Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
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PZM21
CAS:1997387-43-5
PZM21 is an effective and selective μ opioid receptor agonist (EC50: 1.8 nM).
Formula:
C19H27N3O2S
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
361.5
Ref: TM-T4386
| 1mg | 47.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 127.00 € | ||
| 25mg | 205.00 € | ||
| 50mg | 298.00 € | ||
| 100mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 97.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
BMS986187
CAS:684238-37-7
BMS986187 is a novel Potent and Selective Positive Allosteric Modulators of the delta-Opioid Receptor.
Formula:
C31H34O4
Purity:
99.09%
Color and Shape:
Solid
Molecular weight:
470.6
Ref: TM-T8991
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 84.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 227.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 512.00 € | ||
| 500mg | 1,093.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
GR103545
CAS:126766-43-6
GR103545 is a selective agonist of the κ-opioid receptor, which is a radiotracer that can …
Formula:
C23H29Cl2N3O7
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
530.4
Ref: TM-T9459
| 1mg | 87.00 € | ||
| 2mg | 143.00 € | ||
| 5mg | 188.00 € | ||
| 10mg | 283.00 € | ||
| 25mg | 509.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,017.00 € | ||
| 1mL*10mM (DMSO) | 250.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
LY2795050
CAS:1346133-08-1
LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).
Formula:
C23H22ClN3O2
Purity:
97.77%
Color and Shape:
Solid
Molecular weight:
407.89
Ref: TM-TQ0091
| 1mg | 52.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 116.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 298.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 127.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
DAMGO
CAS:78123-71-4
DAMGO (DAGO) is an opioid receptor agonist with the ability to affect the locomotive activity …
Formula:
C26H35N5O6
Purity:
98.83% - 99.92%
Color and Shape:
Solid
Molecular weight:
513.59
Ref: TM-T4351
| 1mg | 50.00 € | ||
| 2mg | 60.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 140.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 423.00 € | ||
| 100mg | 623.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Spinorphin
CAS:137201-62-8
Spinorphin is a heptapeptide, and is a potent enkephalin-degrading enzymes inhibitor.
Formula:
C45H64N8O10
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
877
Ref: TM-T8455
| 1mg | 130.00 € | ||
| 5mg | 245.00 € | ||
| 10mg | 378.00 € | ||
| 25mg | 630.00 € | ||
| 50mg | 898.00 € | ||
| 100mg | 1,216.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Adrenorphin 3TFA(88377-68-8(free base))
Adrenorphin 3TFA(88377-68-8(free base)) (Metorphamide) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C50H72N15O15S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
1326.26
Ref: TM-T7567L
| 1mg | 48.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 180.00 € | ||
| 25mg | 325.00 € | ||
| 50mg | 467.00 € | ||
| 100mg | 645.00 € | ||
| 200mg | 868.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
![[D-Ala2]leucine-enkephalin](https://static.cymitquimica.com/products/TM/thumb/TP1367.jpg)
[D-Ala2]leucine-enkephalin
CAS:64963-01-5
[D-Ala2]-Leucine enkephalin is a delta opioid agonist used to study the signaling pathway of delta …
Formula:
C29H39N5O7
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
569.65
Ref: TM-TP1367
| 2mg | 42.00 € | ||
| 5mg | 63.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 465.00 € | ||
| 200mg | 650.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
N-Desmethylclozapine
CAS:6104-71-8
N-Desmethylclozapine: 5-HT2C antagonist (IC50: 7.1 nM), dopamine D4 antagonist, δ-opioid agonist.
Formula:
C17H17ClN4
Purity:
97.25%
Color and Shape:
Yellow Crystalline Solid
Molecular weight:
312.8
Ref: TM-T5158
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 160.00 € | ||
| 50mg | 248.00 € | ||
| 100mg | 364.00 € | ||
| 200mg | 517.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
Sec-O-Glucosylhamaudol
CAS:80681-44-3
Sec-O-Glucosylhamaudol has anti-inflammatory and strong antinociceptive properties, acting on p38 MAPK and opioid receptors.
Formula:
C21H26O10
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
438.43
Ref: TM-T5S0581
| 20mg | 88.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
GSK1521498 free base
CAS:1007573-18-3
GSK1521498 free base is a potent and selective antagonist of the μ-opioid receptor.
Formula:
C24H20F2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
402.44
Ref: TM-T11478L
| 25mg | 1,206.00 € | ||
| 50mg | 1,568.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
ORL1 antagonist 1
CAS:1174985-59-1
ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 …
Formula:
C20H22ClN5
Purity:
97.87%
Color and Shape:
Solid
Molecular weight:
367.88
Ref: TM-T12320
| 1mg | 77.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 225.00 € | ||
| 25mg | 338.00 € | ||
| 50mg | 475.00 € | ||
| 100mg | 638.00 € | ||
| 200mg | 845.00 € | ||
| 1mL*10mM (DMSO) | 163.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
Opioid receptor modulator 1
CAS:77514-44-4
Opioid receptor modulator 1 is a modulator of opioid receptor.
Formula:
C18H23NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T12314
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
CP-866087
CAS:519052-04-1
CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female …
Formula:
C24H28N2O2
Purity:
100% - 99.44%
Color and Shape:
Soild
Molecular weight:
376.49
Ref: TM-T31081
| 1mg | 723.00 € | ||
| 5mg | 1,510.00 € | ||
| 25mg | 2,023.00 € | ||
| 50mg | 2,452.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
GR 89696 fumarate
CAS:126766-32-3
GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with …
Formula:
C23H29Cl2N3O7
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
530.4
Ref: TM-T22810
| 5mg | 64.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 162.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 334.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
NNC 63-0532
CAS:250685-44-0
NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.
Formula:
C27H29N3O3
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
443.54
Ref: TM-T23074
| 1mg | 49.00 € | ||
| 2mg | 64.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 283.00 € | ||
| 50mg | 447.00 € | ||
| 100mg | 638.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
SCH 221510
CAS:322473-89-2
SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.
Formula:
C28H31NO
Purity:
99.10%
Color and Shape:
Solid
Molecular weight:
397.55
Ref: TM-T23335
| 1mg | 78.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 264.00 € | ||
| 25mg | 533.00 € | ||
| 50mg | 847.00 € | ||
| 100mg | 1,378.00 € | ||
| 200mg | 1,853.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
GSK1521498 free base (hydrochloride)
CAS:1007578-24-6
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H21ClF2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.9
Ref: TM-T11478
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
SCH-486757
CAS:524019-25-8
SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used …
Formula:
C24H23Cl2N3O
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
440.37
Ref: TM-T28728
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
Trimebutine CTB salt
CAS:1456509-46-8
Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.
Formula:
C29H36N2O8S2
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
604.74
Ref: TM-T27413
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,537.00 € |
Estimated delivery in United States, on Monday 2 Jun 2025
