G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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JNJ-20788560
CAS:825649-28-3
JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective …
Formula:
C25H28N2O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
388.5
Ref: TM-T27667
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,549.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
SLP9101555
SLP9101555 is a potent and selective sphingosine kinase 2 (SphK2) inhibitor with a Ki of …
Formula:
C16H22BrClN2
Purity:
99%
Color and Shape:
Liquid
Molecular weight:
357.72
Ref: TM-T63047
| 1mg | 326.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,336.00 € | ||
| 500mg | 4,568.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
OPC-51803
CAS:192514-54-8
OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of …
Formula:
C26H32ClN3O2
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
454
Ref: TM-T28257
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,053.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,568.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
KI-7
CAS:1489263-00-4
KI-7 is an adenosine A2B receptor positive allosteric modulator.
Formula:
C23H18N2O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
354.4
Ref: TM-T9238
| 2mg | 38.00 € | ||
| 5mg | 58.00 € | ||
| 10mg | 90.00 € | ||
| 25mg | 181.00 € | ||
| 50mg | 277.00 € | ||
| 100mg | 419.00 € | ||
| 200mg | 589.00 € | ||
| 1mL*10mM (DMSO) | 65.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
RG 7152
CAS:107813-63-8
RG 7152 is a leukotriene D4 antagonist with anti-asthmatic properties and can be used in …
Formula:
C20H19N5O2
Purity:
98.00%
Color and Shape:
Solid
Molecular weight:
361.4
Ref: TM-T28529
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Sinitrodil
CAS:143248-63-9
Sinitrodil (ITF-296) is a guanylate cyclase stimulant that may be used in the treatment of …
Formula:
C10H10N2O5
Purity:
99%
Color and Shape:
Solid
Molecular weight:
238.2
Ref: TM-T34648
| 1mg | 137.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 492.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,095.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,980.00 € | ||
| 1mL*10mM (DMSO) | 400.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
ML-335
CAS:1069498-96-9
ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief …
Formula:
C25H32N2O3
Purity:
98.52%
Color and Shape:
Solid
Molecular weight:
408.53
Ref: TM-T23002
| 1mg | 46.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 144.00 € | ||
| 25mg | 269.00 € | ||
| 50mg | 430.00 € | ||
| 100mg | 621.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AT-121
CAS:2099681-31-7
AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, …
Formula:
C24H38N4O3S
Purity:
97% - 97.95%
Color and Shape:
Solid
Molecular weight:
462.65
Ref: TM-T37610
| 1mg | 325.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,049.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 1,850.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Seridopidine
CAS:883631-51-4
Seridopidine (ACR343) is a modulator of dopaminergic activity that is used as an oral therapy …
Formula:
C14H20FNO2S
Purity:
99.11%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T34616
| 1mg | 137.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 797.00 € | ||
| 50mg | 1,103.00 € | ||
| 100mg | 1,477.00 € | ||
| 500mg | 2,962.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
PNU-282987 free base
CAS:711085-63-1
PNU-282987 is an α7 nAChR agonist (EC50=154 nM) and a 5-HT3 antagonist (IC50=4541 nM) for …
Formula:
C14H17ClN2O
Purity:
99.64%
Color and Shape:
Liquid
Molecular weight:
264.75
Ref: TM-T60437
| 1mg | 55.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 201.00 € | ||
| 25mg | 392.00 € | ||
| 50mg | 727.00 € | ||
| 100mg | 1,020.00 € | ||
| 500mg | 2,039.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
GS-9667
CAS:618380-90-8
GS-9667, a selective and partial agonist of the A(1) adenosine receptor (AR), represents an effective …
Formula:
C21H24FN5O4S
Purity:
99.76% - 99.76%
Color and Shape:
Solid
Molecular weight:
461.51
Ref: TM-T27439
| 1mg | 107.00 € | ||
| 5mg | 265.00 € | ||
| 10mg | 363.00 € | ||
| 25mg | 598.00 € | ||
| 50mg | 817.00 € | ||
| 100mg | 1,126.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Ordopidine
CAS:871351-60-9
Ordopidine (ACR325) is a dopaminergic stabilizer that suppresses psychostimulant-induced hyperactivity disorder and stimulates behavior during …
Formula:
C14H20FNO2S
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
285.38
Ref: TM-T33816
| 1mg | 137.00 € | ||
| 5mg | 327.00 € | ||
| 10mg | 493.00 € | ||
| 25mg | 798.00 € | ||
| 50mg | 1,100.00 € | ||
| 100mg | 1,483.00 € | ||
| 500mg | 2,980.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Lecozotan HCl
CAS:433282-68-9
Lecozotan HCl is a selective 5-HT antagonist boosting glutamate and acetylcholine release without causing 5-HT(1A) …
Formula:
C28H30ClN5O3
Purity:
99.47%
Color and Shape:
Solid
Molecular weight:
520.02
Ref: TM-T27806
| 1mg | 156.00 € | ||
| 5mg | 363.00 € | ||
| 10mg | 552.00 € | ||
| 25mg | 875.00 € | ||
| 50mg | 1,189.00 € | ||
| 100mg | 1,616.00 € | ||
| 500mg | 3,211.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Clovoxamine
CAS:54739-19-4
Clovoxamine fumarate (DU 23811 fumarate) is a 5-HT reuptake, serotonin and norepinephrine inhibitor with antidepressant …
Formula:
C14H21ClN2O2
Purity:
98.88% - 99.16%
Color and Shape:
Solid
Molecular weight:
284.78
Ref: TM-T27047
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
RO3244794
CAS:361457-01-4
RO3244794 is a selective prostacyclin (IP) receptor antagonist that can be used to study liver …
Formula:
C25H19F2NO5
Purity:
99.36%
Color and Shape:
Liquid
Molecular weight:
451.42
Ref: TM-T69360
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Rafabegron
CAS:244081-42-3
Rafabegron (TAK677) is a potent and selective β3 adrenergic receptor agonist for the study of …
Formula:
C21H23ClN2O4
Purity:
100%
Color and Shape:
Solid
Molecular weight:
402.87
Ref: TM-T34256
| 1mg | 270.00 € | ||
| 5mg | 663.00 € | ||
| 10mg | 917.00 € | ||
| 25mg | 1,380.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,550.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
AZD8797
CAS:911715-90-7
AZD8797 (KAND567) is a CX3CR1 antagonist with potential protective effects against neuronal damage and prevents …
Formula:
C19H25N5OS2
Purity:
98.73% - 99.68%
Color and Shape:
Solid
Molecular weight:
403.56
Ref: TM-T14384
| 1mg | 91.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 346.00 € | ||
| 25mg | 733.00 € | ||
| 50mg | 918.00 € | ||
| 100mg | 1,329.00 € | ||
| 1mL*10mM (DMSO) | 216.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Palmitoyl serinol
CAS:126127-31-9
Palmitoyl serinol (N-Palmitoyl serinol), an analog of the cannabinoid N-palmitoylethanolamine, stimulates an IL-4-mediated decrease in …
Formula:
C19H39NO3
Color and Shape:
Liquid
Molecular weight:
329.52
Ref: TM-T60957
| 5mg | 93.00 € | ||
| 10mg | 178.00 € | ||
| 50mg | 719.00 € | ||
| 100mg | 1,277.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
GSK1521498 free base (hydrochloride)
CAS:1007578-24-6
GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).
Formula:
C24H21ClF2N4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
438.9
Ref: TM-T11478
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
Taprizosin
CAS:210538-44-6
Taprizosin(UK-338003) is a selective and orally active α1-adrenoceptor antagonist for vasodilatation in the treatment of …
Formula:
C25H26N6O4S
Purity:
97.01% - 99.11%
Color and Shape:
Solid
Molecular weight:
506.58
Ref: TM-T28922
| 1mg | 355.00 € | ||
| 5mg | 832.00 € | ||
| 10mg | 1,169.00 € | ||
| 25mg | 1,787.00 € | ||
| 50mg | 2,410.00 € | ||
| 100mg | 3,176.00 € |
Estimated delivery in United States, on Monday 27 Jan 2025
