Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Found 358 products of "Histamine Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Fexofenadine-d6
CAS:<p>Fexofenadine D6 is an antihistamine pharmaceutical drug.Fexofenadine D6 is deuterium labeled is Fexofenadine.</p>Formula:C32H39NO4Purity:98%Color and Shape:SolidMolecular weight:507.69Cetirizine D4
CAS:<p>Cetirizine D4 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Formula:C21H25ClN2O3Purity:98%Color and Shape:SolidMolecular weight:392.91Diphenylpyraline
CAS:<p>Diphenylpyridine is the first generation antihistamine, which has the anticholinergic effect of diphenylpiperidine.</p>Formula:C19H23NOColor and Shape:SolidMolecular weight:281.39WZ4141
CAS:<p>WZ4141 is an intermediate in compound synthesis.</p>Formula:C16H13N3O2Purity:98%Color and Shape:SolidMolecular weight:279.29Acrivastine D7
CAS:<p>Acrivastine D7 is a deuterium labeled Acrivastine. Acrivastine is a short acting antagonist of histamine 1 receptor.</p>Formula:C22H24N2O2Purity:98%Color and Shape:SolidMolecular weight:355.48Doxepin D3 Hydrochloride
CAS:<p>Doxepin D3 Hydrochloride is a deuterium-labeled doxepin hydrochloride.Doxepin hydrochloride is an oral active tricyclic antidepressant used as a sedative.Doxepin hydrochloride is also an effective CYP450 inhibitor, significantly inhibiting CYP450 2C19 and</p>Formula:C19H22ClNOPurity:98%Color and Shape:SolidMolecular weight:318.86Emedastine Difumarate
CAS:<p>Emedastine Difumarate, an H1 receptor blocker for allergic conjunctivitis, reduces histamine-induced eye inflammation.</p>Formula:C25H34N4O9Color and Shape:SolidMolecular weight:534.56Cetirizine D8
CAS:<p>Cetirizine D8 is a deuterium-labeled Cetirizine. Cetirizine is a second-generation antihistamine and a long-acting histamine H1-receptor antagonist.</p>Formula:C21H25ClN2O3Purity:98%Color and Shape:SolidMolecular weight:396.94Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Formula:C8H12N2Purity:99.87% - 99.87%Color and Shape:Yellowish Liquid Liquid LiquidMolecular weight:136.19S 38093
CAS:<p>S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).</p>Formula:C17H24N2O2Purity:99.95%Color and Shape:SolidMolecular weight:288.38GSK189254A
CAS:<p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>Formula:C21H25N3O2Purity:98.71% - 99.858%Color and Shape:SolidMolecular weight:351.44Emedastine
CAS:<p>Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.</p>Formula:C17H26N4OPurity:97.1% - 97.76%Color and Shape:OilMolecular weight:302.41Fexofenadine hydrochloride
CAS:<p>Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the treatment of allergic rhinitis,</p>Formula:C32H39NO4·HClPurity:99.39% - ≥95%Color and Shape:SolidMolecular weight:538.13Buclizine dihydrochloride
CAS:<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Formula:C28H33ClN2·2HClPurity:98.05%Color and Shape:Off-White PowderMolecular weight:505.95Conessine
CAS:<p>Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor and has anti-malarial activity.</p>Formula:C24H40N2Purity:99.65%Color and Shape:SolidMolecular weight:356.59Chlorpheniramine
CAS:<p>Chlorpheniramine is an H1 anti-histamine agent for IgE-mediated inflammation that is commonly used for allergic diseases.</p>Formula:C16H19ClN2Color and Shape:SolidMolecular weight:274.79Dioxopromethazine hydrochloride
CAS:<p>Dioxopromethazine is a target-based classification of drug and available in a number of countries worldwide.</p>Formula:C17H20N2O2S·HClPurity:99.58%Color and Shape:SolidMolecular weight:352.88Hydroxyzine
CAS:<p>Hydroxyzine (Hydroxyzine free base) is an antagonist of histamine H1-receptor.</p>Formula:C21H27ClN2O2Purity:99.54% - ≥95%Color and Shape:Oil SolidMolecular weight:374.9SCH-37370
CAS:<p>SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.</p>Formula:C21H21ClN2OPurity:99.07%Color and Shape:SolidMolecular weight:352.86H4 Receptor antagonist 1
CAS:<p>H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.</p>Formula:C16H17ClN4OPurity:98.81%Color and Shape:SolidMolecular weight:316.79Triprolidine
CAS:<p>Triprolidine: oral H1 receptor blocker with motor/sensory spinal effects, for allergy research.</p>Formula:C19H22N2Color and Shape:SolidMolecular weight:278.39Fenspiride
CAS:<p>Fenspiride: oral non-steroidal anti-inflammatory, treats respiratory infections/otitis, inhibits H1-histamine receptors and PDE 3, 4, 5.</p>Formula:C15H20N2O2Color and Shape:SolidMolecular weight:260.33Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Formula:C15H19N3Purity:≥95%Color and Shape:SolidMolecular weight:241.33Bilastine
CAS:<p>Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration of</p>Formula:C28H37N3O3Purity:99.86% - >99.99%Color and Shape:SolidMolecular weight:463.61Clemizole hydrochloride
CAS:<p>Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.</p>Formula:C19H21Cl2N3Purity:>99.99%Color and Shape:SolidMolecular weight:362.3Clobenpropit dihydrobromide
CAS:<p>Clobenpropit dihydrobromide is a potent antagonist and inverse agonist of histamine H3R (histamine H3LR,pEC50 of 8.07)</p>Formula:C14H19Br2ClN4SPurity:99.86%Color and Shape:SolidMolecular weight:470.7Ritanserin
CAS:<p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>Formula:C27H25F2N3OSPurity:99.77% - 99.89%Color and Shape:SolidMolecular weight:477.57Antazoline
CAS:<p>Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.</p>Formula:C17H19N3Purity:≥95%Color and Shape:White Crystalline Powder SolidMolecular weight:265.35Psoralenoside
CAS:<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Formula:C17H18O9Purity:99.03% - 99.49%Color and Shape:SolidMolecular weight:366.32Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Formula:C21H28N2O2Purity:99.53%Color and Shape:White Or Similar To White PowderMolecular weight:340.46Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Formula:C20H25FN4OPurity:99.56%Color and Shape:SolidMolecular weight:356.442-Pyridylethylamine dihydrochloride
CAS:<p>2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.</p>Formula:C7H12Cl2N2Purity:99.42%Color and Shape:SolidMolecular weight:195.09Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Formula:C18H18ClNOSPurity:99.78%Color and Shape:SolidMolecular weight:331.86Clobenpropit 2HBr
CAS:<p>Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.</p>Formula:C14H17ClN4SColor and Shape:SolidMolecular weight:308.83Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Formula:C11H6ClN3O6Purity:99.13% - 99.81%Color and Shape:SolidMolecular weight:311.63cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Formula:C16H14O2Purity:98.15%Color and Shape:SolidMolecular weight:238.2812Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Formula:C9H7N5O3Purity:98.25%Color and Shape:SolidMolecular weight:233.18Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Formula:C15H19Cl2N3O3SPurity:98.48%Color and Shape:SolidMolecular weight:392.3HTMT dimaleate
CAS:<p>HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.</p>Formula:C27H33F3N4O9Purity:99.51%Color and Shape:SolidMolecular weight:614.57Triprolidine hydrochloride
CAS:<p>Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.</p>Formula:C19H23ClN2Color and Shape:SolidMolecular weight:314.852Tribenoside
CAS:<p>Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.</p>Formula:C29H34O6Purity:≥98%Color and Shape:LiquidMolecular weight:478.58Dioxopromethazine
CAS:<p>Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.</p>Formula:C17H20N2O2SPurity:98%Color and Shape:SolidMolecular weight:316.42Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Formula:C14H20F6N4O7Purity:98.18%Color and Shape:SolidMolecular weight:470.32Buclizine
CAS:<p>Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.</p>Formula:C28H33ClN2Color and Shape:SolidMolecular weight:433.03Desloratadine
CAS:<p>Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.</p>Formula:C19H19ClN2Purity:99.79% - >99.99%Color and Shape:SolidMolecular weight:310.82Fexofenadine
CAS:<p>Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.</p>Formula:C32H39NO4Purity:99.35%Color and Shape:White To Off-White SolidMolecular weight:501.66JNJ-5207852 dihydrochloride
CAS:<p>JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor</p>Formula:C20H34Cl2N2OPurity:99.51%Color and Shape:SolidMolecular weight:389.4Bepotastine Besilate
CAS:<p>Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).</p>Formula:C21H25ClN2O3·C6H6O3SPurity:99.83% - 99.9%Color and Shape:Brown Viscous LiquidMolecular weight:547.06Talastine HCl
CAS:<p>Talastine is an antihistamine drug.</p>Formula:C19H22ClN3OPurity:98%Color and Shape:SolidMolecular weight:343.86VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Formula:C15H19N5Purity:99.44% - 99.57%Color and Shape:SolidMolecular weight:269.34
