G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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SEP-363856 hydrochloride
CAS:1310422-41-3
SEP-363856 hydrochloride is an oral, CNS-active psychotropic for schizophrenia with a non-D2/5-HT2A mechanism.
Formula:
C9H14ClNOS
Purity:
99.86% - 99.99%
Color and Shape:
Solid
Molecular weight:
219.73
Ref: TM-T12899L
| 1mg | 70.00 € | ||
| 2mg | 92.00 € | ||
| 5mg | 154.00 € | ||
| 10mg | 243.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 628.00 € | ||
| 100mg | 938.00 € | ||
| 500mg | 1,882.00 € | ||
| 1mL*10mM (DMSO) | 169.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Venlafaxine hydrochloride
CAS:99300-78-4
Venlafaxine HCl, a cyclohexanol phenethylamine, acts as an SNRI antidepressant.
Formula:
C17H28ClNO2
Purity:
99.86%
Color and Shape:
White Crystalline Powder
Molecular weight:
313.863
Ref: TM-T0472
| 5mg | 38.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 79.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 164.00 € | ||
| 500mg | 264.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Ondansetron hydrochloride dihydrate
CAS:103639-04-9
Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported …
Formula:
C18H19N3O·HCl·2H2O
Purity:
99.92%
Color and Shape:
White Crystal Powder
Molecular weight:
365.86
Ref: TM-T1478
| 25mg | 43.00 € | ||
| 50mg | 50.00 € | ||
| 100mg | 60.00 € | ||
| 200mg | 74.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
(R)-Elagolix
CAS:834153-87-6
(R)-Elagolix (NBI-56418) is an orally active, highly selective, short-term potent antagonist of the non-peptide gonadotropin-releasing …
Formula:
C32H30F5N3O5
Purity:
97.63%
Color and Shape:
Solid
Molecular weight:
631.59
Ref: TM-T11174
| 1mg | 38.00 € | ||
| 2mg | 49.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 188.00 € | ||
| 50mg | 329.00 € | ||
| 100mg | 487.00 € | ||
| 200mg | 695.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Salmeterol
CAS:89365-50-4
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
Formula:
C25H37NO4
Purity:
99.87% - 99.9%
Color and Shape:
Solid
Molecular weight:
415.57
Ref: TM-T12829
| 5mg | 55.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 154.00 € | ||
| 50mg | 274.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Loxapine succinate
CAS:27833-64-3
Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.
Formula:
C22H24ClN3O5
Purity:
99.92%
Color and Shape:
White To Of-White Solid
Molecular weight:
445.9
Ref: TM-T1412
| 50mg | 39.00 € | ||
| 100mg | 51.00 € | ||
| 200mg | 84.00 € | ||
| 500mg | 164.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Tetrahydrozoline
CAS:84-22-0
Tetrahydrozoline (Tetryzoline) is an alpha-adrenergic agonist that causes vasoconstriction and is widely used in the …
Formula:
C13H16N2
Purity:
97.85% - 99.77%
Color and Shape:
Solid
Molecular weight:
200.28
Ref: TM-T0397
| 50mg | 39.00 € | ||
| 100mg | 52.00 € | ||
| 500mg | 127.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Reparixin L-lysine salt
CAS:266359-93-7
Reparixin L-lysine salt (Repertaxin L-lysine salt) is an allosteric chemokine receptor 1/2 (CXCR1/2) activation inhibitor.
Formula:
C20H35N3O5S
Purity:
99%
Color and Shape:
Solid
Molecular weight:
429.57
Ref: TM-T12705
| 5mg | 47.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Sulpiride
CAS:15676-16-1
Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as …
Formula:
C15H23N3O4S
Purity:
99.94%
Color and Shape:
White Crystalline Powder
Molecular weight:
341.43
Ref: TM-T1201
| 50mg | 43.00 € | ||
| 100mg | 55.00 € | ||
| 200mg | 70.00 € | ||
| 500mg | 97.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Evatanepag
CAS:223488-57-1
Evatanepag (CP-533536) is a selective EP2 agonist for bone formation with 0.3 nM EC50, promoting …
Formula:
C25H28N2O5S
Purity:
97.09%
Color and Shape:
Solid
Molecular weight:
468.57
Ref: TM-T15259
| 1mg | 70.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 432.00 € | ||
| 50mg | 620.00 € | ||
| 100mg | 847.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
GR 103691
CAS:162408-66-4
GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).
Formula:
C30H35N3O3
Purity:
98.94% - 99.29%
Color and Shape:
Solid
Molecular weight:
485.62
Ref: TM-T11463
| 2mg | 46.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 197.00 € | ||
| 50mg | 311.00 € | ||
| 100mg | 505.00 € | ||
| 500mg | 1,121.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Droperidol
CAS:548-73-2
Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as …
Formula:
C22H22FN3O2
Purity:
97.16% - 98%
Color and Shape:
Solid
Molecular weight:
379.43
Ref: TM-T0990
| 100mg | 47.00 € | ||
| 200mg | 60.00 € | ||
| 500mg | 89.00 € | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Famotidine
CAS:76824-35-6
Famotidine, a histamine H2-blocker, curbs gastric acid production, lowering volume and acidity.
Formula:
C8H15N7O2S3
Purity:
98.93% - 99.75%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
337.45
Ref: TM-T1627
| 2g | 55.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Degarelix acetate(214766-78-6 free base)
CAS:934016-19-0
Degarelix acetate is a competitive and reversible antagonist of gonadotropin-releasing hormone receptor (GnRHR) .
Formula:
C84H107ClN18O18
Purity:
98.66%
Color and Shape:
Liquid
Molecular weight:
1692.34
Ref: TM-T10988L
| 1mg | 77.00 € | ||
| 2mg | 99.00 € | ||
| 5mg | 165.00 € | ||
| 10mg | 266.00 € | ||
| 25mg | 477.00 € | ||
| 50mg | 695.00 € | ||
| 100mg | 938.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
HJC0197
CAS:1383539-73-8
HJC0197 is a selective Epac antagonist; blocks cAMP-induced activation with IC50=5.9 μM for Epac2.
Formula:
C19H21N3OS
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
339.45
Ref: TM-T15485
| 2mg | 38.00 € | ||
| 5mg | 54.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 135.00 € | ||
| 50mg | 188.00 € | ||
| 100mg | 283.00 € | ||
| 200mg | 426.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Balovaptan
CAS:1228088-30-9
Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism …
Formula:
C22H24ClN5O
Purity:
99.34%
Color and Shape:
Solid
Molecular weight:
409.91
Ref: TM-T14494
| 5mg | 66.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 303.00 € | ||
| 100mg | 472.00 € | ||
| 1mL*10mM (DMSO) | 73.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Hydroxyzine Pamoate
CAS:10246-75-0
Hydroxyzine Pamoate (Bobsule) is a histamine H1 receptor antagonist that is effective in the treatment …
Formula:
C44H43ClN2O8
Purity:
99.49%
Color and Shape:
Solid
Molecular weight:
763.27
Ref: TM-T0053
| 10mg | 35.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 131.00 € | ||
| 200mg | 170.00 € | ||
| 500mg | 283.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Acebutolol hydrochloride
CAS:34381-68-5
Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.
Formula:
C18H29ClN2O4
Purity:
100% - 99.92%
Color and Shape:
White Or Slightly Off-White Crystalline Powder Solid
Molecular weight:
372.89
Ref: TM-T1012
| 50mg | 49.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 66.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Fenspiride hydrochloride
CAS:5053-08-7
Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.
Formula:
C15H20N2O2·HCl
Purity:
99.64% - 99.78%
Color and Shape:
Solid
Molecular weight:
296.79
Ref: TM-T0383
| 50mg | 35.00 € | ||
| 100mg | 48.00 € | ||
| 500mg | 94.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
Mianserin hydrochloride
CAS:21535-47-7
Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce …
Formula:
C18H21ClN2
Purity:
99.63% - 99.82%
Color and Shape:
White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film Coated
Molecular weight:
300.83
Ref: TM-T0783
| 1g | 157.00 € | ||
| 50mg | 35.00 € | ||
| 100mg | 42.00 € | ||
| 500mg | 106.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 28 Mar 2025
