CymitQuimica logo
Endothelin Receptor

Endothelin Receptor

Endothelin receptors are GPCRs that mediate the effects of endothelins, potent vasoconstrictor peptides that play a significant role in vascular tone regulation, blood pressure control, and cell proliferation. Endothelin receptor antagonists are used in the treatment of conditions such as pulmonary arterial hypertension and heart failure. These receptors are also important targets in research on cardiovascular diseases and cancer. At CymitQuimica, we offer a selection of high-quality endothelin receptor modulators to support your research in cardiovascular biology, oncology, and vascular physiology.

Found 86 products for "Endothelin Receptor".

Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
products per page.
  • K-8794
    Targetmol
    + Info

    K-8794

    CAS:
    K-8794 is an orally active and selective endothelin receptor ETB antagonist that can be utilized in cardiovascular disease research.
    Formula:C36H38N6O6S
    Color and Shape:Solid
    Molecular weight:682.789

    Ref: TM-T204123

    10mg
    To inquire
    50mg
    To inquire
  • Diosuxentan
    Targetmol
    + Info

    Diosuxentan

    CAS:
    Diosuxentan is an inhibitor of ETA and is utilized in research pertaining to cardiovascular, renal, and neuronal inflammatory diseases.
    Formula:C20H21BrN6O7S
    Color and Shape:Solid
    Molecular weight:569.39

    Ref: TM-T211846

    25mg
    1,504.00€
    50mg
    1,963.00€
    100mg
    2,520.00€
  • BMS-248360
    Targetmol
    + Info

    BMS-248360

    CAS:
    BMS-248360: Oral dual hAT1/hETA antagonist with Kis of 10nM & 1.9nM, respectively; treats hypertension.
    Formula:C36H45N5O5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.84

    Ref: TM-T14672

    25mg
    To inquire
    50mg
    To inquire
    100mg
    To inquire
  • JKC 302
    Targetmol
    + Info

    JKC 302

    CAS:
    JKC 302 is an ET-A receptor antagonist that partially inhibits the contraction of tracheal rings in asthmatic rats induced by ET-1.
    Formula:C30H42N6O6
    Color and Shape:Solid
    Molecular weight:582.69

    Ref: TM-TP3818

    10mg
    To inquire
    50mg
    To inquire
  • Tezosentan
    Targetmol
    + Info

    Tezosentan

    CAS:
    Tezosentan is an antagonist of the endothelin receptor (pA2s: 9.5, 7.7 for ETA and ETB receptors, respectively).
    Formula:C27H27N9O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:605.63

    Ref: TM-T17064

    25mg
    2,025.00€
    50mg
    2,737.00€
    100mg
    3,565.00€
  • BQ-788
    Targetmol
    + Info

    BQ-788

    CAS:
    BQ-788 is an ETB receptor antagonist with potential hypertensive activity that inhibits exogenous ET-1-induced elevation of coronary perfusion pressure.
    Formula:C34H51N5O7
    Purity:98.81%
    Color and Shape:Yellow Solid
    Molecular weight:641.8

    Ref: TM-T10595

    1mg
    130.00€
    2mg
    178.00€
    5mg
    313.00€
    1mL*10mM (DMSO)
    341.00€
    10mg
    447.00€
    25mg
    713.00€
    50mg
    964.00€
    100mg
    1,305.00€
    500mg
    2,592.00€