G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
Read more
Timonacic
CAS:444-27-9
Timonacic (Thioproline) has been used in trials studying the treatment of HIV Infections.
Formula:
C4H7NO2S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
133.17
Ref: TM-T0221
| 1ml | 57.00 € | ||
| 200mg | 34.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Clomipramine hydrochloride
CAS:17321-77-6
Clomipramine HCl (Anafranil) is a serotonin-inhibiting tricyclic antidepressant, well-absorbed and metabolized to desmethylclomipramine in the …
Formula:
C19H23ClN2·HCl
Purity:
99.07% - 99.47%
Color and Shape:
White To Slightly Yellow Crystalline Powder
Molecular weight:
351.31
Ref: TM-T0255
| 25mg | 43.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 72.00 € | ||
| 500mg | 94.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Carbinoxamine Maleate Salt
CAS:3505-38-2
Carbinoxamine Maleate Salt (Lergefin) is an ethanolamine class of H1 antihistamines with mild antimuscarinic and …
Formula:
C20H23ClN2O5
Purity:
99.81%
Color and Shape:
Off-White Solid
Molecular weight:
406.86
Ref: TM-T2222
| 1g | 160.00 € | ||
| 1ml | 34.00 € | ||
| 50mg | 34.00 € | ||
| 100mg | 45.00 € | ||
| 200mg | 62.00 € | ||
| 500mg | 110.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Diphenylpyraline hydrochloride
CAS:132-18-3
Diphenylpyraline hydrochloride treats Parkinsonism. It's an antihistamine with anticholinergic properties and inhibits dopamine reuptake.
Formula:
C19H23NO·HCl
Purity:
99.22%
Color and Shape:
Solid
Molecular weight:
317.85
Ref: TM-T0059
| 1g | 52.00 € | ||
| 1ml | 49.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Phenothiazine
CAS:92-84-2
Phenothiazine (ENT 38) is a class of agents exhibiting antiemetic, antipsychotic, antihistaminic, and anticholinergic activities.
Formula:
C12H9NS
Purity:
99.94%
Color and Shape:
Yellow Solid Pellets
Molecular weight:
199.27
Ref: TM-T0776
| 1ml | 51.00 € | ||
| 500mg | 49.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
KGA-2727
CAS:666842-36-0
KGA-2727: potent, selective SGLT1 inhibitor (human Ki 97.4 nM, rat 43.5 nM), with high selectivity …
Formula:
C26H40N4O8
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
536.62
Ref: TM-T15656
| 1mg | 84.00 € | ||
| 1ml | 182.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 264.00 € | ||
| 25mg | 434.00 € | ||
| 50mg | 595.00 € | ||
| 100mg | 815.00 € | ||
| 200mg | 1,092.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Isoxsuprine hydrochloride
CAS:579-56-6
Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular …
Formula:
C18H24ClNO3
Purity:
99.31%
Color and Shape:
Crystals From Water Solid
Molecular weight:
337.84
Ref: TM-T0324
| 1ml | 60.00 € | ||
| 100mg | 41.00 € | ||
| 200mg | 54.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Granisetron hydrochloride
CAS:107007-99-8
Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used …
Formula:
C18H25ClN4O
Purity:
99.88% - 99.94%
Color and Shape:
White To Off-White Crystalline Solid
Molecular weight:
348.87
Ref: TM-T1042
| 1ml | 89.00 € | ||
| 10mg | 38.00 € | ||
| 25mg | 55.00 € | ||
| 50mg | 80.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 176.00 € | ||
| 500mg | 298.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Haloperidol
CAS:52-86-8
Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve …
Formula:
C21H23ClFNO2
Purity:
99.69% - 99.76%
Color and Shape:
Crystals Solid
Molecular weight:
375.86
Ref: TM-T0025
| 1ml | 55.00 € | ||
| 25mg | 40.00 € | ||
| 50mg | 52.00 € | ||
| 100mg | 59.00 € | ||
| 200mg | 75.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Acetophenazine dimaleate
CAS:5714-00-1
Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the …
Formula:
C31H37N3O10S
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
643.71
Ref: TM-T10232
| 1ml | 87.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 125.00 € | ||
| 50mg | 181.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Naphazoline hydrochloride
CAS:550-99-2
Naphazoline hydrochloride (Naphazoline HCl) is an adrenergic vasoconstrictor agent used as a decongestant.
Formula:
C14H15ClN2
Purity:
97.6%
Color and Shape:
White Crystalline Powder White Crystalline Powder
Molecular weight:
246.74
Ref: TM-T0446
| 1g | 34.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Nicergoline
CAS:27848-84-6
Nicergoline (Nicergolinum) is an ergot derivative used to treat senile dementia and other disorders with …
Formula:
C24H26BrN3O3
Purity:
100% - 99.53%
Color and Shape:
Solid
Molecular weight:
484.39
Ref: TM-T1132
| 1ml | 34.00 € | ||
| 10mg | 34.00 € | ||
| 25mg | 43.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 68.00 € | ||
| 500mg | 141.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Ticagrelor
CAS:274693-27-5
Ticagrelor (AR-C 126532XX), produced by AstraZeneca, is an inhibitor of platelet aggregation.
Formula:
C23H28F2N6O4S
Purity:
100%
Color and Shape:
Solid
Molecular weight:
522.57
Ref: TM-T0179
| 1g | 356.00 € | ||
| 1ml | 59.00 € | ||
| 10mg | 47.00 € | ||
| 25mg | 65.00 € | ||
| 50mg | 80.00 € | ||
| 100mg | 107.00 € | ||
| 200mg | 151.00 € | ||
| 500mg | 240.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
JNJ-39758979
CAS:1046447-90-8
JNJ-39758979: selective H4 receptor antagonist, Kis 12.5/5.3/25 nM (human/mouse/monkey), blocks histamine cAMP inhibition (pA2 7.9).
Formula:
C11H19N5
Purity:
98.00% - 98.3%
Color and Shape:
Solid
Molecular weight:
221.3
Ref: TM-T11723L
| 1mg | 45.00 € | ||
| 1ml | 101.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 244.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 521.00 € | ||
| 200mg | 707.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Centanafadine hydrochloride
CAS:923981-14-0
Centanafadine HCl is a NE/DA reuptake inhibitor, also affects serotonin (IC50: NE 6 nM, DA …
Formula:
C15H16ClN
Purity:
99.66%
Color and Shape:
Solid
Molecular weight:
245.75
Ref: TM-T10758L
| 1mg | 59.00 € | ||
| 1ml | 140.00 € | ||
| 5mg | 123.00 € | ||
| 10mg | 198.00 € | ||
| 25mg | 399.00 € | ||
| 50mg | 639.00 € | ||
| 100mg | 1,003.00 € | ||
| 200mg | 1,346.00 € | ||
| 500mg | 2,006.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
BP 897 hydrochloride
CAS:314776-92-6
BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low …
Formula:
C26H32ClN3O2
Purity:
99.42%
Color and Shape:
Solid
Molecular weight:
454
Ref: TM-T14767
| 1mg | 36.00 € | ||
| 1ml | 87.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 109.00 € | ||
| 25mg | 212.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 553.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Aniracetam
CAS:72432-10-1
Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and …
Formula:
C12H13NO3
Purity:
99.8%
Color and Shape:
White Crystalline Or Crystalline Powde
Molecular weight:
219.24
Ref: TM-T0333
| 1g | 51.00 € | ||
| 1ml | 34.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
AMG 487
CAS:473719-41-4
AMG 487: potent CXCR3 antagonist, blocks CXCL10/CXCL11 binding, IC50s: 8.0/8.2 nM.
Formula:
C32H28F3N5O4
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
603.59
Ref: TM-T10297L
| 1mg | 52.00 € | ||
| 1ml | 153.00 € | ||
| 2mg | 75.00 € | ||
| 5mg | 113.00 € | ||
| 10mg | 161.00 € | ||
| 25mg | 262.00 € | ||
| 50mg | 391.00 € | ||
| 100mg | 577.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Chlorprothixene hydrochloride
CAS:6469-93-8
Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.
Formula:
C18H18ClNS·HCl
Purity:
99.16%
Color and Shape:
White Powder
Molecular weight:
352.32
Ref: TM-T0074L
| 1ml | 47.00 € | ||
| 100mg | 37.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
Domperidone
CAS:57808-66-9
Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.
Formula:
C22H24ClN5O2
Purity:
98% - 99.73%
Color and Shape:
Solid
Molecular weight:
425.91
Ref: TM-T0082
| 1ml | 55.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 63.00 € | ||
| 200mg | 93.00 € | ||
| 500mg | 149.00 € |
Estimated delivery in United States, on Friday 4 Oct 2024
