G-protein Coupled Receptors and 7-TM Receptors
G-protein coupled receptors (GPCRs) and 7-transmembrane (7-TM) receptors are a large family of membrane proteins that play key roles in cellular communication and signal transduction. These receptors are involved in a wide range of physiological processes, including sensory perception, immune response, and hormone regulation. GPCRs are major targets in drug discovery, making them essential for research in pharmacology and medicine. At CymitQuimica, we offer a comprehensive selection of high-quality reagents and compounds related to GPCRs and 7-TM receptors to support your research and drug development efforts.
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G-Protein antagonist peptide acetate
G-Protein antagonist peptide acetate is a truncated substance P-related peptide, competes with receptor for G …
Formula:
C59H68N12O11S
Purity:
98.06%
Color and Shape:
Solid
Molecular weight:
1153.33
Ref: TM-TP1902L1
| 1mg | 134.00 € | ||
| 2mg | 217.00 € | ||
| 5mg | 341.00 € | ||
| 10mg | 540.00 € | ||
| 25mg | 853.00 € | ||
| 50mg | 1,161.00 € | ||
| 100mg | 1,570.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Valorphin
CAS:144313-54-2
Valorphin (Valorphin TFAsalt) has opioid analgesic activity, binds to rat mu-opioid receptor, with an IC50 …
Formula:
C44H61N9O11
Purity:
98%
Color and Shape:
Solid
Molecular weight:
892.01
Ref: TM-T7306
| 2mg | 79.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 438.00 € | ||
| 100mg | 656.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
AC-264613
CAS:1051487-82-1
AC-264613 is an agonist of the GPCR protease-activated receptor 2 (PAR2). AC-264613 suppresses interferon regulatory …
Formula:
C19H18BrN3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
400.28
Ref: TM-T4186
| 1mg | 92.00 € | ||
| 5mg | 275.00 € | ||
| 10mg | 506.00 € | ||
| 25mg | 1,148.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
NPC 567 acetate
NPC 567 acetate is a bradykinin B2 antagonist and can be used in studies about …
Formula:
C62H91N19O15
Purity:
97.72%
Color and Shape:
Liquid
Molecular weight:
1342.5
Ref: TM-T21060L
| 1mg | 182.00 € | ||
| 5mg | 406.00 € | ||
| 10mg | 600.00 € | ||
| 25mg | 920.00 € | ||
| 50mg | 1,290.00 € | ||
| 100mg | 1,728.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BMY-14802
CAS:105565-56-8
BMY-14802 (alpha-(4-fluorophenyl)-4-(5-fluoro-2-pyrimidinyl)-1-piperazine butanol) is a selective and orally active sigma-1 antagonist with an IC50 of …
Formula:
C18H22F2N4O
Purity:
98.93%
Color and Shape:
Soild
Molecular weight:
348.39
Ref: TM-T67739
| 1mg | 40.00 € | ||
| 5mg | 89.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 267.00 € | ||
| 50mg | 437.00 € | ||
| 100mg | 645.00 € | ||
| 500mg | 1,327.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Latanoprost acid
CAS:41639-83-2
Latanoprost acid is a prostanoid receptor agonist that blocks RANKL and can be used to …
Formula:
C23H34O5
Purity:
96.97%
Color and Shape:
Pale Yellow Oil
Molecular weight:
390.51
Ref: TM-T15718
| 1mg | 56.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 220.00 € | ||
| 25mg | 440.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 897.00 € | ||
| 200mg | 1,190.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
PIT
CAS:56583-49-4
PIT (2,2'-Pyridylisatogen tosylate) is a specific and non-competitive antagonist of the Purinergic receptor P2Y1 with …
Formula:
C20H16N2O5S
Purity:
99.01%
Color and Shape:
Solid
Molecular weight:
396.42
Ref: TM-T23164
| 5mg | 40.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 183.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Drinabant
CAS:358970-97-5
Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.
Formula:
C23H20Cl2F2N2O2S
Purity:
99.8%
Color and Shape:
Solid
Molecular weight:
497.38
Ref: TM-T21861
| 1mg | 85.00 € | ||
| 2mg | 114.00 € | ||
| 5mg | 171.00 € | ||
| 10mg | 254.00 € | ||
| 25mg | 416.00 € | ||
| 50mg | 585.00 € | ||
| 100mg | 791.00 € | ||
| 500mg | 1,588.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
![[D-Ala2]leucine-enkephalin acetate](https://static.cymitquimica.com/products/TM/thumb/TP1367L.jpg)
[D-Ala2]leucine-enkephalin acetate
[D-Ala2]leucine-enkephalin acetate ([D-Ala2]leucine-enkephalin acetate (64963-01-5 free base)) is a delta opioid agonist used to study …
Formula:
C31H43N5O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
629.65
Ref: TM-TP1367L
| 5mg | 55.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 99.00 € | ||
| 50mg | 160.00 € | ||
| 100mg | 232.00 € | ||
| 200mg | 349.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Neurokinin A(4-10)
CAS:97559-35-8
Neurokinin A(4-10)(TFA) is an agonist of tachykinin NK2 receptor .
Formula:
C34H54N8O10S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
766.91
Ref: TM-T7559
| 1mg | 123.00 € | ||
| 5mg | 243.00 € | ||
| 10mg | 427.00 € | ||
| 25mg | 850.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BIMU 8
CAS:134296-40-5
BIMU 8 is a selective agonist of 5-HT4 with EC50s of 18 nM, 77 nM, …
Formula:
C19H27ClN4O2
Purity:
99.36%
Color and Shape:
Solid
Molecular weight:
378.9
Ref: TM-T21946
| 1mg | 88.00 € | ||
| 5mg | 169.00 € | ||
| 10mg | 244.00 € | ||
| 25mg | 410.00 € | ||
| 50mg | 601.00 € | ||
| 100mg | 854.00 € | ||
| 500mg | 1,734.00 € | ||
| 1mL*10mM (DMSO) | 184.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Eledoisin
CAS:69-25-0
Eledoisin (Eledone peptide) is a specific agonist of NK2 and NK3 receptors.Eledoisin is an undecapeptide …
Formula:
C54H85N13O15S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1188.4
Ref: TM-TP1177
| 1mg | 204.00 € | ||
| 5mg | 797.00 € | ||
| 10mg | 1,394.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Licoarylcoumarin
CAS:125709-31-1
Licoarylcoumarin inhibits cAMP phosphodiesterase, fights VRE bacteria, has anti-HIV properties, and blocks xanthine oxidase.
Formula:
C21H20O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
368.38
Ref: TM-TN4433
| 5mg | 850.00 € | ||
| 1mL*10mM (DMSO) | 869.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
UCM-1306
CAS:2258608-78-3
UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive …
Formula:
C14H14FNO2S
Purity:
100%
Color and Shape:
Soild
Molecular weight:
279.33
Ref: TM-T67729
| 1mg | 36.00 € | ||
| 5mg | 78.00 € | ||
| 10mg | 112.00 € | ||
| 25mg | 218.00 € | ||
| 50mg | 324.00 € | ||
| 100mg | 464.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
BMS-903452
CAS:1339944-47-6
BMS-903452: potent GPR119 agonist, EC50 = 14 nM, treats rodent diabetes, no P450 inhibition, safe …
Formula:
C21H19Cl2FN4O4S
Purity:
100% - 100%
Color and Shape:
Liquid
Molecular weight:
513.37
Ref: TM-T67791
| 1mg | 149.00 € | ||
| 5mg | 359.00 € | ||
| 10mg | 510.00 € | ||
| 25mg | 766.00 € | ||
| 50mg | 1,035.00 € | ||
| 100mg | 1,398.00 € | ||
| 500mg | 2,739.00 € | ||
| 1mL*10mM (DMSO) | 426.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Adrenorphin
CAS:88377-68-8
Adrenorphin (Metorphamide)(3TFA) is an agonist of μ-opioid receptor(Ki :12 nM).
Formula:
C44H69N15O9S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
984.18
Ref: TM-T7567
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Monday 16 Dec 2024
Octodrine
CAS:543-82-8
Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as …
Formula:
C8H19N
Purity:
99.98%
Color and Shape:
Clear Colorless To Light Yellow Liquid
Molecular weight:
129.24
Ref: TM-T0043
| 1g | 77.00 € | ||
| 5g | 166.00 € | ||
| 500mg | 51.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
GPCR agonist-2
CAS:291528-35-3
GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.
Formula:
C10H10N2O4
Purity:
99.94%
Color and Shape:
Liquid
Molecular weight:
222.2
Ref: TM-T60074
| 10mg | 35.00 € | ||
| 25mg | 47.00 € | ||
| 50mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
Misoprostol
CAS:59122-46-2
Misoprostol is a useful organic compound for research related to life sciences. The catalog number …
Formula:
C22H38O5
Purity:
100%
Color and Shape:
Water-Soluble Viscous Liquid
Molecular weight:
382.53
Ref: TM-T2573
| 1mg | 59.00 € | ||
| 5mg | 181.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 551.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Formula:
C141H221N33O42S
Purity:
96.52%
Color and Shape:
Liquid
Molecular weight:
3082.52
Ref: TM-T38193L
| 1mg | 111.00 € | ||
| 2mg | 157.00 € | ||
| 5mg | 240.00 € | ||
| 10mg | 355.00 € | ||
| 25mg | 542.00 € | ||
| 50mg | 758.00 € | ||
| 100mg | 1,016.00 € | ||
| 200mg | 1,354.00 € |
Estimated delivery in United States, on Monday 16 Dec 2024
