesoridazine Besylate (Serentil), a piperidine antipsychotic and phenothiazine, treats schizophrenia; it's a thioridazine metabolite.</p>
    Formula:C27H32N2O4S3
    Purity:99.58%
    Color and Shape:Solid
    Molecular weight:544.75
  • 5-MeO-pyr-T

    CAS:
    <p>5-MeO-pyr-T (5-Methoxy pyrrolidinyltryptamine) acts as a 5-HT1AR agonist, exhibiting Ki values of 0.577 μM and 373 μM for 5-HT1AR and 5-HT2AR, respectively. It inhibits the reuptake of 5-HT and triggers its release. Additionally, 5-MeO-pyr-T can induce reduced motor activity.</p>
    Formula:C15H20N2O
    Color and Shape:Solid
    Molecular weight:244.33
  • SKF-83566 hydrochloride

    CAS:
    <p>SKF-83566 hydrochloride is a D1-like dopamine receptor antagonist, inhibiting dopamine transporters and mitigating GBP-induced CPP.</p>
    Formula:C17H19BrClNO
    Purity:99.27%
    Color and Shape:Soild
    Molecular weight:368.69
  • LY-53857 free base

    CAS:
    <p>LY-53857 free base is a bioactive chemical.</p>
    Formula:C23H32N2O3
    Color and Shape:Solid
    Molecular weight:384.51
  • MR33317


    <p>MR33317 is an inhibitor of acetylcholinesterase with an IC50 value of 41 nM. Additionally, it acts as an agonist for brain 5-HT4 receptors.</p>
    Formula:C22H28ClN3O2
    Molecular weight:401.187
  • Methamnetamine hydrochloride

    CAS:
    <p>Methamnetamine (PAL-1046) hydrochloride is a psychoactive substance derived from phenethylamine, known to cause excessive serotonin release.</p>
    Formula:C14H18ClN
    Color and Shape:Solid
    Molecular weight:235.75
  • 25E-NBOMe hydrochloride

    CAS:
    <p>25E-NBOMe hydrochloride is a derivative of 2C-E, featuring an N-(2-methoxybenzyl) addition to the amine group, and acts as a selective agonist of the 5-HT2A receptor.</p>
    Formula:C20H28ClNO3
    Color and Shape:Solid
    Molecular weight:365.89
  • 1,8-Cineole

    CAS:
    <p>Eucalyptol, a natural monoterpenoid and cyclic ether found in eucalyptus species, effectively controls excessive airway mucus secretion and asthma by inhibiting pro-inflammatory cytokines. It serves as an efficacious treatment for non-purulent sinusitis, reducing inflammation and pain when applied topically, and demonstrating leukemic cell-killing capabilities in vitro.</p>
    Formula:C10H18O
    Purity:97.44% - 97.44%
    Color and Shape:Solid
    Molecular weight:154.25
  • LY 293284

    CAS:
    <p>LY 293284 is a potent, selective full agonist of 5-HT1A receptor with anxiogenic effects in animal studies.</p>
    Formula:C19H26N2O
    Color and Shape:Solid
    Molecular weight:298.42
  • BMY-14802

    CAS:
    <p>BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol) is a selective and orally active sigma-1 antagonist with an IC50 of 112 nM.</p>
    Formula:C18H22F2N4O
    Purity:99.84%
    Color and Shape:Soild
    Molecular weight:348.39
  • 4-hydroxy DiPT hydrochloride

    CAS:
    <p>4-hydroxy DiPT (hydrochloride) is a 5-HT2A agonist that can induce head twitch response (HTR) in mice, indicating its hallucinogenic potential. This compound holds promise for research into hallucinogens.</p>
    Formula:C16H25ClN2O
    Color and Shape:Solid
    Molecular weight:296.84
  • 5-HT6R antagonist 6


    <p>5-HT6R antagonist 6 (Compound PP15) exhibits high affinity and selectivity for the 5-HT6R receptor, with a Ki of 42 nM. It demonstrates weak antiproliferative activity on tumor cells and low toxicity toward normal cells. 5-HT6R antagonist 6 is applicable in tumor research.</p>
    Formula:C24H26N4O2S
    Color and Shape:Solid
    Molecular weight:434.55
  • Mosapride citrate dihydrate

    CAS:
    <p>Mosapride Citrate, a 5-HT4 agonist, boosts gut movement by enhancing acetylcholine release.</p>
    Formula:C27H35ClFN3O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:632.04
  • SB 699551

    CAS:
    <p>SB 699551 is a selective 5-HT5A antagonist (Ki=6.31 nM) that enhances 5-HT neuronal function. It inhibits SERT (Ki=25.12 nM),inhibit breast cancer.</p>
    Formula:C34H45N3O
    Purity:99.83%
    Molecular weight:511.74
  • 7-Methyl DMT

    CAS:
    <p>7-Methyl DMT (7-TMT) acts as a 5-HT2 receptor agonist. Structurally, it is a tryptamine derivative and serves as an analytical reference for the psychoactive substance DOM. It is also applicable in research related to neurological disorders.</p>
    Formula:C13H18N2
    Color and Shape:Solid
    Molecular weight:202.3
  • Arotinolol hydrochloride

    CAS:
    <p>Arotinolol HCl is a non-selective α/β-blocker, anti-hypertensive, anti-obesity, and improves aortic stiffness.</p>
    Formula:C15H22ClN3O2S3
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:408
  • 4-Chloromethamphetamine hydrochloride

    CAS:
    <p>4-Chloromethamphetamine hydrochloride is a novel psychoactive substance belonging to the amphetamine class.</p>
    Formula:C10H15Cl2N
    Color and Shape:Solid
    Molecular weight:220.14
  • Jatrorrhizine hydroxide

    CAS:
    <p>Jatrorrhizine hydroxide: alkaloid from Coptis chinensis; neuroprotective, antimicrobial, antiplasmodial, antioxidant; AChE inhibitor, affects 5-HT/NE uptake.</p>
    Formula:C20H21NO5
    Color and Shape:Solid
    Molecular weight:355.38
  • Femoxetine

    CAS:
    <p>Femoxetine: antidepressant, enhances morphine, inhibits MAO-A/B, boosts mice's exercise capacity.</p>
    Formula:C20H25NO2
    Purity:99.1% - 99.35%
    Color and Shape:Solid
    Molecular weight:311.42
  • Tiflucarbine

    CAS:
    <p>Tiflucarbine is a potential non-selective 5-HT agonist with antidepressant activity.Tiflucarbine dose-dependently increased the specific activity of soluble</p>
    Formula:C16H17FN2S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:288.38
  • Alosetron-d3

    CAS:
    <p>Alosetron D3 (GR 68755 D3) is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>
    Formula:C17H18N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.37
  • Eletriptan

    CAS:
    <p>Eletriptan, second-generation triptans used to treat migraines, is used as an abortion drug.</p>
    Formula:C22H26N2O2S
    Color and Shape:Solid
    Molecular weight:382.52
  • DOAM

    CAS:
    <p>DOAM is an antagonist of the 5-HT2 receptor.</p>
    Formula:C16H27NO2
    Color and Shape:Solid
    Molecular weight:265.39
  • R 50595

    CAS:
    <p>R 50595 is a selective non-competitive cisapride antagonist.</p>
    Formula:C30H35Cl2F2N3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:594.52
  • Tryptamine hydrochloride

    CAS:
    <p>Tryptamine hydrochloride is a monoamine alkaloid, metabolite of tryptophan and CNS active substance, agonist of 5-HT4 receptor, TAAR1, AHR.</p>
    Formula:C10H13ClN2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:196.68
  • Naratriptan D3 Hydrochloride

    CAS:
    <p>Naratriptan D3 Hydrochloride is the deuterium labeled Naratriptan, is a selective agonist of 5-HT1 receptor subtype.</p>
    Formula:C17H26ClN3O2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:374.94
  • AMI-193

    CAS:
    <p>AMI-193 (Spiramide) is a selective 5-HT2 &amp; D2 receptor antagonist with antipsychotic properties.</p>
    Formula:C22H26FN3O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:383.46
  • PF-03382792

    CAS:
    <p>PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.</p>
    Formula:C23H32FN3O4
    Purity:99.64%
    Color and Shape:Solid
    Molecular weight:433.52
  • Dapoxetine

    CAS:
    <p>Dapoxetine (Dapoxetina) is a selective serotonin reuptake inhibitor, for the treatment of premature ejaculation.</p>
    Formula:C21H23NO
    Purity:99.73%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:305.42
  • 4-Hydroxy MET

    CAS:
    <p>4-Hydroxy MET (4-HO-MET) is a tryptamine-based new psychoactive substance (NPS), structurally similar to the endogenous neurotransmitter serotonin. It has hallucinogenic properties that affect mood, movement, and cognitive functions.</p>
    Formula:C13H18N2O
    Color and Shape:Solid
    Molecular weight:218.3
  • Zicronapine fumarate

    CAS:
    <p>Zicronapine fumarate, an antipsychotic, targets D1/D2 &amp; 5-HT2A receptors; may treat neuropsychiatric conditions.</p>
    Formula:C26H31ClN2O4
    Color and Shape:Solid
    Molecular weight:470.99
  • Minesapride

    CAS:
    <p>Minesapride: novel 5-HT4 partial agonist, may treat constipation-predominant IBS.</p>
    Formula:C21H31ClN4O5
    Purity:99.85% - 99.88%
    Color and Shape:Solid
    Molecular weight:454.95
  • Vortioxetine D8

    CAS:
    <p>Vortioxetine D8 is a deuterium-labeled antidepressant inhibiting 5-HT1A/B, 5-HT3A, 5-HT7 receptors &amp; SERT (Ki: 15-1.6 nM).</p>
    Formula:C18H22N2S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:306.5
  • Cabergoline

    CAS:
    <p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>
    Formula:C26H37N5O2
    Purity:97.69% - 99.86%
    Color and Shape:White Crystalline Solid
    Molecular weight:451.6
  • 4-Butyl-α-agarofuran

    CAS:
    <p>4-Butyl-alpha-agarofuran, a Gharu-wood derivative, is an anxiolytic, antidepressant, and aids neurological research.</p>
    Formula:C18H30O
    Color and Shape:Solid
    Molecular weight:262.43
  • Ethylpropyltryptamine

    CAS:
    <p>Ethylpropyltryptamine (EPT) is an orally active novel psychoactive substance. It is predicted to act as a partial agonist of the 5-HT2A receptor.</p>
    Formula:C15H22N2
    Color and Shape:Solid
    Molecular weight:230.35
  • ECPLA

    CAS:
    <p>ECPLA is an LSD analog and a potent 5-HT2A agonist (EC50 of 14.6 nM), capable of stimulating Gq-mediated calcium flux. It exhibits high affinity for most serotonin receptors, α2-adrenergic receptors, and D2-like dopamine receptors.</p>
    Formula:C21H25N3O
    Color and Shape:Solid
    Molecular weight:335.44
  • Xylamidine

    CAS:
    <p>Xylamidine is a biochemical.</p>
    Formula:C19H24N2O2
    Color and Shape:Solid
    Molecular weight:312.41
  • Quetiapine-d4 fumarate

    CAS:
    <p>Deuterium-labeled Quetiapine fumarate; an antidepressant and anxiolytic 5-HT agonist, dopamine antagonist.</p>
    Formula:C25H29N3O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:503.61
  • Mirtazapine N-oxide

    CAS:
    <p>Mirtazapine N-oxide, a mirtazapine metabolite, is produced by CYP1A2 and CYP3A4 in human liver.</p>
    Formula:C17H19N3O
    Color and Shape:Solid
    Molecular weight:281.359
  • HTR2A antagonist 1


    <p>HTR2A antagonist 1 (Compound 15f) is an HTR2A antagonist with an IC50 of 42.79 nM. It induces sub-G1 cell cycle arrest and apoptosis in colorectal cancer cells by activating the p53/p21/caspase 3 signaling pathway. HTR2A antagonist 1 exhibits good liver microsomal stability and is useful for colorectal cancer research.</p>
    Formula:C35H43Cl2F2N5O4
    Color and Shape:Solid
    Molecular weight:706.65
  • GM-60186


    <p>GM-60186, a potent inhibitor of the 5-HT receptor 2B (HTR2B) with an IC50 of 257 nM, effectively suppresses the proliferation and migration of colorectal cancer cells.</p>
    Formula:C30H33FN2O4
    Color and Shape:Solid
    Molecular weight:504.59
  • 1-Phenylbiguanide HCl

    CAS:
    <p>Compound PDK0269, as 5-HT3 receptor agonists(3–100 μM, pEC50 5.05±0.06), acutely increased XII (hypoglossal) burst frequency and regularity, and decreased bursts/episode . Phenylbiguanide produced a dose-related (10-500 microM) increase in the release of dopamine (280-2000%). When nomifensine (5 microM) was included in the Ringer solution, the effect of Compound PDK0269 on the release of dopamine was ameliorated or inhibited.</p>
    Formula:C8H12ClN5
    Purity:99.31%
    Color and Shape:Solid
    Molecular weight:213.67
  • Tegaserod

    CAS:
    <p>Tegaserod is a 5-HT4R agonist and 5-HT2B receptor antagonist with antitumor activity used in the treatment of irritable bowel syndrome (IBS).</p>
    Formula:C16H23N5O
    Purity:99.20% - 99.89%
    Color and Shape:Solid
    Molecular weight:301.39
  • Clothiapine

    CAS:
    <p>Clothiapine is an atypical antipsychotic of the dibenzothiazepine chemical class.</p>
    Formula:C18H18ClN3S
    Purity:99.93%
    Color and Shape:Solid
    Molecular weight:343.87
  • Thioridazine

    CAS:
    <p>Thioridazine: an antipsychotic, anti-anxiety drug, blocks dopamine D2, PI3K-Akt-mTOR; halts angiogenesis, kills cancer cells, targets CSCs.</p>
    Formula:C21H26N2S2
    Color and Shape:Solid
    Molecular weight:370.57
  • Altanserin

    CAS:
    <p>Altanserin, a 5-HT2A receptor binder, is tagged with F-18 for brain PET scans.</p>
    Formula:C22H22FN3O2S
    Color and Shape:Solid
    Molecular weight:411.49
  • Setiptiline maleate

    CAS:
    <p>Setiptiline maleate is a norepinephrine reuptake inhibitor, 2-adrenergic receptor antagonist, H1 receptor inverse agonist, 5-HT serotonin receptor antagonist.</p>
    Formula:C23H23NO4
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:377.43
  • SB-269970 hydrochloride

    CAS:
    <p>SB-269970 hydrochloride (SB-269970A) , a hydrochloride salt form of SB-269970, is a 5-HT7 receptor antagonist (pKi of 8.3) and exhibits &gt;50-fold selectivity</p>
    Formula:C18H28N2O3S·HCl
    Purity:98.45%
    Color and Shape:Solid
    Molecular weight:388.95
  • Fluvoxamine

    CAS:
    <p>Fluvoxamine (DU-23000) is a selective, orally available 5-HT and serotonin reuptake inhibitor (SSRI) exhibiting antidepressant effects.</p>
    Formula:C15H21F3N2O2
    Color and Shape:Solid
    Molecular weight:318.33
  • SB-277011 hydrochloride

    CAS:
    <p>SB-277011 hydrochloride (SB-277011A hydrochloride) is a D3R antagonist, which induces delayed ejaculation in rats.</p>
    Formula:C28H31ClN4O
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:475.03
  • Cefaclor

    CAS:
    <p>Cefaclor (Panoral) is a cephalosporin antibiotic.</p>
    Formula:C15H14ClN3O4S
    Purity:99.03% - 99.98%
    Color and Shape:Solid
    Molecular weight:367.81
  • Ziprasidone D8

    CAS:
    <p>Ziprasidone D8, deuterium-labeled, is a potent antipsychotic, antagonizing 5-HT and dopamine receptors.</p>
    Formula:C21H21ClN4OS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:420.99
  • 3-Hydroxy agomelatine

    CAS:
    <p>3-Hydroxy agomelatine (3-Hydroxyagomelatine) is a 5-HT2C receptor antagonist used in the study of neurological disorders.</p>
    Formula:C15H17NO3
    Color and Shape:Solid
    Molecular weight:259.3
  • cis-(Z)-Flupentixol dihydrochloride

    CAS:
    <p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>
    Formula:C23H27Cl2F3N2OS
    Purity:98.07%
    Color and Shape:Solid
    Molecular weight:507.44
  • Agomelatine (L(+)-Tartaric acid)

    CAS:
    <p>Agomelatine (S-20098) L(+)-Tartaric acid is a specific agonist of MT1 and MT2 receptors (Kis: 0.1, 0.06, 0.12, and 0.27 nM for CHO-hMT1, HEK-hMT1, CHO-hMT2, and</p>
    Formula:C19H23NO8
    Color and Shape:Solid
    Molecular weight:393.39
  • Granisetron

    CAS:
    <p>Granisetron, a serotonin receptor (5HT-3 selective) antagonist, is used as an antinauseant and antiemetic for cancer chemotherapy.</p>
    Formula:C18H24N4O
    Color and Shape:Solid
    Molecular weight:312.41
  • (R)-Praziquantel-d11

    CAS:
    <p>(R)-Praziquantel D11 is the deuterium labeled (R)-Praziquantel.</p>
    Formula:C19H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:323.47
  • Olanzapine D3

    CAS:
    <p>Olanzapine D3 is the deuterium labeled Olanzapine.</p>
    Formula:C17H20N4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:315.45
  • Eplivanserin (mixture)

    CAS:
    <p>Eplivanserin mixture is a selective serotonin reuptake inhibitor and a 5-HT2A receptor antagonist,</p>
    Formula:C19H21FN2O2
    Color and Shape:Solid
    Molecular weight:328.387
  • Aripiprazole (D8)

    CAS:
    <p>Aripiprazole D8 (OPC-14597 D8) is the deuterium-labeled Aripiprazole. Aripiprazole is a human 5-HT1A receptor partial agonist (Ki: 4.2 nM).</p>
    Formula:C23H27Cl2N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:456.44
  • BW 723C86

    CAS:
    <p>BW 723C86 is a 5-HT2B receptor agonist with anxiolytic effects, inducing overeating and reduced grooming in rats, useful in studying neurological disorders.</p>
    Formula:C16H19ClN2OS
    Purity:99.35%
    Color and Shape:Solid
    Molecular weight:322.85
  • SB-200646A

    CAS:
    <p>SB-200646A: oral 5-HT2B/2C antagonist; higher affinity than 5-HT2A (pKi: 7.5, 6.9 vs 5.2); anxiolytic with in vivo effects.</p>
    Formula:C15H15ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:302.76
  • Agomelatine-d6

    CAS:
    <p>Agomelatine D6 (S-20098 D6) is a deuterium-labeled Agomelatine. Agomelatine is a specific agonist of MT1 and MT2 receptors.</p>
    Formula:C15H17NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:249.34
  • Quetiapine-d4 hemifumarate

    CAS:
    <p>Quetiapine D4 hemifumarate is the deuterium labeled Quetiapine hemifumarate. Quetiapine hemifumarate is a agonist of 5-HT receptors and a antagonist of dopamine receptor,with ntidepressant and anxiolytic.</p>
    Formula:C25H29N3O6S
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:503.61
  • Flibanserin-d4

    CAS:
    <p>Flibanserin: Serotonin 5-HT1A agonist (Ki=1 nM), 5-HT2A antagonist (49 nM). Flibanserin D4 is deuterium-labeled.</p>
    Formula:C20H21F3N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:394.43
  • Sumatriptan

    CAS:
    <p>Sumatriptan (GR 43175 free base) is a 5-HT1 receptor agonist with anti-inflammatory activity used in acute migraine and acute myocardial infarction.</p>
    Formula:C14H21N3O2S
    Purity:99.93%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:295.4
  • Paliperidone Palmitate

    CAS:
    <p>Paliperidone: atypical antipsychotic, dopamine &amp; serotonin antagonist, affects α1/α2 adrenergic and H1 histamine receptors.</p>
    Formula:C39H57FN4O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:664.89
  • Spiroxatrine

    CAS:
    <p>Spiroxatrine (R 5188) is a 5-HT1α and α2-adrenergic dual antagonist with sedative activity for the study of diseases related to the cardiovascular system.</p>
    Formula:C22H25N3O3
    Purity:99.94%
    Color and Shape:Solid
    Molecular weight:379.45
  • Clozapine-d8

    CAS:
    <p>Clozapine-d8 is a deuterium-labeled analog of Clozapine, used as an internal standard for mass spectrometric analysis of this atypical antipsychotic.</p>
    Formula:C18H19ClN4
    Color and Shape:Solid
    Molecular weight:334.87
  • Dehydroaripiprazole

    CAS:
    <p>Dehydroaripiprazole (DM-14857), aripiprazole's active metabolite, is formed by CYP3A4 and CYP2D6, with similar antipsychotic effects.</p>
    Formula:C23H25Cl2N3O2
    Purity:98.7%
    Color and Shape:Solid
    Molecular weight:446.37
  • Asenapine hydrochloride

    CAS:
    <p>Asenapine hydrochloride (Org 5222 hydrochloride) is an antagonist of 5-hydroxytryptamine, adrenergic, dopamine, and histamine receptors with antipsychotic effects.</p>
    Formula:C17H17Cl2NO
    Color and Shape:Solid
    Molecular weight:322.23
  • Alosetron D3 Hydrochloride

    CAS:
    <p>Alosetron D3 (GR 68755 D3) Hydrochloride is a deuterium-labeled Alosetron. Alosetron is an antagonist of 5HT3-receptor.</p>
    Formula:C17H19ClN4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:333.83
  • Nefazodone

    CAS:
    <p>Nefazodone (Nefadar) is an oral antidepressant that is an antagonist of postsynaptic 5-HT 2A receptors and 5-HT 2C receptors, and SNDRI.</p>
    Formula:C25H32ClN5O2
    Purity:99.85%
    Color and Shape:White To Off-White Crystalline Powder
    Molecular weight:470.01
  • Cariprazine D6

    CAS:
    <p>Cariprazine D6 (RGH-188 D6) is a deuterium-labeled Cariprazine. Cariprazine is an antipsychotic agent (D3 receptors, Ki: 0.085 nM; D2 receptors, Ki: 0.49 nM).</p>
    Formula:C21H26D6Cl2N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:433.45
  • Ziprasidone amino acid

    CAS:
    <p>Ziprasidone Impurity C is a byproduct of Ziprasidone, an antipsychotic that blocks 5-HT and dopamine receptors.</p>
    Formula:C21H23ClN4O2S
    Color and Shape:Solid
    Molecular weight:430.95
  • Levomepromazine

    CAS:
    <p>Levomepromazine (Methotrimeprazine) is a Ca2+ release inducer with antiviral, anti-inflammatory, neuroprotective, sedative, and anti-nociceptive activities.</p>
    Formula:C19H24N2OS
    Purity:99.15%
    Color and Shape:Solid
    Molecular weight:328.47
  • Vilazodone-d8

    CAS:
    <p>Vilazodone D8 is a deuterium-labeled vilazodone. Vilazodone is a combined inhibitor of serotonin specific reuptake (SSRI) and agonist of 5-HT1A receptor partial.</p>
    Formula:C26H27N5O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:449.57
  • 3-Hydroxy agomelatine D3

    CAS:
    <p>3-Hydroxy agomelatine D3 is a deuterated metabolite of Agomelatine and a 5-HT2C antagonist (IC50: 3.2 μM, Ki: 1.8 μM).</p>
    Formula:C15H17NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:262.32
  • 5-HT2B antagonist-1

    CAS:
    <p>Orally active 5-HT2B antagonist; IC50 = 33.4 nM; potential for hepatocellular, cardiovascular, GI disease research.</p>
    Formula:C11H14BrN5
    Purity:99.965%
    Color and Shape:Solid
    Molecular weight:296.17
  • Asenapine

    CAS:
    <p>Asenapine (Org 5222) is a 5-HT receptor, adrenergic receptor, and histamine receptor antagonist with antipsychotic properties for the treatment of schizophrenia</p>
    Formula:C17H16ClNO
    Purity:99.64%
    Color and Shape:Coa
    Molecular weight:285.77
  • 5-HT3 antagonist 5

    CAS:
    <p>5-HT3 antagonist 5, a quinoxalin-2-carboxamide, blocks 5-HT3 receptors and has antidepressant effects in mice.</p>
    Formula:C16H13N3O2
    Purity:99.84%
    Color and Shape:Solid
    Molecular weight:279.29
  • 4,4-Diphenylbutylamine hydrochloride

    CAS:
    <p>4,4-Diphenylbutylamine shows affinity for the 5-HT2A and H1 receptors with Kis of 2589 and 1670 nM, respectively[1].</p>
    Formula:C16H20ClN
    Color and Shape:Solid
    Molecular weight:261.79
  • WAY-100635

    CAS:
    <p>WAY-100635 is a potent 5-HT 1A receptor antagonist pyramidal neuron firing frequency during conditioned reflexes; a dopamine D4 receptor agonist .</p>
    Formula:C25H34N4O2
    Purity:98.972%
    Color and Shape:Solid
    Molecular weight:422.56
  • LY310762

    CAS:
    <p>LY310762 is a 5-HT1D receptor antagonist with Ki of 249 nM.</p>
    Formula:C24H27FN2O2·HCl
    Purity:99.8%
    Color and Shape:Solid
    Molecular weight:430.94
  • Melperone

    CAS:
    <p>Melperone, a butyrophenone tranquillizer, caused bradycardia in vivo and in vitro.</p>
    Formula:C16H22FNO
    Purity:98.84%
    Color and Shape:Solid
    Molecular weight:263.35