PDGFR
PDGFR (platelet-derived growth factor receptor) inhibitors are compounds that block the signaling of PDGFR, a receptor involved in cell growth, proliferation, and angiogenesis. PDGFR plays a significant role in the development of the blood vessels that supply tumors. Inhibiting PDGFR can therefore prevent angiogenesis, making these inhibitors valuable in cancer therapy. At CymitQuimica, we provide a selection of high-quality PDGFR inhibitors to support your research in oncology, vascular biology, and angiogenesis.
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PD168393
CAS:194423-15-9
PD168393 is an irreversible EGFR inhibitor (IC50: 0.70 nM), irreversibly alkylate Cys-773; inactive against PKC, …
Formula:
C17H13BrN4O
Purity:
99.13% - 99.7%
Color and Shape:
Solid
Molecular weight:
369.22
Ref: TM-T6932
| 1mg | 39.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 304.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Lenvatinib mesylate
CAS:857890-39-2
Lenvatinib mesylate (E7080 (mesylate)) is an oral and multi-targeted inhibitor of VEGFR1-3, FGFR1-4, PDGFR, KIT, …
Formula:
C22H23ClN4O7S
Purity:
99.03% - 99.79%
Color and Shape:
Solid
Molecular weight:
522.96
Ref: TM-T8541
| 10mg | 40.00 € | ||
| 25mg | 59.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 162.00 € | ||
| 500mg | 263.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Regorafenib monohydrate
CAS:1019206-88-2
Regorafenib Monohydrate is a novel oral multikinase inhibitor with IC50 values of 13, 4.2, 46, …
Formula:
C21H17ClF4N4O4
Purity:
99.69%
Color and Shape:
Solid
Molecular weight:
500.83
Ref: TM-T1792L
| 5mg | 36.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 138.00 € | ||
| 200mg | 204.00 € | ||
| 500mg | 348.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Methylnissolin
CAS:73340-41-7
Methylnissolin (3-Hydroxy-9,10-dimethoxyptercarpan) is derived from Astragalus and has antibacterial and anti-cancer effects.
Formula:
C17H16O5
Purity:
99.68% - 99.98%
Color and Shape:
Solid
Molecular weight:
300.31
Ref: TM-TN2354
| 1mg | 87.00 € | ||
| 5mg | 198.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 513.00 € | ||
| 50mg | 732.00 € | ||
| 1mL*10mM (DMSO) | 185.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tyrphostin AG1296
CAS:146535-11-7
Tyrphostin AG1296 (Tyrphostin AG 1296) is an inhibitor of PDGFR with IC50 of 0.3-0.5 μM, …
Formula:
C16H14N2O2
Purity:
99.66% - 99.68%
Color and Shape:
Solid
Molecular weight:
266.29
Ref: TM-T6711
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 174.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 397.00 € | ||
| 200mg | 565.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Cediranib
CAS:288383-20-0
Cediranib (AZD2171) is a potent KDR tyrosine kinase inhibitor (IC50 < 1nM), also targets Flt1/4, PDGFRβ, …
Formula:
C25H27FN4O3
Purity:
97.21% - 99.94%
Color and Shape:
Solid
Molecular weight:
450.51
Ref: TM-T2500
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 134.00 € | ||
| 50mg | 175.00 € | ||
| 100mg | 248.00 € | ||
| 200mg | 454.00 € | ||
| 500mg | 729.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Dovitinib lactate hydrate
CAS:915769-50-5
Dovitinib lactate hydrate (TKI258) is the Lactate of Dovitinib, which is a multitargeted RTK inhibitor, …
Formula:
C24H27FN6O4
Purity:
99.17%
Color and Shape:
Solid
Molecular weight:
482.51
Ref: TM-T6479
| 5mg | 54.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 378.00 € | ||
| 200mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Amuvatinib
CAS:850879-09-3
Amuvatinib (MP470) is an orally bioavailable synthetic carbothioamide with potential antineoplastic activity.
Formula:
C23H21N5O3S
Purity:
98.48% - 99.54%
Color and Shape:
Solid
Molecular weight:
447.51
Ref: TM-T2516
| 1mg | 52.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 257.00 € | ||
| 50mg | 411.00 € | ||
| 100mg | 519.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bisindolylmaleimide I
CAS:133052-90-1
Bisindolylmaleimide I (GF109203X) is a potent and highly selective protein kinase C (PKC) inhibitor with …
Formula:
C25H24N4O2
Purity:
98.19% - 99.08%
Color and Shape:
Orange Solid
Molecular weight:
412.48
Ref: TM-T6513
| 5mg | 66.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 184.00 € | ||
| 50mg | 345.00 € | ||
| 100mg | 460.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
TAK-593
CAS:1005780-62-0
TAK-593 is an effective VEGFR and PDGFR family inhibitor (IC50s: 3.2, 0.95, 1.1, 4.3, and …
Formula:
C23H23N7O3
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
445.47
Ref: TM-T16975
| 2mg | 43.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 292.00 € | ||
| 100mg | 421.00 € | ||
| 200mg | 591.00 € | ||
| 1mL*10mM (DMSO) | 75.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Masitinib mesylate
CAS:1048007-93-7
Masitinib mesylate (AB-1010 mesylate) is a selective and orally bioavailable c-Kit inhibitor (IC50 of 200 …
Formula:
C29H34N6O4S2
Purity:
100% - 99.92%
Color and Shape:
Solid
Molecular weight:
594.75
Ref: TM-T8544
| 5mg | 35.00 € | ||
| 10mg | 51.00 € | ||
| 25mg | 75.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 220.00 € | ||
| 500mg | 364.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PP121
CAS:1092788-83-4
PP-121 inhibits PDGFR, Hck, mTOR, VEGFR2, Src, Abl, and DNA-PK with IC50 values ranging from …
Formula:
C17H17N7
Purity:
99.19% - 99.67%
Color and Shape:
Solid
Molecular weight:
319.36
Ref: TM-T2415
| 5mg | 60.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 237.00 € | ||
| 100mg | 344.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SU4312
CAS:5812-07-7
SU-4312 (DMBI) inhibits VEGFR & PDGFR (IC50: 0.8, 19.4 μM) and shields neurons from MPP(+)-induced …
Formula:
C17H16N2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
264.32
Ref: TM-T3570
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 375.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
N-(p-Coumaroyl) serotonin
CAS:68573-24-0
N-(p-Coumaroyl) Serotonin, from safflower seeds, has antioxidant, antitumor properties and improves vascular health.
Formula:
C19H18N2O3
Purity:
98.78%
Color and Shape:
Solid
Molecular weight:
322.36
Ref: TM-TN1969
| 1mg | 42.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 185.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 407.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Toceranib Phosphate
CAS:874819-74-6
Toceranib Phosphate (SU11654 phosphate), is a selective inhibitor of the tyrosine kinase activity of several …
Formula:
C22H28FN4O6P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
494.45
Ref: TM-T7394
| 10mg | 48.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 107.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
SU14813
CAS:627908-92-3
SU14813: inhibits multiple kinases (VEGFR2, VEGFR1, PDGFRβ, KIT) with IC50s of 50, 2, 4, 15 …
Formula:
C23H27FN4O4
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
442.48
Ref: TM-T7945
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 220.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Avapritinib
CAS:1703793-34-3
Avapritinib (BLU-285) is a selective, highly potent, and orally active inhibitor of KIT and PDGFRA …
Formula:
C26H27FN10
Purity:
96.59% - 99.7%
Color and Shape:
Solid
Molecular weight:
498.56
Ref: TM-T5109
| 1mg | 86.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 510.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,003.00 € | ||
| 500mg | 2,024.00 € | ||
| 1mL*10mM (DMSO) | 204.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Nintedanib esylate
CAS:656247-18-6
Nintedanib esylate (BIBF 1120 esylate) is a potent triple angiokinase inhibitor for VEGFR1/2/3, FGFR1/2/3 and …
Formula:
C31H33N5O4·C2H6O3S
Purity:
99.43% - 99.96%
Color and Shape:
Solid
Molecular weight:
649.76
Ref: TM-T5001
| 5mg | 42.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 83.00 € | ||
| 100mg | 103.00 € | ||
| 200mg | 161.00 € | ||
| 500mg | 310.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Multi-kinase inhibitor 1
CAS:778274-97-8
Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.
Formula:
C20H17F3N4O3
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
418.37
Ref: TM-T4191
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 505.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ki20227
CAS:623142-96-1
Ki-20227 is a specific c-Fms tyrosine kinase(CSF1R) inhibitor (IC50: 2 nM).
Formula:
C24H24N4O5S
Purity:
97.16% - 99.37%
Color and Shape:
Solid
Molecular weight:
480.54
Ref: TM-T4315
| 1mg | 46.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 730.00 € | ||
| 200mg | 994.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
