Bradykinin Receptor

Bradykinin receptors are GPCRs that mediate the effects of bradykinin, a peptide involved in inflammatory responses, pain sensation, and blood pressure regulation. There are two main types of bradykinin receptors, B1 and B2, each playing distinct roles in pathophysiological processes. Bradykinin receptor antagonists are used in the treatment of conditions such as hereditary angioedema, chronic pain, and hypertension. At CymitQuimica, we offer a variety of high-quality bradykinin receptor modulators to support your research in inflammation, pain management, and cardiovascular biology.

Found 59 products of "Bradykinin Receptor"

Purity (%)

100

products per page.

+ Info
Anatibant 2HCl
CAS:
- 209788-45-4
Anatibant 2HCl is a small molecule bradykinin B2 receptor antagonist for the treatment of neurological disorders and may be used in the study of brain injury.
Formula:C₃₄H₃₆Cl₂N₆O₅S·2ClH
Purity:99.17% - 99.58%
Color and Shape:Soild
Molecular weight:784.58
Ref: TM-T26627L
+ Info
[Des-Arg9]-Bradykinin acetate
CAS:
- 23827-91-0
[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.
Formula:C₄₆H₆₅N₁₁O₁₂
Purity:99.05%
Color and Shape:Solid
Molecular weight:964.07
Ref: TM-TP1445
+ Info
Fasitibant chloride
CAS:
- 1157852-02-2
Fasitibant chloride, a potent B2R blocker, alleviates pain and swelling in arthritis.
Formula:C₃₆H₄₉Cl₃N₆O₆S
Color and Shape:Solid
Molecular weight:800.23
Ref: TM-T38544
+ Info
Icatibant
CAS:
- 130308-48-4
Icatibant is a selective and specific antagonist of the bradykinin B2 receptor (IC50 and Ki: 1.07 nM and 0.798 nM respectively).
Formula:C₅₉H₈₉N₁₉O₁₃S
Purity:98%
Color and Shape:White Solid
Molecular weight:1304.52
Ref: TM-T15547
+ Info
[Phe8Ψ(CH-NH)-Arg9]-Bradykinin
CAS:
- 118122-39-7
Selective bradykinin B2 receptor agonist that is resistant to carboxypeptidase cleavage.
Formula:C₅₀H₇₅N₁₅O₁₀
Purity:98%
Color and Shape:Solid
Molecular weight:1046.23
Ref: TM-TP2076
+ Info
Bombinakinin M
CAS:
- 509151-65-9
Potent, selective bradykinin receptor agonist 50x stronger than bradykinin, contracts guinea pig ileum muscle at EC50 4.0 nM.
Formula:C₁₀₀H₁₅₉N₃₁O₂₄
Purity:98%
Color and Shape:Solid
Molecular weight:2179.55
Ref: TM-TP2075
+ Info
Lys-(Des-Arg9,Leu8)-Bradykinin
CAS:
- 71800-37-8
Lys-(Des-Arg9,Leu8)-Bradykinin is a selective antagonist of the bradykinin B1 receptor [1].
Formula:C₄₇H₇₅N₁₃O₁₁
Purity:98%
Color and Shape:Solid
Molecular weight:998.18
Ref: TM-T80117
+ Info
(Hyp³)-Bradykinin acetate
(Hyp³)-Bradykinin acetate is an agonist of bradykinin B2 receptor and stimulates inositol phosphate production in cultured human fibroblasts.
Formula:C₅₂H₇₇N₁₅O₁₄
Purity:99.46%
Color and Shape:Solid
Molecular weight:1136.26
Ref: TM-T36442L
+ Info
Sar-[D-Phe8]-des-Arg9-Bradykinin
CAS:
- 126959-88-4
Potent bradykinin B1 agonist, EC50 = 9.02 nM, enzyme resistant, induces hypotension and angiogenesis.
Formula:C₄₇H₆₆N₁₂O₁₁
Purity:98%
Color and Shape:Solid
Molecular weight:975.11
Ref: TM-TP1917
+ Info
[Des-Arg9]-Bradykinin
CAS:
- 15958-92-6
[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.
Formula:C₄₄H₆₁N₁₁O₁₀
Purity:98%
Color and Shape:Solid
Molecular weight:904.02
Ref: TM-T7645
+ Info
B-Raf IN 14
CAS:
- 326918-98-3
B-Raf IN 14 is a BRAF inhibitor.
Formula:C₁₅H₁₄BrN₅O₃S
Purity:98.32%
Color and Shape:Solid
Molecular weight:424.27
Ref: TM-T72070
+ Info
Labradimil
CAS:
- 159768-75-9
Labradimil, a bradykinin B2 agonist, boosts brain drug delivery and tumor survival rates.
Formula:C₄₉H₇₅N₁₅O₁₂S
Purity:98%
Color and Shape:Solid
Molecular weight:1098.29
Ref: TM-T27790
+ Info
[Des-Arg10]-HOE I40 TFA
[Des-Arg10]-HOE I40 TFA is a potent antagonist of the bradykinin B1 receptor.
Formula:C₅₃H₇₇N₁₅O₁₂S·xC₂HF₃O₂
Color and Shape:Solid
Ref: TM-T207446
+ Info
Des-Arg9-[Leu8]-Bradykinin acetate
CAS:
- 115035-45-5
Des-Arg9-[Leu8]-Bradykinin acetate is a potent antagonist of the bradykinin receptor 1 (B1R), utilized in renal fibrosis research [1].
Formula:C₄₃H₆₇N₁₁O₁₂
Purity:98%
Color and Shape:Solid
Molecular weight:930.06
Ref: TM-T80072
+ Info
Bombinakinin M acetate
Bombinakinin M acetate is a potent bradykinin receptor agonist with high selectivity for mammalian arterial smooth muscle bradykinin receptors and is
Formula:C₁₀₂H₁₆₃N₃₁O₂₆
Purity:99.80%
Color and Shape:Solid
Molecular weight:2239.58
Ref: TM-TP2075L
+ Info
NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about the treatment of allergic airway disease.
Formula:C₆₂H₉₁N₁₉O₁₅
Purity:97.72%
Color and Shape:Solid
Molecular weight:1342.5
Ref: TM-T21060L
+ Info
FR190997
CAS:
- 193344-25-1
FR190997 is an agonist of bradykinin B2 receptor.
Formula:C₃₇H₃₃Cl₂N₅O₅
Color and Shape:Solid
Molecular weight:698.59
Ref: TM-T27377
+ Info
Fasitibant chloride hydrochloride
CAS:
- 869880-33-1
Fasitibant chloride( MEN16132) is an effective and selective non-peptide antagonist of kinin B2 receptor.
Formula:C₃₆H₅₀Cl₄N₆O₆S
Color and Shape:Solid
Molecular weight:836.7
Ref: TM-T31747
+ Info
Lys-Bradykinin
CAS:
- 342-10-9
Endogenous bradykinin receptor agonist
Formula:C₅₆H₈₅N₁₇O₁₂
Purity:98%
Color and Shape:Solid
Molecular weight:1188.38
Ref: TM-TP2268
+ Info
Zoliprofen
CAS:
- 56355-17-0
Zoliprofen: potent, oral NSAID with anti-inflammatory, antipyretic, analgesic effects. Exceeds ibuprofen's efficacy in rats and rabbits.
Formula:C₁₂H₁₁NO₃S
Purity:99.62%
Color and Shape:Solid
Molecular weight:249.29
Ref: TM-T68025
+ Info
NPC 567
CAS:
- 109333-26-8
NPC 567 is an antagonist of the bradykinin receptor.
Formula:C₆₀H₈₇N₁₉O₁₃
Purity:98%
Color and Shape:Solid
Molecular weight:1282.48
Ref: TM-T21060
+ Info
L 366811
CAS:
- 127819-95-8
L 366811 is a potent oxytocin antagonist.
Formula:C₄₃H₅₆N₈O₆
Color and Shape:Solid
Molecular weight:780.95
Ref: TM-T24291
+ Info
FR167344 free base
CAS:
- 215258-13-2
FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.
Formula:C₃₀H₂₈BrCl₂N₅O₄
Purity:98%
Color and Shape:Solid
Molecular weight:673.38
Ref: TM-T15347
+ Info
Bradykinin (1-3)
CAS:
- 23815-91-0
Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Formula:C₁₆H₂₈N₆O₄
Purity:98%
Color and Shape:Solid
Molecular weight:368.43
Ref: TM-TP1780
+ Info
JMV-1645
CAS:
- 284037-77-0
JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.
Formula:C₄₉H₆₉N₁₃O₁₂S
Purity:98%
Color and Shape:Solid
Molecular weight:1064.23
Ref: TM-T25555
+ Info
Lys-[Des-Arg9]Bradykinin TFA
CAS:
- 2763588-90-3
Lys-[Des-Arg9]Bradykinin TFA: natural kinin, selective B1 agonist; Ki: 0.12 nM (human), 1.7 nM (mouse), 0.23 nM (rabbit); weak on B2 receptors.
Formula:C₅₄H₇₅F₆N₁₃O₁₅
Color and Shape:Solid
Molecular weight:1260.24
Ref: TM-T73646
+ Info
MEN 11270
CAS:
- 235082-52-7
B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.
Formula:C₆₀H₉₀N₂₀O₁₁S
Purity:98%
Color and Shape:Solid
Molecular weight:1299.56
Ref: TM-TP1999
+ Info
Methionyl-Lysyl-Bradykinin
CAS:
- 550-19-6
Methionyl-Lysyl-Bradykinin (Met-Lys-Bradykinin), a Bradykinin analogue, is a kinin [1] [2] .
Formula:C₆₁H₉₄N₁₈O₁₃S
Color and Shape:Solid
Molecular weight:1319.58
Ref: TM-T76384
+ Info
Bradykinin (1-7)
CAS:
- 23815-87-4
Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.
Formula:C₃₅H₅₂N₁₀O₉
Purity:98%
Color and Shape:White Lyophilized Powder
Molecular weight:756.85
Ref: TM-TP1210
+ Info
Bradykinin (1-6)
CAS:
- 23815-88-5
Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.
Formula:C₃₀H₄₅N₉O₈
Purity:98%
Color and Shape:Solid
Molecular weight:659.73
Ref: TM-TP1747
+ Info
Lys-[Des-Arg9]Bradykinin
CAS:
- 71800-36-7
Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.
Formula:C₅₀H₇₃N₁₃O₁₁
Purity:98%
Color and Shape:Solid
Molecular weight:1032.21
Ref: TM-TP1918
+ Info
Retrobradykinin
CAS:
- 5991-13-9
Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.
Formula:C₅₀H₇₃N₁₅O₁₁
Color and Shape:Solid
Molecular weight:1060.228
Ref: TM-T37795
+ Info
Lys-[Hyp3]-Bradykinin
CAS:
- 113662-39-8
Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.
Formula:C₅₆H₈₅N₁₇O₁₃
Color and Shape:Solid
Molecular weight:1204.38
Ref: TM-T76293
+ Info
Bradykinin (1-5)
CAS:
- 23815-89-6
Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.
Formula:C₂₇H₄₀N₈O₆
Color and Shape:Solid
Molecular weight:572.66
Ref: TM-TP1725
+ Info
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant to
Formula:C₄₉H₇₀N₁₂O₁₃
Purity:99.93%
Color and Shape:Solid
Molecular weight:1035.15
Ref: TM-TP1917L1
+ Info
Icatibant Acetate
CAS:
- 138614-30-9
Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.
Formula:C₆₁H₉₃N₁₉O₁₅S
Purity:99.68%
Color and Shape:Solid
Molecular weight:1364.57
Ref: TM-T22344
+ Info
5-Hydroxy-1-methylhydantoin
CAS:
- 84210-26-4
5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.
Formula:C₄H₆N₂O₃
Purity:99.99%
Color and Shape:Solid
Molecular weight:130.1
Ref: TM-T28222
+ Info
Bradykinin
CAS:
- 58-82-2
Bradykinin is an inflammatory mediator.
Formula:C₅₀H₇₃N₁₅O₁₁
Purity:99.68%
Color and Shape:Solid
Molecular weight:1060.21
Ref: TM-TP1277
+ Info
Emorfazone
CAS:
- 38957-41-4
Emorfazone (PH011085) has an anti-nociceptive effect.
Formula:C₁₁H₁₇N₃O₃
Purity:99.89%
Color and Shape:Solid
Molecular weight:239.27
Ref: TM-T9132
+ Info
ELN-441958
CAS:
- 913064-47-8
ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.
Formula:C₂₉H₂₉ClN₄O₂
Purity:99.88%
Color and Shape:Solid
Molecular weight:501.02
Ref: TM-T2086
+ Info
SSR240612
CAS:
- 464930-42-5
SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,
Formula:C₄₂H₅₃ClN₄O₇S
Purity:98.59% - 99.16%
Color and Shape:Solid
Molecular weight:793.41
Ref: TM-T5048
+ Info
Bradykinin (acetate)
CAS:
- 6846-03-3
Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.
Formula:C₅₂H₇₇N₁₅O₁₃
Purity:>99.99%
Color and Shape:Solid
Molecular weight:1120.26
Ref: TM-T21610
+ Info
Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2
Formula:C₅₄H₇₅F₆N₁₃O₁₅
Purity:97.35%
Color and Shape:Solid
Molecular weight:1260.24
Ref: TM-TP1918L
+ Info
[Des-Arg9]-Bradykinin TFA
CAS:
- 199433-70-0
[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.
Formula:C₄₆H₆₂F₃N₁₁O₁₂
Purity:>99.99%
Color and Shape:Solid
Molecular weight:1018.05
Ref: TM-T8809
+ Info
Bradykinin (2-9)
CAS:
- 16875-11-9
Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.
Formula:C₄₄H₆₁N₁₁O₁₀
Purity:>99.99%
Color and Shape:Solid
Molecular weight:904.02
Ref: TM-TP1181
+ Info
R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).
Formula:C₅₉H₈₂F₃N₁₃O₁₄
Purity:>99.99%
Color and Shape:Solid
Molecular weight:1254.36
Ref: TM-TP1933
+ Info
Lys-Bradykinin acetate(342-10-9 free base)
CAS:
- 84640-50-6
Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.
Formula:C₅₈H₈₉N₁₇O₁₄
Purity:99.86%
Color and Shape:Solid
Molecular weight:1248.43
Ref: TM-TP2268L
+ Info
Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and
Formula:C₅₂H₇₇N₁₃O₁₃
Purity:99.93%
Color and Shape:Solid
Molecular weight:1092.27
Ref: TM-TP1918L1
+ Info
BKM-570
CAS:
- 259885-54-6
BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.
Formula:C₃₄H₃₄Cl₂F₅N₃O₃
Purity:98%
Color and Shape:Solid
Molecular weight:698.55
Ref: TM-T26833
+ Info
Anatibant
CAS:
- 209733-45-9
Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.
Formula:C₃₄H₃₆Cl₂N₆O₅S
Purity:98%
Color and Shape:Solid
Molecular weight:711.66
Ref: TM-T26627

Bradykinin Receptor

Found 59 products of "Bradykinin Receptor"

Anatibant 2HCl

Ref: TM-T26627L

[Des-Arg9]-Bradykinin acetate

Ref: TM-TP1445

Fasitibant chloride

Ref: TM-T38544

Icatibant

Ref: TM-T15547

[Phe8Ψ(CH-NH)-Arg9]-Bradykinin

Ref: TM-TP2076

Bombinakinin M

Ref: TM-TP2075

Lys-(Des-Arg9,Leu8)-Bradykinin

Ref: TM-T80117

(Hyp³)-Bradykinin acetate

Ref: TM-T36442L

Sar-[D-Phe8]-des-Arg9-Bradykinin

Ref: TM-TP1917

[Des-Arg9]-Bradykinin

Ref: TM-T7645

B-Raf IN 14

Ref: TM-T72070

Labradimil

Ref: TM-T27790

[Des-Arg10]-HOE I40 TFA

Ref: TM-T207446

Des-Arg9-[Leu8]-Bradykinin acetate

Ref: TM-T80072

Bombinakinin M acetate

Ref: TM-TP2075L

NPC 567 acetate

Ref: TM-T21060L

FR190997

Ref: TM-T27377

Fasitibant chloride hydrochloride

Ref: TM-T31747

Lys-Bradykinin

Ref: TM-TP2268

Zoliprofen

Ref: TM-T68025

NPC 567

Ref: TM-T21060

L 366811

Ref: TM-T24291

FR167344 free base

Ref: TM-T15347

Bradykinin (1-3)

Ref: TM-TP1780

JMV-1645

Ref: TM-T25555

Lys-[Des-Arg9]Bradykinin TFA

Ref: TM-T73646

MEN 11270

Ref: TM-TP1999

Methionyl-Lysyl-Bradykinin

Ref: TM-T76384

Bradykinin (1-7)

Ref: TM-TP1210

Bradykinin (1-6)

Ref: TM-TP1747

Lys-[Des-Arg9]Bradykinin

Ref: TM-TP1918

Retrobradykinin

Ref: TM-T37795

Lys-[Hyp3]-Bradykinin

Ref: TM-T76293

Bradykinin (1-5)

Ref: TM-TP1725

Sar-[D-Phe8]-des-Arg9-Bradykinin acetate

Ref: TM-TP1917L1

Icatibant Acetate

Ref: TM-T22344

5-Hydroxy-1-methylhydantoin

Ref: TM-T28222

Bradykinin

Ref: TM-TP1277

Emorfazone

Ref: TM-T9132