G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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AT-121
CAS:2099681-31-7
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, …
Formula:
C24H38N4O3S
Purity:
97% - 97.95%
Color and Shape:
Solid
Molecular weight:
462.65
Ref: TM-T37610
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Seridopidine
CAS:883631-51-4
Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy …
Formula:
C14H20FNO2S
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T34616
| 1mg | 137.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,103.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,962.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ASP-4058
CAS:952565-91-2
ASP-4058: Safe, oral S1P1/S1P5 agonist; improves autoimmune encephalomyelitis in mice.
Formula:
C19H12F6N4O2
Purity:
99.5% - 99.51%
Color and Shape:
Solid
Molecular weight:
442.31
Ref: TM-T10385
| 1mg | 95.00 € | ||
| 5mg | 226.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 654.00 € | ||
| 50mg | 896.00 € | ||
| 100mg | 1,262.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Ordopidine
CAS:871351-60-9
Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during …
Formula:
C14H20FNO2S
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T33816
| 1mg | 137.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SCH 221510
CAS:322473-89-2
SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.
Formula:
C28H31NO
Purity:
99.10%
Color and Shape:
Solid
Molecular weight:
397.55
Ref: TM-T23335
| 1mg | 77.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 260.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 834.00 € | ||
| 100mg | 1,355.00 € | ||
| 200mg | 1,822.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Clonidine
CAS:4205-90-7
Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.
Formula:
C9H9Cl2N3
Purity:
99.44% - 99.88%
Color and Shape:
Crystals Solid
Molecular weight:
230.09
Ref: TM-T7045
| 50mg | 89.00 € | ||
| 100mg | 128.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Trimebutine CTB salt
CAS:1456509-46-8
Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.
Formula:
C29H36N2O8S2
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
604.74
Ref: TM-T27413
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,499.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SCH-486757
CAS:524019-25-8
SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used …
Formula:
C24H23Cl2N3O
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
440.37
Ref: TM-T28728
| 1mg | 278.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 936.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
AVN-322
CAS:1194574-68-9
AVN-322 is a 5-HT6 receptor antagonist. 5-HT6R antagonists improves cognition in animal models of cognitive …
Formula:
C17H20ClN5O2S
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
393.89
Ref: TM-T26691
| 1mg | 276.00 € | ||
| 5mg | 679.00 € | ||
| 10mg | 928.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Imiloxan
CAS:81167-16-0
Imiloxan (RS-21361) is an α2 adrenergic receptor antagonist used in the treatment of major depressive …
Formula:
C14H16N2O2
Purity:
100% - 98.89%
Color and Shape:
Solid
Molecular weight:
244.29
Ref: TM-T27599
| 1mg | 392.00 € | ||
| 5mg | 932.00 € | ||
| 25mg | 1,827.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CCX777
CAS:1226686-36-7
CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer …
Formula:
C31H43N7O3S
Purity:
98.73%
Color and Shape:
Solid
Molecular weight:
593.78
Ref: TM-T23866
| 1mg | 278.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
BGC201531
CAS:1186532-61-5
BGC201531 (AP-1531) is a EP4 antagonist for the treatment of acute migraine.
Formula:
C26H28N2O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
496.58
Ref: TM-T8993
| 25mg | 762.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
JNJ 10191584 maleate
CAS:869497-75-6
JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor …
Formula:
C17H19ClN4O5
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
394.81
Ref: TM-T22879
| 1mg | 53.00 € | ||
| 2mg | 81.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 14 Jan 2025
AZD8797
CAS:911715-90-7
AZD8797 (KAND567) is a CX3CR1 antagonist with potential protective effects against neuronal damage and prevents …
Formula:
C19H25N5OS2
Purity:
98.73% - 99.68%
Color and Shape:
Solid
Molecular weight:
403.56
Ref: TM-T14384
| 1mg | 91.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 733.00 € | ||
| 50mg | 918.00 € | ||
| 100mg | 1,329.00 € | ||
| 1mL*10mM (DMSO) | 216.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Sigma-LIGAND-1
CAS:139652-01-0
Sigma-LIGAND-1 is a selective Sigma Receptor ligand with an IC50s of 16 nM, 19 nM …
Formula:
C27H33NO4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
435.56
Ref: TM-T13510
| 1mg | 94.00 € | ||
| 5mg | 236.00 € | ||
| 10mg | 350.00 € | ||
| 25mg | 548.00 € | ||
| 50mg | 738.00 € | ||
| 100mg | 1,015.00 € | ||
| 500mg | 2,019.00 € | ||
| 1mL*10mM (DMSO) | 276.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L 674573
CAS:127481-29-2
L 674573 is an inhibitor of leukotriene biosynthesis.
Formula:
C28H27NO3S
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
457.58
Ref: TM-T24327
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 270.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
QS11
CAS:944328-88-5
QS11, a GTPase ARFGAP1, modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling pathway to …
Formula:
C36H33N5O2
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
567.68
Ref: TM-T4022
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 331.00 € | ||
| 200mg | 453.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
CP 316311
CAS:175139-41-0
CP 316311 is a specific CRF1 receptor antagonist with potential antidepressant activity and may be …
Formula:
C21H29NO2
Purity:
99.47% - 99.60%
Color and Shape:
Solid
Molecular weight:
327.46
Ref: TM-T15008
| 1mg | 277.00 € | ||
| 5mg | 497.00 € | ||
| 10mg | 637.00 € | ||
| 25mg | 865.00 € | ||
| 50mg | 1,174.00 € | ||
| 100mg | 1,565.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
SB-215505
CAS:162100-15-4
SB215505: potent 5-HT2B/2C blocker, enhances rat wakefulness/motor activity. (pKi: 5-HT2B - 8.3, 5-HT2C - 7.66, …
Formula:
C19H16ClN3O
Purity:
98.33%
Color and Shape:
Solid
Molecular weight:
337.8
Ref: TM-T28680
| 1mg | 209.00 € | ||
| 5mg | 521.00 € | ||
| 10mg | 726.00 € | ||
| 25mg | 1,081.00 € | ||
| 50mg | 1,493.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Taprizosin
CAS:210538-44-6
Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of …
Formula:
C25H26N6O4S
Purity:
97.01% - 99.11%
Color and Shape:
Solid
Molecular weight:
506.58
Ref: TM-T28922
| 1mg | 355.00 € | ||
| 5mg | 832.00 € | ||
| 10mg | 1,169.00 € | ||
| 25mg | 1,787.00 € | ||
| 50mg | 2,410.00 € | ||
| 100mg | 3,176.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
