PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
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PI3K/mTOR Inhibitor-2
CAS:1848242-58-9
Potent PI3K/mTOR Inhibitor-2 targets PI3Kα/β/δ/γ & mTOR (IC50: 3.4, 34, 16,1, 4.7 nM); exhibits antitumor …
Formula:
C20H13ClF2N4O4S
Purity:
96.16%
Color and Shape:
Solid
Molecular weight:
478.86
Ref: TM-T12459
| 1mg | 56.00 € | ||
| 5mg | 141.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 520.00 € | ||
| 100mg | 703.00 € | ||
| 200mg | 903.00 € | ||
| 1mL*10mM (DMSO) | 147.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
IHMT-PI3Kδ-372
CAS:2429889-62-1
IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can …
Formula:
C26H23F2N7O2
Purity:
99.54%
Color and Shape:
Liquid
Molecular weight:
503.5
Ref: TM-T35530
| 1mg | 50.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 274.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 551.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Vps34-IN-2
CAS:1523404-29-6
Vps34-IN-2 is a potent and selective Vps34 inhibitor (IC50s: 2 and 82 nM on the …
Formula:
C18H25F3N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
402.41
Ref: TM-T13311
| 25mg | 1,549.00 € | ||
| 50mg | 2,031.00 € | ||
| 100mg | 2,609.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Dactolisib Tosylate
CAS:1028385-32-1
Dactolisib Tosylate (BEZ235 Tosylate) is a dual kinase inhibitor that targets PI3K and mTOR.
Formula:
C37H31N5O4S
Purity:
99.85%
Color and Shape:
Solid
Molecular weight:
641.74
Ref: TM-T14552
| 25mg | 49.00 € | ||
| 50mg | 64.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
TGX-115
CAS:351071-62-0
TGX-115 inhibits PI 3-K p110β (IC50=0.13μM) & p110δ (IC50=0.63μM), treats various cardiovascular diseases.
Formula:
C20H20N2O3
Purity:
99.2%
Color and Shape:
Solid
Molecular weight:
336.38
Ref: TM-T24873
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,846.00 € | ||
| 100mg | 2,331.00 € | ||
| 500mg | 4,547.00 € | ||
| 1mL*10mM (DMSO) | 645.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PI3K-IN-10
CAS:2211922-64-2
PI3K-IN-10 is a potent inhibitor of pan-PI3K .
Formula:
C23H19ClN6O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
430.89
Ref: TM-T12456
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 27 Jan 2025
PI3Kγ inhibitor 1
CAS:1172118-03-4
PI3Kγ inhibitor 1 is a inhibitor of PI3Kδ and PI3Kγ.
Formula:
C32H26N8O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
586.67
Ref: TM-T12464
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PI3K/HDAC-IN-1
CAS:2361418-52-0
PI3K/HDAC-IN-1 is a potent PI3K and HDAC dual inhibitor(IC50s of 8.1 nM and 1.4 nM, …
Formula:
C22H25FN4O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
428.46
Ref: TM-T12455
| 25mg | 1,545.00 € | ||
| 50mg | 2,033.00 € | ||
| 100mg | 2,611.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PI3K-IN-38
CAS:1382979-64-7
PI3K-IN-38: oral PI3K inhibitor, IC50 of 0.541 µM, anticancer, anti-inflammatory, halts tumors in vivo.
Formula:
C20H24N6O2
Purity:
99.74%
Color and Shape:
Liquid
Molecular weight:
380.44
Ref: TM-T61618
| 1mg | 181.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,262.00 € | ||
| 100mg | 1,698.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
NVP-BAG956
CAS:853910-02-8
NVP-BAG956 is an ATP-competitive PI3K inhibitor (IC50s: 34/56/112/444 nM for PI3Kδ/PI3Kα/PI3Kγ/PI3Kβ).
Formula:
C28H21N5
Purity:
99.71% - 99.80%
Color and Shape:
Solid
Molecular weight:
427.5
Ref: TM-TQ0313
| 50mg | 700.00 € | ||
| 100mg | 1,273.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PI3Kα/mTOR-IN-1
CAS:1013098-90-2
PI3Kα/mTOR-IN-1 is a potent dual inhibitor of PI3Kα/mTOR.
Formula:
C16H18N6O
Purity:
99.3%
Color and Shape:
Solid
Molecular weight:
310.35
Ref: TM-T12589
| 1mg | 609.00 € | ||
| 5mg | 1,203.00 € | ||
| 10mg | 1,616.00 € | ||
| 25mg | 2,413.00 € | ||
| 50mg | 3,229.00 € | ||
| 100mg | 4,409.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PI3K-IN-6
CAS:1842380-77-1
PI3K-IN-6 is an oral active and highly selective inhibitor of phosphoinositide 3-kinase (PI3K) β/δ(IC50 values …
Formula:
C17H14Cl2FN9O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
450.26
Ref: TM-T12457
| 25mg | 1,406.00 € | ||
| 50mg | 1,847.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CHMFL-PI3KD-317
CAS:2244992-76-3
CHMFL-PI3KD-317: potent PI3Kδ inhibitor, IC50=6 nM, orally active, >10x selective vs. PI3K isoforms, anti-cancer.
Formula:
C21H24ClN5O3S2
Purity:
97.8%
Color and Shape:
Solid
Molecular weight:
494.03
Ref: TM-T10804
| 1mg | 91.00 € | ||
| 5mg | 214.00 € | ||
| 10mg | 326.00 € | ||
| 25mg | 587.00 € | ||
| 50mg | 881.00 € | ||
| 100mg | 1,201.00 € | ||
| 1mL*10mM (DMSO) | 233.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
GS-9901
CAS:1640247-87-5
GS-9901 is a selective, orally active and potent PI3Kδ inhibitor (IC50: 1 nM) for the …
Formula:
C22H17ClFN9O
Purity:
99.12% - 99.14%
Color and Shape:
Solid
Molecular weight:
477.88
Ref: TM-T15420
| 1mg | 90.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 322.00 € | ||
| 25mg | 691.00 € | ||
| 50mg | 915.00 € | ||
| 100mg | 1,270.00 € | ||
| 500mg | 2,559.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ON 146040
CAS:1404231-34-0
ON 146040 is an effective inhibitor of PI3K isoforms with IC50s of 14 and 20 …
Formula:
C24H23N7O3S
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
489.55
Ref: TM-T12310
| 1mg | 61.00 € | ||
| 5mg | 140.00 € | ||
| 10mg | 217.00 € | ||
| 25mg | 354.00 € | ||
| 50mg | 498.00 € | ||
| 100mg | 666.00 € | ||
| 200mg | 899.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PQR514
CAS:1927857-55-3
PQR514: more potent pan-PI3K inhibitor than predecessor PQR309, exhibits strong anticancer activity in vitro and …
Formula:
C16H20F2N8O2
Purity:
98.76% - 99.29%
Color and Shape:
Liquid
Molecular weight:
394.38
Ref: TM-T70058
| 1mg | 315.00 € | ||
| 5mg | 746.00 € | ||
| 10mg | 1,057.00 € | ||
| 25mg | 1,576.00 € | ||
| 50mg | 2,057.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PI4KIII β inhibitor 3
CAS:1245319-54-3
PI4KIII beta inhibitor 3 is a novel and high effective inhibitor of PI4KIIIβ (IC50 of …
Formula:
C22H22N8OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
446.53
Ref: TM-T12467
| 1mg | 456.00 € | ||
| 500µg | 240.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
CAL-130 Hydrochloride
CAS:1431697-78-7
CAL-130 Hydrochloride is a PI3Kδ and PI3Kγ inhibitor (IC50s: 1.3 and 6.1 nM).
Formula:
C23H23ClN8O
Color and Shape:
Solid
Molecular weight:
462.94
Ref: TM-T10660L
| 2mg | 122.00 € | ||
| 5mg | 234.00 € | ||
| 25mg | 708.00 € | ||
| 50mg | 929.00 € | ||
| 100mg | 1,395.00 € | ||
| 1mL*10mM (DMSO) | 271.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Zandelisib
CAS:1401436-95-0
Zandelisib is an inhibitor of phosphatidylinositol 3-kinase (PI3K)(p110δ, IC50 of 3.5 nM), and with antineoplastic …
Formula:
C31H38F2N8O
Purity:
99.15%
Color and Shape:
Solid
Molecular weight:
576.68
Ref: TM-T13386
| 1mg | 94.00 € | ||
| 5mg | 174.00 € | ||
| 10mg | 290.00 € | ||
| 25mg | 470.00 € | ||
| 50mg | 634.00 € | ||
| 100mg | 872.00 € | ||
| 200mg | 1,171.00 € | ||
| 1mL*10mM (DMSO) | 217.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
PI3Kγ inhibitor 2
CAS:1315538-79-4
PI3Kγ inhibitor 2 is an orally bioavailable inhibitor of PI3Kγ(Ki of 4 nM).
Formula:
C20H18F3N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
433.38
Ref: TM-T12465
| 25mg | 1,688.00 € | ||
| 50mg | 2,226.00 € | ||
| 100mg | 2,899.00 € |
Estimated delivery in United States, on Monday 10 Feb 2025
