G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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AC-099 hydrochloride
CAS:849335-07-5
AC-099 hydrochloride is a full agonist of neuropeptide FF2 receptor NPFF2R and a partial agonist …
Formula:
C9H9Cl2F3N4
Purity:
99.86%
Color and Shape:
Liquid
Molecular weight:
301.1
Ref: TM-T83212
| 5mg | 48.00 € | ||
| 10mg | 71.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 127.00 € | ||
| 100mg | 198.00 € | ||
| 1mL*10mM (DMSO) | 53.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
Dihydrexidine
CAS:123039-93-0
Dihydrexidine is a full efficacy D1-like dopamine receptor (D1/D5) agonist (IC50: 10 nM for D1 …
Formula:
C17H17NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
267.32
Ref: TM-T13463L
| 25mg | 1,827.00 € | ||
| 50mg | 2,412.00 € | ||
| 100mg | 3,178.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
(S)-Bexicaserin
CAS:2035818-21-2
(S)-Bexcaserin (compound 2) serves as a 5-HT2C receptor agonist, presenting research possibilities in obesity and …
Formula:
C15H19F2N3O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
295.33
Ref: TM-T79838
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Feb 2025
NK3R-IN-1
CAS:2854331-14-7
NK3R-IN-1 (compound 16x), an orally active imidazolepiperazine derivative, acts as a Neurokinin Receptor NK3R inhibitor …
Formula:
C17H16FN5OS
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
357.41
Ref: TM-T78757
| 5mg | 1,290.00 € | ||
| 50mg | 2,618.00 € | ||
| 100mg | 3,484.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
DG-041
CAS:861238-35-9
DG-041: EP3 receptor antagonist, high affinity (IC50: 4.6 & 8.1 nM), inhibits PGE2 in platelets, …
Formula:
C23H15Cl4FN2O3S2
Purity:
97.25%
Color and Shape:
Solid
Molecular weight:
592.32
Ref: TM-T15108
| 1mg | 50.00 € | ||
| 2mg | 66.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 295.00 € | ||
| 50mg | 530.00 € | ||
| 100mg | 760.00 € | ||
| 500mg | 1,570.00 € | ||
| 1mL*10mM (DMSO) | 110.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
Fiduxosin
CAS:208993-54-8
Fiduxosin is a selective and potent α1-adrenoceptor antagonist with inhibitory effects on α1a-adrenoceptor, α1b-adrenoceptor and …
Formula:
C30H29N5O4S
Purity:
99.73%
Color and Shape:
Solid
Molecular weight:
555.65
Ref: TM-T11286
| 1mg | 650.00 € | ||
| 5mg | 1,678.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
Pentiapine
CAS:81382-51-6
Pentiapine (CGS 10746) is a novel inhibitor of dopamine release.
Formula:
C15H17N5S
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
299.39
Ref: TM-T12405
| 1mg | 469.00 € | ||
| 5mg | 725.00 € | ||
| 10mg | 1,171.00 € | ||
| 25mg | 1,628.00 € | ||
| 50mg | 2,176.00 € | ||
| 100mg | 2,953.00 € | ||
| 1mL*10mM (DMSO) | 932.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
H3 receptor antagonist 1
CAS:935840-13-4
H3 receptor antagonist 1 is used in the study of neurological diseases, histamine H3 receptor …
Formula:
C20H28F2N2O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
350.45
Ref: TM-T10911
| 25mg | 1,410.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
GV150013
CAS:167355-22-8
GV150013 is an antagonist of cholecystokinin-2 (CCK2) receptor.
Formula:
C33H34N4O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
534.65
Ref: TM-T27503
| 1mg | 182.00 € | ||
| 5mg | 443.00 € | ||
| 10mg | 604.00 € | ||
| 25mg | 915.00 € | ||
| 50mg | 1,229.00 € | ||
| 100mg | 1,617.00 € | ||
| 200mg | 2,189.00 € | ||
| 1mL*10mM (DMSO) | 627.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
Nolomirole HCl
CAS:138531-51-8
Nolomirole HCl (CHF 1035) is a novel selective dopamine agonist with oral activity and inhibitory …
Formula:
C19H28ClNO4
Purity:
100% - 99.12%
Color and Shape:
Solid
Molecular weight:
369.88
Ref: TM-T33711L
| 1mg | 493.00 € | ||
| 5mg | 1,093.00 € | ||
| 25mg | 1,683.00 € | ||
| 50mg | 2,224.00 € | ||
| 100mg | 2,877.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
Pentixafor
CAS:1341207-62-2
Pentixafor is a peptide that selectively targets the CXCR4 receptor and can be labeled with …
Formula:
C60H80N14O14
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
1221.36
Ref: TM-T79070
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Feb 2025
Xanthine amine congener
CAS:96865-92-8
Xanthine amine congener is an Adenosine receptor antagonist.
Formula:
C21H28N6O4
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
428.48
Ref: TM-T23535
| 10mg | 361.00 € | ||
| 50mg | 1,499.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
GPR120 Agonist 1
CAS:1628448-77-0
GPR120 Agonist 1 selectively activates human/mouse GPR120 with EC50 of 42/77 nM in HEK293 cells.
Formula:
C20H12ClF6NO3S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
495.82
Ref: TM-T11452
| 25mg | 1,683.00 € | ||
| 50mg | 2,219.00 € | ||
| 100mg | 2,891.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
Mu opioid receptor antagonist 7
CAS:2378397-30-7
Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid …
Formula:
C22H27ClN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
386.91
Ref: TM-T79431
| 25mg | 1,410.00 € | ||
| 50mg | 1,851.00 € | ||
| 100mg | 2,337.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
H4R antagonist 2
CAS:1148115-99-4
H4R Antagonist 2, a potent Furo[3,2-d]pyrimidine derivative, serves as a histamine H4 receptor antagonist and …
Formula:
C13H17N5O
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
259.31
Ref: TM-T79786
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Feb 2025
CGP-20712
CAS:137888-49-4
CGP-20712 is a selective β 1-adrenoceptor antagonist with an IC50 of 0.7 nM.
Formula:
C23H25F3N4O5
Purity:
100% - 99.40%
Color and Shape:
Solid
Molecular weight:
494.46
Ref: TM-T30846
| 1mg | 327.00 € | ||
| 5mg | 774.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,481.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,322.00 € | ||
| 500mg | 4,577.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
5-HT3-In-1
CAS:186348-68-5
5-HT3-In-1 (compound example 8) exhabits with 5-HT3 inhibition activity.
Formula:
C16H21ClN4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
352.82
Ref: TM-T10006
| 25mg | 1,827.00 € | ||
| 50mg | 2,404.00 € | ||
| 100mg | 3,168.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
CCG-63808
CAS:620113-73-7
CCG-63808 is a reversible inhibitor of regulator of G-protein signaling (RGS) proteins.
Formula:
C25H15FN4O2S
Purity:
90%
Color and Shape:
Solid
Molecular weight:
454.48
Ref: TM-T14898
| 1mg | 51.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 137.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Feb 2025
Wf-516
CAS:310392-94-0
Wf-516 is a 5-HT reuptake inhibitor (Kis: 5 nM and 40 nM for 5-HT1A receptor …
Formula:
C25H25Cl2N3O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
502.39
Ref: TM-T13339
| 25mg | 1,688.00 € | ||
| 50mg | 2,225.00 € | ||
| 100mg | 2,897.00 € |
Estimated delivery in United States, on Friday 7 Feb 2025
5-HT2 agonist-1
CAS:2708279-78-9
Compound 24, a 5-HT2 agonist-1, selectively activates 5-HT2A, 5-HT2B, and 5-HT2C receptors with IC50 values …
Formula:
C19H23ClN2O2
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
346.85
Ref: TM-T79804
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Friday 7 Feb 2025
