G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Anti-inflammatory agent 49
CAS:851471-44-8
Compound SC9, an anti-inflammatory agent, serves as a potent and selective inhibitor of the Drp1-Fis1 …
Formula:
C21H22N8O3S
Purity:
99.62% - 99.74%
Color and Shape:
Solid
Molecular weight:
466.52
Ref: TM-T83057
| 1mg | 96.00 € | ||
| 5mg | 201.00 € | ||
| 10mg | 328.00 € | ||
| 25mg | 656.00 € | ||
| 50mg | 1,029.00 € | ||
| 100mg | 1,397.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ebrotidine
CAS:100981-43-9
Ebrotidine (FI3542) is a competitive H2-receptor antagonist with Ki of 127.5 nM. Ebrotidine has a …
Formula:
C14H17BrN6O2S3
Purity:
97.5%
Color and Shape:
Solid
Molecular weight:
477.42
Ref: TM-T15195
| 1ml | 71.00 € | ||
| 2mg | 44.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 94.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Abaperidone
CAS:183849-43-6
Abaperidone is an atypical antipsychotic, antagonizes 5-HT2A (IC50=6.2 nM) and D2 receptors (IC50=17 nM), reduces …
Formula:
C25H25FN2O5
Purity:
94.35%
Color and Shape:
Solid
Molecular weight:
452.47
Ref: TM-T14083
| 1mg | 326.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,053.00 € | ||
| 25mg | 1,477.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
DPI-3290
CAS:182417-73-8
DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 …
Formula:
C30H34FN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
487.61
Ref: TM-T15165
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
PSNCBAM-1
CAS:877202-74-9
PSNCBAM-1 (PSNCBAM 1) is a CB1 receptor negative allosteric modulator (EC50 = 0.1 μM) with …
Formula:
C22H21ClN4O
Purity:
98.18%
Color and Shape:
Solid
Molecular weight:
392.88
Ref: TM-T28468
| 1mg | 34.00 € | ||
| 1ml | 82.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 102.00 € | ||
| 25mg | 169.00 € | ||
| 50mg | 255.00 € | ||
| 100mg | 612.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Gestonorone Capronate
CAS:1253-28-7
Gestonorone Capronate is a progesterone used in benign prostatic hyperplasia and endometrial cancer studies.
Formula:
C26H38O4
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
414.58
Ref: TM-T13703
| 1mg | 143.00 € | ||
| 1ml | 360.00 € | ||
| 5mg | 312.00 € | ||
| 10mg | 462.00 € | ||
| 25mg | 736.00 € | ||
| 50mg | 1,054.00 € | ||
| 100mg | 1,411.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bunazosin Hydrochloride
CAS:52712-76-2
Bunazosin Hydrochloride (E 1015) is an alpha(1)-adrenoceptor antagonist used as a systemic antihypertensive and an …
Formula:
C19H28ClN5O3
Purity:
98.48%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T26923
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 211.00 € | ||
| 100mg | 383.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Adomeglivant
CAS:1488363-78-5
Adomeglivant (LY2409021) is a potent and selective glucagon receptor antagonist. Which is used in clinical …
Formula:
C32H36F3NO4
Purity:
99.97%
Color and Shape:
Solid
Molecular weight:
555.63
Ref: TM-T14130
| 1mg | 38.00 € | ||
| 1ml | 87.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 351.00 € | ||
| 100mg | 584.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
MRS 1754
CAS:264622-58-4
MRS 1754 is a selective antagonist radioligand for the A2B adenosine receptor. It has a …
Formula:
C26H26N6O4
Purity:
96.12% - 97.48%
Color and Shape:
Solid
Molecular weight:
486.52
Ref: TM-T16140
| 2mg | 37.00 € | ||
| 5mg | 56.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 177.00 € | ||
| 50mg | 272.00 € | ||
| 100mg | 411.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Dihydrexidine
CAS:123039-93-0
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 …
Formula:
C17H17NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
267.32
Ref: TM-T13463L
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GV150013
CAS:167355-22-8
GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
534.65
Ref: TM-T27503
| 1mg | 306.00 € | ||
| 1ml | 1,067.00 € | ||
| 5mg | 742.00 € | ||
| 10mg | 1,013.00 € | ||
| 25mg | 1,532.00 € | ||
| 50mg | 2,083.00 € | ||
| 100mg | 2,737.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AC-099 hydrochloride
CAS:849335-07-5
AC-099 hydrochloride is a full agonist of neuropeptide FF2 receptor NPFF2R and a partial agonist …
Formula:
C9H9Cl2F3N4
Purity:
99.86%
Color and Shape:
Solid
Molecular weight:
301.1
Ref: TM-T83212
| 1ml | 53.00 € | ||
| 5mg | 48.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 127.00 € | ||
| 100mg | 198.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GS-6201
CAS:752222-83-6
GS-6201 (CVT-6883) is a selective antagonist of adenosine A2B receptor.
Formula:
C21H21F3N6O2
Purity:
98.32% - 99.74%
Color and Shape:
Solid
Molecular weight:
446.43
Ref: TM-T15418
| 1mg | 43.00 € | ||
| 1ml | 115.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 307.00 € | ||
| 50mg | 485.00 € | ||
| 100mg | 705.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Lotiglipron
CAS:2401892-75-7
Lotiglipron (PF-07081532) is a GLP-1R agonist that lowers blood glucose and may be used in …
Formula:
C31H31ClN4O5
Purity:
98.3%
Color and Shape:
Solid
Molecular weight:
575.05
Ref: TM-T77781
| 1mg | 69.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 203.00 € | ||
| 25mg | 406.00 € | ||
| 50mg | 610.00 € | ||
| 100mg | 915.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
H3 receptor antagonist 1
CAS:935840-13-4
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor …
Formula:
C20H28F2N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
350.45
Ref: TM-T10911
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CB 65
CAS:913534-05-1
CB 65 is a high affinity and selective CB2 receptor agonist with Ki values of …
Formula:
C22H28ClN3O3
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
417.93
Ref: TM-T41230
| 1mg | 63.00 € | ||
| 5mg | 134.00 € | ||
| 10mg | 193.00 € | ||
| 25mg | 328.00 € | ||
| 50mg | 487.00 € | ||
| 100mg | 693.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CCG-63808
CAS:620113-73-7
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.
Formula:
C25H15FN4O2S
Purity:
90%
Color and Shape:
Solid
Molecular weight:
454.48
Ref: TM-T14898
| 1mg | 51.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 10 Dec 2024
WAY-639889
CAS:432506-24-6
WAY-639889 is a small molecule compound with selective and potent inhibitory effects on neuropeptide Y-5 …
Formula:
C25H27N5O
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
413.51
Ref: TM-T77783
| 1mg | 52.00 € | ||
| 5mg | 115.00 € | ||
| 10mg | 173.00 € | ||
| 25mg | 337.00 € | ||
| 50mg | 499.00 € | ||
| 100mg | 711.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GW 833972A
CAS:1092502-33-4
GW 833972A: selective CB2 agonist; reduces neural depolarization and citric acid cough in animals.
Formula:
C44H57NO8
Purity:
98%
Color and Shape:
Soild
Molecular weight:
727.93
Ref: TM-T64394
| 1mg | 327.00 € | ||
| 1ml | 933.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,321.00 € | ||
| 500mg | 4,568.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Deriglidole
CAS:122830-14-2
Deriglidole (SL 86-0715), an alpha2 receptor inhibitor, blocks colistin/Idazoxan but not prazosin/α2-adrenergic receptors.
Formula:
C16H21N3
Purity:
98.24% - 99.45%
Color and Shape:
Solid
Molecular weight:
255.36
Ref: TM-T10998
| 1mg | 427.00 € | ||
| 1ml | 748.00 € | ||
| 5mg | 991.00 € | ||
| 10mg | 1,327.00 € | ||
| 25mg | 1,950.00 € | ||
| 50mg | 2,396.00 € | ||
| 100mg | 3,158.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
