G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Aplindore Fumarate
CAS:189681-71-8
Aplindore Fumarate (DAB-452), a selective dopamine D2/D3 partial agonist, is used in Parkinson's and schizophrenia …
Formula:
C22H22N2O7
Purity:
100%
Color and Shape:
Solid
Molecular weight:
426.42
Ref: TM-T30098
| 1mg | 274.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,421.00 € | ||
| 50mg | 1,839.00 € | ||
| 100mg | 2,601.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
VA-K-14 hydrochloride
CAS:1171341-19-7
VA-K-14 hydrochloride(VAK14 HCl) is a selective thyrotropin receptor (TSHR) antagonist (IC50= 12.3 μM) that inhibits …
Formula:
C18H16ClN3S
Purity:
98.01%
Color and Shape:
Solid
Molecular weight:
341.86
Ref: TM-T29087
| 1mg | 58.00 € | ||
| 5mg | 122.00 € | ||
| 10mg | 182.00 € | ||
| 25mg | 368.00 € | ||
| 50mg | 599.00 € | ||
| 100mg | 916.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
ML192
CAS:460331-61-7
ML192 (CID1434953) is a selective GPR55 ligand antagonist.
Formula:
C20H22N4O2S
Purity:
99.79%
Color and Shape:
Solid
Molecular weight:
382.48
Ref: TM-T33452
| 1mg | 50.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 297.00 € | ||
| 50mg | 427.00 € | ||
| 100mg | 602.00 € | ||
| 500mg | 1,198.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
SKF83959
CAS:80751-85-5
SKF83959: dopamine D1 partial agonist, Ki: D1(1.18 nM), D5(7.56 nM), D2(920 nM), D3(399 nM); improves …
Formula:
C18H20ClNO2
Purity:
98.45%
Color and Shape:
Liquid
Molecular weight:
317.81
Ref: TM-T60835
| 1mg | 52.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 353.00 € | ||
| 50mg | 522.00 € | ||
| 100mg | 741.00 € | ||
| 1mL*10mM (DMSO) | 113.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
A 61603
CAS:107756-30-9
Cixutumumab (IMC-A12) is a humanized IgG monoclonal antibody targeting the IGF1R with anticancer activity.
Formula:
C14H20BrN3O3S
Color and Shape:
Solid
Molecular weight:
390.3
Ref: TM-T21927
| 1mg | 86.00 € | ||
| 5mg | 237.00 € | ||
| 10mg | 329.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
SPD-473 citrate
CAS:161190-26-7
SPD-473 citrate is an inhibitior of serotonin/dopamine/norepinephrine reuptake.
Formula:
C23H31Cl2NO8S
Purity:
99.37%
Color and Shape:
Solid
Molecular weight:
552.47
Ref: TM-T13898
| 1mg | 230.00 € | ||
| 5mg | 575.00 € | ||
| 10mg | 806.00 € | ||
| 25mg | 1,290.00 € | ||
| 50mg | 1,735.00 € | ||
| 100mg | 2,347.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Clonidine
CAS:4205-90-7
Clonidine (Kapvay): central alpha-adrenergic agonist, antihypertensive, often combined, not tied to liver issues.
Formula:
C9H9Cl2N3
Purity:
99.44% - 99.88%
Color and Shape:
Crystals Solid
Molecular weight:
230.09
Ref: TM-T7045
| 50mg | 89.00 € | ||
| 100mg | 128.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
JNJ 10191584 maleate
CAS:869497-75-6
JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor …
Formula:
C17H19ClN4O5
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
394.81
Ref: TM-T22879
| 1mg | 53.00 € | ||
| 2mg | 81.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 130.00 € | ||
| 25mg | 278.00 € | ||
| 50mg | 403.00 € | ||
| 100mg | To inquire |
Estimated delivery in United States, on Wednesday 29 Jan 2025
L 674573
CAS:127481-29-2
L 674573 is an inhibitor of leukotriene biosynthesis.
Formula:
C28H27NO3S
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
457.58
Ref: TM-T24327
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 270.00 € | ||
| 1mL*10mM (DMSO) | 82.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
QS11
CAS:944328-88-5
QS11, a GTPase ARFGAP1, modulates ARF-GTP levels and synergizes with the Wnt/β-catenin signaling pathway to …
Formula:
C36H33N5O2
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
567.68
Ref: TM-T4022
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 220.00 € | ||
| 100mg | 331.00 € | ||
| 200mg | 453.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
FRG8701
CAS:108498-50-6
FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to …
Formula:
C22H30N2O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
418.55
Ref: TM-T11324
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
S 16924
CAS:734513-52-1
S 16924 is a 5-HT 1A agonist with potential anxiolytic effects and may be useful …
Formula:
C22H24FNO4
Purity:
98.23% - 99.45%
Color and Shape:
Solid
Molecular weight:
385.43
Ref: TM-T28638
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
A2AR-agonist-1
CAS:41552-95-8
A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).
Formula:
C20H22N6O4
Purity:
99.82%
Color and Shape:
Solid
Molecular weight:
410.43
Ref: TM-T10212
| 1mg | 94.00 € | ||
| 2mg | 131.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 277.00 € | ||
| 25mg | 441.00 € | ||
| 50mg | 630.00 € | ||
| 100mg | 847.00 € | ||
| 500mg | 1,653.00 € | ||
| 1mL*10mM (DMSO) | 217.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Foscarbidopa
CAS:1907685-81-7
Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.
Formula:
C10H15N2O7P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
306.21
Ref: TM-T15339
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
PNU-177864 hydrochloride
CAS:1783978-03-9
PNU-177864 hydrochloride is a potent, selective and orally active antagonist of dopamine D3 receptor.
Formula:
C18H22ClF3N2O3S
Purity:
99.20%
Color and Shape:
Solid
Molecular weight:
438.89
Ref: TM-T12510
| 5mg | 35.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 111.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
L-902688
CAS:634193-54-7
L-902688 is an orally active EP4 receptor agonist (Ki: 0.38 nM; EC50: 0.6 nM).
Formula:
C21H27F2N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
419.47
Ref: TM-T15690
| 1mg | 503.00 € | ||
| 5mg | 2,238.00 € | ||
| 10mg | 3,955.00 € | ||
| 500µg | 266.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Cetrorelix Acetate
CAS:145672-81-7
Cetrorelix Acetate is gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM.
Formula:
C70H92ClN17O14·xC2H4O2
Purity:
97.96%
Color and Shape:
Solid
Molecular weight:
1491.11
Ref: TM-T5520
| 1mg | 46.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 117.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 388.00 € | ||
| 100mg | 606.00 € | ||
| 1mL*10mM (DMSO) | 173.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Masupirdine free base
CAS:701205-60-9
Masupirdine free base (SUVN-502 free base) is a 5-HT6 receptor antagonist that can be used …
Formula:
C21H24BrN3O3S
Purity:
97.40% - 98.67%
Color and Shape:
Solid
Molecular weight:
478.4
Ref: TM-T11948
| 1mg | 274.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 1mL*10mM (DMSO) | 736.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
N 0861
CAS:141696-90-4
N 0861 is a selective adenosine A1 receptor antagonist that attenuates renal insufficiency during adenosine-controlled …
Formula:
C13H17N5
Purity:
99.81%
Color and Shape:
Liquid
Molecular weight:
243.31
Ref: TM-T70722
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
Undecylenoyl phenylalanine
CAS:175357-18-3
Undecylenoyl phenylalanine (Sepiwhite msh QD) is a novel depigmenting agent, which possibly acts as an …
Formula:
C20H29NO3
Purity:
≥98%
Color and Shape:
White To Pinkish Solid Powder
Molecular weight:
331.45
Ref: TM-T20501
| 5mg | 34.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 72.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 140.00 € | ||
| 200mg | 182.00 € | ||
| 1mL*10mM (DMSO) | 43.00 € |
Estimated delivery in United States, on Wednesday 29 Jan 2025
