G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Levocetirizine
CAS:130018-77-8
Levocetirizine is a Histamine-1 Receptor Antagonist. The mechanism of action of levocetirizine is as a …
Formula:
C21H25ClN2O3
Purity:
98% - 99.9%
Color and Shape:
White Powder
Molecular weight:
388.89
Ref: TM-T1469
| 5mg | 38.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 94.00 € | ||
| 100mg | 169.00 € | ||
| 200mg | 253.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Phentolamine mesylate
CAS:65-28-1
Phentolamine mesylate: nonselective alpha-blocker for hypertension, pheochromocytoma, Raynaud's, frostbite, impotence, and vascular issues.
Formula:
C17H19N3O·CH4O3S
Purity:
99.77% - 99.9%
Color and Shape:
By The Metabolic Processes Of Bacillus Subtilis And Licheniformis
Molecular weight:
377.46
Ref: TM-T1275
| 100mg | 60.00 € | ||
| 200mg | 78.00 € | ||
| 500mg | 152.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Alosetron hydrochloride
CAS:122852-69-1
Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin …
Formula:
C17H19ClN4O
Purity:
100%
Color and Shape:
Off-White Powder
Molecular weight:
330.81
Ref: TM-T2525
| 10mg | 36.00 € | ||
| 25mg | 76.00 € | ||
| 50mg | 110.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 256.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Clonidine hydrochloride
CAS:4205-91-8
Clonidine hydrochloride (Catapres) is a centrally active α-adrenergic agonist used predominantly as an antihypertensive agent.
Formula:
C9H10Cl3N3
Purity:
100% - 99.99%
Color and Shape:
Solid
Molecular weight:
266.55
Ref: TM-T1247
| 50mg | 45.00 € | ||
| 100mg | 58.00 € | ||
| 200mg | 72.00 € | ||
| 500mg | 138.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Xylometazoline hydrochloride
CAS:1218-35-5
Xylometazoline hydrochloride (Xylometazoline HCl) is an α-adrenoceptor agonist usually used as nasal decongestant.
Formula:
C16H24N2·HCl
Purity:
100% - 99.83%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
280.84
Ref: TM-T0042
| 1g | 36.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LY2940094
CAS:1307245-86-8
LY2940094 (LY-2940094) decreases ethanol self-administration in animal models.
Formula:
C22H23ClF2N4O2S
Purity:
99.40%
Color and Shape:
Solid
Molecular weight:
480.96
Ref: TM-T15799
| 1mg | 80.00 € | ||
| 2mg | 105.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 270.00 € | ||
| 25mg | 533.00 € | ||
| 50mg | 764.00 € | ||
| 100mg | 1,054.00 € | ||
| 1mL*10mM (DMSO) | 179.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Acebutolol hydrochloride
CAS:34381-68-5
Acebutolol HCl: cardioselective beta-blocker, minimal bronchial impact, intrinsic sympathomimetic, treats hypertension & ventricular arrhythmias.
Formula:
C18H29ClN2O4
Purity:
100% - 100%
Color and Shape:
White Or Slightly Off-White Crystalline Powder Solid
Molecular weight:
372.89
Ref: TM-T1012
| 50mg | 49.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 66.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Desipramine hydrochloride
CAS:58-28-6
Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of …
Formula:
C18H23ClN2
Purity:
99.58% - 99.94%
Color and Shape:
White To Off-White Powder
Molecular weight:
302.842
Ref: TM-T0991
| 50mg | 41.00 € | ||
| 100mg | 52.00 € | ||
| 200mg | 66.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Isoxsuprine hydrochloride
CAS:579-56-6
Isoxsuprine hydrochloride (Isolait) is a beta-adrenergic agonist that causes direct relaxation of uterine and vascular …
Formula:
C18H24ClNO3
Purity:
99.31%
Color and Shape:
Crystals From Water Solid
Molecular weight:
337.84
Ref: TM-T0324
| 200mg | 35.00 € | ||
| 500mg | 51.00 € | ||
| 1mL*10mM (DMSO) | 39.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Moxisylyte hydrochloride
CAS:964-52-3
Moxisylyte hydrochloride (Thymoxamine hydrochloride) is an alpha-adrenergic blocking agent that is used in Raynaud's disease.
Formula:
C16H26ClNO3
Purity:
99.93% - ≥95%
Color and Shape:
Solid
Molecular weight:
315.84
Ref: TM-T0394
| 50mg | 42.00 € | ||
| 100mg | 54.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Fenspiride hydrochloride
CAS:5053-08-7
Fenspiride HCl treats respiratory diseases including asthma and ENT inflammation in Russia.
Formula:
C15H20N2O2·HCl
Purity:
99.18% - 99.78%
Color and Shape:
Solid
Molecular weight:
296.79
Ref: TM-T0383
| 50mg | 35.00 € | ||
| 100mg | 47.00 € | ||
| 500mg | 91.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Naftopidil
CAS:57149-07-2
Naftopidil (KT-611) (INN, marketed under the brand name Flivas), an antihypertensive medicine, is used as …
Formula:
C24H28N2O3
Purity:
99.4% - 99.97%
Color and Shape:
White Crystalline Powder
Molecular weight:
392.49
Ref: TM-T0696
| 1g | 68.00 € | ||
| 500mg | 46.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
LY2510924 acetate(1088715-84-7 free base)
Ly2510924 acetate is an potent and selective CXCR4 antagonist. It prevents the binding of SDF-1 …
Formula:
C64H91N13O13
Purity:
97.32%
Color and Shape:
Solid
Molecular weight:
1250.49
Ref: TM-T15805L
| 1mg | 156.00 € | ||
| 5mg | 300.00 € | ||
| 10mg | 449.00 € | ||
| 25mg | 735.00 € | ||
| 50mg | 1,006.00 € | ||
| 100mg | 1,389.00 € | ||
| 1mL*10mM (DMSO) | 725.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Prucalopride
CAS:179474-81-8
Prucalopride (R-93877), a selective 5-HT4A/4B agonist (Ki: 2.5/8 nM), is >290x more specific for these …
Formula:
C18H26ClN3O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
367.87
Ref: TM-T2542
| 10mg | 45.00 € | ||
| 25mg | 57.00 € | ||
| 50mg | 73.00 € | ||
| 100mg | 109.00 € | ||
| 200mg | 162.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Salmeterol
CAS:89365-50-4
Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
Formula:
C25H37NO4
Purity:
99.87% - 99.9%
Color and Shape:
Solid
Molecular weight:
415.57
Ref: TM-T12829
| 5mg | 54.00 € | ||
| 10mg | 86.00 € | ||
| 25mg | 151.00 € | ||
| 50mg | 270.00 € | ||
| 1mL*10mM (DMSO) | 77.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Blonanserin
CAS:132810-10-7
Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like …
Formula:
C23H30FN3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
367.5
Ref: TM-T1180
| 5mg | 42.00 € | ||
| 10mg | 57.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 127.00 € | ||
| 100mg | 174.00 € | ||
| 200mg | 300.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mizolastine
CAS:108612-45-9
Mizolastine (SL 850324), an antihistamine with IC50 of 47 nM, treats allergies like hay fever …
Formula:
C24H25FN6O
Purity:
98% - 99.77%
Color and Shape:
Solid
Molecular weight:
432.49
Ref: TM-T0118
| 10mg | 41.00 € | ||
| 25mg | 63.00 € | ||
| 50mg | 78.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 179.00 € | ||
| 500mg | 291.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Mianserin hydrochloride
CAS:21535-47-7
Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce …
Formula:
C18H21ClN2
Purity:
99.63% - 99.82%
Color and Shape:
White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film Coated
Molecular weight:
300.83
Ref: TM-T0783
| 1g | 152.00 € | ||
| 50mg | 35.00 € | ||
| 100mg | 41.00 € | ||
| 500mg | 104.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Urapidil hydrochloride
CAS:64887-14-5
Urapidil hydrochloride (Urapidil HCl) is 5-HT1A receptor agonist and an α1-adrenoceptor antagonist.
Formula:
C20H29N5O3·HCl
Purity:
99.93%
Color and Shape:
White Or Off-White Crystalline Powder
Molecular weight:
423.94
Ref: TM-T0088
| 1g | 132.00 € | ||
| 100mg | 45.00 € | ||
| 200mg | 60.00 € | ||
| 500mg | 90.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AM095 free acid
CAS:1228690-36-5
AM095 (free acid) is a potent LPA1 receptor antagonist (IC50s: 0.98 and 0.73 μM for …
Formula:
C27H24N2O5
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
456.49
Ref: TM-T10293
| 1mg | 39.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 83.00 € | ||
| 10mg | 119.00 € | ||
| 25mg | 209.00 € | ||
| 50mg | 349.00 € | ||
| 100mg | 542.00 € | ||
| 200mg | 782.00 € | ||
| 1mL*10mM (DMSO) | 91.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
