Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
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Dermorphin TFA
CAS:78331-26-7
Dermorphin TFA is a new class of opioids-like peptides
Formula:
C42H51F3N8O12
Purity:
100% - 98%
Color and Shape:
Solid
Molecular weight:
916.89
Ref: TM-T7748
| 1mg | 89.00 € | ||
| 2mg | 138.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 277.00 € | ||
| 25mg | 518.00 € | ||
| 50mg | 741.00 € | ||
| 100mg | 1,016.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Gluten Exorphin C
CAS:142479-62-7
Gluten exorphin C is an opioid peptide derived from wheat gluten.
Formula:
C29H45N5O8
Purity:
100%
Color and Shape:
Solid
Molecular weight:
591.7
Ref: TM-TP1832
| 1mg | 46.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 344.00 € | ||
| 100mg | 504.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
![[Leu5]-Enkephalin TFA(58822-25-6(free bas))](https://static.cymitquimica.com/products/TM/thumb/T7665.jpg)
[Leu5]-Enkephalin TFA(58822-25-6(free bas))
CAS:73563-78-7
[Leu5]-Enkephalin TFA(58822-25-6(free bas)) (Leucyl-enkephalin) is the most potent δ-receptor ago
Formula:
C30H38F3N5O9
Purity:
97.03% - 99.78%
Color and Shape:
Solid
Molecular weight:
669.64
Ref: TM-T7665
| 10mg | 51.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 144.00 € | ||
| 100mg | 209.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
ADL-5859
CAS:850173-95-4
ADL-5859 (ADL5859 Hydrochloride) is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against …
Formula:
C24H28N2O3·HCl
Purity:
99.11% - 99.71%
Color and Shape:
Solid
Molecular weight:
428.95
Ref: TM-T6175
| 1mg | 52.00 € | ||
| 2mg | 70.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 167.00 € | ||
| 25mg | 333.00 € | ||
| 50mg | 513.00 € | ||
| 100mg | 739.00 € | ||
| 500mg | 1,514.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
MCOPPB triHydrochloride
CAS:1108147-88-1
MCOPPB triHydrochloride (MCOPPB 3HCl) is a nociceptin receptor agonist.
Formula:
C26H43Cl3N4
Purity:
99.89% - 99.91%
Color and Shape:
Solid
Molecular weight:
518.01
Ref: TM-T2071
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 158.00 € | ||
| 50mg | 246.00 € | ||
| 100mg | 362.00 € | ||
| 200mg | 516.00 € | ||
| 1mL*10mM (DMSO) | 56.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Deltorphin I
CAS:122752-15-2
Deltorphin I is an agonist of δ-opioid receptor.
Formula:
C37H52N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
768.86
Ref: TM-T7637
| 1mg | 62.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 343.00 € | ||
| 50mg | 505.00 € | ||
| 100mg | 720.00 € | ||
| 1mL*10mM (DMSO) | 199.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Tyr-Gly-Gly-Phe-Met-OH
CAS:58569-55-4
Tyr-Gly-Gly-Phe-Met-OH (Met-Enkephalin), is a naturally occurring, endogenous opioid peptide that inhibits tumor growth via binding …
Formula:
C27H35N5O7S
Purity:
≥95%
Color and Shape:
White Lyophilised Solid
Molecular weight:
573.66
Ref: TM-T7211
| 10mg | 35.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 177.00 € | ||
| 1mL*10mM (DMSO) | 37.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Endomorphin 2
CAS:141801-26-5
EM-2 reduces sEPSC frequency/amplitude in lamina IX motoneurons; CTOP reverses this. EM-2-IR affects limb muscles …
Formula:
C32H37N5O5
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
571.67
Ref: TM-T7218
| 1mg | 48.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 310.00 € | ||
| 100mg | 466.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
EST73502 HCl
CAS:2307458-82-6
EST73502 is an agonist of μ-opioid receptor(Ki = 64 nM) agonist and an antagonist of …
Formula:
C19H27ClF2N2O2
Purity:
97.66%
Color and Shape:
Solid
Molecular weight:
388.88
Ref: TM-T39284
| 1mg | 89.00 € | ||
| 5mg | 176.00 € | ||
| 10mg | 251.00 € | ||
| 25mg | 413.00 € | ||
| 50mg | 582.00 € | ||
| 100mg | 770.00 € | ||
| 200mg | 1,044.00 € | ||
| 1mL*10mM (DMSO) | 193.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
JTC-801
CAS:244218-51-7
JTC-801 is a selective opioid receptor-like1 (ORL1) receptor antagonist with IC50 of 94 nM, weakly …
Formula:
C26H25N3O2·HCl
Purity:
98% - 99.27%
Color and Shape:
Solid
Molecular weight:
447.96
Ref: TM-T6553
| 5mg | 48.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 139.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BMS-986122
CAS:313669-88-4
BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment …
Formula:
C16H15BrClNO3S2
Purity:
98.42%
Color and Shape:
Solid
Molecular weight:
448.78
Ref: TM-T26869
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 158.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 539.00 € | ||
| 100mg | 772.00 € | ||
| 500mg | 1,537.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Sinomenine
CAS:115-53-7
Sinomenine (Kukoline) is a pure alkaloid isolated from the Sinomenium acutum, is utilized in the …
Formula:
C19H23NO4
Purity:
99.02% - 99.89%
Color and Shape:
White Powder
Molecular weight:
329.39
Ref: TM-T2726
| 100mg | 59.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PZM21
CAS:1997387-43-5
PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).
Formula:
C19H27N3O2S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
361.5
Ref: TM-T4386
| 1mg | 46.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 203.00 € | ||
| 50mg | 295.00 € | ||
| 100mg | 468.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BMS986187
CAS:684238-37-7
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
Formula:
C31H34O4
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
470.6
Ref: TM-T8991
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 118.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 503.00 € | ||
| 500mg | 1,068.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
GR103545
CAS:126766-43-6
GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can …
Formula:
C23H29Cl2N3O7
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
530.4
Ref: TM-T9459
| 1mg | 96.00 € | ||
| 2mg | 141.00 € | ||
| 5mg | 185.00 € | ||
| 10mg | 278.00 € | ||
| 25mg | 499.00 € | ||
| 50mg | 715.00 € | ||
| 100mg | 994.00 € | ||
| 1mL*10mM (DMSO) | 249.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
LY2795050
CAS:1346133-08-1
LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).
Formula:
C23H22ClN3O2
Purity:
97.77%
Color and Shape:
Solid
Molecular weight:
407.89
Ref: TM-TQ0091
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 114.00 € | ||
| 10mg | 177.00 € | ||
| 25mg | 292.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 126.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
DAMGO
CAS:78123-71-4
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity …
Formula:
C26H35N5O6
Purity:
98.83% - 99.92%
Color and Shape:
Solid
Molecular weight:
513.59
Ref: TM-T4351
| 1mg | 50.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 416.00 € | ||
| 100mg | 609.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Spinorphin
CAS:137201-62-8
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
Formula:
C45H64N8O10
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
877
Ref: TM-T8455
| 1mg | 129.00 € | ||
| 5mg | 241.00 € | ||
| 10mg | 373.00 € | ||
| 25mg | 622.00 € | ||
| 50mg | 887.00 € | ||
| 100mg | 1,201.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C50H72N15O15S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1326.26
Ref: TM-T7567L
| 1mg | 47.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 314.00 € | ||
| 50mg | 450.00 € | ||
| 100mg | 621.00 € | ||
| 200mg | 836.00 € | ||
| 1mL*10mM (DMSO) | 180.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
![[D-Ala2]leucine-enkephalin](https://static.cymitquimica.com/products/TM/thumb/TP1367.jpg)
[D-Ala2]leucine-enkephalin
CAS:64963-01-5
[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta …
Formula:
C29H39N5O7
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-TP1367
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 326.00 € | ||
| 100mg | 460.00 € | ||
| 200mg | 643.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
