Proteasome
Proteasome inhibitors are compounds that inhibit the proteasome, a large protein complex responsible for degrading unwanted or damaged proteins within the cell. Inhibition of the proteasome leads to the accumulation of proteins, which can induce cell cycle arrest and apoptosis, particularly in rapidly dividing cells like cancer cells. Proteasome inhibitors are crucial in cancer research and therapy, especially in the treatment of multiple myeloma and other hematologic malignancies. At CymitQuimica, we offer proteasome inhibitors to support your research in oncology, cell biology, and drug development.
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Phepropeptin B
CAS:396729-24-1
Phepropeptin B is a secondary metabolite derived from microorganisms, functioning as a proteasome (proteasome) inhibitor …
Formula:
C40H56N6O6
Color and Shape:
Solid
Molecular weight:
716.91
Ref: TM-T203201
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
Phepropeptin C
CAS:396729-25-2
Phepropeptin C is a microbial secondary metabolite that acts as a proteasome (proteasome) inhibitor, with …
Formula:
C38H60N6O6
Color and Shape:
Solid
Molecular weight:
696.92
Ref: TM-T203422
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
Phepropeptin A
CAS:396729-23-0
Phepropeptin A is a secondary metabolite produced by microorganisms and acts as a proteasome (proteasome) …
Formula:
C37H58N6O6
Color and Shape:
Solid
Molecular weight:
682.89
Ref: TM-T203547
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
Phepropeptin D
CAS:396729-26-3
Phepropeptin D is a secondary metabolite produced by microorganisms and acts as a proteasome (proteasome) …
Formula:
C41H58N6O6
Color and Shape:
Solid
Molecular weight:
730.94
Ref: TM-T203581
| 10mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
β5i-IN-1
β5i-IN-1 is a selective inhibitor of β5i, exhibiting potent activity with an IC50 of 8.463 …
Purity:
98%
Color and Shape:
Odour Solid
Ref: TM-T80697
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
Antitrypanosomal agent 15
Antitrypanosomal Agent 15 (Compound 26) is an orally active, brain-penetrant, selective inhibitor of the Trypanosoma …
Formula:
C21H19FN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
410.4
Ref: TM-T79316
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 13 May 2025
PR-924
CAS:1416709-79-9
PR-924 is a selective inhibitor of tripeptide epoxyketone immunoproteasome subunit LMP-7 (IC50: 22 nM).
Formula:
C37H38N4O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
618.72
Ref: TM-T16568
| 2mg | 685.00 € | ||
| 1mL*10mM (DMSO) | 1,730.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
Sitagliptin phosphate monohydrate
CAS:654671-77-9
Sitagliptin phosphate monohydrate (MK-0431 phosphate monohydrate) is a potent inhibitor of DPP-IV with IC50 of …
Formula:
C16H15F6N5O·H3PO4·H2O
Purity:
99.65% - 99.85%
Color and Shape:
White Or Almost White Crystalline Powder
Molecular weight:
523.33
Ref: TM-T0242L
| 100mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 13 May 2025
RA375
CAS:2649154-57-2
RA375 inhibits RPN13, enhances UPR, ROS, apoptosis, and is 10x more potent against cancer than …
Formula:
C30H25ClN4O7
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
588.99
Ref: TM-T36902
| 2mg | 37.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 147.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 294.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 19 May 2025
4'-Hydroxychalcone
CAS:2657-25-2
4'-Hydroxychalcone (2-Benzal-4-Hydroxyacetophenone) is a chalcone metabolite with hepatoprotective activity
Formula:
C15H12O2
Purity:
99.71% - 99.86%
Color and Shape:
Yellow-Cream Powder
Molecular weight:
224.25
Ref: TM-T7917
| 5g | 365.00 € | ||
| 100mg | 51.00 € | ||
| 500mg | 105.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 19 May 2025
ONX-0914
CAS:960374-59-8
ONX-0914 (PR-957) is an effective and specific immunoproteasome inhibitor, which has minimal cross-reactivity for the …
Formula:
C31H40N4O7
Purity:
98.35% - 99.31%
Color and Shape:
Solid
Molecular weight:
580.67
Ref: TM-T6029
| 1mg | 52.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 315.00 € | ||
| 50mg | 474.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Monday 19 May 2025
Bortezomib
CAS:179324-69-7
Bortezomib (LDP 341) is a 20S proteasome inhibitor (Ki=0.6 nM) that is reversible and selective.
Formula:
C19H25BN4O4
Purity:
100% - 99.97%
Color and Shape:
Yellow Solid
Molecular weight:
384.24
Ref: TM-T2399
| 5mg | 52.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 80.00 € | ||
| 50mg | 96.00 € | ||
| 100mg | 144.00 € | ||
| 200mg | 225.00 € | ||
| 500mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 19 May 2025
TPCK
CAS:402-71-1
TPCK is an irreversible inhibitor of chymotrypsin-like proteases that affect cell proliferation, apoptosis, and tumorigenesis
Formula:
C17H18ClNO3S
Purity:
97.33%
Color and Shape:
Powder
Molecular weight:
351.85
Ref: TM-T8350
| 25mg | 47.00 € | ||
| 50mg | 60.00 € | ||
| 100mg | 88.00 € | ||
| 200mg | 113.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 19 May 2025
(R)-MG-132
CAS:1211877-36-9
(R)-MG-132 (Z-Leu-D-leu-leu-al) is the enantiomer of MG-132. (R)-MG-132 stereoisomer is a more potent proteasome inhibitor …
Formula:
C26H41N3O5
Purity:
98.45%
Color and Shape:
Solid
Molecular weight:
475.62
Ref: TM-T12628
| 1g | 1,103.00 € | ||
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | 329.00 € | ||
| 500mg | 797.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Monday 19 May 2025
Omarigliptin
CAS:1226781-44-7
Omarigliptin is a potent and selective oral dipeptidyl peptidase 4 (DPP4) inhibitor with IC50 value …
Formula:
C17H20F2N4O3S
Purity:
100% - 99.77%
Color and Shape:
Solid
Molecular weight:
398.43
Ref: TM-T2316
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 505.00 € | ||
| 500mg | 1,121.00 € | ||
| 1mL*10mM (DMSO) | 138.00 € |
Estimated delivery in United States, on Monday 19 May 2025
Saxagliptin
CAS:361442-04-8
Saxagliptin (BMS-477118) is a selective and reversible DPP4 inhibitor with IC50 of 26 nM.
Formula:
C18H25N3O2
Purity:
98.05% - 99.95%
Color and Shape:
Solid
Molecular weight:
315.41
Ref: TM-T6203
| 10mg | 42.00 € | ||
| 25mg | 74.00 € | ||
| 50mg | 105.00 € | ||
| 100mg | 164.00 € | ||
| 200mg | 239.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 19 May 2025
Teneligliptin hydrobromide
CAS:906093-29-6
Teneligliptin hydrobromide: potent, novel DPP-4 inhibitor; inhibits human/rat plasma DPP-4 with ~1 nM IC50.
Formula:
C22H30N6OSBrH
Purity:
97.83% - 99.92%
Color and Shape:
Solid
Molecular weight:
628.86
Ref: TM-T6999
| 5mg | 37.00 € | ||
| 10mg | 48.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 111.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 274.00 € | ||
| 500mg | 462.00 € |
Estimated delivery in United States, on Monday 19 May 2025
Alloxan monohydrate
CAS:2244-11-3
Alloxan Monohydrate is a glucose analog used to induce diabetes by destroying beta-cells.
Formula:
C4H4N2O5
Purity:
99.42%
Color and Shape:
Off-White To Beige-Yellowish Crystalline Powder
Molecular weight:
160.09
Ref: TM-T7814
| 1g | 34.00 € |
Estimated delivery in United States, on Monday 19 May 2025
MG-132
CAS:133407-82-6
View and buy MG-132 from TargetMol.MG-132 is a potent cell-permeable 26S proteasome inhibitor (IC50: 100 …
Formula:
C26H41N3O5
Purity:
95% - 99.99%
Color and Shape:
White To Off-White Powder
Molecular weight:
475.62
Ref: TM-T2154
| 10mg | 48.00 € | ||
| 25mg | 88.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 216.00 € | ||
| 200mg | 376.00 € | ||
| 500mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Monday 19 May 2025
Tomatine
CAS:17406-45-0
Tomatine (lycopersicin) is an antiproliferatve agent of breast adenocarcinoma cells.
Formula:
C50H83NO21
Purity:
98.42% - 99.94%
Color and Shape:
White To Light Yellow
Molecular weight:
1034.19
Ref: TM-T3786
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 208.00 € | ||
| 100mg | 309.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Monday 19 May 2025
