Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
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LY2444296
CAS:1346133-11-6
LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 …
Formula:
C24H22F2N2O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
408.44
Ref: TM-T11909
| 5mg | 46.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 3 Feb 2025
IPAG
CAS:193527-91-2
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
Formula:
C17H22IN3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
395.28
Ref: TM-T22870
| 1mg | 45.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 449.00 € | ||
| 100mg | 647.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
ICI 199,441 hydrochloride
CAS:115199-84-3
ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
Formula:
C21H25Cl3N2O
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
427.8
Ref: TM-T22849
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 320.00 € | ||
| 200mg | 449.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
GSK1521498 free base
CAS:1007573-18-3
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor.
Formula:
C24H20F2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
402.44
Ref: TM-T11478L
| 25mg | 1,178.00 € | ||
| 50mg | 1,537.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
ICI 204,448
CAS:121264-04-8
ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of …
Formula:
C23H27Cl3N2O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
501.83
Ref: TM-T22850
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 606.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
GSK1521498
CAS:1426543-84-1
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H23F2N4O4P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.43
Ref: TM-T11479
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
Bevenopran
CAS:676500-67-7
Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies …
Formula:
C20H26N4O4
Purity:
98.14% - 98.76%
Color and Shape:
Solid
Molecular weight:
386.44
Ref: TM-T14551
| 1mg | 95.00 € | ||
| 5mg | 217.00 € | ||
| 10mg | 323.00 € | ||
| 25mg | 518.00 € | ||
| 50mg | 705.00 € | ||
| 100mg | 920.00 € | ||
| 500mg | 1,845.00 € | ||
| 1mL*10mM (DMSO) | 242.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
JNJ-20788560
CAS:825649-28-3
JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective …
Formula:
C25H28N2O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
388.5
Ref: TM-T27667
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,549.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
ML-335
CAS:1069498-96-9
ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief …
Formula:
C25H32N2O3
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
408.53
Ref: TM-T23002
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 621.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
AT-121
CAS:2099681-31-7
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, …
Formula:
C24H38N4O3S
Purity:
97% - 97.95%
Color and Shape:
Solid
Molecular weight:
462.65
Ref: TM-T37610
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Monday 3 Feb 2025
MOR agonist-1
CAS:2305781-14-8
MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and …
Formula:
C22H26ClFN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
404.91
Ref: TM-T79060
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
μ opioid receptor agonist 3
CAS:2378397-91-0
Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that …
Formula:
C22H28N2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
352.47
Ref: TM-T79430
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Icalcaprant
CAS:2227384-17-8
Icalcaprant is a kappa-opioid receptor antagonist [1].
Formula:
C23H26N4O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
406.48
Ref: TM-T79848
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
DPI-3290
CAS:182417-73-8
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 …
Formula:
C30H34FN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
487.61
Ref: TM-T15165
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Mu opioid receptor antagonist 7
CAS:2378397-30-7
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid …
Formula:
C22H27ClN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
386.91
Ref: TM-T79431
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Nalmefene
CAS:55096-26-9
Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study …
Formula:
C21H25NO3
Color and Shape:
Liquid
Molecular weight:
339.43
Ref: TM-T86954
| 5mg | 61.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 179.00 € |
Estimated delivery in United States, on Monday 17 Mar 2025
Norbinaltorphimine dihydrochloride
CAS:113158-34-2
Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses …
Formula:
C40H45Cl2N3O6
Purity:
99%
Color and Shape:
Solid
Molecular weight:
734.71
Ref: TM-T12241
| 1mg | 40.00 € | ||
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 17 Mar 2025
Naloxone hydrochloride
CAS:357-08-4
Naloxone hydrochloride (Naloxone HCl) is a specific opiate antagonist that has no agonist activity. It …
Formula:
C19H21NO4·HCl
Purity:
97.91%
Color and Shape:
White To Off-White/Powder
Molecular weight:
363.84
Ref: TM-T0102
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 200mg | Discontinued | Request information |
Nalfurafine
CAS:152657-84-6
Nalfurafine (TRK-820) is an effective and selective agonist of G protein-biased κ-opioid receptor with high …
Formula:
C28H32N2O5
Purity:
99.18%
Color and Shape:
Solid
Molecular weight:
476.56
Ref: TM-T41284
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 100mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
Nalfurafine hydrochloride
CAS:152658-17-8
Nalfurafine hydrochloride (TRK-820 hydrochloride) is an opioid κ-selective agonist; has been approved in Japan for …
Formula:
C28H33ClN2O5
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
513.03
Ref: TM-T2388
| 1mg | Discontinued | Request information | |
| 2mg | Discontinued | Request information | |
| 5mg | Discontinued | Request information | |
| 10mg | Discontinued | Request information | |
| 25mg | Discontinued | Request information | |
| 50mg | Discontinued | Request information | |
| 1ml*10 (DMSO) | Discontinued | Request information |
