Cannabinoid Receptor
Cannabinoid receptors are GPCRs that mediate the effects of endogenous cannabinoids (endocannabinoids) and phytocannabinoids, such as those found in cannabis. The two main types of cannabinoid receptors, CB1 and CB2, are involved in regulating a wide range of physiological processes, including pain perception, appetite, mood, and immune function. Cannabinoid receptor modulators have therapeutic potential in treating conditions such as chronic pain, epilepsy, and multiple sclerosis. At CymitQuimica, we offer a wide range of high-quality cannabinoid receptor modulators to support your research in neuropharmacology, pain management, and immunology.
Found 226 products for "Cannabinoid Receptor".
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AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Formula:C21H19Cl2IN4O2Purity:98.6% - >99.99%Color and Shape:SolidMolecular weight:557.21Olivetol
CAS:Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.Formula:C11H16O2Purity:99.98%Color and Shape:(Melting Point 102-106°F) (Ntp 1992)Molecular weight:180.24(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Formula:C23H20Cl2N4O2SPurity:99.75% - 99.83%Color and Shape:SolidMolecular weight:487.4RVD-Hpα acetate
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Formula:C67H109N19O19Purity:99.87%Color and Shape:SolidMolecular weight:1484.71RTICBM-189
CAS:RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Formula:C15H14Cl2N2OPurity:99.96%Color and Shape:SolidMolecular weight:309.19Ref: TM-T9466
2mg34.00€5mg52.00€1mL*10mM (DMSO)67.00€10mg84.00€25mg161.00€50mg250.00€100mg369.00€200mg522.00€Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Formula:C20H37NO2Purity:99.97%Color and Shape:SolidMolecular weight:323.51Ref: TM-T8425
1mg34.00€5mg64.00€1mL*10mM (DMSO)80.00€10mg95.00€25mg156.00€50mg225.00€100mg329.00€200mg495.00€AM1241
CAS:AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Formula:C22H22IN3O3Purity:98.93% - 99.1%Color and Shape:SolidMolecular weight:503.33Ref: TM-T6755
2mg35.00€5mg49.00€10mg84.00€1mL*10mM (DMSO)87.00€25mg168.00€50mg275.00€100mg495.00€500mg1,071.00€LY2828360
CAS:LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Formula:C22H27ClN6OPurity:99.45% - 99.51%Color and Shape:White SolidMolecular weight:426.94Ref: TM-T7316
2mg35.00€5mg49.00€1mL*10mM (DMSO)57.00€10mg80.00€25mg137.00€50mg192.00€100mg281.00€200mg419.00€Voacamine
CAS:Voacamine: an indole alkaloid, CB1 antagonist, inhibits P-gp, may affect rhythm.Formula:C43H52N4O5Purity:98.54% - 99.97%Color and Shape:White SolidMolecular weight:704.9GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFormula:C23H24Cl2N2O3Purity:99.82% - 99.93%Color and Shape:SolidMolecular weight:447.35A-836339
CAS:A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.Formula:C16H26N2O2SPurity:99.94%Color and Shape:SolidMolecular weight:310.45AM251
CAS:AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).Formula:C22H21Cl2IN4OPurity:97.43% - 99.24%Color and Shape:A Crystalline SolidMolecular weight:555.24CID 16020046
CAS:CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.Formula:C25H19N3O4Purity:99.03%Color and Shape:SolidMolecular weight:425.44CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Formula:C33H31Cl2F3N6O3S2Purity:99.08% - 99.76%Color and Shape:SolidMolecular weight:751.67Ref: TM-T5996
1mg82.00€2mg110.00€5mg180.00€1mL*10mM (DMSO)215.00€10mg258.00€25mg423.00€50mg588.00€100mg793.00€500mg1,594.00€GW842166X
CAS:GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Formula:C18H17Cl2F3N4O2Purity:99.89%Color and Shape:SolidMolecular weight:449.25Org 27569
CAS:Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity andFormula:C24H28ClN3OPurity:99.91% - ≥95%Color and Shape:White SolidMolecular weight:409.95WIN 55,212-2 Mesylate
CAS:WIN 55,212-2 Mesylate ((R)-(+)-WIN 55212) is a potent aminoalkylindole cannabinoid (CB) receptor agonist with Kis of 62.3 and 3.3 nM for human recombinant CB1 and CB2 receptors, respectively. Cannabinoid analogue WIN 55,212-2 Mesylate exhibited a novel anticancer effect against human tumors.Formula:C28H30N2O6SPurity:98% - 99.71%Color and Shape:SolidMolecular weight:522.61ML-184
CAS:ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.Formula:C25H34N4O3SPurity:99.45% - 99.45%Color and Shape:SolidMolecular weight:470.63BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Formula:C23H23ClN2O4Purity:97.70%Color and Shape:SolidMolecular weight:426.89β-Caryophyllene
CAS:β-Caryophyllene ((-)-(E)-Caryophyllene) acts as an CB2 receptor agonist.Formula:C15H24Purity:95.43% - 99.67%Color and Shape:Transparent LiquidMolecular weight:204.35
