G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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MrgprX2 antagonist-8
CAS:2768216-96-0
MrgprX2 antagonist-8 is an MrgprX2 antagonist that can be used to study inflammatory diseases.
Formula:
C24H24ClF3N4O3S
Purity:
98.87%
Color and Shape:
Liquid
Molecular weight:
540.99
Ref: TM-T63812
| 1mg | 100.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 344.00 € | ||
| 25mg | 564.00 € | ||
| 50mg | 745.00 € | ||
| 100mg | 992.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
KUL-7211 racemate
CAS:911196-40-2
KUL 7211, a selective β-adrenoceptor agonist, exists as a racemate, referred to as KUL 7211 …
Formula:
C19H23NO5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
345.39
Ref: TM-T11786
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
A2AR-agonist-1
CAS:41552-95-8
A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).
Formula:
C20H22N6O4
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
410.43
Ref: TM-T10212
| 1mg | 94.00 € | ||
| 2mg | 131.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 277.00 € | ||
| 25mg | 441.00 € | ||
| 50mg | 630.00 € | ||
| 100mg | 847.00 € | ||
| 500mg | 1,653.00 € | ||
| 1mL*10mM (DMSO) | 217.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Laropiprant
CAS:571170-77-9
Laropiprant (MK-0524) is a potent and selective antagonist of prostaglandin D2 (PGD2) receptor (DP) such …
Formula:
C21H19ClFNO4S
Purity:
98.24% - 99.97%
Color and Shape:
Solid
Molecular weight:
435.9
Ref: TM-T15712
| 1mg | 37.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 110.00 € | ||
| 25mg | 214.00 € | ||
| 50mg | 328.00 € | ||
| 100mg | 469.00 € | ||
| 200mg | 640.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Foscarbidopa
CAS:1907685-81-7
Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
Formula:
C10H15N2O7P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
306.21
Ref: TM-T15339
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Ro 363
CAS:74513-77-2
RO 363: Potent β1-adrenoceptor agonist, boosts heart contractility, lowers diastolic pressure.
Formula:
C19H25NO6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
363.4
Ref: TM-T16769
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L-365260
CAS:118101-09-0
L-365260 is a nonpeptide gastrin and cerebral cholecystokinin receptor (CCK-B) antagonist used in the study …
Formula:
C24H22N4O2
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
398.46
Ref: TM-T22895
| 2mg | 293.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
LY2881835
CAS:1292290-38-0
LY2881835 is a potent and selective GPR40 agonist.
Formula:
C33H33NO3
Purity:
97.65% - 97.65%
Color and Shape:
Solid
Molecular weight:
491.62
Ref: TM-T27937
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
ReN-1869 hydrochloride
CAS:170149-76-5
ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.
Formula:
C24H28ClNO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
397.94
Ref: TM-T12703
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Bedoradrine
CAS:194785-19-8
Bedoradrine (MN-221) free base is a novel, highly selective β2-adrenoceptor agonist.Cost-effective and quality-assured.
Formula:
C24H32N2O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
428.52
Ref: TM-T70047
| 1mg | 724.00 € | ||
| 5mg | 1,477.00 € | ||
| 25mg | 2,556.00 € | ||
| 50mg | 3,139.00 € | ||
| 100mg | 4,272.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
PNU-177864 hydrochloride
CAS:1783978-03-9
PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor.
Formula:
C18H22ClF3N2O3S
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
438.89
Ref: TM-T12510
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 111.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L-902688
CAS:634193-54-7
L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).
Formula:
C21H27F2N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
419.47
Ref: TM-T15690
| 1mg | 503.00 € | ||
| 5mg | 2,238.00 € | ||
| 10mg | 3,955.00 € | ||
| 500µg | 266.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Rilapine
CAS:79781-95-6
Rilapine (Rilapinum) is an antipsychotic compound that shows high affinity for 5-HT6 receptors and can …
Formula:
C22H20ClN3
Purity:
99% - 99.66%
Color and Shape:
Solid
Molecular weight:
361.87
Ref: TM-T26085
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Cetrorelix Acetate
CAS:145672-81-7
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
Formula:
C70H92ClN17O14·xC2H4O2
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
1491.11
Ref: TM-T5520
| 1mg | 46.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 117.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 388.00 € | ||
| 100mg | 606.00 € | ||
| 1mL*10mM (DMSO) | 173.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
L 651896
CAS:99134-29-9
L 651896 is an inhibitor of 5-lipoxygenase.
Formula:
C18H18O3
Purity:
95.87% - 99.70%
Color and Shape:
Solid
Molecular weight:
282.33
Ref: TM-T24306
| 1mg | 311.00 € | ||
| 5mg | 747.00 € | ||
| 10mg | 1,059.00 € | ||
| 25mg | 1,549.00 € | ||
| 50mg | 2,127.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
EPAC 5376753
CAS:302826-61-5
EPAC 5376753 is an allosteric inhibitor of EPAC1 with an IC50 of 4 µM in …
Formula:
C15H8Cl2N2O3S
Purity:
90%
Color and Shape:
Solid
Molecular weight:
367.21
Ref: TM-T11212
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 152.00 € | ||
| 25mg | 296.00 € | ||
| 1mL*10mM (DMSO) | 111.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
Anpirtoline hydrochloride
CAS:99201-87-3
Anpirtoline hydrochloride (D-16949 hydrochloride) is a 5-HT1B receptor agonist and 5-HT3 receptor antagonist used in …
Formula:
C10H14Cl2N2S
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
265.20
Ref: TM-T22576
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 276.00 € | ||
| 50mg | 421.00 € | ||
| 100mg | 606.00 € | ||
| 500mg | 1,253.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
(S)-(+)-Niguldipine hydrochloride
CAS:113145-69-0
(S)-(+)-Niguldipine hydrochloride is a selective α1A-AR antagonist used in the study of depression and epilepsy.
Formula:
C36H40ClN3O6
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
646.17
Ref: TM-T23301
| 1mg | 82.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 249.00 € | ||
| 25mg | 586.00 € | ||
| 50mg | 1,021.00 € | ||
| 100mg | 1,371.00 € | ||
| 500mg | 2,732.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
![N-[(4-Aminophenyl)methyl]adenosine](https://static.cymitquimica.com/products/TM/thumb/T16166.jpg)
N-[(4-Aminophenyl)methyl]adenosine
CAS:95523-13-0
N-[(4-Aminophenyl)methyl]adenosine is an adenosine receptor inhibitor (Ki: 29 nM for Rat ecto-5′-Nucleotidase).
Formula:
C17H20N6O4
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
372.38
Ref: TM-T16166
| 1mg | 90.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 276.00 € | ||
| 25mg | 546.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,395.00 € | ||
| 1mL*10mM (DMSO) | 235.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
PF-03654764
CAS:935840-35-0
PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with …
Formula:
C20H28F2N2O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
350.45
Ref: TM-T61213
| 1mg | 305.00 € | ||
| 5mg | 736.00 € | ||
| 25mg | 1,483.00 € | ||
| 50mg | 2,009.00 € |
Estimated delivery in United States, on Tuesday 14 Jan 2025
