PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
Found 231 products of "PI3K"
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PI3K/mTOR Inhibitor-2
CAS:Potent PI3K/mTOR Inhibitor-2 targets PI3Kα/β/δ/γ & mTOR (IC50: 3.4, 34, 16,1, 4.7 nM); exhibits antitumor effects.Formula:C20H13ClF2N4O4SPurity:96.16%Color and Shape:SolidMolecular weight:478.86Ref: TM-T12459
1mg55.00€5mg138.00€1mL*10mM (DMSO)144.00€10mg215.00€25mg358.00€50mg512.00€100mg692.00€200mg888.00€PI3K-IN-10
CAS:PI3K-IN-10 is a potent inhibitor of pan-PI3K .Formula:C23H19ClN6OPurity:98%Color and Shape:SolidMolecular weight:430.89PI4KIII β inhibitor 3
CAS:PI4KIII beta inhibitor 3 is a novel and high effective inhibitor of PI4KIIIβ (IC50 of 5.7 nM).Formula:C22H22N8OSPurity:98%Color and Shape:SolidMolecular weight:446.53GS-9901
CAS:GS-9901 is a selective, orally active and potent PI3Kδ inhibitor (IC50: 1 nM) for the study of non-Hodgkin's lymphoma and chronic lymphocytic leukemia.Formula:C22H17ClFN9OPurity:98.60% - 99.92%Color and Shape:SolidMolecular weight:477.88NVP-BAG956
CAS:NVP-BAG956 is an ATP-competitive PI3K inhibitor (IC50s: 34/56/112/444 nM for PI3Kδ/PI3Kα/PI3Kγ/PI3Kβ).Formula:C28H21N5Purity:99.25% - 99.80%Color and Shape:SolidMolecular weight:427.5Ref: TM-TQ0313
1mg54.00€5mg114.00€1mL*10mM (DMSO)126.00€10mg200.00€25mg401.00€50mg670.00€100mg1,224.00€200mg1,648.00€AZ044
CAS:AZ044 is a potent, selective inhibitor of type III phosphatidylinositol-4-kinase alpha-subtype (PI4KIIIalpha).Formula:C24H27N3O3SPurity:99.5%Color and Shape:SolidMolecular weight:437.55Ref: TM-T26698
1mg54.00€5mg114.00€1mL*10mM (DMSO)126.00€10mg178.00€25mg409.00€50mg708.00€100mg1,153.00€200mg1,558.00€TGX-115
CAS:TGX-115 inhibits PI 3-K p110β (IC50=0.13μM) & p110δ (IC50=0.63μM), treats various cardiovascular diseases.Formula:C20H20N2O3Purity:99.48%Color and Shape:SolidMolecular weight:336.38Ref: TM-T24873
1mg190.00€1mL*10mM (DMSO)369.00€5mg447.00€10mg610.00€25mg858.00€50mg1,063.00€100mg1,350.00€200mg1,765.00€SRX3207
CAS:SRX3207 is an inhibitor of Syk and PI3K and relieves tumor immunosuppression.Formula:C29H29N7O3SPurity:99.85%Color and Shape:SolidMolecular weight:555.65PQR514
CAS:PQR514: more potent pan-PI3K inhibitor than predecessor PQR309, exhibits strong anticancer activity in vitro and in OVCAR-3 model.
Formula:C16H20F2N8O2Purity:98.77% - 99.19%Color and Shape:SolidMolecular weight:394.38Ginsenoside Rk1
CAS:Ginsenoside Rk1 is a component created by processing the ginseng plant at high temperatures.Formula:C42H70O12Purity:98.46% - 99.13%Color and Shape:SolidMolecular weight:767.00PI3Kδ-IN-1
CAS:PI3Kδ-IN-1 is an efficacious PI3Kδ inhibitor (IC50 of 1.7 nM).Formula:C22H20F3N7O2Purity:99.85%Color and Shape:SolidMolecular weight:471.44GNE-490
CAS:GNE-490 is an effective inhibitor of pan-PI3K with IC50s of 3.5 nM, 25 nM, 5.2 nM, 15 nM for PI3Kα, PI3Kβ, PI3Kδ and PI3Kγ, respectively.Formula:C18H22N6O2SPurity:99.77%Color and Shape:SolidMolecular weight:386.47Ref: TM-T22339
1mg80.00€2mg109.00€5mg178.00€1mL*10mM (DMSO)193.00€10mg304.00€25mg482.00€50mg665.00€100mg883.00€200mg1,215.00€CAL-130 Racemate
CAS:CAL-130 Racemate is the racemate of CAL-130. CAL-130 is a PI3Kδ and PI3Kγ inhibitor (IC50s: 1.3 and 6.1 nM).Formula:C23H22N8OPurity:98%Color and Shape:SolidMolecular weight:426.47NVP-QAV-572
CAS:NVP-QAV-572 is a inhibitor of PI3K(IC50 of 10 nM).Formula:C17H19F2N7O3S2Purity:98%Color and Shape:SolidMolecular weight:471.5Zandelisib
CAS:Zandelisib is an inhibitor of phosphatidylinositol 3-kinase (PI3K)(p110δ, IC50 of 3.5 nM), and with antineoplastic activity.Formula:C31H38F2N8OPurity:99.88%Color and Shape:SolidMolecular weight:576.68Ref: TM-T13386
1mg80.00€5mg168.00€1mL*10mM (DMSO)213.00€10mg264.00€25mg462.00€50mg620.00€100mg853.00€PIK-inhibitors
CAS:PIK-inhibitors (MDK34597) is a pan PI3K inhibitors, an analog of PI-103.Formula:C19H17N5O2Purity:96.98%Color and Shape:SolidMolecular weight:347.37SAR-260301
CAS:SAR-260301 is an orally available and selective inhibitor of PI3Kβ (IC50: 23 nM).Formula:C19H22N4O3Purity:99.74%Color and Shape:SolidMolecular weight:354.4Ref: TM-T16841
2mg43.00€5mg65.00€1mL*10mM (DMSO)71.00€10mg87.00€25mg173.00€50mg264.00€100mg371.00€200mg523.00€MIPS-21335
CAS:MIPS-21335 is a potent PI3KC2α inhibitor with an IC50 value of 7 nM and additionally exhibits inhibitory activity against PI3KC2β, p110α, p110β, and p110δ withFormula:C24H21N7O5Purity:98%Color and Shape:SolidMolecular weight:487.47LAS191954
CAS:LAS191954 is a selective, potent and orally active PI3Kδ inhibitor for inflammatory diseases treatment(IC50 : 2.6 nM).Formula:C20H15N9OPurity:98%Color and Shape:SolidMolecular weight:397.39MSC2360844
CAS:MSC2360844 is a potent, orally active and selective inhibitor of PI3Kδ(IC50 of 145 nM).Formula:C26H27FN4O5SPurity:99.54% - 99.9%Color and Shape:SolidMolecular weight:526.58Ref: TM-T12115
1mg52.00€5mg116.00€1mL*10mM (DMSO)135.00€10mg182.00€25mg354.00€50mg568.00€100mg900.00€200mg1,206.00€
