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Bradykinin Receptor

Bradykinin Receptor

Bradykinin receptors are GPCRs that mediate the effects of bradykinin, a peptide involved in inflammatory responses, pain sensation, and blood pressure regulation. There are two main types of bradykinin receptors, B1 and B2, each playing distinct roles in pathophysiological processes. Bradykinin receptor antagonists are used in the treatment of conditions such as hereditary angioedema, chronic pain, and hypertension. At CymitQuimica, we offer a variety of high-quality bradykinin receptor modulators to support your research in inflammation, pain management, and cardiovascular biology.

Found 59 products of "Bradykinin Receptor"

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  • Anatibant 2HCl

    CAS:
    <p>Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.</p>
    Formula:C34H36Cl2N6O5S·2ClH
    Purity:99.17% - 99.58%
    Color and Shape:Soild
    Molecular weight:784.58
  • Bradykinin (1-7)

    CAS:
    <p>Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.</p>
    Formula:C35H52N10O9
    Purity:98%
    Color and Shape:White Lyophilized Powder
    Molecular weight:756.85
  • FR167344 free base

    CAS:
    <p>FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.</p>
    Formula:C30H28BrCl2N5O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:673.38
  • Bradykinin (1-6)

    CAS:
    <p>Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.</p>
    Formula:C30H45N9O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:659.73
  • Labradimil

    CAS:
    <p>Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.</p>
    Formula:C49H75N15O12S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1098.29
  • MEN 11270

    CAS:
    <p>B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.</p>
    Formula:C60H90N20O11S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1299.56
  • Bradykinin (1-3)

    CAS:
    <p>Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.</p>
    Formula:C16H28N6O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:368.43
  • [Des-Arg9]-Bradykinin

    CAS:
    <p>[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.</p>
    Formula:C44H61N11O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:904.02
  • Sar-[D-Phe8]-des-Arg9-Bradykinin

    CAS:
    <p>Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.</p>
    Formula:C47H66N12O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:975.11
  • Icatibant

    CAS:
    <p>Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).</p>
    Formula:C59H89N19O13S
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:1304.52
  • Lys-[Des-Arg9]Bradykinin

    CAS:
    <p>Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (&gt;30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.</p>
    Formula:C50H73N13O11
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1032.21
  • [Des-Arg10]-HOE I40 TFA


    <p>[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.</p>
    Formula:C53H77N15O12S·xC2HF3O2
    Color and Shape:Solid
  • Bombinakinin M

    CAS:
    <p>Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.</p>
    Formula:C100H159N31O24
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2179.55
  • [Phe8Ψ(CH-NH)-Arg9]-Bradykinin

    CAS:
    <p>Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.</p>
    Formula:C50H75N15O10
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1046.23
  • Fasitibant chloride

    CAS:
    <p>Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.</p>
    Formula:C36H49Cl3N6O6S
    Color and Shape:Solid
    Molecular weight:800.23
  • NPC 567

    CAS:
    <p>NPC 567 is an antagonist of the bradykinin receptor.</p>
    Formula:C60H87N19O13
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1282.48
  • Fasitibant chloride hydrochloride

    CAS:
    <p>Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.</p>
    Formula:C36H50Cl4N6O6S
    Color and Shape:Solid
    Molecular weight:836.7
  • Lys-Bradykinin

    CAS:
    <p>Endogenous bradykinin receptor agonist</p>
    Formula:C56H85N17O12
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1188.38
  • Zoliprofen

    CAS:
    <p>Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.</p>
    Formula:C12H11NO3S
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:249.29
  • Retrobradykinin

    CAS:
    <p>Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.</p>
    Formula:C50H73N15O11
    Color and Shape:Solid
    Molecular weight:1060.228