G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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Ezlopitant
CAS:147116-64-1
Ezlopitant (CJ-11974) is a small molecule neurokinin-1-receptor (NK1) antagonist used to treat nausea, vomiting and …
Formula:
C31H38N2O
Purity:
97.03%
Color and Shape:
Solid
Molecular weight:
454.65
Ref: TM-T68068
| 1mg | 91.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 729.00 € | ||
| 100mg | 1,013.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Misoprostol
CAS:59122-46-2
Misoprostol is a useful organic compound for research related to life sciences. The catalog number …
Formula:
C22H38O5
Purity:
100%
Color and Shape:
Water-Soluble Viscous Liquid
Molecular weight:
382.53
Ref: TM-T2573
| 1mg | 59.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 551.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
N,N′-Diferuloylputrescine
CAS:42369-86-8
N,N′-Diferuloylputrescine acts as a pigment inhibitor, showing a 57% reduction in pigmentation.
Formula:
C24H28N2O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
440.49
Ref: TM-T79996
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Losulazine
CAS:72141-57-2
Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.
Formula:
C27H22F4N4O3S
Purity:
99.80%
Color and Shape:
Solid
Molecular weight:
558.55
Ref: TM-T68095
| 1mg | 92.00 € | ||
| 5mg | 195.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 725.00 € | ||
| 100mg | 1,013.00 € | ||
| 500mg | 2,023.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
GPCR agonist-2
CAS:291528-35-3
GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.
Formula:
C10H10N2O4
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
222.2
Ref: TM-T60074
| 1ml | 34.00 € | ||
| 10mg | 35.00 € | ||
| 25mg | 47.00 € | ||
| 50mg | 60.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(S, R)-LSN 3318839
CAS:2765539-92-0
(S,R)-LSN 3318839 enhances GLP-1R, shows strong blood sugar lowering in animals, works with sitagliptin.
Formula:
C26H23Cl2N3O2
Purity:
99.57%
Color and Shape:
Soild
Molecular weight:
480.39
Ref: TM-T63166L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,268.00 € | ||
| 100mg | 1,699.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Octodrine
CAS:543-82-8
Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as …
Formula:
C8H19N
Purity:
99.98%
Color and Shape:
Clear Colorless To Light Yellow Liquid
Molecular weight:
129.24
Ref: TM-T0043
| 1g | 77.00 € | ||
| 5g | 166.00 € | ||
| 500mg | 51.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
PF-03382792
CAS:1400811-63-3
PF-03382792 is a small molecule 5-HT4 receptor activator for the study of Alzheimer's disease.
Formula:
C23H32FN3O4
Purity:
98.09%
Color and Shape:
Solid
Molecular weight:
433.52
Ref: TM-T33940
| 1mg | 224.00 € | ||
| 5mg | 558.00 € | ||
| 10mg | 794.00 € | ||
| 25mg | 1,189.00 € | ||
| 50mg | 1,635.00 € | ||
| 100mg | 2,192.00 € | ||
| 500mg | 4,419.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
(R)-CJ 11974
CAS:187281-35-2
(R)-CJ 11974: non-peptide NK1 receptor antagonist, may relieve pain and prevent chemo-induced vomiting.
Formula:
C31H38N2O
Purity:
97.03%
Color and Shape:
Soild
Molecular weight:
454.65
Ref: TM-T68068L
| 1mg | 182.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 591.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,706.00 € | ||
| 500mg | 3,418.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Adrenorphin
CAS:88377-68-8
Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C44H69N15O9S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
984.18
Ref: TM-T7567
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
DPTN dihydrochloride
CAS:325767-87-1
DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 …
Formula:
C22H20Cl2N4OS
Purity:
100%
Color and Shape:
Soild
Molecular weight:
459.39
Ref: TM-T72067
| 1mg | 50.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 162.00 € | ||
| 25mg | 339.00 € | ||
| 50mg | 524.00 € | ||
| 100mg | 738.00 € | ||
| 500mg | 1,557.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
D3R/MOR antagonist 1
Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and …
Formula:
C22H27Cl2N3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
420.38
Ref: TM-T78778
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
hNTS1R agonist-1
Compound 10, an hNTS1R agonist-1, acts as a full agonist with a strong affinity for …
Formula:
C37H62N10O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
790.95
Ref: TM-T78954
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Lintopride HCl
CAS:268548-31-8
Lintopride HCl is a 5HT-4 antagonist.
Formula:
C14H20Cl2N4O2
Purity:
97.70% - 98.42%
Color and Shape:
Soild
Molecular weight:
347.24
Ref: TM-T15760L
| 1mg | 96.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 292.00 € | ||
| 25mg | 493.00 € | ||
| 50mg | 713.00 € | ||
| 100mg | 998.00 € | ||
| 500mg | 2,004.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
CB2R agonist 3
CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value …
Purity:
98%
Ref: TM-T82769
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Isobutyryl-L-carnitine
CAS:25518-49-4
Isobutyryl-L-carnitine is a member of the class of compounds known as acylcarnitines. Isobutyryl-L-carnitine is a …
Formula:
C11H21NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
231.29
Ref: TM-T19381
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Adrenocorticotropic Hormone (ACTH) (4-10), human
CAS:4037-01-8
Adrenocorticotropic Hormone (ACTH) (4-10) is an agonist of potent melanocortin(MC4R) receptor .
Formula:
C44H59N13O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
962.09
Ref: TM-T7627
| 2mg | 52.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 226.00 € | ||
| 50mg | 293.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
LHRH
CAS:35263-73-1
Luteinizing hormone-releasing hormone (LHRH) is a neuropeptide produced in the hypothalamus that plays a pivotal …
Formula:
C55H74N16O14
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1183.27
Ref: TM-T80116
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 8 Oct 2024
BMS-903452
CAS:1339944-47-6
BMS-903452: potent GPR119 agonist, EC50 = 14 nM, treats rodent diabetes, no P450 inhibition, safe …
Formula:
C21H19Cl2FN4O4S
Purity:
100% - 100%
Color and Shape:
Solid
Molecular weight:
513.37
Ref: TM-T67791
| 1mg | 149.00 € | ||
| 1ml | 426.00 € | ||
| 5mg | 359.00 € | ||
| 10mg | 510.00 € | ||
| 25mg | 766.00 € | ||
| 50mg | 1,035.00 € | ||
| 100mg | 1,398.00 € | ||
| 500mg | 2,739.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
Semaglutide TFA (910463-68-2 free base)
Semaglutide TFA is a agonist of glucagon-like peptide-1 (GLP-1) receptor,with a potential for type 2 …
Formula:
NA
Purity:
98%
Color and Shape:
Solid
Molecular weight:
4210.63
Ref: TM-T12878
| 1mg | 219.00 € | ||
| 5mg | 758.00 € |
Estimated delivery in United States, on Tuesday 8 Oct 2024
