Histamine Receptor
Histamine receptors are GPCRs that mediate the effects of histamine, a biogenic amine involved in immune responses, gastric acid secretion, and neurotransmission. There are four subtypes of histamine receptors (H1, H2, H3, and H4), each playing distinct roles in allergic reactions, gastric function, and central nervous system activity. Histamine receptor antagonists are widely used in the treatment of allergies, peptic ulcers, and motion sickness. At CymitQuimica, we provide a comprehensive selection of high-quality histamine receptor modulators to support your research in immunology, gastroenterology, and neuropharmacology.
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WZ4141
CAS:1222776-76-2
WZ4141 is an intermediate in compound synthesis.
Formula:
C16H13N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
279.29
Ref: TM-T19604
| 5mg | 439.00 € | ||
| 1mL*10mM (DMSO) | 433.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Betahistine dihydrochloride
CAS:5579-84-0
Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as …
Formula:
C8H14Cl2N2
Purity:
99.34% - 99.88%
Color and Shape:
White To Light Yellow Crystalline Powder
Molecular weight:
209.12
Ref: TM-T0246
| 1g | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
H4 Receptor antagonist 1
CAS:848217-00-5
H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with …
Formula:
C16H17ClN4O
Purity:
98.81%
Color and Shape:
Solid
Molecular weight:
316.79
Ref: TM-T5829
| 2mg | 45.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 176.00 € | ||
| 50mg | 302.00 € | ||
| 100mg | 435.00 € | ||
| 500mg | 931.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Mebhydrolin
CAS:524-81-2
Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.
Formula:
C19H20N2
Purity:
99.73% - ≥98%
Color and Shape:
Solid
Molecular weight:
276.38
Ref: TM-T7085
| 100mg | 43.00 € | ||
| 200mg | 64.00 € | ||
| 500mg | 124.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Fexofenadine
CAS:83799-24-0
Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.
Formula:
C32H39NO4
Purity:
99.87%
Color and Shape:
White To Off-White Solid
Molecular weight:
501.66
Ref: TM-T21390
| 10mg | 50.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 143.00 € | ||
| 200mg | 208.00 € | ||
| 500mg | 364.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Conessine
CAS:546-06-5
Conessine (Conessinum), a steroidal alkaloid isolated from Holarrhena floribunda, interacts with the histamine H3 receptor …
Formula:
C24H40N2
Purity:
99.65%
Color and Shape:
Solid
Molecular weight:
356.59
Ref: TM-T20712
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 330.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Fexofenadine hydrochloride
CAS:153439-40-8
Fexofenadine hydrochloride (Terfenidine carboxylate hydrochloride) is a second generation antihistamine that is used for the …
Formula:
C32H39NO4·HCl
Purity:
99.39% - ≥95%
Color and Shape:
Solid
Molecular weight:
538.13
Ref: TM-T1470
| 10mg | 49.00 € | ||
| 25mg | 77.00 € | ||
| 50mg | 95.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Acrivastine
CAS:87848-99-5
Acrivastine (Acrivastin) is a short-acting histamine 1 receptor antagonist.
Formula:
C22H24N2O2
Purity:
100% - 99.85%
Color and Shape:
Solid
Molecular weight:
348.44
Ref: TM-T4551
| 1g | 774.00 € | ||
| 5mg | 41.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 102.00 € | ||
| 50mg | 162.00 € | ||
| 100mg | 222.00 € | ||
| 500mg | 541.00 € | ||
| 1mL*10mM (DMSO) | 41.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Chlorphenoxamine
CAS:77-38-3
Chlorphenoxamine (Contristamine) is an antihistamine and anticholinergic used as an antipruritic and antiparkinsonian agent.
Formula:
C18H22ClNO
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
303.83
Ref: TM-T7564
| 5mg | 51.00 € | ||
| 10mg | 80.00 € | ||
| 50mg | 145.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Alcaftadine
CAS:147084-10-4
Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated …
Formula:
C19H21N3O
Purity:
98% - 99.99%
Color and Shape:
Solid
Molecular weight:
307.39
Ref: TM-T2533
| 10mg | 34.00 € | ||
| 25mg | 67.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 130.00 € | ||
| 200mg | 200.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Bepotastine Besilate
CAS:190786-44-8
Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).
Formula:
C21H25ClN2O3·C6H6O3S
Purity:
99.83% - 99.90%
Color and Shape:
Brown Viscous Liquid
Molecular weight:
547.06
Ref: TM-T6405
| 100mg | 46.00 € | ||
| 500mg | 90.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Desloratadine
CAS:100643-71-8
Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.
Formula:
C19H19ClN2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
310.82
Ref: TM-T2520
| 1g | 356.00 € | ||
| 25mg | 41.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 68.00 € | ||
| 200mg | 97.00 € | ||
| 500mg | 225.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Lodoxamide
CAS:53882-12-5
Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in …
Formula:
C11H6ClN3O6
Purity:
99.13% - 99.81%
Color and Shape:
Solid
Molecular weight:
311.63
Ref: TM-T4566
| 5mg | 46.00 € | ||
| 10mg | 59.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 183.00 € | ||
| 200mg | 319.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Niaprazine
CAS:27367-90-4
Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.
Formula:
C20H25FN4O
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
356.44
Ref: TM-T36949
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 299.00 € | ||
| 200mg | 429.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ritanserin
CAS:87051-43-2
Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective …
Formula:
C27H25F2N3OS
Purity:
99.45% - 99.89%
Color and Shape:
Solid
Molecular weight:
477.57
Ref: TM-T16759
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 182.00 € | ||
| 50mg | 268.00 € | ||
| 100mg | 403.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Emedastine
CAS:87233-61-2
Emedastine (LY188695) is a second generation, selective histamine H1 receptor antagonist with anti-allergic activity.
Formula:
C17H26N4O
Purity:
97.1% - 97.1%
Color and Shape:
Oil
Molecular weight:
302.41
Ref: TM-T3979
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 113.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 409.00 € | ||
| 500mg | 912.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Tesmilifene fumarate
CAS:1185241-83-1
Tesmilifene fumarate (DPPE fumarate) (DPPE fumarate) is an H1C receptor antagonist。
Formula:
C23H29NO5
Purity:
99.38%
Color and Shape:
Solid
Molecular weight:
399.48
Ref: TM-T22746
| 5mg | 45.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 112.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 240.00 € | ||
| 200mg | 355.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Diphenhydramine
CAS:58-73-1
Diphenhydramine (Syntedril): first-gen antihistamine for allergies, antiemetic, antitussive, anticholinergic, sedative, treats drug-induced parkinsonism.
Formula:
C17H21NO
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
255.35
Ref: TM-T21419
| 200mg | 40.00 € | ||
| 500mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ebastine
CAS:90729-43-4
Ebastine (Kestine) (trade names Evastin, Kestine, Ebastel, Aleva) is a non-sedating H1 antihistamine.
Formula:
C32H39NO2
Purity:
100% - 99.93%
Color and Shape:
White To Off-White Powder
Molecular weight:
469.66
Ref: TM-T2335
| 500mg | 56.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Pitolisant hydrochloride
CAS:903576-44-3
Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki …
Formula:
C17H27Cl2NO
Purity:
99.26% - 99.72%
Color and Shape:
Solid
Molecular weight:
332.31
Ref: TM-T7176
| 5mg | 51.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 193.00 € | ||
| 100mg | 305.00 € | ||
| 200mg | 460.00 € | ||
| 500mg | 731.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
