Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
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SNC 80
CAS:156727-74-1
SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 …
Formula:
C28H39N3O2
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
449.63
Ref: TM-T8414
| 1mg | 41.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 389.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
BPR1M97
CAS:2059904-66-2
BPR1M97 is a mu opioid receptor (MOP) and neuropeptide-orphin FQ (NOP) receptor agonist with blood-brain …
Formula:
C18H18Cl2N2O
Purity:
98.13% - 99.15%
Color and Shape:
Solid
Molecular weight:
349.25
Ref: TM-T10593
| 1mg | 94.00 € | ||
| 5mg | 223.00 € | ||
| 10mg | 352.00 € | ||
| 25mg | 647.00 € | ||
| 50mg | 1,014.00 € | ||
| 100mg | 1,423.00 € | ||
| 500mg | 2,762.00 € | ||
| 1mL*10mM (DMSO) | 215.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Dermorphin
CAS:77614-16-5
Dermorphin is agonist of μ-opioid receptor (MOR) agonist.
Formula:
C40H50N8O10
Purity:
98.82%
Color and Shape:
Solid
Molecular weight:
802.87
Ref: TM-T7404
| 1mg | 44.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
LY255582
CAS:119193-09-8
LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta …
Formula:
C22H35NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.52
Ref: TM-T27934
| 5mg | 463.00 € | ||
| 50mg | 1,840.00 € | ||
| 100mg | 3,586.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Propiram fumarate HCl
CAS:945013-73-0
Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study …
Formula:
C16H25N3O·xClH
Purity:
99.25%
Color and Shape:
Soild
Ref: TM-T28453L
| 1mg | 183.00 € | ||
| 5mg | 401.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,271.00 € | ||
| 100mg | 1,710.00 € | ||
| 500mg | 3,416.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
DuP 747 HCl
CAS:115904-74-0
DuP 747 HCl is a selective kappa agonist with analgesic activity.DuP 747 consists of two …
Formula:
C24H29Cl3N2O2
Purity:
99.81%
Color and Shape:
Soild
Molecular weight:
483.86
Ref: TM-T25354L
| 1mg | 241.00 € | ||
| 5mg | 600.00 € | ||
| 10mg | 853.00 € | ||
| 25mg | 1,279.00 € | ||
| 50mg | 1,727.00 € | ||
| 100mg | 2,334.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
MOR agonist-2
Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist …
Formula:
C37H47Cl2N5O3
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
680.71
Ref: TM-T79547
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Apitegromab
CAS:2278276-46-1
Apitegromab (SRK-015) is a new myostatin inhibitor, an antibody targeting myostatin precursor, which can be …
Purity:
95%
Color and Shape:
Liquid
Ref: TM-T77445
| 1mg | 207.00 € | ||
| 5mg | 608.00 € | ||
| 10mg | 917.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
![[DPro10] Dynorphin A (1-11)acetate,porcine](https://static.cymitquimica.com/products/TM/thumb/T76341L.jpg)
[DPro10] Dynorphin A (1-11)acetate,porcine
[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value …
Formula:
C65H107N21O15
Purity:
99.05%
Color and Shape:
Soild
Molecular weight:
1422.7
Ref: TM-T76341L
| 1mg | 60.00 € | ||
| 5mg | 124.00 € | ||
| 10mg | 176.00 € | ||
| 25mg | 296.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 646.00 € | ||
| 500mg | 1,364.00 € |
Estimated delivery in United States, on Tuesday 18 Feb 2025
Adrenorphin
CAS:88377-68-8
Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C44H69N15O9S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
984.18
Ref: TM-T7567
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 18 Feb 2025
![[Leu5]-Enkephalin](https://static.cymitquimica.com/products/TM/thumb/T7173.jpg)
[Leu5]-Enkephalin
CAS:58822-25-6
[Leu5]-Enkephalin (Leu-enkephalin) is an endogenous neuropeptide involved in nociception and an agonist of δ-opioid and …
Formula:
C28H37N5O7
Purity:
99.87%
Color and Shape:
Solid
Molecular weight:
555.62
Ref: TM-T7173
| 10mg | 47.00 € | ||
| 25mg | 83.00 € | ||
| 50mg | 112.00 € | ||
| 100mg | 157.00 € |
Estimated delivery in United States, on Thursday 20 Feb 2025
Asimadoline
CAS:153205-46-0
Asimadoline (EMD-61753) is a proprietary small molecule therapeutic, originally discovered by Merck KGaA of Darmstadt, …
Formula:
C27H30N2O2
Color and Shape:
Solid
Molecular weight:
414.54
Ref: TM-T4633
| 5mg | 73.00 € | ||
| 25mg | 278.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Thursday 20 Feb 2025
BAN ORL 24 dihydrochloride
CAS:1401463-54-4
BAN ORL 24 dihydrochloride is a highly potent nociceptin/orphan FQ (N/OFQ) receptor (NOP) antagonist that …
Formula:
C27H37Cl2N3O2
Purity:
95.03%
Color and Shape:
Solid
Molecular weight:
506.51
Ref: TM-T10457
| 2mg | 78.00 € |
Estimated delivery in United States, on Thursday 20 Feb 2025
(R,S)-Ivosidenib
CAS:2070009-31-1
(R,S)-Ivosidenib is the less active enantiomer of Ivosidenib .
Formula:
C28H22ClF3N6O3
Color and Shape:
Solid
Molecular weight:
582.96
Ref: TM-T13438
| 2mg | 392.00 € |
Estimated delivery in United States, on Thursday 20 Feb 2025
Deltorphin 2
CAS:122752-16-3
Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of …
Formula:
C38H54N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
782.88
Ref: TM-T7639
| 1mg | 62.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 307.00 € | ||
| 25mg | 521.00 € | ||
| 50mg | 749.00 € | ||
| 100mg | 1,023.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Methylnaltrexone bromide
CAS:73232-52-7
Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to …
Formula:
C21H26BrNO4
Purity:
99.02%
Color and Shape:
Solid
Molecular weight:
436.35
Ref: TM-T21422
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 266.00 € | ||
| 100mg | 462.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Corydaline
CAS:518-69-4
Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits …
Formula:
C22H27NO4
Purity:
98.01% - 99.86%
Color and Shape:
Solid
Molecular weight:
369.45
Ref: TM-T5S2360
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 303.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Nociceptin
CAS:170713-75-4
Nociceptin (Orphanin FQ) is a 17-amino-acid polypeptide that is structurally related to the opioid peptide …
Formula:
C79H129N27O22
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
1809.04
Ref: TM-TP1071
| 1mg | 80.00 € | ||
| 5mg | 222.00 € | ||
| 10mg | 360.00 € | ||
| 25mg | 603.00 € | ||
| 50mg | 861.00 € | ||
| 100mg | 1,170.00 € | ||
| 500mg | 2,341.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
N-Desmethylclozapine
CAS:6104-71-8
N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.
Formula:
C17H17ClN4
Purity:
97.25%
Color and Shape:
Yellow Crystalline Solid
Molecular weight:
312.8
Ref: TM-T5158
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 155.00 € | ||
| 50mg | 238.00 € | ||
| 100mg | 351.00 € | ||
| 200mg | 499.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
Sec-O-Glucosylhamaudol
CAS:80681-44-3
Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.
Formula:
C21H26O10
Purity:
99.35%
Color and Shape:
Solid
Molecular weight:
438.43
Ref: TM-T5S0581
| 20mg | 86.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 24 Feb 2025
