G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
ABT-080
CAS:189498-57-5
ABT-080 (VML 530), a leukotriene synthesis inhibitor, is used potentially for treatment of asthma.
Formula:
C37H31N2NaO4
Purity:
98.15%
Color and Shape:
Solid
Molecular weight:
590.64
Ref: TM-T26524
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 270.00 € | ||
| 200mg | 405.00 € | ||
| 1mL*10mM (DMSO) | 90.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Itasetron
CAS:123258-84-4
Itasetron, a 5-HT3 antagonist, prevents memory loss in rats and has antiemetic effects in cancer …
Formula:
C16H20N4O2
Purity:
100% - 99.63%
Color and Shape:
Solid
Molecular weight:
300.36
Ref: TM-T24184
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,050.00 € | ||
| 25mg | 1,486.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,547.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
PF-03654746 Tosylate
CAS:1039399-17-1
PF-03654746 Tosylate is selective antagonist of histamine H3 receptor with high brain penetration.
Formula:
C25H32F2N2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
494.6
Ref: TM-T12416
| 25mg | 854.00 € | ||
| 50mg | 1,096.00 € | ||
| 100mg | 1,668.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Quinpirole Hydrochloride
CAS:85798-08-9
Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has …
Formula:
C13H22ClN3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
255.79
Ref: TM-T12606
| 1mg | 107.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
GPR84 antagonist 8
CAS:1445846-30-9
GPR84 antagonist 8 is a selective GPR84 antagonist.
Formula:
C23H23N3O5
Color and Shape:
Solid
Molecular weight:
421.45
Ref: TM-T11462
| 25mg | 4,212.00 € | ||
| 50mg | 5,896.00 € | ||
| 100mg | 8,259.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
PNU-177864
CAS:250266-51-4
PNU-177864 is a selective dopamine D3 receptor antagonist.
Formula:
C18H21F3N2O3S
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
402.43
Ref: TM-T23167
| 1mg | 63.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 121.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 330.00 € | ||
| 50mg | 462.00 € | ||
| 100mg | 638.00 € | ||
| 500mg | 1,291.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
BAY-1316957
CAS:1613264-40-6
BAY-1316957 is a highly potent and selective EP4 receptor antagonist. With an IC50 of 15.3 …
Formula:
C27H27N3O3
Color and Shape:
Solid
Molecular weight:
441.52
Ref: TM-T14500
| 50mg | 739.00 € | ||
| 100mg | 1,198.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
JP1302
CAS:80259-18-3
JP1302: α2C adrenoceptor antagonist, Kb 16 nM, Ki 28 nM, antidepressant, FACT disruptor, studies: neuropsychiatric, …
Formula:
C24H24N4
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
368.47
Ref: TM-T22882
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 128.00 € | ||
| 25mg | 234.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 604.00 € | ||
| 500mg | 1,287.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Imetit dihydrobromide
CAS:32385-58-3
Imetit dihydrobromide is a high affinity and effective agonist of histamine H3 and H4 receptors …
Formula:
C6H12Br2N4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
332.06
Ref: TM-T15565
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Licogliflozin
CAS:1291094-73-9
Licogliflozin (LIK066) is an inhibitor of sodium-glucose cotransporter (SGLT1 and SGLT2).
Formula:
C23H28O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
416.46
Ref: TM-T15752
| 25mg | 800.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,741.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
L-692429
CAS:145455-23-8
L-692429 (MK-0751) is a GHS agonist with high affinity for G protein-coupled receptors and can …
Formula:
C29H31N7O2
Purity:
98.64% - 99.9%
Color and Shape:
Solid
Molecular weight:
509.614
Ref: TM-T11798
| 1mg | 152.00 € | ||
| 5mg | 371.00 € | ||
| 10mg | 546.00 € | ||
| 25mg | 890.00 € | ||
| 50mg | 1,208.00 € | ||
| 100mg | 1,623.00 € | ||
| 1mL*10mM (DMSO) | 420.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
(S)-Terazosin
CAS:109351-33-9
(S)-Terazosin is an active S-enantiomer of Terazosin.
Formula:
C19H25N5O4
Color and Shape:
Solid
Molecular weight:
387.43
Ref: TM-T12815
| 2mg | 115.00 € | ||
| 5mg | 186.00 € | ||
| 50mg | 739.00 € | ||
| 100mg | 1,161.00 € | ||
| 1mL*10mM (DMSO) | 214.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Lorglumide sodium salt
CAS:1021868-76-7
Lorglumide sodium salt (CR-1409 sodium salt) is an antagonist of cholecystokinin receptors (CCK).
Formula:
C22H31Cl2N2NaO4
Purity:
99.32%
Color and Shape:
Solid
Molecular weight:
481.39
Ref: TM-T11868
| 5mg | 34.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
JTE-907
CAS:282089-49-0
JTE-907 is a CB2 receptor inverse agonist with high selectivity and oral activity.JTE-907 exhibits anti-inflammatory …
Formula:
C24H26N2O6
Purity:
100%
Color and Shape:
Solid
Molecular weight:
438.47
Ref: TM-T19705
| 1mg | 55.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 323.00 € | ||
| 50mg | 482.00 € | ||
| 100mg | 688.00 € | ||
| 1mL*10mM (DMSO) | 150.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Landipirdine
CAS:1000308-25-7
Landipirdine (RO-5025181) is a selective 5-HT6R antagonist for the study of central nervous system disorders …
Formula:
C18H19FN2O3S
Purity:
97.50% - 99.33%
Color and Shape:
Solid
Molecular weight:
362.42
Ref: TM-T27795
| 1mg | 227.00 € | ||
| 5mg | 541.00 € | ||
| 10mg | 726.00 € | ||
| 25mg | 1,172.00 € | ||
| 50mg | 1,493.00 € | ||
| 100mg | 2,124.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
T-0509
CAS:96843-99-1
T-0509 is a selective beta 1 receptor agonist that increases inotropy in canine ventricular muscle …
Formula:
C18H23NO5
Purity:
97.46% - 98.21%
Color and Shape:
Solid
Molecular weight:
333.38
Ref: TM-T28895
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,331.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
BTB09089
CAS:245728-44-3
BTB09089 (GPR65 agonist ) is a T cell death-associated gene 8 (TDAG8/GPR65)-specific agonist.BTB09089 induces TDAG8 …
Formula:
C14H12Cl2N4OS2
Purity:
100%
Color and Shape:
Soild
Molecular weight:
387.31
Ref: TM-T67892
| 1mg | 71.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 184.00 € | ||
| 25mg | 336.00 € | ||
| 50mg | 510.00 € | ||
| 100mg | 733.00 € | ||
| 500mg | 1,514.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
ReN-1869
CAS:170149-99-2
ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity …
Formula:
C24H27NO2
Purity:
99.87% - 99.89%
Color and Shape:
Solid
Molecular weight:
361.48
Ref: TM-T28516
| 1mg | 201.00 € | ||
| 5mg | 502.00 € | ||
| 10mg | 725.00 € | ||
| 25mg | 1,117.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
SLM6031434 HCl
CAS:1897379-34-8
SLM6031434 HCl (SLM-6031434 HCl) is a SphK2 inhibitor that reduces LPS-induced TNF伪 and IL-1尾 production.
Formula:
C22H31ClF3N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
489.96
Ref: TM-T28806
| 1mg | 126.00 € | ||
| 5mg | 397.00 € | ||
| 10mg | 546.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
p-MPPF dihydrochloride
CAS:223699-41-0
p-MPPF dihydrochloride is a 5-HT antagonist that can be used to study neurological diseases.
Formula:
C25H29Cl2FN4O2
Purity:
99.78%
Color and Shape:
Liquid
Molecular weight:
507.43
Ref: TM-T69750
| 1mg | 266.00 € | ||
| 5mg | 655.00 € | ||
| 10mg | 896.00 € | ||
| 25mg | 1,437.00 € | ||
| 50mg | 1,872.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
