c-Kit
c-Kit inhibitors are compounds that block the activity of the Stem Cell Factor Receptor (c-Kit), a tyrosine kinase that plays a pivotal role in cell survival, proliferation, and differentiation, particularly in hematopoietic cells. Mutations in c-Kit are linked to various cancers, including gastrointestinal stromal tumors (GIST) and leukemia. At CymitQuimica, we provide c-Kit inhibitors to support your research in oncology, hematology, and stem cell biology.
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JNJ-38158471
CAS:951151-97-6
JNJ-38158471 (CS-2660), a highly selective, orally available, well tolerated VEGFR2 inhibitor, inhibits closely related tyrosine …
Formula:
C15H17ClN6O3
Purity:
97.08%
Color and Shape:
Solid
Molecular weight:
364.79
Ref: TM-T22349
| 1mg | 51.00 € | ||
| 2mg | 72.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 250.00 € | ||
| 50mg | 364.00 € | ||
| 100mg | 490.00 € | ||
| 200mg | 673.00 € | ||
| 1mL*10mM (DMSO) | 109.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
OSI-930
CAS:728033-96-3
OSI-930 is an oral c-Kit/VEGFR-2 inhibitor targeting tumor growth and angiogenesis.
Formula:
C22H16F3N3O2S
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
443.44
Ref: TM-T2624
| 1mg | 51.00 € | ||
| 5mg | 100.00 € | ||
| 10mg | 143.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 605.00 € | ||
| 1mL*10mM (DMSO) | 100.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Masitinib
CAS:790299-79-5
Masitinib (AB1010) is a tyrosine-kinase inhibitor used in the treatment of mast cell tumors in …
Formula:
C28H30N6OS
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
498.64
Ref: TM-T2609
| 5mg | 36.00 € | ||
| 10mg | 52.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 156.00 € | ||
| 200mg | 236.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Toceranib Phosphate
CAS:874819-74-6
Toceranib Phosphate (SU11654 phosphate), is a selective inhibitor of the tyrosine kinase activity of several …
Formula:
C22H28FN4O6P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
494.45
Ref: TM-T7394
| 10mg | 48.00 € | ||
| 25mg | 73.00 € | ||
| 50mg | 92.00 € | ||
| 100mg | 107.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BLU-263
CAS:2505078-08-8
BLU-263 is an investigational, potent, and selective oral small molecule inhibitor of KIT with sub-nanomolar …
Formula:
C27H29FN10O
Purity:
99.67%
Color and Shape:
Solid
Molecular weight:
528.58
Ref: TM-T9295
| 1mg | 64.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 220.00 € | ||
| 25mg | 423.00 € | ||
| 50mg | 553.00 € | ||
| 100mg | 793.00 € | ||
| 200mg | 1,063.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ripretinib
CAS:1442472-39-0
Ripretinib (DCC-2618) is an orally bioavailable inhibitor of KIT and PDGFRA.
Formula:
C24H21BrFN5O2
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
510.36
Ref: TM-T8482
| 1mg | 391.00 € | ||
| 2mg | 585.00 € | ||
| 5mg | 930.00 € | ||
| 10mg | 1,274.00 € | ||
| 25mg | 1,722.00 € | ||
| 50mg | 2,401.00 € | ||
| 100mg | 3,353.00 € | ||
| 500mg | 5,402.00 € | ||
| 1mL*10mM (DMSO) | 427.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SU14813
CAS:627908-92-3
SU14813: inhibits multiple kinases (VEGFR2, VEGFR1, PDGFRβ, KIT) with IC50s of 50, 2, 4, 15 …
Formula:
C23H27FN4O4
Purity:
99.72%
Color and Shape:
Solid
Molecular weight:
442.48
Ref: TM-T7945
| 5mg | 35.00 € | ||
| 10mg | 52.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 220.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Avapritinib
CAS:1703793-34-3
Avapritinib (BLU-285) is a selective, highly potent, and orally active inhibitor of KIT and PDGFRA …
Formula:
C26H27FN10
Purity:
96.59% - 99.7%
Color and Shape:
Solid
Molecular weight:
498.56
Ref: TM-T5109
| 1mg | 86.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 510.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,003.00 € | ||
| 500mg | 2,024.00 € | ||
| 1mL*10mM (DMSO) | 204.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Multi-kinase inhibitor 1
CAS:778274-97-8
Multi-kinase inhibitor 1 (Multi-kinase inhibitor I) is a Multi-kinase inhibitor.
Formula:
C20H17F3N4O3
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
418.37
Ref: TM-T4191
| 1mg | 39.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 230.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 505.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Ki20227
CAS:623142-96-1
Ki-20227 is a specific c-Fms tyrosine kinase(CSF1R) inhibitor (IC50: 2 nM).
Formula:
C24H24N4O5S
Purity:
97.16% - 99.37%
Color and Shape:
Solid
Molecular weight:
480.54
Ref: TM-T4315
| 1mg | 46.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 458.00 € | ||
| 100mg | 730.00 € | ||
| 200mg | 994.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Flumatinib
CAS:895519-90-1
Flumatinib (HHGV678) is an orally bioavailable tyrosine kinase inhibitor flumatinib, with potential antineoplastic activity.
Formula:
C29H29F3N8O
Purity:
99.52% - 99.95%
Color and Shape:
Solid
Molecular weight:
562.59
Ref: TM-T4320
| 1mg | 35.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 85.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 267.00 € | ||
| 200mg | 402.00 € | ||
| 500mg | 666.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AZD2932
CAS:883986-34-3
AZD2932 is a potent and multi-targeted kinase inhibitor VEGFR2, PDGFβ, Flt-3, and c-Kit.
Formula:
C24H25N5O4
Purity:
97.71% - 98.37%
Color and Shape:
Solid
Molecular weight:
447.49
Ref: TM-T1836
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 150.00 € | ||
| 100mg | 232.00 € | ||
| 200mg | 344.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Midostaurin
CAS:120685-11-2
PKC412(Midostaurin (PKC412); CGP41231; CGP41251) is a broad spectrum protein kinase inhibitor.
Formula:
C35H30N4O4
Purity:
100% - 99.56%
Color and Shape:
Solid
Molecular weight:
570.64
Ref: TM-T3211
| 1mg | 51.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 213.00 € | ||
| 50mg | 321.00 € | ||
| 100mg | 477.00 € | ||
| 500mg | 1,072.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Dovitinib lactate
CAS:692737-80-7
Dovitinib lactate (TKI-258 lactate)(TKI258) lactate is a potent inhibitor of fibroblast growth factor receptor 3 …
Formula:
C24H27FN6O4
Purity:
98.44% - 99.54%
Color and Shape:
Solid
Molecular weight:
482.51
Ref: TM-T7104
| 5mg | 51.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 350.00 € | ||
| 200mg | 523.00 € | ||
| 500mg | 828.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tandutinib
CAS:387867-13-2
Tandutinib (CT53518) (MLN518, CT53518), an effective FLT3 antagonist (IC50: 0.22 μM), can also inhibit c-Kit …
Formula:
C31H42N6O4
Purity:
99.45% - ≥98%
Color and Shape:
White Solid
Molecular weight:
562.7
Ref: TM-T1667
| 25mg | 50.00 € | ||
| 50mg | 63.00 € | ||
| 100mg | 84.00 € | ||
| 200mg | 104.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Vimseltinib
CAS:1628606-05-2
Vimseltinib (DCC-3014) is a c-FMS (CSF-IR) and c-Kit dual inhibitor (IC50s: <0.01 μM and 0.1-1 …
Formula:
C23H25N7O2
Purity:
98.98% - 99.57%
Color and Shape:
Solid
Molecular weight:
431.49
Ref: TM-T10652
| 1mg | 91.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 308.00 € | ||
| 25mg | 527.00 € | ||
| 50mg | 719.00 € | ||
| 100mg | 926.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
SKLB4771
CAS:1370256-78-2
SKLB4771 (FLT3-IN-1) is a novel potent and selective Flt3 inhibitor.
Formula:
C25H27N7O3S2
Purity:
100% - 98.27%
Color and Shape:
Solid
Molecular weight:
537.66
Ref: TM-T2051
| 1mg | 66.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 129.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 386.00 € | ||
| 50mg | 577.00 € | ||
| 100mg | 817.00 € | ||
| 500mg | 1,661.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
c-Kit-IN-3
CAS:2363169-01-9
c-Kit-IN-3 is a selective inhibitor of c-KIT kinase with IC50s of 4 nM and 8 …
Formula:
C26H20ClF3N2O4
Purity:
99.43%
Color and Shape:
Solid
Molecular weight:
516.9
Ref: TM-T10651
| 1mg | 85.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 411.00 € | ||
| 50mg | 551.00 € | ||
| 100mg | 771.00 € | ||
| 500mg | 1,545.00 € | ||
| 1mL*10mM (DMSO) | 333.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Chiauranib
CAS:1256349-48-0
Chiauranib, a potent anticancer agent, inhibits angiogenesis kinases (VEGFR1-3, PDGFRα, c-Kit), Aurora B, and CSF1R …
Formula:
C27H21N3O3
Purity:
96.25%
Color and Shape:
Solid
Molecular weight:
435.47
Ref: TM-T35570
| 1mg | 89.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 300.00 € | ||
| 25mg | 508.00 € | ||
| 50mg | 732.00 € | ||
| 100mg | 1,003.00 € | ||
| 1mL*10mM (DMSO) | 213.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Bezuclastinib
CAS:1616385-51-3
Bezuclastinib (CGT9486) is a novel, potent and highly selective tyrosine kinase and c-kit D816V inhibitor …
Formula:
C19H17N5O
Purity:
99.81%
Color and Shape:
Liquid
Molecular weight:
331.37
Ref: TM-T60976
| 1mg | 172.00 € | ||
| 5mg | 422.00 € | ||
| 10mg | 675.00 € | ||
| 25mg | 1,344.00 € | ||
| 50mg | 2,151.00 € | ||
| 100mg | 3,421.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
