PI3K
PI3K inhibitors are compounds that block the activity of Phosphoinositide 3-Kinases (PI3Ks), a family of enzymes involved in a wide range of cellular processes, including growth, proliferation, survival, and metabolism. The PI3K/Akt/mTOR pathway is often dysregulated in cancer, making PI3K a key target for cancer therapy. PI3K inhibitors are critical tools for studying signal transduction, cancer biology, and the development of targeted therapies. At CymitQuimica, we provide a variety of PI3K inhibitors to support your research in cell signaling, oncology, and therapeutic development.
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KU-0060648
CAS:881375-00-4
KU-0060648 is a dual inhibitor of DNA-PK and PI3Kα, PI3Kβ, PI3Kδ with IC50 of 8.6 …
Formula:
C33H34N4O4S
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
582.71
Ref: TM-T6557
| 1mg | 59.00 € | ||
| 2mg | 81.00 € | ||
| 5mg | 104.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 298.00 € | ||
| 50mg | 444.00 € | ||
| 100mg | 635.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Desmethyl-VS-5584
CAS:1246535-95-4
Desmethyl-VS-5584 is a dimethyl analog of VS-5584, which is a novel and highly selective PI3K/mTOR …
Formula:
C16H20N8O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
340.38
Ref: TM-T4199
| 1mg | 59.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 150.00 € | ||
| 10mg | 256.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 635.00 € | ||
| 100mg | 902.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Duvelisib
CAS:1201438-56-3
Duvelisib (INK1197, IPI-145) is a selective inhibitor of phosphatidylinositol 3-kinase (PI3K) and p100δ.Cost-effective and quality-assured.
Formula:
C22H17ClN6O
Purity:
99.38% - 99.74%
Color and Shape:
Solid
Molecular weight:
416.86
Ref: TM-T1988
| 2mg | 48.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 93.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 244.00 € |
Estimated delivery in United States, on Friday 16 May 2025
PIK-75
CAS:372196-67-3
PIK-75, a DNA-PK and PI3K inhibitor, suppresses DNA-PK(IC50=2 nM), p110α(IC50=5.8 nM) and p110γ(IC50=76 nM).
Formula:
C16H14BrN5O4S
Purity:
100% - 99.88%
Color and Shape:
Solid
Molecular weight:
452.28
Ref: TM-T2667
| 5mg | 46.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 183.00 € | ||
| 100mg | 283.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Vacuolin-1
CAS:351986-85-1
Vacuolin-1 is a cell-permeable inhibitor of Ca2+ dependent fusion of lysosomes to the cell membrane.
Formula:
C26H24IN7O
Purity:
97.20% - 98.45%
Color and Shape:
Solid
Molecular weight:
577.42
Ref: TM-T21992
| 1mg | 37.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 550.00 € |
Estimated delivery in United States, on Friday 16 May 2025
CZC24832
CAS:1159824-67-5
CZC24832 is a selective inhibitor of PI 3-kinase γ.
Formula:
C15H17FN6O2S
Purity:
99.08% - 99.12%
Color and Shape:
Solid
Molecular weight:
364.4
Ref: TM-T1949
| 1mg | 50.00 € | ||
| 2mg | 66.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 356.00 € | ||
| 100mg | 525.00 € | ||
| 1mL*10mM (DMSO) | 110.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Deoxyelephantopin
CAS:29307-03-7
Deoxyelephantopin: anti-inflammatory, hepatoprotective, wound healing, antitumor; blocks NF-κB, MAPK, PI3K/Akt, β-catenin pathways.
Formula:
C19H20O6
Purity:
99.6% - 99.71%
Color and Shape:
Solid
Molecular weight:
344.36
Ref: TM-TN1079
| 1mg | 96.00 € | ||
| 5mg | 235.00 € | ||
| 10mg | 349.00 € | ||
| 25mg | 567.00 € | ||
| 50mg | 820.00 € | ||
| 1mL*10mM (DMSO) | 240.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Acalisib
CAS:870281-34-8
Acalisib (CAL-120) (GS-9820) is a potent and selective inhibitor of PI3Kδ.
Formula:
C21H16FN7O
Purity:
98.99% - ≥95%
Color and Shape:
Solid
Molecular weight:
401.4
Ref: TM-T2682
| 5mg | 51.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 138.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 283.00 € | ||
| 200mg | 424.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Parsaclisib hydrochloride
CAS:1995889-48-9
Parsaclisib hydrochloride (INCB050465 HCl) is a selectve PI3Kδ inhibitor with antitumor activity. Parsaclisib demonstrates potent …
Formula:
C20H23Cl2FN6O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
469.34
Ref: TM-T28297
| 25mg | 1,169.00 € | ||
| 50mg | 1,529.00 € | ||
| 100mg | 2,442.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Umbralisib hydrochloride
CAS:1532533-78-0
Umbralisib hydrochloride: PI3Kδ inhibitor; IC50=22.2 nM, EC50=24.3 nM; active vs CK1ε, EC50=6.0 μM.
Formula:
C31H25ClF3N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
608.01
Ref: TM-T17066
| 2mg | 58.00 € |
Estimated delivery in United States, on Friday 16 May 2025
BGT226 maleate
CAS:1245537-68-1
BGT226 maleate (NVP-BGT226) is a class I PI3K/mTOR inhibitor for PI3Kα/β/γ (IC50: 4/63/38 nM) .
Formula:
C28H25F3N6O2·C4H4O4
Purity:
97.75% - 98.78%
Color and Shape:
Solid
Molecular weight:
650.6
Ref: TM-T6072
| 1mg | 38.00 € | ||
| 5mg | 77.00 € | ||
| 10mg | 114.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 359.00 € | ||
| 100mg | 512.00 € | ||
| 200mg | 702.00 € | ||
| 1mL*10mM (DMSO) | 99.00 € |
Estimated delivery in United States, on Tuesday 27 May 2025
GSK2292767
CAS:1254036-66-2
GSK2292767 is a potent and selective PI3Kδ inhibitor.
Formula:
C24H28N6O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
512.58
Ref: TM-T6850
| 1mg | To inquire | ||
| 5mg | To inquire | ||
| 10mg | To inquire | ||
| 25mg | To inquire |
Estimated delivery in United States, on Friday 13 Jun 2025
CNX-1351
CAS:1276105-89-5
CNX-1351 is a potent and isoform-selective targeted covalent PI3Kα inhibitor.
Formula:
C30H35N7O3S
Purity:
98.83% - 99.69%
Color and Shape:
Solid
Molecular weight:
573.71
Ref: TM-T2256
| 1mg | 48.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 281.00 € | ||
| 50mg | 520.00 € | ||
| 100mg | 750.00 € | ||
| 500mg | 1,549.00 € |
Estimated delivery in United States, on Friday 13 Jun 2025
TGX-115
CAS:351071-62-0
TGX-115 inhibits PI 3-K p110β (IC50=0.13μM) & p110δ (IC50=0.63μM), treats various cardiovascular diseases.
Formula:
C20H20N2O3
Purity:
99.2%
Color and Shape:
Solid
Molecular weight:
336.38
Ref: TM-T24873
| 1mg | 200.00 € | ||
| 5mg | 472.00 € | ||
| 10mg | 645.00 € | ||
| 25mg | 905.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,425.00 € | ||
| 200mg | 1,863.00 € | ||
| 1mL*10mM (DMSO) | 389.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
PI3K-IN-10
CAS:2211922-64-2
PI3K-IN-10 is a potent inhibitor of pan-PI3K .
Formula:
C23H19ClN6O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
430.89
Ref: TM-T12456
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 27 Jun 2025
PI3K/mTOR Inhibitor-2
CAS:1848242-58-9
Potent PI3K/mTOR Inhibitor-2 targets PI3Kα/β/δ/γ & mTOR (IC50: 3.4, 34, 16,1, 4.7 nM); exhibits antitumor …
Formula:
C20H13ClF2N4O4S
Purity:
96.16%
Color and Shape:
Solid
Molecular weight:
478.86
Ref: TM-T12459
| 1mg | 58.00 € | ||
| 5mg | 145.00 € | ||
| 10mg | 226.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 540.00 € | ||
| 100mg | 730.00 € | ||
| 200mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 153.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
PI3Kdelta inhibitor 1
CAS:2242109-74-4
PI3Kdelta inhibitor 1 is a potent, selective and orally available inhibitor of PI3Kδ with an …
Formula:
C27H38N6O5S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
558.69
Ref: TM-T12461
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
IHMT-PI3Kδ-372
CAS:2429889-62-1
IHMT-PI3Kδ-372 is a selective inhibitor of PI3Kδ with an IC50 of 14 nM and can …
Formula:
C26H23F2N7O2
Purity:
99.54%
Color and Shape:
Liquid
Molecular weight:
503.5
Ref: TM-T35530
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 105.00 € | ||
| 25mg | 167.00 € | ||
| 50mg | 249.00 € | ||
| 100mg | 338.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
PI3Kγ inhibitor 1
CAS:1172118-03-4
PI3Kγ inhibitor 1 is a inhibitor of PI3Kδ and PI3Kγ.
Formula:
C32H26N8O2S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
586.67
Ref: TM-T12464
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
PI3Kα-IN-13
CAS:2955529-67-4
PI3Kα-IN-13 (Compound 18a), a PI3Kα inhibitor with an IC50 of 2.5 nM, effectively induces apoptosis …
Formula:
C21H19N5O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
389.41
Ref: TM-T79685
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Friday 27 Jun 2025
