G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Timonacic
CAS:444-27-9
Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.
Formula:
C4H7NO2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
133.17
Ref: TM-T0221
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Clomipramine hydrochloride
CAS:17321-77-6
Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the …
Formula:
C19H23ClN2·HCl
Purity:
99.07% - 99.47%
Color and Shape:
White To Slightly Yellow Crystalline Powder
Molecular weight:
351.31
Ref: TM-T0255
| 1g | 62.00 € | ||
| 200mg | 35.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
GSK256073
CAS:862892-90-8
GSK256073 is an orally active GPR109A agonist.
Formula:
C10H13ClN4O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
256.69
Ref: TM-T15432
| 1mg | 73.00 € | ||
| 2mg | 97.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 439.00 € | ||
| 50mg | 647.00 € | ||
| 100mg | 920.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Ziprasidone hydrochloride
CAS:122883-93-6
Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows …
Formula:
C21H22CL2N4OS
Purity:
98.37% - 99.34%
Color and Shape:
Solid
Molecular weight:
449.4
Ref: TM-T0031L
| 5mg | 44.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 133.00 € | ||
| 100mg | 166.00 € | ||
| 500mg | 398.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Carbinoxamine Maleate Salt
CAS:3505-38-2
Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and …
Formula:
C20H23ClN2O5
Purity:
99.81%
Color and Shape:
Off-White Solid
Molecular weight:
406.86
Ref: TM-T2222
| 25mg | 42.00 € | ||
| 50mg | 55.00 € | ||
| 100mg | 72.00 € | ||
| 200mg | 96.00 € | ||
| 500mg | 183.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Promazine hydrochloride
CAS:53-60-1
Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.
Formula:
C17H21ClN2S
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
320.88
Ref: TM-T0766
| 500mg | 55.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Ursodeoxycholic acid
CAS:128-13-2
Ursodeoxycholic acid (UDCA) can be used to dissolve gallstones and reduce cholesterol absorption.
Formula:
C24H40O4
Purity:
99.74% - ≥95%
Color and Shape:
White - Almost White Solid Powder
Molecular weight:
392.57
Ref: TM-T0700
| 1g | 35.00 € | ||
| 5g | 55.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Pizotifen
CAS:15574-96-6
Pizotifen is a serotonin antagonist with mild anticholinergic effects, used in migraine prevention. Not available …
Formula:
C19H21NS
Purity:
99.91%
Color and Shape:
Solid
Molecular weight:
295.44
Ref: TM-T1442
| 50mg | 43.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 124.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
N6-Cyclohexyladenosine
CAS:36396-99-3
N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.
Formula:
C16H23N5O4
Purity:
99.84% - 99.98%
Color and Shape:
Solid
Molecular weight:
349.38
Ref: TM-T12160
| 10mg | 34.00 € | ||
| 25mg | 62.00 € | ||
| 50mg | 104.00 € | ||
| 100mg | 156.00 € | ||
| 200mg | 220.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
MRS-1706
CAS:264622-53-9
MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.
Formula:
C27H29N5O5
Purity:
97.95%
Color and Shape:
Solid
Molecular weight:
503.55
Ref: TM-T16136
| 1mg | 37.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 472.00 € | ||
| 100mg | 687.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Alverine citrate
CAS:5560-59-8
Alverine citrate (NSC 35459) is utilized in functional gastrointestinal disorders.
Formula:
C26H35NO7
Purity:
100% - 99.83%
Color and Shape:
Coa
Molecular weight:
473.57
Ref: TM-T0428
| 1g | 81.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Atenolol
CAS:29122-68-7
Atenolol (Tenormin) is a selective β1 receptor antagonist.
Formula:
C14H22N2O3
Purity:
99.07%
Color and Shape:
White Crystalline Powder Solid
Molecular weight:
266.3361
Ref: TM-T0007
| 1ml | 54.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Metipranolol
CAS:22664-55-7
Metipranolol (Betamann) is a type of β- Adrenergic receptors( β- A potent antagonist of adrenergic …
Formula:
C17H27NO4
Purity:
98.54%
Color and Shape:
Solid
Molecular weight:
309.4
Ref: TM-T8899
| 5mg | 51.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 296.00 € | ||
| 100mg | 480.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Vincamine
CAS:1617-90-9
Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain …
Formula:
C21H26N2O3
Purity:
99.52%
Color and Shape:
White To Almost White Fine Crystalline Powder
Molecular weight:
354.44
Ref: TM-T1286
| 1g | 62.00 € | ||
| 500mg | 48.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Rimonabant hydrochloride
CAS:158681-13-1
Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。
Formula:
C22H22Cl4N4O
Purity:
100% - 99.5%
Color and Shape:
Off-White To White Crystalline Powder
Molecular weight:
500.25
Ref: TM-T1519
| 5mg | 46.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 116.00 € | ||
| 50mg | 207.00 € | ||
| 100mg | 310.00 € | ||
| 500mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 74.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Naphazoline hydrochloride
CAS:550-99-2
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
Formula:
C14H15ClN2
Purity:
97.6%
Color and Shape:
White Crystalline Powder White Crystalline Powder
Molecular weight:
246.74
Ref: TM-T0446
| 1g | 34.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Citalopram hydrobromide
CAS:59729-32-7
Citalopram hydrobromide (XU-62-320) , a selective serotonin reuptake inhibitor (SSRI), selectively inhibits the CNS neuronal …
Formula:
C20H22BrFN2O
Purity:
99.35%
Color and Shape:
White Crystalline Powder
Molecular weight:
405.304
Ref: TM-T1483
| 10mg | 48.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 89.00 € | ||
| 100mg | 110.00 € | ||
| 200mg | 155.00 € | ||
| 500mg | 246.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Zolmitriptan
CAS:139264-17-8
Zolmitriptan targets 5-HT 1B/1D receptors, constricts cranial vessels, inhibits pain signals, and stops pro-inflammatory neuropeptides, …
Formula:
C16H21N3O2
Purity:
98.8% - 99.91%
Color and Shape:
White Or Kind Of White Powder
Molecular weight:
287.36
Ref: TM-T1092
| 10mg | 58.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 141.00 € | ||
| 100mg | 216.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Anamorelin
CAS:249921-19-5
Anamorelin (ONO-7643) is a novel ghrelin receptor agonist (EC50: 0.74 nM in the FLIPR assay).
Formula:
C31H42N6O3
Purity:
99.35% - 99.88%
Color and Shape:
Solid
Molecular weight:
546.7
Ref: TM-T10319
| 5mg | 60.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 127.00 € | ||
| 50mg | 177.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
Tripelennamine hydrochloride
CAS:154-69-8
Tripelennamine hydrochloride (Pyribenzamine hydrochloride) is a histamine H1 antagonist with low sedative action but frequent …
Formula:
C16H21N3·HCl
Purity:
100% - 100%
Color and Shape:
White Solid
Molecular weight:
291.82
Ref: TM-T1269
| 1g | 139.00 € | ||
| 100mg | 37.00 € | ||
| 500mg | 97.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 4 Mar 2025
