PI3K/Akt/mTOR Signaling
Subcategories of "PI3K/Akt/mTOR Signaling"
Show 2 more subcategories
Products of "PI3K/Akt/mTOR Signaling"
PS10
CAS:1564265-82-2
PS10 is a ATP-competitive inhibitor of pan-PDK(PDK2, PDK4, PDK1, and PDK3 with IC50 of 0.8 …
Formula:
C14H13NO6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
323.32
Ref: TM-T12566
1mg | 40.00 € | ||
2mg | To inquire |
Estimated delivery in United States, on Wednesday 7 Aug 2024
NV-5138
CAS:2095886-80-7
NV-5138 is a selective and orally active activator of brain mTORC1, with antidepressant effects.
Formula:
C7H13F2NO2
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
181.18
Ref: TM-T12270
1mg | 88.00 € | ||
1ml | 168.00 € | ||
5mg | 211.00 € | ||
10mg | 339.00 € | ||
25mg | 725.00 € | ||
50mg | 1,148.00 € | ||
100mg | 1,662.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
9-ING-41
CAS:1034895-42-5
9-ING-41 is a glycogen synthase kinase-3 inhibitor.
Formula:
C22H13FN2O5
Purity:
99.25%
Color and Shape:
Solid
Molecular weight:
404.35
Ref: TM-T14066
1mg | 49.00 € | ||
1ml | 116.00 € | ||
2mg | 69.00 € | ||
5mg | 98.00 € | ||
10mg | 160.00 € | ||
25mg | 320.00 € | ||
50mg | 462.00 € | ||
100mg | 689.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Lidocaine Hydrochloride hydrate
CAS:6108-05-0
Lidocaine Hydrochloride hydrate is an amide local anesthetic, has anti-inflammatory property.
Formula:
C14H22N2O·HCl·H2O
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
288.82
Ref: TM-T1144L
1ml | 49.00 € | ||
50mg | 63.00 € | ||
100mg | 81.00 € | ||
200mg | 100.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Epertinib hydrochloride
CAS:2071195-74-7
Epertinib hydrochloride (S-22611 hydrochloride) shows potent antitumor activity.
Formula:
C30H28Cl2FN5O3
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
596.48
Ref: TM-T11213
1mg | 95.00 € | ||
1ml | 301.00 € | ||
2mg | 138.00 € | ||
5mg | 230.00 € | ||
10mg | 368.00 € | ||
25mg | 621.00 € | ||
50mg | 885.00 € | ||
100mg | 1,205.00 € | ||
500mg | 2,404.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Erlotinib hydrochloride
CAS:183319-69-9
Erlotinib hydrochloride (NSC 718781) is an EGFR inhibitor (IC50: 2 nM). It is used for …
Formula:
C22H23N3O4·HCl
Purity:
99.79%
Color and Shape:
White Or Off-White Powder
Molecular weight:
429.9
Ref: TM-T0373L
1g | 115.00 € | ||
1ml | 65.00 € | ||
50mg | 41.00 € | ||
100mg | 52.00 € | ||
500mg | 82.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
MELK-IN-1
CAS:2095596-44-2
MELK-IN-1 (MELK inhibitor 17) is a potent inhibitor of maternal embryonic leucine zipper kinase (MELK),(IC50:3nm;Ki:0.39 …
Formula:
C31H33N5O4
Purity:
99.14%
Color and Shape:
Solid
Molecular weight:
539.62
Ref: TM-T11997
1mg | 55.00 € | ||
1ml | 142.00 € | ||
2mg | 80.00 € | ||
5mg | 118.00 € | ||
10mg | 184.00 € | ||
25mg | 424.00 € | ||
50mg | 626.00 € | ||
100mg | 891.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Mevastatin
CAS:73573-88-3
Mevastatin (ML236B) is an HMG-CoA reductase inhibitor that was initially isolated from the mold Pythium …
Formula:
C23H34O5
Purity:
97.96%
Color and Shape:
White-Yellowish To Yellow Powder Solid Powder
Molecular weight:
390.51
Ref: TM-T0683
1ml | 59.00 € | ||
50mg | 55.00 € | ||
100mg | 83.00 € | ||
500mg | 207.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Cyanoacetohydrazide
CAS:140-87-4
Cyanoacetohydrazide (Cyanoacetic hydrazide) is an anti-TB drug. It has also been used to derive compounds …
Formula:
C3H5N3O
Purity:
99.9%
Color and Shape:
Stout Prisms From Alcohol Slightly Brown Powder
Molecular weight:
99.09
Ref: TM-T0704
1g | 34.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
NSC781406
CAS:1676893-24-5
NSC781406 is a highly effective inhibitor of PI3K and mTOR (IC50: 2 nM for PI3Kα).
Formula:
C29H27F2N5O5S2
Purity:
99.08%
Color and Shape:
Solid
Molecular weight:
627.68
Ref: TM-T16355
1mg | 51.00 € | ||
1ml | 132.00 € | ||
5mg | 94.00 € | ||
10mg | 157.00 € | ||
25mg | 277.00 € | ||
50mg | 456.00 € | ||
100mg | 664.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Isoprenaline hydrochloride
CAS:51-30-9
Isoprenaline hydrochloride (NCI-c55630) is a potent beta-adrenergic agonist with the peripheral vasodilator, bronchodilator, and cardiac …
Formula:
C11H18ClNO3
Purity:
100%
Color and Shape:
Turn Brownish-Pink Upon Prolonged Exposure To Air (Ntp 1992)
Molecular weight:
247.719
Ref: TM-T1056
1g | 44.00 € | ||
1ml | 36.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Mutated EGFR-IN-1
CAS:1421372-66-8
Mutated EGFR-IN-1 (Osimertinib analog) is a useful intermediate for the inhibitors design for mutated EGFR, …
Formula:
C25H31N7O
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
445.56
Ref: TM-T16162
1ml | 49.00 € | ||
25mg | 57.00 € | ||
50mg | 66.00 € | ||
100mg | 88.00 € | ||
200mg | 114.00 € | ||
500mg | 183.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Erlotinib
CAS:183321-74-6
Erlotinib (NSC-718781) is an EGFR inhibitor (IC50: 2 nM). It is used for the treatment …
Formula:
C22H23N3O4
Purity:
99.98%
Color and Shape:
White To Off-White Powder
Molecular weight:
393.44
Ref: TM-T0373
1ml | 55.00 € | ||
50mg | 47.00 € | ||
100mg | 52.00 € | ||
500mg | 78.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
O-Desmethyl gefitinib
CAS:847949-49-9
O-Desmethyl gefitinib is an active EGFR inhibitor (IC50: 36 nM), a metabolite of Gefitinib, formed …
Formula:
C21H22ClFN4O3
Purity:
99.6%
Color and Shape:
Solid
Molecular weight:
432.88
Ref: TM-T16369
1mg | 55.00 € | ||
1ml | 121.00 € | ||
5mg | 109.00 € | ||
10mg | 167.00 € | ||
25mg | 335.00 € | ||
50mg | 535.00 € | ||
100mg | 766.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
CGS 15943
CAS:104615-18-1
CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.
Formula:
C13H8ClN5O
Purity:
99.63%
Color and Shape:
Solid
Molecular weight:
285.69
Ref: TM-T14944
1mg | 46.00 € | ||
1ml | 91.00 € | ||
5mg | 88.00 € | ||
10mg | 128.00 € | ||
25mg | 207.00 € | ||
50mg | 310.00 € | ||
100mg | 463.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
STL127705
CAS:1326852-06-5
STL127705 inhibits Ku 70/80 protein & DNA-PKCS kinase, IC50s: 3.5 μM & 2.5 μM.
Formula:
C22H20FN5O4
Purity:
97.41%
Color and Shape:
Solid
Molecular weight:
437.42
Ref: TM-T13017
1mg | 112.00 € | ||
1ml | 315.00 € | ||
5mg | 269.00 € | ||
10mg | 423.00 € | ||
25mg | 700.00 € | ||
50mg | 984.00 € | ||
100mg | 1,333.00 € | ||
500mg | 2,655.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Adenosine 5'-monophosphate monohydrate
CAS:18422-05-4
Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is …
Formula:
C10H14N5O7P·H2O
Purity:
98.36%
Color and Shape:
White Powder
Molecular weight:
365.24
Ref: TM-T0853L
1g | 52.00 € | ||
1ml | 49.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
Lapatinib Ditosylate
CAS:388082-77-7
Lapatinib Ditosylate (Tykerb ditosylate) is an effective EGFR and ErbB2 inhibitor (IC50: 10.8/9.2 nM for …
Formula:
C29H26ClFN4O4S·2C7H8O3S
Purity:
99.71%
Color and Shape:
Yellow Solid
Molecular weight:
925.46
Ref: TM-T6235
1g | 145.00 € | ||
1ml | 63.00 € | ||
25mg | 46.00 € | ||
50mg | 58.00 € | ||
100mg | 73.00 € | ||
200mg | 94.00 € | ||
500mg | 126.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
PI4KIIIbeta-IN-9
CAS:1429624-84-9
PI4KIIIbeta-IN-9 is a potent inhibitor of PI4KIIIβ(IC50 of 7 nM). .
Formula:
C23H25N3O5S2
Purity:
98.22%
Color and Shape:
Solid
Molecular weight:
487.59
Ref: TM-T12469
1mg | 78.00 € | ||
1ml | 202.00 € | ||
5mg | 183.00 € | ||
10mg | 275.00 € | ||
25mg | 498.00 € | ||
50mg | 696.00 € | ||
100mg | 913.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024
LTURM34
CAS:1879887-96-3
LTURM34 is an inhibitor of DNA-PK with IC50 of 34 nM.
Formula:
C24H18N2O3S
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
414.48
Ref: TM-T15789
1ml | 77.00 € | ||
5mg | 69.00 € | ||
10mg | 109.00 € | ||
25mg | 230.00 € | ||
50mg | 398.00 € | ||
100mg | 594.00 € |
Estimated delivery in United States, on Friday 9 Aug 2024