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Tyrosine Kinase/Adaptors

Tyrosine Kinase/Adaptors

Tyrosine kinase and adaptor inhibitors are compounds that target tyrosine kinases and their associated adaptor proteins, which play pivotal roles in cell signaling, growth, and differentiation. These inhibitors are essential tools in cancer research, as many tyrosine kinases are involved in the signaling pathways that drive tumor growth and metastasis. By inhibiting tyrosine kinases, these compounds can block critical signaling cascades, offering potential therapeutic strategies for various cancers and other diseases involving abnormal cell signaling. At CymitQuimica, we provide a comprehensive range of high-quality tyrosine kinase and adaptor inhibitors to support your research in oncology, molecular biology, and targeted therapy development.

Subcategories of "Tyrosine Kinase/Adaptors"

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Found 1370 products of "Tyrosine Kinase/Adaptors"

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  • TPX-0046
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    TPX-0046

    CAS:
    <p>TPX-0046 is a RET inhibitor designed to overcome resistance to Selpercatinib and Pralsetinib.</p>
    Formula:C21H21FN6O3
    Purity:99.95%
    Color and Shape:Solid
    Molecular weight:424.43

    Ref: TM-T35384

  • Canertinib
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    Canertinib

    CAS:
    <p>Canertinib (CI-1033), a pan-erbB inhibitor, effectively targets esophageal cancer in vitro/vivo, altering metabolism and reducing growth and hypoxia.</p>
    Formula:C24H25ClFN5O3
    Purity:98% - >99.99%
    Color and Shape:White Or Similar To White Crystalline Powder
    Molecular weight:485.94

    Ref: TM-T6136

  • Entrectinib
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    Entrectinib

    CAS:
    <p>Entrectinib (RXDX-101) is an orally Trk, ROS1, and ALK inhibitor. Entrectinib exhibits antitumor activity. Cost-effective and quality-assured.</p>
    Formula:C31H34F2N6O2
    Purity:98.03% - 99.61%
    Color and Shape:Solid
    Molecular weight:560.64

    Ref: TM-T3678

  • Desmethyl Erlotinib hydrochloride
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    Desmethyl Erlotinib hydrochloride

    CAS:
    <p>Desmethyl Erlotinib hydrochloride (OSI 420) is an active metabolite of erlotinib which is an orally active EGFR tyrosin kinase inhibitor.</p>
    Formula:C21H21N3O4·HCl
    Purity:99.49%
    Color and Shape:Solid
    Molecular weight:415.87

    Ref: TM-T6619

  • (E)-AG 99
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    (E)-AG 99

    CAS:
    <p>(E)-AG 99 ((E)-Tyrphostin AG 99) is an inhibitor of EGFR kinase (IC50: 10 μM in the human epidermoid carcinoma cell line A431).</p>
    Formula:C10H8N2O3
    Purity:99.23%
    Color and Shape:Solid
    Molecular weight:204.18

    Ref: TM-T5155

  • EGFR/ErbB-2/ErbB-4 inhibitor-2
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    EGFR/ErbB-2/ErbB-4 inhibitor-2

    CAS:
    <p>EGFR/ErbB-2/ErbB-4 inhibitor-2 (EGFR/ErbB2 Inhibitor) is a cell-permeable inhibitor of EGFR and c-ErbB2 (IC50s = 20 and 79 nM, respectively)</p>
    Formula:C23H21N3O3
    Purity:99.55%
    Color and Shape:Solid
    Molecular weight:387.43

    Ref: TM-T21954

  • 5'-Fluoroindirubinoxime
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    5'-Fluoroindirubinoxime

    CAS:
    <p>5'-Fluoroindirubinoxime (5'-FIO) is a potent FLT3 inhibitor( IC50 : 15 nM).</p>
    Formula:C16H10FN3O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:295.27

    Ref: TM-T8317

  • JCN037
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    JCN037

    CAS:
    <p>JCN037 is potent, non-covalent and brain-penetrant inhibitor of EGFR(EGFR, p-wtEGFR and pEGFRvⅢ with IC50 of 2.49 nM, 3.95 nM, 4.48 nM , respectively).</p>
    Formula:C16H11BrFN3O2
    Purity:99.5%
    Color and Shape:Solid
    Molecular weight:376.18

    Ref: TM-T8431

  • ALK-IN-1
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    ALK-IN-1

    CAS:
    <p>ALK-IN-1 is a potent ALK inhibitor, demonstrating the ability to overcome Crizotinib resistance mediated by an L1196M mutation.</p>
    Formula:C26H34ClN6O2P
    Purity:99.74% - 99.80%
    Color and Shape:Solid
    Molecular weight:529.01

    Ref: TM-T3059

  • Fostamatinib Disodium
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    Fostamatinib Disodium

    CAS:
    <p>Fostamatinib Disodium (R788 Disodium) is an orally available Syk kinase inhibitor with potential anti-inflammatory and immunomodulating activities.</p>
    Formula:C23H24FN6O9P·2Na
    Purity:96.13% - 99.09%
    Color and Shape:Solid
    Molecular weight:624.42

    Ref: TM-T2605

  • FLT3-IN-2
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    FLT3-IN-2

    CAS:
    <p>FLT3-IN-2 is an FLT3 inhibitor (IC50&lt;1 μM).</p>
    Formula:C21H16ClF3N4
    Purity:97.57% - 98.53%
    Color and Shape:Solid
    Molecular weight:416.83

    Ref: TM-T1938

  • Rebastinib
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    Rebastinib

    CAS:
    <p>DCC-2036 (Rebastinib (DCC-2036)) is a conformational control Bcr-Abl inhibitor for Abl1(WT, IC50: 0.8 nM) and Abl1(T315I, IC50: 4 nM), also inhibits LYN, SRC,</p>
    Formula:C30H28FN7O3
    Purity:99.53% - 99.79%
    Color and Shape:Solid
    Molecular weight:553.59

    Ref: TM-T2640

  • ASP5878
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    ASP5878

    CAS:
    <p>ASP5878 potently inhibited the tyrosine kinase activities of recombinant FGFR1, 2, 3, and 4 with IC50 values of 0.47, 0.60, 0.74, and 3.5 nmol/L.</p>
    Formula:C18H19F2N5O4
    Purity:99.8% - 99.89%
    Color and Shape:Solid
    Molecular weight:407.37

    Ref: TM-T5473

  • Avapritinib
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    Avapritinib

    CAS:
    <p>Avapritinib (BLU-285) is a selective, highly potent, and orally active inhibitor of KIT and PDGFRA activation loop mutant kinases.Cost-effective and quality-assured.</p>
    Formula:C26H27FN10
    Purity:96.59% - 99.7%
    Color and Shape:Solid
    Molecular weight:498.56

    Ref: TM-T5109

  • Bacitracin Zinc
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    Bacitracin Zinc

    CAS:
    <p>Bacitracin Zinc is a dephosphorylated disruptor of C55-isoprene pyrophosphate that inhibits Tyr cleavage in Met-enkephalin with an IC50 of 10 μM.</p>
    Formula:C66H101N17O16SZn
    Purity:63.98%
    Color and Shape:Light-Colored Free-Flowing Powders
    Molecular weight:1486.07

    Ref: TM-T2208

  • Naquotinib
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    Naquotinib

    CAS:
    <p>Naquotinib (ASP8273) (ASP8273) is an orally available, mutant-selective and irreversible EGFR inhibitor; (IC50s: 8-33 nM and 230 nM toward EGFR mutants and EGFR</p>
    Formula:C30H42N8O3
    Purity:97.49%
    Color and Shape:Solid
    Molecular weight:562.71

    Ref: TM-TQ0092

  • lavendustin C
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    lavendustin C

    CAS:
    <p>lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine kinase.</p>
    Formula:C14H13NO5
    Purity:98.06%
    Color and Shape:Yellow To Tan Powder
    Molecular weight:275.26

    Ref: TM-T4185

  • Futibatinib
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    Futibatinib

    CAS:
    <p>Futibatinib (TAS-120) is an orally active, potent,and irreversible FGFR inhibitor of FGFR1, FGFR2, FGFR3, and FGFR4.Cost-effective and quality-assured.</p>
    Formula:C22H22N6O3
    Purity:97.66% - 99.44%
    Color and Shape:Solid
    Molecular weight:418.45

    Ref: TM-T5044

  • Dovitinib lactate hydrate
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    Dovitinib lactate hydrate

    CAS:
    <p>Dovitinib lactate hydrate (TKI258) is the Lactate of Dovitinib, which is a multitargeted RTK inhibitor, mostly for class III (FLT3/c-Kit).</p>
    Formula:C24H27FN6O4
    Purity:99.82%
    Color and Shape:Solid
    Molecular weight:482.51

    Ref: TM-T6479

  • Methyl 2,5-dihydroxycinnamate
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    Methyl 2,5-dihydroxycinnamate

    CAS:
    <p>Methyl 2,5-dihydroxycinnamate is an EGF receptor-associated tyrosine kinases inhibitor.</p>
    Formula:C10H10O4
    Purity:99.60%
    Color and Shape:Crystalline
    Molecular weight:194.18

    Ref: TM-T22974