G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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CCX777
CAS:1226686-36-7
CCX777 is a partial agonist recruited to ACKR3 by β-arrestin-2 and is used in cancer …
Formula:
C31H43N7O3S
Purity:
98.73%
Color and Shape:
Solid
Molecular weight:
593.78
Ref: TM-T23866
| 1mg | 278.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Repinotan
CAS:144980-29-0
Repinotan (BAY x 3702 free base) is a 5-HT1A receptor agonist used in acute ischemic …
Formula:
C21H24N2O4S
Purity:
99%
Color and Shape:
Solid
Molecular weight:
400.49
Ref: TM-T61934
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
AZ12216052
CAS:1290628-31-7
AZ12216052 is a GRP8 antagonist with anxiolytic and anti-inflammatory activity and can be used to …
Formula:
C19H22BrNOS
Purity:
99.29%
Color and Shape:
Solid
Molecular weight:
392.35
Ref: TM-T26701
| 1mg | 56.00 € | ||
| 5mg | 118.00 € | ||
| 10mg | 183.00 € | ||
| 25mg | 321.00 € | ||
| 50mg | 476.00 € | ||
| 100mg | 678.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Levobunolol hydrochloride
CAS:27912-14-7
Levobunolol hydrochloride is a non-selective blocker of β-adrenergic receptor and can be used in studies …
Formula:
C17H26ClNO3
Purity:
100% - 98.49%
Color and Shape:
Solid
Molecular weight:
327.85
Ref: TM-T15742
| 1ml | 70.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 95.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Atrasentan hydrochloride
CAS:195733-43-8
Atrasentan hydrochloride (ABT-627 hydrochloride) is an antagonist of the endothelin receptor(IC50 = 55.1 μM for …
Formula:
C29H39ClN2O6
Purity:
98.64%
Color and Shape:
Solid
Molecular weight:
547.08
Ref: TM-TQ0270
| 1ml | 74.00 € | ||
| 2mg | 41.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 159.00 € | ||
| 50mg | To inquire |
Estimated delivery in United States, on Monday 25 Nov 2024
Aganepag
CAS:910562-18-4
Aganepag: Potent EP2 agonist, EC50 0.19 nM, inactive at EP4, used in wound healing and …
Formula:
C24H31NO4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
429.57
Ref: TM-T14139
| 25mg | 2,106.00 € | ||
| 50mg | 2,785.00 € | ||
| 100mg | 3,739.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Pancopride
CAS:121650-80-4
Pancopride(LAS 30451) is a novel, orally available, long-acting, selective 5-HT3 receptor antagonist that blocks nitrogen …
Formula:
C18H24ClN3O2
Purity:
93.64%
Color and Shape:
Solid
Molecular weight:
349.86
Ref: TM-T16433
| 1mg | 650.00 € | ||
| 5mg | 1,682.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
SARS-CoV-2-IN-57
CAS:1265624-68-7
SARS-CoV-2-IN-57 (compound (+)-R-26) is a potent inhibitor of SARS-CoV-2 with an IC50 of 80 nM …
Formula:
C23H37N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
371.56
Ref: TM-T79356
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
APNEA
CAS:89705-21-5
APNEA ((2R,3R,4S,5R)-2-[6-[2-(4-aminophenyl)ethylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol) is a non-selective agonist of adenosine A3 receptor.
Formula:
C18H22N6O4
Purity:
99.58%
Color and Shape:
Solid
Molecular weight:
386.41
Ref: TM-T12159
| 1ml | 34.00 € | ||
| 25mg | 50.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
KSK68
CAS:2566715-91-9
KSK68 is a sigma-1 and histamine H3 receptor antagonist with analgesic activity, inhibits H3 receptors …
Formula:
C23H28N2O2
Purity:
97.22%
Color and Shape:
Solid
Molecular weight:
364.48
Ref: TM-T79499
| 1mg | 74.00 € | ||
| 5mg | 159.00 € | ||
| 10mg | 224.00 € | ||
| 25mg | 372.00 € | ||
| 50mg | 558.00 € | ||
| 100mg | 796.00 € | ||
| 500mg | 2,210.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
KSK94
CAS:2566716-07-0
KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value …
Formula:
C25H26N4O
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
398.5
Ref: TM-T79500
| 1mg | 59.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 277.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 623.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Moprolol
CAS:5741-22-0
Moprolol ((±)-Moprolol) is a beta-adrenergic receptor antagonist utilized in research pertaining to essential hypertension [1] …
Formula:
C13H21NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
239.31
Ref: TM-T78567
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
CXCR4-IN-1
CAS:2304750-48-7
CXCR4-IN-1 (Example C5), with an IC50 of 20 nM, is a potent inhibitor of CXCR4, …
Formula:
C23H32N6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
392.54
Ref: TM-T79059
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
PSB-16133 sodium
CAS:2089035-40-3
PSB-16133 sodium is a selective P2Y purine receptor variant antagonist with an IC of 233 …
Formula:
C28H21N2NaO5S2
Purity:
98.08% - 99.36%
Color and Shape:
Solid
Molecular weight:
552.60
Ref: TM-T28463
| 1mg | 273.00 € | ||
| 2mg | 406.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 919.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,838.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
A-77636
CAS:778546-51-3
A-77636 is a potent, selective, and long-acting oral dopamine D1 receptor agonist with an effective …
Formula:
C20H27NO3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
329.43
Ref: TM-T78644
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
GPR81 agonist 1
CAS:1620992-67-7
GPR81 agonist 1 is a GPR81 agonist that improves glycaemic control in insulin-resistant mouse models …
Formula:
C22H30N4O2S2
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
446.63
Ref: TM-T62656
| 1mg | 127.00 € | ||
| 1ml | 276.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 521.00 € | ||
| 25mg | 974.00 € | ||
| 50mg | 1,474.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
AMX12006
CAS:2639775-01-0
AMX12006, a potent and selective EP4 antagonist, exhibits cytotoxic and antitumor activity, demonstrating oral activity …
Formula:
C26H22F3N3O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
481.47
Ref: TM-T78710
| 1mg | 141.00 € | ||
| 5mg | 601.00 € | ||
| 10mg | 1,063.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
5-HT2 antagonist 1
CAS:191592-09-3
5-HT2 antagonist 1 is a potent 5-HT2 receptor antagonist, has weak α1 adrenoceptor blocking activity.
Formula:
C22H29FN4O2
Purity:
99.25%
Color and Shape:
Solid
Molecular weight:
400.49
Ref: TM-T12597
| 1mg | 663.00 € | ||
| 1ml | 1,595.00 € | ||
| 5mg | 1,328.00 € | ||
| 10mg | 1,792.00 € | ||
| 25mg | 2,665.00 € | ||
| 50mg | 3,593.00 € | ||
| 100mg | 4,855.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Sarizotan HCl
CAS:195068-07-6
Sarizotan HCl (EMD 128130 HCl) is a 5-HT1A receptor and dopamine receptor agonist and an …
Formula:
C22H22ClFN2O
Purity:
96%
Color and Shape:
Solid
Molecular weight:
384.87
Ref: TM-T70044
| 1mg | 272.00 € | ||
| 2mg | 405.00 € | ||
| 5mg | 671.00 € | ||
| 10mg | 917.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,845.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
Fallypride
CAS:166173-78-0
Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.
Formula:
C20H29FN2O3
Purity:
100% - 99.17%
Color and Shape:
Solid
Molecular weight:
364.45
Ref: TM-T70302
| 1mg | 429.00 € | ||
| 5mg | 998.00 € | ||
| 10mg | 1,225.00 € | ||
| 25mg | 1,623.00 € | ||
| 50mg | 2,033.00 € | ||
| 100mg | 2,611.00 € |
Estimated delivery in United States, on Monday 25 Nov 2024
