PDGFR
PDGFR (platelet-derived growth factor receptor) inhibitors are compounds that block the signaling of PDGFR, a receptor involved in cell growth, proliferation, and angiogenesis. PDGFR plays a significant role in the development of the blood vessels that supply tumors. Inhibiting PDGFR can therefore prevent angiogenesis, making these inhibitors valuable in cancer therapy. At CymitQuimica, we provide a selection of high-quality PDGFR inhibitors to support your research in oncology, vascular biology, and angiogenesis.
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PDGF R β/CD140b Protein, Human, Recombinant (His & Avi)
PDGF R beta/CD140b Protein, Human, Recombinant (His & Avi) is expressed in HEK293 mammalian cells …
Color and Shape:
Liquid
Molecular weight:
59 kDa (predicted). Due to glycosylation, the protein migrates to 78-115 kDa based on Tris-Bis PAGE result.
Ref: TM-TMPK-00421
| 1mg | 2,212.00 € | ||
| 100µg | 348.00 € | ||
| 500µg | 1,372.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Telatinib
CAS:332012-40-5
Telatinib (Bay 57-9352) inhibits VEGFR2/3, c-Kit, PDGFRα with IC50s: 6 nM, 4 nM, 1 nM, …
Formula:
C20H16ClN5O3
Purity:
97.61% - 99.81%
Color and Shape:
Solid
Molecular weight:
409.83
Ref: TM-T6166
| 10mg | 39.00 € | ||
| 25mg | 78.00 € | ||
| 50mg | 113.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Linifanib
CAS:796967-16-3
Linifanib (AL-39324) (ABT-869) is a novel, potent ATP-competitive VEGFR/PDGFR inhibitor for KDR (IC50: 4 nM), …
Formula:
C21H18FN5O
Purity:
98% - 98.24%
Color and Shape:
Solid
Molecular weight:
375.4
Ref: TM-T2514
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 184.00 € | ||
| 100mg | 268.00 € | ||
| 200mg | 493.00 € | ||
| 500mg | 802.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pazopanib Hydrochloride
CAS:635702-64-6
Pazopanib HCl (Votrient) inhibits VEGFR1-3, PDGFR, FGFR, c-Kit, c-Fms with IC50 range 10-146 nM in …
Formula:
C21H23N7O2S·HCl
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
473.98
Ref: TM-T6930
| 10mg | 52.00 € | ||
| 25mg | 90.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 139.00 € | ||
| 200mg | 225.00 € | ||
| 500mg | 355.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CHIR-124
CAS:405168-58-3
CHIR-124 is an effective Chk1 inhibitor (IC50: 0.3 nM). It has 2, 000-fold selectivity against …
Formula:
C23H22ClN5O
Purity:
96.33% - 98.35%
Color and Shape:
Solid
Molecular weight:
419.91
Ref: TM-T6350
| 1mg | 41.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 350.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ponatinib
CAS:943319-70-8
Ponatinib (AP24534) is an orally available, multitargeted kinase inhibitor (IC50s: 0.37/1.1/1.5/2.2/5.4 nM for Abl, PDGFRα, …
Formula:
C29H27F3N6O
Purity:
98% - 99.74%
Color and Shape:
Solid
Molecular weight:
532.56
Ref: TM-T2372
| 10mg | 54.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 136.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
XL 999
CAS:705946-27-6
Tyrosine kinase-IN-1 is a multi-targeted tyrosine kinase inhibitor(KDR, Flt-1, FGFR1 and PDGFRα with IC50s of …
Formula:
C26H28FN5O
Purity:
99.55%
Color and Shape:
Solid
Molecular weight:
445.53
Ref: TM-T5466
| 1mg | 41.00 € | ||
| 5mg | 61.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 398.00 € | ||
| 1mL*10mM (DMSO) | 68.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Regorafenib Hydrochloride
CAS:835621-07-3
Regorafenib HCl (BAY73-4506) is an oral inhibitor targeting angiogenic, stromal, and cancer kinases with strong …
Formula:
C21H16Cl2F4N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
519.28
Ref: TM-T8402
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 142.00 € | ||
| 500mg | 343.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Flumatinib mesylate
CAS:895519-91-2
Flumatinib mesylate (HHGV678 mesylate) is a selective inhibitor of c-Abl, PDGFRβ and c-Kit, effectively overcomes …
Formula:
C30H33F3N8O4S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
658.69
Ref: TM-T7861
| 1mg | 37.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 131.00 € | ||
| 25mg | 247.00 € | ||
| 50mg | 388.00 € | ||
| 100mg | 621.00 € | ||
| 500mg | 1,285.00 € | ||
| 1mL*10mM (DMSO) | 138.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Nintedanib
CAS:656247-17-5
Nintedanib (Intedanib) is a triple vascular kinase inhibitor that inhibits VEGFR1, VEGFR2, and VEGFR3 (IC50=34/13/13 …
Formula:
C31H33N5O4
Purity:
98% - 99.92%
Color and Shape:
Solid
Molecular weight:
539.62
Ref: TM-T1777
| 5mg | 45.00 € | ||
| 10mg | 58.00 € | ||
| 50mg | 69.00 € | ||
| 100mg | 90.00 € | ||
| 200mg | 139.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
NVP-ACC789
CAS:300842-64-2
ACC-789 (NVP-ACC789 (ZK202650); ZK-202650) is an effective, specific and orally active inhibitor of the VEGF …
Formula:
C21H17BrN4
Purity:
99.44% - 99.63%
Color and Shape:
Solid
Molecular weight:
405.29
Ref: TM-T3463
| 10mg | 44.00 € | ||
| 25mg | 56.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 145.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Dovitinib
CAS:405169-16-6
Dovitinib is an orally active, multi-targeted tyrosine kinase (RTK) inhibitor with anti-tumor effects.Cost-effective and quality-assured.
Formula:
C21H21FN6O
Purity:
98% - 99.78%
Color and Shape:
Solid
Molecular weight:
392.43
Ref: TM-T6289
| 5mg | 46.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 123.00 € | ||
| 50mg | 199.00 € | ||
| 100mg | 321.00 € | ||
| 200mg | 479.00 € | ||
| 500mg | 766.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
ENMD-2076
CAS:934353-76-1
ENMD-2076, a multi-targeted kinase inhibitor, has specific activity against Aurora A, Flt3, KDR/VEGFR2, Flt4/VEGFR3, FGFR1, …
Formula:
C21H25N7
Purity:
97.63% - ≥95%
Color and Shape:
Solid
Molecular weight:
375.47
Ref: TM-T2358
| 1mg | 51.00 € | ||
| 2mg | 71.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 156.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 452.00 € | ||
| 100mg | 638.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PD-089828
CAS:179343-17-0
PD 089828 inhibits FGFR1, PDGFRβ, EGFR (IC50s: 0.15-5.47 μM), and c-Src (IC50: 0.18 μM).
Formula:
C18H18Cl2N6O
Purity:
96.78%
Color and Shape:
Solid
Molecular weight:
405.28
Ref: TM-T8976
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 245.00 € | ||
| 50mg | 365.00 € | ||
| 100mg | 537.00 € | ||
| 500mg | 1,137.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tandutinib
CAS:387867-13-2
Tandutinib (CT53518) (MLN518, CT53518), an effective FLT3 antagonist (IC50: 0.22 μM), can also inhibit c-Kit …
Formula:
C31H42N6O4
Purity:
99.45% - ≥98%
Color and Shape:
White Solid
Molecular weight:
562.7
Ref: TM-T1667
| 25mg | 50.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 84.00 € | ||
| 200mg | 104.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Vorolanib
CAS:1013920-15-4
Vorolanib (X-82) is an orally active VEGFR/PDGFR dual inhibitor.
Formula:
C23H26FN5O3
Purity:
97.35%
Color and Shape:
Solid
Molecular weight:
439.48
Ref: TM-T8491
| 1mg | 111.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 369.00 € | ||
| 25mg | 618.00 € | ||
| 50mg | 877.00 € | ||
| 100mg | 1,189.00 € | ||
| 1mL*10mM (DMSO) | 257.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Masitinib
CAS:790299-79-5
Masitinib (AB1010) is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in …
Formula:
C28H30N6OS
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
498.64
Ref: TM-T2609
| 5mg | 36.00 € | ||
| 10mg | 52.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 156.00 € | ||
| 200mg | 236.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CP-673451
CAS:343787-29-1
CP-673451 is a specific inhibitor of PDGFRα/β (IC50: 10/1 nM) with antiangiogenic and antitumor activity …
Formula:
C24H27N5O2
Purity:
99.88% - 99.93%
Color and Shape:
Solid
Molecular weight:
417.5
Ref: TM-T6091
| 1mg | 52.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 346.00 € | ||
| 50mg | 529.00 € | ||
| 100mg | 761.00 € | ||
| 500mg | 1,576.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ripretinib
CAS:1442472-39-0
Ripretinib (DCC-2618) is an orally bioavailable inhibitor of KIT and PDGFRA.
Formula:
C24H21BrFN5O2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
510.36
Ref: TM-T8482
| 1mg | 391.00 € | ||
| 2mg | 585.00 € | ||
| 5mg | 930.00 € | ||
| 10mg | 1,274.00 € | ||
| 25mg | 1,722.00 € | ||
| 50mg | 2,401.00 € | ||
| 100mg | 3,353.00 € | ||
| 500mg | 5,402.00 € | ||
| 1mL*10mM (DMSO) | 427.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Regorafenib
CAS:755037-03-7
Regorafenib (BAY 73-4506) is a multi-targeted receptor tyrosine kinase inhibitor that inhibits RET, C-RAF, VEGFR2, …
Formula:
C21H15ClF4N4O3
Purity:
98% - 99.95%
Color and Shape:
Solid
Molecular weight:
482.82
Ref: TM-T1792
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 79.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 142.00 € | ||
| 200mg | 181.00 € | ||
| 500mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
