Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
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AR-M 1000390 hydrochloride
CAS:209808-47-9
ARM-390 HCl is a δ-opioid receptor agonist, brain-penetrant, nonpeptidic, prevents hyperalgesia without desensitization. Derived from …
Formula:
C23H29ClN2O
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
384.94
Ref: TM-T4236
| 5mg | 69.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 368.00 € | ||
| 100mg | 553.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Bisacodyl
CAS:603-50-9
Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for …
Formula:
C22H19NO4
Purity:
97.13% - 99.78%
Color and Shape:
Smaller Than 50 Microns Predominate White To Off-White Crystalline Powder
Molecular weight:
361.39
Ref: TM-T6414
| 500mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BRL 52537 hydrochloride
CAS:112282-24-3
BRL 52537 hydrochloride: selective KOR agonist, may protect against ischemic brain injury, used in stroke …
Formula:
C18H25Cl3N2O
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
391.76
Ref: TM-T21757
| 1mg | 41.00 € | ||
| 2mg | 53.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 215.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 490.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Aticaprant
CAS:1174130-61-0
Aticaprant (CERC-501) is a potent and centrally-penetrant antagonist of the kappa-opioid receptor (Ki: 0.807 nM).Cost-effective …
Formula:
C26H27FN2O2
Purity:
99.53% - 99.93%
Color and Shape:
Solid
Molecular weight:
418.5
Ref: TM-TQ0082
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 254.00 € | ||
| 50mg | 398.00 € | ||
| 100mg | 593.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Deltorphin 2
CAS:122752-16-3
Deltorphin 2 ([D-Ala2]-Deltorphin II) is an agonist of δ opioid receptor with an IC50 of …
Formula:
C38H54N8O10
Purity:
100%
Color and Shape:
Solid
Molecular weight:
782.88
Ref: TM-T7639
| 1mg | 62.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 307.00 € | ||
| 25mg | 521.00 € | ||
| 50mg | 749.00 € | ||
| 100mg | 1,023.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BMS986188
CAS:1776115-10-6
BMS986188 is a novel Potent and Selective Positive Allosteric Modulator of the delta-Opioid Receptor.
Formula:
C30H31BrO4
Purity:
98.76%
Color and Shape:
Solid
Molecular weight:
535.47
Ref: TM-T8992
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 133.00 € | ||
| 50mg | 191.00 € | ||
| 100mg | 284.00 € | ||
| 200mg | 397.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BW-180C
CAS:63631-40-3
BW-180C (DADLE) is a prototypical δ-opioid receptor agonist that also displays activity at the μ-opioid …
Formula:
C29H39N5O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-TP1905
| 1mg | 46.00 € | ||
| 2mg | 61.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | 249.00 € | ||
| 50mg | 392.00 € | ||
| 100mg | 582.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
DAMGO TFA (78123-71-4(Free base))
DAMGO TFA (78123-71-4(Free base)) is a potent and selective agonist of the Mu-opioid receptor.Cost-effective and …
Formula:
C28H36F3N5O8
Purity:
98.67% - 99.76%
Color and Shape:
Solid
Molecular weight:
627.6
Ref: TM-T4411
| 1mg | 63.00 € | ||
| 2mg | 96.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 282.00 € | ||
| 25mg | 536.00 € | ||
| 50mg | 733.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Asimadoline hydrochloride
CAS:185951-07-9
Asimadoline HCl (EMD-61753) is a kappa-opioid receptor agonist for pruritus and IBS treatment.
Formula:
C27H31ClN2O2
Purity:
98.63% - 98.94%
Color and Shape:
Solid
Molecular weight:
451.01
Ref: TM-T4691
| 1mg | 35.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 222.00 € | ||
| 50mg | 330.00 € | ||
| 100mg | 488.00 € | ||
| 500mg | 1,048.00 € | ||
| 1mL*10mM (DMSO) | 81.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Endomorphin 1
CAS:189388-22-5
Endomorphin 1 is a high affinity and selective agonist of the μ-opioid receptor and displays …
Formula:
C34H38N6O5
Purity:
95.92%
Color and Shape:
Solid (Solid Powder )
Molecular weight:
610.7
Ref: TM-TQ0267
| 5mg | 49.00 € | ||
| 10mg | 68.00 € | ||
| 25mg | 94.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
CP-866087
CAS:519052-04-1
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female …
Formula:
C24H28N2O2
Purity:
100% - 99.44%
Color and Shape:
Soild
Molecular weight:
376.49
Ref: TM-T31081
| 1mg | 707.00 € | ||
| 5mg | 1,486.00 € | ||
| 25mg | 1,976.00 € | ||
| 50mg | 2,412.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
ML-335
CAS:1069498-96-9
ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief …
Formula:
C25H32N2O3
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
408.53
Ref: TM-T23002
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 621.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
LY2444296
CAS:1346133-11-6
LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 …
Formula:
C24H22F2N2O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
408.44
Ref: TM-T11909
| 5mg | 46.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 22 Jan 2025
IPAG
CAS:193527-91-2
IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.
Formula:
C17H22IN3
Purity:
98.8%
Color and Shape:
Solid
Molecular weight:
395.28
Ref: TM-T22870
| 1mg | 45.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 261.00 € | ||
| 50mg | 449.00 € | ||
| 100mg | 647.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
ADL-5747
CAS:850176-30-6
ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the …
Formula:
C24H28N2O3
Purity:
100% - 99.44%
Color and Shape:
Solid
Molecular weight:
392.49
Ref: TM-T29663
| 1mg | 138.00 € | ||
| 5mg | 335.00 € | ||
| 10mg | 495.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,971.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
GSK1521498 free base (hydrochloride)
CAS:1007578-24-6
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H21ClF2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.9
Ref: TM-T11478
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
ICI 199,441 hydrochloride
CAS:115199-84-3
ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.
Formula:
C21H25Cl3N2O
Purity:
99.46%
Color and Shape:
Solid
Molecular weight:
427.8
Ref: TM-T22849
| 2mg | 34.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 141.00 € | ||
| 50mg | 218.00 € | ||
| 100mg | 320.00 € | ||
| 200mg | 449.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
SCH 221510
CAS:322473-89-2
SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.
Formula:
C28H31NO
Purity:
99.10%
Color and Shape:
Solid
Molecular weight:
397.55
Ref: TM-T23335
| 1mg | 77.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 260.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 834.00 € | ||
| 100mg | 1,355.00 € | ||
| 200mg | 1,822.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
GSK1521498
CAS:1426543-84-1
GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H23F2N4O4P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
500.43
Ref: TM-T11479
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Trimebutine CTB salt
CAS:1456509-46-8
Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.
Formula:
C29H36N2O8S2
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
604.74
Ref: TM-T27413
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,499.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
