Bombesin Receptor
Bombesin receptors are a group of GPCRs that are activated by bombesin-like peptides, which are involved in regulating gastrointestinal function, energy balance, and cell proliferation. These receptors are of particular interest in cancer research, as they are often overexpressed in certain types of tumors. Bombesin receptor antagonists are studied for their potential as cancer therapeutics. At CymitQuimica, we provide a selection of high-quality bombesin receptor modulators to support your research in oncology, gastrointestinal physiology, and receptor signaling.
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CD80-IN-3
CAS:486449-65-4
CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 …
Formula:
C17H10FN3O3
Purity:
98.08%
Color and Shape:
Solid
Molecular weight:
323.28
Ref: TM-T10722
| 1mg | 79.00 € | ||
| 5mg | 183.00 € | ||
| 10mg | 299.00 € | ||
| 25mg | 482.00 € | ||
| 50mg | 666.00 € | ||
| 100mg | 828.00 € | ||
| 1mL*10mM (DMSO) | 202.00 € |
Estimated delivery in United States, on Friday 3 Jan 2025
RC-3095 TFA
CAS:1217463-61-0
RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.
Formula:
C58H80F3N15O11
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1220.34
Ref: TM-TP1701
| 1mg | 345.00 € | ||
| 5mg | 768.00 € | ||
| 10mg | 1,208.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 7 Jan 2025
PD176252
CAS:204067-01-6
PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the …
Formula:
C32H36N6O5
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
584.67
Ref: TM-T16449
| 1mg | 35.00 € | ||
| 5mg | 67.00 € | ||
| 10mg | To inquire | ||
| 25mg | To inquire | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
kuwanon G
CAS:75629-19-5
Kuwanon G (Moracenin B) may be used to treat the type II diabetes mellitus as …
Formula:
C40H36O11
Purity:
98% - 98.47%
Color and Shape:
Solid
Molecular weight:
692.71
Ref: TM-T3S1612
| 1mg | 67.00 € | ||
| 5mg | 148.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 344.00 € | ||
| 50mg | 498.00 € | ||
| 100mg | 670.00 € | ||
| 200mg | 902.00 € | ||
| 1mL*10mM (DMSO) | 191.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
Kuwanon H
CAS:76472-87-2
Kuwanon H is a potent non-peptide GRP receptor antagonist with a Ki of 290 nM, …
Formula:
C45H44O11
Purity:
97.99%
Color and Shape:
Solid
Molecular weight:
760.82
Ref: TM-TN1849
| 1mg | 61.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 215.00 € | ||
| 25mg | 413.00 € | ||
| 1mL*10mM (DMSO) | 211.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
ML-18
CAS:1422269-30-4
ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.
Formula:
C32H35N5O5
Purity:
100% - 98.53%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-T4540
| 1mg | 35.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 89.00 € | ||
| 25mg | 173.00 € | ||
| 50mg | 269.00 € | ||
| 100mg | 434.00 € | ||
| 200mg | 598.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Friday 10 Jan 2025
MK-5046
CAS:1022152-70-0
MK-5046 is a novel BRS-3 agonist, binding to BRS-3 with high affinity (mouse Ki = …
Formula:
C20H18F6N4O
Purity:
98.56%
Color and Shape:
Solid
Molecular weight:
444.37
Ref: TM-T2126
| 1mg | 82.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 246.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
PD 168368
CAS:204066-82-0
PD 168368 is a mixed neuromodulin B receptor (NMB-R) antagonist and potent FPR1/FPR2/FPR3 agonist that …
Formula:
C31H34N6O4
Purity:
98.44%
Color and Shape:
Solid
Molecular weight:
554.64
Ref: TM-T8691
| 1mg | 97.00 € | ||
| 25mg | To inquire |
Estimated delivery in United States, on Friday 7 Mar 2025
