Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
Read more
Pheniramine maleate
CAS:132-20-7
Pheniramine maleate (Trimetose), an alkylamine derivative with antihistaminic and vasodilatory properties, binds to histamine H1 …
Formula:
C16H20N2·C4H4O4
Purity:
99.79%
Color and Shape:
Physical Description White Powder With A Faint Amine-Like Odor Melting Point 107°C
Molecular weight:
356.42
Ref: TM-T0370
| 25mg | 36.00 € | ||
| 50mg | 45.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 65.00 € | ||
| 500mg | 91.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
JNJ-39758979
CAS:1046447-90-8
JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).
Formula:
C11H19N5
Purity:
98.00% - 98.3%
Color and Shape:
Solid
Molecular weight:
221.3
Ref: TM-T11723L
| 1mg | 74.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 247.00 € | ||
| 25mg | 419.00 € | ||
| 50mg | 608.00 € | ||
| 100mg | 894.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Carbinoxamine Maleate Salt
CAS:3505-38-2
Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and …
Formula:
C20H23ClN2O5
Purity:
99.81%
Color and Shape:
Off-White Solid
Molecular weight:
406.86
Ref: TM-T2222
| 25mg | 46.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 72.00 € | ||
| 200mg | 95.00 € | ||
| 500mg | 181.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Amitriptyline hydrochloride
CAS:549-18-8
Amitriptyline hydrochloride (Annoyltin) is the hydrochloride salt of the tricyclic dibenzocycloheptadiene amitriptyline with antidepressant and …
Formula:
C20H24ClN
Purity:
97% - 99.94%
Color and Shape:
Crystals White To Off-White Powder
Molecular weight:
313.86
Ref: TM-T0678
| 1g | 57.00 € | ||
| 500mg | 49.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Mizolastine
CAS:108612-45-9
Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever …
Formula:
C24H25FN6O
Purity:
98% - 99.77%
Color and Shape:
Solid
Molecular weight:
432.49
Ref: TM-T0118
| 10mg | 41.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 179.00 € | ||
| 500mg | 291.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
(+)-Dropropizine
CAS:99291-24-4
(+)-Dropropizine can inhibit histamine receptor, anti-allergic, and reduce a cough by modulation of neuropeptides involved …
Formula:
C13H20N2O2
Purity:
99.92%
Color and Shape:
White Or Off White Crystalline Powder
Molecular weight:
236.31
Ref: TM-T0217L
| 1g | 49.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Doxepin hydrochloride
CAS:1229-29-4
Doxepin hydrochloride, a dibenzoxepin tricyclic, blocks monoamine reuptake and has anticholinergic and antihistaminic effects. Mechanism …
Formula:
C19H22ClNO
Purity:
99.57% - 99.91%
Color and Shape:
White To Off-White Powder
Molecular weight:
315.837
Ref: TM-T1540
| 1g | 59.00 € | ||
| 5g | 123.00 € | ||
| 10g | 152.00 € | ||
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Perphenazine
CAS:58-39-9
Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.
Formula:
C21H26ClN3OS
Purity:
99.3% - 99.72%
Color and Shape:
Solid
Molecular weight:
403.97
Ref: TM-T1090
| 50mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Terfenadine
CAS:50679-08-8
Terfenadine, metabolized to fexofenadine by CYP3A4, is a non-sedative antihistamine targeting H1 receptors.
Formula:
C32H41NO2
Purity:
98.76% - 99.75%
Color and Shape:
Solid
Molecular weight:
471.67
Ref: TM-T1266
| 50mg | 42.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 81.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Brompheniramine maleate
CAS:980-71-2
Brompheniramine maleate (Dimotane) is an antagonist against histamine H1 receptors.
Formula:
C16H19BrN2·C4H4O4
Purity:
99.3%
Color and Shape:
Crystal Powder
Molecular weight:
435.31
Ref: TM-T0205
| 25mg | 34.00 € | ||
| 50mg | 43.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 94.00 € | ||
| 500mg | 144.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Betahistine mesylate
CAS:54856-23-4
Betahistine mesylate (Extovyl), an H1 agonist and vasodilator, treats Meniere's disease and vascular headaches; risks …
Formula:
C8H12N2·2(CH4O3S)
Purity:
98%
Color and Shape:
Coa
Molecular weight:
328.4
Ref: TM-T0246L
| 10mg | 35.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Triprolidine hydrochloride monohydrate
CAS:6138-79-0
Triprolidine hydrochloride monohydrate is a histamine H1 antagonist used in allergic rhinitis, asthma.
Formula:
C19H25ClN2O
Purity:
99.68% - ≥95%
Color and Shape:
White Crystalline Powder
Molecular weight:
332.87
Ref: TM-T1030
| 10mg | 35.00 € | ||
| 25mg | 69.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 138.00 € | ||
| 500mg | 331.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Benztropine mesylate
CAS:132-17-2
Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in …
Formula:
C21H25NO·CH4SO3
Purity:
100% - 99.52%
Color and Shape:
White Crystalline Powder; Odourless Or Almost Odourless
Molecular weight:
403.53
Ref: TM-T1336
| 500mg | 39.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Azacyclonol
CAS:115-46-8
Azacyclonol (MER 17) is a drug used to diminish hallucinations in psychotic individuals.
Formula:
C18H21NO
Purity:
99.61%
Color and Shape:
Solid Powder
Molecular weight:
267.37
Ref: TM-T0318
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Tripelennamine hydrochloride
CAS:154-69-8
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent …
Formula:
C16H21N3·HCl
Purity:
100% - 100%
Color and Shape:
White Solid
Molecular weight:
291.82
Ref: TM-T1269
| 1g | 138.00 € | ||
| 100mg | 37.00 € | ||
| 500mg | 93.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Chlorpheniramine maleate
CAS:113-92-8
Chlorpheniramine maleate (NCI-C55265) is a histamine H1 antagonist used in allergic reactions, hay fever, rhinitis, …
Formula:
C20H23ClN2O4
Purity:
99.67%
Color and Shape:
Odorless White Crystalline Solid Or White Powder With A Bitter Taste
Molecular weight:
390.87
Ref: TM-T1553
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Loratadine
CAS:79794-75-5
Loratadine (SCH 29851) is a second-generation histamine H1 receptor antagonist used in the treatment of …
Formula:
C22H23ClN2O2
Purity:
99.49% - 99.75%
Color and Shape:
White Powder
Molecular weight:
382.88
Ref: TM-T1097
| 500mg | 48.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Pimethixene
CAS:314-03-4
Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 & muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.
Formula:
C19H19NS
Purity:
99.1%
Color and Shape:
Solid
Molecular weight:
293.43
Ref: TM-T12489
| 2mg | 34.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 63.00 € | ||
| 25mg | 103.00 € | ||
| 50mg | 152.00 € | ||
| 100mg | 218.00 € | ||
| 200mg | 326.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Chloropyramine hydrochloride
CAS:6170-42-9
Chloropyramine hydrochloride (Alergosan) is a histamine receptor H1 antagonist.
Formula:
C16H20ClN3·HCl
Purity:
99.45% - 99.8%
Color and Shape:
Solid
Molecular weight:
326.26
Ref: TM-T0263
| 25mg | 39.00 € | ||
| 50mg | 51.00 € | ||
| 100mg | 74.00 € | ||
| 200mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Cinnarizine
CAS:298-57-7
Cinnarizine is a piperazine, blocks H1-receptor & Ca-channels, has vasodilating & antiemetic effects, may cause …
Formula:
C26H28N2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
368.51
Ref: TM-T0903
| 50mg | 46.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 85.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
