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Bombesin Receptor

Bombesin Receptor

Bombesin receptors are a group of GPCRs that are activated by bombesin-like peptides, which are involved in regulating gastrointestinal function, energy balance, and cell proliferation. These receptors are of particular interest in cancer research, as they are often overexpressed in certain types of tumors. Bombesin receptor antagonists are studied for their potential as cancer therapeutics. At CymitQuimica, we provide a selection of high-quality bombesin receptor modulators to support your research in oncology, gastrointestinal physiology, and receptor signaling.

Found 30 products of "Bombesin Receptor"

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  • CD80-IN-3
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    CD80-IN-3

    CAS:
    <p>CD80-IN-3 is a potent CD80 inhibitor and inhibits CD80/CD28 interaction (Kd: 125 nM; EC50: 630 nM).</p>
    Formula:C17H10FN3O3
    Purity:98.08%
    Color and Shape:Solid
    Molecular weight:323.28

    Ref: TM-T10722

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    AMTG-DA1

    <p>AMTG-DA1 is a ligand for the gastrin-releasing peptide receptor (GRPR), and it can be utilized in cancer research.</p>
    Formula:C101H149IN22O25
    Color and Shape:Solid
    Molecular weight:2197.0109

    Ref: TM-T207222

  • RC-3095
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    RC-3095

    CAS:
    <p>RC-3095, a selective GRPR antagonist, has been shown to have anti-inflammatory properties in different models of inflammation.</p>
    Formula:C56H79N15O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1106.32

    Ref: TM-TP1470

  • BA 1
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    BA 1

    CAS:
    <p>Potent BB1, BB2, and BB3 agonist; IC50: 0.26, 1.55, 2.52 nM. Boosts glucose transport in myocytes, promotes cancer cell growth in vitro.</p>
    Formula:C57H76N14O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1133.32

    Ref: TM-TP1913

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    PSMA/GRPR ligand 1

    <p>PSMA/GRPR ligand 1 (compound 3) is a bispecific ligand with dual targeting capabilities for tumors that express PSMA(+) and GRPR(+).</p>
    Color and Shape:Odour Solid

    Ref: TM-T206782

  • [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P
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    [D-Arg1,D-Phe5,D-Trp7,9,Leu11]-Substance P

    CAS:
    <p>Broad-spectrum inverse agonist; potent at ghrelin receptor (EC50=5.2 nM); blocks other neuropeptide receptors; induces apoptosis; inhibits tumor growth.</p>
    Formula:C79H109N19O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1516.85

    Ref: TM-TP1931

  • [D-Phe12]-Bombesin
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    [D-Phe12]-Bombesin

    CAS:
    <p>Bombesin receptor antagonist</p>
    Formula:C74H112N22O18S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1629.88

    Ref: TM-TP2239

  • [D-Phe12,Leu14]-Bombesin
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    [D-Phe12,Leu14]-Bombesin

    CAS:
    <p>Bombesin receptor blocker; stops binding in rat brain (IC50=2 μM), hinders amylase release (IC50=4 μM), reduces appetite suppression in vivo.</p>
    Formula:C77H113F3N22O20
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1724.9

    Ref: TM-TP1916

  • (D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14)
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    (D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14)

    CAS:
    <p>(D-Phe6,Leu-NHEt13,des-Met14)-Bombesin (6-14), a bombesin (BBN) antagonist, holds potential for cancer research applications [1].</p>
    Formula:C49H69N13O9
    Color and Shape:Solid
    Molecular weight:984.15

    Ref: TM-T76601

  • CymitQuimica logo
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    BA 1 TFA

    <p>BA1 TFA agonizes BB receptors; binds BRS3, GRPR, NMBR with IC50s of 6, 0.4, 2.5 nM.</p>
    Formula:C59H77F3N14O13
    Color and Shape:Solid
    Molecular weight:1247.32

    Ref: TM-T75945

  • Ici 216140
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    Ici 216140

    CAS:
    <p>ICI 216140: GRP/bombesin receptor 2 blocker, potent at 2 nM. Reduces amylase at 2 mg/kg and lowers bombesin-induced blood pressure at 1 mM in rats.</p>
    Formula:C45H65N13O8
    Color and Shape:Solid
    Molecular weight:916.08

    Ref: TM-T25522

  • GRP (14-27) (human, porcine, canine)
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    GRP (14-27) (human, porcine, canine)

    CAS:
    <p>GRP (14-27) (human, porcine, canine) functions as a ligand for bombesin receptors, with its specific binding being inhibited by GTP and GDP, while GMP does not</p>
    Formula:C75H110N24O16S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1667.96

    Ref: TM-T80148

  • GB-6
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    GB-6

    CAS:
    <p>GB-6, a short linear peptide that selectively binds to the gastrin releasing peptide receptor (GRPR), shows potential as a high-contrast imaging probe due to</p>
    Formula:C32H45N11O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:711.77

    Ref: TM-T80266

  • RC-3095 TFA
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    RC-3095 TFA

    CAS:
    <p>RC-3095 TFA (RC-3095 (TFA)) is a bombesin/gastrin-releasing peptide (BN/GRP) antagonist with potential anticancer activity.</p>
    Formula:C58H80F3N15O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1220.34

    Ref: TM-TP1701

  • Bombesin
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    Bombesin

    CAS:
    <p>Bombesin: 14-amino acid peptide from toad skin with two mammalian homologs, neuromedin B and gastrin-releasing peptide.</p>
    Formula:C71H110N24O18S
    Color and Shape:While Lyophilized Powder
    Molecular weight:1619.85

    Ref: TM-TP1281

  • PD176252
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    PD176252

    CAS:
    <p>PD176252 is a BB1 and BB2 antagonist, GRPR inhibitor, and FPR1/FPR2 agonist that inhibits the growth and proliferation of a wide range of cancer cells.</p>
    Formula:C32H36N6O5
    Purity:99.18%
    Color and Shape:Solid
    Molecular weight:584.67

    Ref: TM-T16449

  • ML-18
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    ML-18

    CAS:
    <p>ML-18 is a non-peptide bombesin receptor subtype-3 (BRS-3) antagonist with an IC50 of 4.8 μM.</p>
    Formula:C32H35N5O5
    Purity:98.62% - >99.99%
    Color and Shape:Solid
    Molecular weight:569.65

    Ref: TM-T4540

  • kuwanon G
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    kuwanon G

    CAS:
    <p>Kuwanon G (Moracenin B) may be used to treat the type II diabetes mellitus as a dual inhibitor of PTP1B and α-glucosidase and as an insulin sensitiser.</p>
    Formula:C40H36O11
    Purity:98% - 99.57%
    Color and Shape:Solid
    Molecular weight:692.71

    Ref: TM-T3S1612

  • Litorin acetate(55749-97-8 Free base)
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    Litorin acetate(55749-97-8 Free base)

    <p>Litorin acetate, an amphibian bombesin peptide derivative, is an bombesin receptor agonist.</p>
    Formula:C53H72N14O13S
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:1145.29

    Ref: TM-T20604L

  • Bombesin acetate(31362-50-2 free base)
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    Bombesin acetate(31362-50-2 free base)

    CAS:
    <p>Bombesin acetate is a 14-amino acid peptide originally isolated from the skin of the European fire-bellied toad (Bombina bombina).</p>
    Formula:C73H114N24O20S
    Purity:98.44%
    Color and Shape:Solid
    Molecular weight:1679.92

    Ref: TM-TP1281L1