PKA
Protein kinase A (PKA) is a key enzyme in the GPCR signaling cascade, activated by cyclic AMP (cAMP) in response to various extracellular signals. PKA regulates a wide range of cellular processes, including metabolism, gene expression, and cell growth. Dysregulation of PKA activity is associated with various diseases, including cancer, metabolic disorders, and cardiovascular conditions. PKA modulators are valuable tools in research aimed at understanding GPCR signaling pathways and developing new therapeutic strategies. At CymitQuimica, we provide a selection of high-quality PKA modulators to support your research in signal transduction, cellular regulation, and disease mechanisms.
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CCG215022
CAS:1813527-81-9
CCG215022 is a G protein-coupled receptor kinases (GRKs) inhibitor with IC50s of 0.15±0.07 μM, 0.38±0.06 …
Formula:
C26H22FN7O3
Purity:
97.63% - 99.69%
Color and Shape:
Solid
Molecular weight:
499.5
Ref: TM-T3498
| 1mg | 96.00 € | ||
| 2mg | 140.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 378.00 € | ||
| 25mg | 630.00 € | ||
| 50mg | 898.00 € | ||
| 100mg | 1,216.00 € | ||
| 500mg | 2,442.00 € | ||
| 1mL*10mM (DMSO) | 259.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
AT7867
CAS:857531-00-1
AT7867 inhibits Akt1/2/3 & p70S6K/PKA (IC50: 32/17/47 nM & 85/20 nM), minimal effect beyond AGC …
Formula:
C20H20ClN3
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
337.85
Ref: TM-T6304
| 2mg | 44.00 € | ||
| 5mg | 65.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 210.00 € | ||
| 100mg | 313.00 € | ||
| 200mg | 452.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
Daphnetin
CAS:486-35-1
Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR …
Formula:
C9H6O4
Purity:
97.47% - 99.8%
Color and Shape:
Solid
Molecular weight:
178.14
Ref: TM-T2851
| 10mg | 50.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 166.00 € | ||
| 100mg | 244.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
Bilobetin
CAS:521-32-4
Bilobetin ameliorates insulin resistance by PKA-mediated phosphorylation of PPARα in rats fed a high-fat diet.
Formula:
C31H20O10
Purity:
97.74% - 99.73%
Color and Shape:
Solid
Molecular weight:
552.48
Ref: TM-T4S2128
| 1mg | 47.00 € | ||
| 2mg | 70.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 613.00 € | ||
| 100mg | 843.00 € | ||
| 1mL*10mM (DMSO) | 187.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
HA-100
CAS:84468-24-6
HA-100 is an inhibitor of protein kinase
Formula:
C13H15N3O2S
Purity:
99.44%
Color and Shape:
Pale Yellow Crystalline Solid
Molecular weight:
277.34
Ref: TM-T7648
| 5mg | 63.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 369.00 € | ||
| 100mg | 540.00 € | ||
| 1mL*10mM (DMSO) | 69.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
PKG drug G1
CAS:374703-78-3
PKG drug G1 targets PKG Iα C42. PKG drug G1 can couple to vasodilation and …
Formula:
C13H11N3OS
Purity:
97.57% - 97.67%
Color and Shape:
Solid
Molecular weight:
257.31
Ref: TM-T4661
| 2mg | 39.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 227.00 € | ||
| 100mg | 344.00 € | ||
| 500mg | 812.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
H-89 dihydrochloride
CAS:130964-39-5
H-89 dihydrochloride (5-Isoquinolinesulfonamide) is a potent inhibitor of protein kinase A (PKA; IC50: 0.14 μM, …
Formula:
C20H20BrN3O2S·2HCl
Purity:
100% - 99.4%
Color and Shape:
Solid
Molecular weight:
519.28
Ref: TM-T6250
| 5mg | 39.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 106.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 344.00 € | ||
| 200mg | 512.00 € | ||
| 500mg | 815.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
Metadoxine
CAS:74536-44-0
Metadoxine (Metadoxil) is a neurotransmitter stimulant.
Formula:
C8H11NO3·C5H7NO3
Purity:
99.19%
Color and Shape:
Off-White Powder
Molecular weight:
298.29
Ref: TM-T3269
| 1g | 114.00 € | ||
| 100mg | 39.00 € | ||
| 200mg | 52.00 € | ||
| 500mg | 86.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 28 Apr 2025
Rp-cAMPS triethylammonium salt
CAS:151837-09-1
Rp-cAMPS triethylammonium salt is a competitive inhibitor of cAMP-dependent protein kinase I and II.
Formula:
C16H27N6O5PS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
446.46
Ref: TM-T12764
| 1mg | 465.00 € | ||
| 5mg | 1,955.00 € | ||
| 500µg | 274.00 € |
Estimated delivery in United States, on Tuesday 10 Jun 2025
